CURRICULUM VITAE VOMMIMA V. SURESHBABU Bangalore … · 2018-09-14 · including native chemical ligation; Development of new synthetic methods Academic assignment : Served as sectional

CURRICULUM VITAE VOMMIMA V. SURESHBABU

Professor in Chemistry Department of Chemistry

Central College Campus

Bangalore University Bangalore-560001, India Ph: + 91 080 22961339

Mob: 08147757961

Email: [email protected], [email protected];

[email protected] Residential Address: Golden Grand, FB 1504,Tumkur Road,

Yeshwanthapur, Bangalore- 560 022, Karnataka,

India Personal

Indian

Male

Married

Birth: 14-07-1961

EDUCATION

Ph.D. Organic chemistry (Peptide chemistry) Bangalore University, 1990.

M.Sc. Chemistry (Organic) S. K. University, Ananthapur, A.P. 1981-83.

B.Sc Chemistry S. V. University, Tirupathi, A.P. 1978-81.

Positions held:

Position Date of Appointment Duration

Research Assistant 24-07-1985 5 Years Bangalore university

Lecturer 11-06-1990 5 years Bangalore university

Sr. Lecturer 11-06-1995 3 years Bangalore university

Reader 01-07-1998 8 years Bangalore university

Professor 01-07-2006 till date Bangalore university

mailto:[email protected]

mailto:[email protected]

Courses Teaching MSc (Chemistry-Organic ), B.E. (1st and 2nd Semester Chemistry).

Research Interest :: Organic Chemistry; Chemistry of Peptides and Peptidomimetics

including native chemical ligation; Development of new synthetic

methods

Academic assignment : Served as sectional president for organic chemistry in

XXXIV -I CC 2017. Awards

Sl. Year Name of award Awarded by

No.

1) 1981-83 National merit scholarship Government of Andhra Pradesh 2) 1983 Junior Research Fellowship Council of Scientific & Industrial

(based on NET examination) Research

3) 1993 Young scientist in organic chemistry Indian Council of Chemists 4) 1993-94 Visiting Summer Fellowship (short Jawaharlal Nehru Center for

term) Advanced Studies, Bangalore

(to work at NCL, Pune) 5) 2001 Professor D. K. Banerjee Memorial Dept. of Organic Chemistry,

Lecture award I.I.Sc., Bangalore (The first

recipient) 6) 2001 The Overseas Associate ship Award Dept. of Biotechnology,

(short term) Govt. of India 7) 2001 Sir C. V. Raman Young Scientist Govt. of Karnataka

Award in

Chemical Sciences 8) 2002 Young Scientist Award in Chemical Karnataka Association for the

Sciences for the year Advancement of Science, Bangalore 9) 2005 Professor S. Siddappa 60th birthday Dept. of Chemistry, Karnatak

commemorative lecture University, Dharwad

10) 2008 CRSI Bronze medal CRSI, Bangalore, India

11) 2009 Prof. Wadia Lecture award University of Pune, Pune

12) 2010 Best research Publication award for

the paper “Chiral N-Fmoc-â-amino

alkyl isonitriles derived from amino

acids- first synthesis and application

in 1-substituted tetrazoles synthesis”

Vision group on Science and

Technology, Govt. of Karnataka

Tetrahedron Letters Most cited paper award for the period 2005-2008 for the paper

entitled “Protonated chiral prolinamide catalyzed enantioselective direct aldol reaction in

water”(Chimni, S. S., Mahajan, D., Sureshbabu, V. V., Tetrahedron Lett., 2005, 46(34), 5617).

Selected to visit UK under bilateral exchange programme from Indian National

Science Academy, New Delhi (2008-2009).

Ongoing/completed project details with funding agency, funding, time frame and title Granting Title of the project and Reference Duration Amount Status agency number & in Rs.

Period

1. DST Studies on glycoopioid peptides related to 1992- 1996 5,80,800 Completed

dermorphin 2. CSIR Studies on the solid phase synthesis of 1992 - 1995 5,39,833 Completed

glycoopioid peptides

3.Jupiter Preparation of industrially useful peptides 2000-2001 50,000 Completed

Org. Ltd

4. DST Studies on chemical synthesis of peptides :

Coupling methods for the incorporation of 2001 - 2004 21,26,134 Completed

non-coded amino acids into peptides

5. CSIR Exploration of synthetically useful Bsmoc

group in solid phase synthesis of 2002- 2005 6,47,500 Completed

cyclosporine

6. DBT Studies on chemical synthesis of partially

modified Retro-Inverso peptides and June 2004- 9,70,000 Completed Peptidyl ureas: Exploration of Urethane June 2007

type protecting groups

7. DST Studies on chemical synthesis of

Ureidopeptides: Ná-Fmoc-peptide 2005- 2008 31,89,000 Completed isocyanates as building blocks for

incorporation of urea and thiourea moieties

as a replacement of amide bond into

peptides

8. CSIR Studies on chemical synthesis of

Peptidomimetics: Protected â-amino 2006 - 2009 11,16,120 Completed alkoxy carbonyl chlorides/ carbonates as

monomeric building blocks for the

incorporation of carbamate and carbonate

moieties

9. UGC Studies on chemical synthesis of peptides: 2006 - 2009 7,68,600 Completed

Incorporation of amino group and

carbohydrate at the â/ã position of Asp/Glu 10. DST Studies on chemical Synthesis of peptides: 2008 - 2011 57,38,800 Completed

Synthesis of backbone modified

peptidomimetics and peptidyl conjugates

through Ugi multi-component reactions

and click chemistry protocols

11. CSIR Synthesis of unnatural amino acids, 2009 - 2012 14,00,000 Completed

peptidomimetics and neoglycopeptides;

Insertion of aromatic heterocycles,

thioureido and selenoamide/carbamate

linkages as peptide/amide bond surrogates

12. UGC Studies on chemical synthesis of 2009-2012 9,76,800 Completed

peptimimetics: Synthesis of novel N-

protected amino alkyl sulfamoyl chlorides

and thiocyanates: insertion of sulfamide,

methylamine, tetrazole, imidazoles and

pyrazole as peptide bond/carboxylic group

isosteres 13. DST- Studies on chemical synthesis of 2009-2012 41,40,400 Completed Nano peptidomimetics based self-assembling

mission organic nano-tubes and application of

carbon nanotubes in peptidomimetic

synthesis

14. DBT A structure-function correlation study to 2010-2013 50,00,000 Completed

unravel the mechanism of action of human

catestatin

(a join collaboration project with Dr.

Nithish Mahapatra, IIT, Chennai

15. Studies on chemical synthesis of 2011-2014 40,70,000 Completed

BRNS selenopeptides, selenoamide/selenourea

linked glycosylated amino acids, insertion

of selenocarboxamide, selenourea and

[CH2SeH] moieties as carboxy group

replacement

16. Studies on chemical synthesis of 2012-2015 55,00,000 Completed

DST

peptidomimetics: Insertion of guanide and

some hybrid tethers in peptide back bone:

preparation of diverse classes of peptoids

and phosphonopeptides

17. Peptides, peptidomimetics based 2012-2015 63,34,000 Completed

hydrogelators and organogelators;

DST- Magnetically separable metal

Nano nanocatalysts, peptidic catalysts and their

mission application in organic, peptide and

peptidomimetics synthesis.

18. CSIR Studies on chemical synthesis of 2013-2017 20,48,000 Completed

peptidomimetics and application of native

chemical ligation for polypeptides

synthesis.

19. UGC Studies on Chemical Synthesis of 2015-2018 15,04,600 Completed

Peptidomimetics: Synthesis of novel

fluorescent amino acids/peptides,

iminohydantoin tethered peptides; Novel

approaches for the insertion of

sulfonamidotetrazoles, amino tetrazoles

and imides into peptide back bone.

20. DST-

Nano

Peptides, peptidomimetics based

hydrogelators and organogelators;

2015-2018 69,41,600 In progress

magnetically separable metal

nanocatalysts, peptidic catalysts and their

application in organic, peptide and

peptidomimetic synthesis

21. DST-

SERB

Studies on chemical synthesis of

peptidomimetics: Phosphonopeptides and

other phosphorous-containing

peptidomimetics, heterocyclic

peptidomimetics, peptidomimetics using

multicomponent reactions

2017-2020 53,53,480 In progress

UGC support under BSR scheme

UGC-BSR Duration Amount in Status

Rs.

One time 2 years 7,50,000 2015

assistance for

strengthening

infracture

Coordinator for departmental project

Granting agency Duration Amount in Rs. Status

DST-FIST

5 years 114.50 lakhs Completed

Research funds obtained in the form of fellowships

No Name of the Student Type of Funding Amount Period

Fellowship Agency utilized

(Rs)

1. Ananda K SRF CSIR 1,79,718 03-10-1999 to

31-10-2001 2. Basanagoud S. Patil SRF CSIR 2,72,245 02-05-2003 to

31-03-2005

22. Synthetic and Biological Peptides: A proposal submitted to INDO-US

INDO- Strategies for developing Drugs, Vaccines, Science and Technology Forum, New

US Biologicas and Materials Delhi (IUSSTF) for arranging a INDO- US international work-shop. Proposed Budget: USD 73,600/- (approx: Rs.

35,32,800/-; sanctioned and not utilized)

3. Kantharaju SRF CSIR 2,84,080 01-04-2004 to 31-03-2006 4. Ramanrao R. V. NET-JRF- CSIR 5,83,728 7-1-2003 to

SRF 31-10-2007

5. G. Chennakrishnareddy SRF CSIR 2,13,200 1-4-2008 to

Resea

rch

guidance

1. Ph.D supervised: awarded: 24; pursuing: 06

Sl. No Name of the Title of the thesis Year of

candidate award

1 H. N. Gopi Applications of some new techniques and 2000

reagents in the synthesis of a -and â-peptides

2 K. Ananda New synthetic routes to â-amino acids and 2001

(CSIR-SRF)

coupling methods for the incorporation of

non-coded amino acids into peptides

3 G.R.Vasantha Studies on chemical synthesis of peptides 2005

kumar

:Efficient Synthetic Methods for â-Amino Acids,

Azides, Amino Acids Hydroxamates and Esters

31-8-2010 6. N. Narendra SRF CSIR 2,13,200 1-4-2010 to

10-5-2010 7. Dr. Ravi S. Lamani Dr. Kothari UGC 8,24,000 15-05-2009 to

Post 14-05-2011 doctoral

Fellowship 8. Madhu C. JRF UGC 13,98,200 30-09-2009 to

29-09-2014 9. Panduranga V. JRF CSIR 14,37,400 26-10-2010 to

25-10-2015 10. Sharanabai K. M. DST- DST 12,65,013 19-04-2011 to

INSPIRE 18-04-2016 11. Vishwanatha T. M. SRF CSIR 11,40,000 01-04-2012 to

31-03-2015 12. Basavaprabhu SRF CSIR 9,02,400 01-04-2013 to

31-03-2016 13 Nageswara Rao P SRF CSIR 9,02,400 01-10-14 to

30-9-17

4 Basanagoud S.

Patil

CSIR-SRF

Studies on chemical synthesis of Peptidomimitics: Synthesis, Characterization and stability of Isocyanates of Fm

amino acids/peptides & their utility in the synthesis of

acids andacetylation of sugars

2006

5 Kantharaju Studies on chemical synthesis of peptidyl ureas, 2007

(CSIR-SRF)

â-amino acids and development of new eco-friendly reaction

6 S. J. Tantry Exploration of new synthetic routes and reagents in 2007

peptide synthesis: Peptides containing both natural and

unnatural amino acids

7 R. V. Ramana Applications of Curtius rearrangement in synthesis 2008

Rao of retro-inverso peptides, peptidyl ureas, unnatural

(CSIR-SRF) amino acids, neoglycopeptides and use of oxazolidin-

ones in the synthesis of N-glycosylated amino acids

8 Sudarshan N. S. Studies on synthesis of N-Fmoc-N’-formyl gem- diamines, 2009

Fmoc/Bsmoc ureidopeptides and new coupling reagents

and methods for peptide synthesis

9 Shankar A. Studies on chemical synthesis of thioureido linked 2010

Naik peptidomimetics, unnatural amino acids containing aromatic

heterocylces, and selenocarbamates

10 Chennakrishna Studies on Synthesis of isoselenocyanates and their 2010

-reddy, G application to the preparation of selenoureido

CSIR-SRF peptidomimetics; new routes to ureido and

thioureidopeptides and development of new co-coupling

agent for peptide synthesis

11 Hemantha, Studies on chemical synthesis of peptidomimetics: 2011

H. P. protected â-aminoalkoxy carbonyl chlorides /

carbonates as monomeric building blocks for the

incorporation of carbamate and carbonate moieties

in to unnatural peptides

12 Nagendra, G Studies on Chemical Synthesis of Peptidomimetics: 2011

Mimetics Related to Endothiopeptides, Peptide

Heterocycles, Selenoureidopeptides and Urea Linked

Glycosylated Amino Acids

13 Lalithamba, Studies on the Application of Coupling Agents for the 2012

H. S Synthesis of Acyl Azides, Ureas, Carbamates; Preparation

of Trithiocarbonate-Linked Peptidomimetics; Selenazoles

derived from Amino Acids and Peptide Synthesis through

Click Approach

14 Narendra, N Chemical synthesis of peptidomimetics: Studies on 2014

CSIR-SRF synthesis of N-Fmoc-â-amino alkyl isonitriles and their

synthetic applications; amino acid analogues and

dipeptitomimetics containing thiazole units; carbon

nanotubes conjugates of á-ureidopeptides and new

methods to á-ureidopeptidses

15 Vasantha B Studies on chemical synthesis of peptidomimetics: 2014

N-protected amino alkyl thiocyanates and selenocyanates

and their utility in the synthesis of S- and Se-linked

tetrazoles 16 Vishwanatha Unnatural amino acids and back bone modified peptides: 2014

T. M. Novel synthetic strategies for selenoxopeptides, chiral

CSIR-SRF â–amino alkyl thiols, chiral â–amino alkyl isonitriles and

their applications for the synthesis of peptidomimetics 17 Basavaprabhu Studies on Chemical Synthesis of Peptidomimetics: 2014

CSIR-SRF Synthesis and characterization of guanidine tethered

peptidomimetics, urea tethered glycosylated amino acids,

Ná-protected amino acid azides and their application for

ureidopeptide synthesis and application of Ritter reaction

to the synthesis of di

and trisusbstituted ureas 18 Madhu Ch. Studies on chemical synthesis of peptidomimetics: 2014

UGC-JRF/SRF Click chemistry aided insertion of 1,2,3-triazoles into

neoglycopeptides 19 Samarasimha

Reddy Studies on chemical synthesis of peptides and

peptidomimetics: human catestatin and its analogues and application of

Pd(0)/PVC nanoparticles for Suzuki cross-coupling

reaction

2014

20 Nageshwara

Rao. P

CSIR-SRF

Studies on chemical synthesis of peptidomimetics:

Synthesis of selenocysteine, chiral β-amino diselenides,

seleninic acids; amino acid azides, ureidopeptides and

amino/peptide hydroxamic acids

2015

21 Veladi

Panduranga

CSIR-JRF/SRF

Studies on chemical synthesis of peptidomimetics: Novel

synthetic strategies for the synthesis of thioxo peptides and

imide tethered mimetics; New methodologies for the

synthesis of dibenzyl-diselenides, disulfides and

application of Ritter reaction to the synthesis of

disusbstituted ureas

2016

22 Girish Prabhu Studies on chemical synthesis of peptidomimetics:

Synthesis of 2-amino-1,3,4-oxadiazoles, 2-

aminohydantoins, and 1,5-disubstituted tetrazoles by

desulfurization/deselenization chemistry

2016

23 Krishnamurthy

M

Studies on chemical synthesis of peptides and

peptidomimetics: Iodine-mediated oxidative peptide bond

formation; Insertion of S-linked 1,3,5-triazine and

dithiocarbonate moieties into peptides

2017

24 Sharnabai. K.

M.

DST-Inspire

fellowship

Studies on chemical synthesis of peptidomemitics:

Synthesis of amino acid derived sulfonyl azides,

cyanomethyl ketones and Weinreb amides and their

applications for the synthesis of novel peptidomimetics

2017

Ph.D pursuing: 05

Sl. Name of the Title of the thesis Year of

No. candidate joining 1 Santhosh L STUDIES ON CHEMICAL SYNTHESIS OF

PEPTIDOMIMETICS: SYNTHESIS OF 1, 5-DISUBSTITUTED TETRAZOLES AND 2-AMINOHYDANTOINS DERIVED FROM AMINO ACID AMIDES/PEPTIDES

2015

2 Roopesh

Kumar L STUDIES ON CHEMICAL SYNTHESIS OF PEPTIDOMIMETICS: NOVEL SYNTHETIC ROUTES FOR THE SYNTHESIS OF THIOUREIDOPEPTIDES EMPLOYING DITHIOCARBAMATES AND AMIDINES USING TPP-I2 SYSTEM AS DEHYDRATING AGENT

2016

3 Sagar N. R STUDIESON CHEMICAL SYNTHESIS OF

PEPTIDOMIMETICS:SYNTHESIS OF

UNSYMMETRICAL /SYMMETRICAL PEPTIDYL

UREAS AND N-ACYL SULFONAMIDE

PEPTIDOMIMETICS

2016

4 Shekharappa STUDIES ON CHEMICAL SYNTHESIS OF PEPTIDOMIMETICS: SYNTHESIS OF Se-TRIAZOLE/TETRAZOLE LINKED GLYCOSYL AND N- PROTECTED AMINO ACIDS

2015

5 Vathsala. U STUDIES ON CHEMICAL SYNTHESIS OF PEPTIDES

AND AMINO ACID DERIVATIVES: SYNTHESIS OF PEPTIDES VIA Nα-PROTECTED DIACYLDISELENIDES; ANILIEDS FROM THIOACIDS; AMINO HYDROXAMIC ACIDS AND THIOUREAS FROM DITHIOCARBAMATE AND AROMATIC ALKYL AZIDE

2015

6 C. Srinivasulu STUDIES ON CHEMICAL SYNTHESIS OF

PEPTIDOMIMETICS: SYNTHESIS OF N-

ACYLPHOSPHORAMIDE TETHERED

PEPTIDOMIMETICS, N- AMINO/ N-HYDROXY

PEPTIDES THROUGH UGI-MULTI COMPONENT

REACTION

2016

2. M.Phil supervised: 03

Sl. No. Name of the Candidate Title of the Dissertation Year of award 1 H.N.Gopi Rapid synthesis of short peptide 1996

fragments mediated by KOBt and KOAt

2 Smt. K. Gayatri Fmoc amino acid chlorides/ AgCN as 1997

coupling agent in peptide synthesis

3 K.Ananda Synthesis of peptides containing á, á- 1998

dialkyl amino acids using KOBt

Conference, Seminar organized-

No Description Date Sponsoring agency 1 Advances in Science and Technology& Global 31st March, Bangalore University,

Higher Education Scenario organized by 2004 Bangalore and Queensland

Bangalore University and Queeensland University, Australia. University, Australia, at Central College,

Bangalore.Organizers: Prof. Katre. S.,

Sureshbabu, V. V. and Dr. P. G. Siddeshwar 2 Intel Science Talent Discovery Fair. 6th Dec, Intel Innovation in India

Local Coordinator: Sureshbabu V. V. 2005 3 In-House Symposium in Chemistry & 26th, 27th UGC-DRS

Biochemistry, Dept. of Chemistry, Central Dec, 2005

College, Bangalore University.Convener:

Sureshbabu, V. V. 4 Workshop on research projects: Conception to 6th Nov Bangalore University

execution for young faculties of Bangalore 2006

University. A training programme for teachers.

Organizers: Sureshbabu V. V. and P. V. Kamath 5 National Conference in Chemistry, Central

College, Bangalore University

Conveners: Sureshbabu, V. V. and P. V. Kamath

27-29, Sep, 2007

DST, CSIR, DIST, ICMR, ISRO, INCASR

6 UGC-DRS Seminar, Dept. of Chemistry, Central 28th, 29th UGC-DRS

College,Bangalore University. Feb, 2008

Convener: Sureshbabu, V. V. 7 DST PAC meeting (Organic Chemistry) at Dept. 8th & 9th DST

of Chemistry, Central College,Bangalore Aug, 2009

University

Local Organizers: Sureshbabu, V. V. and P. V.

Kamath 8 DST PAC meeting (Physical chemistry) at Dept 24-25, July, DST

of Chemistry, Central College, Bangalore 2008

University.

Local Organizers: P. V. Kamath and Sureshbabu 9 Indian Peptide Society, Special Lecture 8th Feb, Jupiter Biosciences Ltd,

programme, Dept. of Chemistry, Central 2008, Hyderabad. College,Bangalore University. Local Organizer: Bio Concept, New Delhi

Sureshbabu V. V. 10 Prof. K. M. Shivanandaiah 75th Birthday Annual Convener : V . V.

Commemorative Lecture Programme event since Sureshbabu & P. V.

2007 Kamath 11 Frontier Lectures in Bio-organic Chemistry 28th & 29th Indian Academy of

Convener : V. V. Sureshbabu May Sciences, Bangalore; 2009 Indian National Science Academy, New Delhi; The National Academy of

Sciences, Allahabad 12 Current trends in organic synthesis April Convenor : Prof. S.

Co- ordinators : V.V Sureshbabu & P. V. Kamath 9&10th 2010 Chandrasekaran IISc

Bangalore 13 DST PAC meeting (Organic Chemistry) at Dept. August 22- DST

of Chemistry, Central College,Bangalore 24, 2013

University

Local Organizer: Sureshbabu, V. V.

14.

DST SCIENCE CAMP UNDER INSPIRE

INTERNSHIP SCHEME

June 23-27,

2015 DST

15.

DST SCIENCE CAMP UNDER INSPIRE

INTERNSHIP SCHEME

November 8-

12, 2016

DST

FOREIGN COUNTRIES VISITED ON ACADEMIC ASSIGNMENTS:

Sl. Name of Purpose Year Sponsoring agency

No. the

Country 1 Dept. of Synthesis of biotinylated analogs of 2001 Dept. of

Chemistry, tridecapeptide á-factor mating Biotechnology, City pheromone of Saccharomyces cerevisiae New Delhi

University, ii. Synthesis and biophysical

NewYork analysis on a trans membrane PCR T-40

fragment.

2

Dept. of Chemistry,

i. Synthesis of Ste2p (á- factor receptor) of Saccharomyces cerevisiae- a G 2002-2003

NIH project sanctioned to Prof.

City protein-coupleled receptor (GPCR) & its Freid Naider by the University, fragments by Native Chemical Ligation US Govt. NewYork ii. Synthesis and biophysical studies of

sixth membrane domain of Ste 2p-four

M62K peptides-each one-33 amino acid

residues

iii. Synthesis of phosphorpeptides

iv. Synthesis of chemokine

receptor-CCR5 peptide and analysis

Details of talks delivered in Japan:

Sl. Date Place Title of Topic

No.

1 27th 42nd Japanese Ná-Fmoc-peptide isocyanates and

Oct. Peptide their utilization in synthesis of

2005

Symposium, ueidopeptides and retro-inverso

Osaka peptides

2 31st Institute for Isocyanates of Ná-Fmoc-amino

Oct. Protein Research, acids and their utility in the

2005 Osaka University, synthesis of peptidomimetics

Osaka

4th International Peptide Symposium in conjunction with the 7th Australian Peptide Conference

and the 2nd Asia-Pacific International Peptide Symposium,Cairns, Queensland, Australia, Oct

21-25, 2007.

Book Chapter “Protection Reactions” to the text book “Amino acids, Peptides and Proteins in Organic

Chemistry” Vol. 4. Protection Reactions, Combinatorial and Medicinal Chemistry: Edited by Prof.

Andrew Hughes, published by the Wiley Publishers, V. V. Sureshbabu,* and N. Narendra. Page

numbers 1-9

Review Articles

Thioacids – synthons for amide bond formation and ligation reactions: assembly of

peptides and peptidomimetics, Narendra. N, Vishwanatha. T. M, Basavaprabhu. H,

Girish prabhu, L. Roopesh Kumar, and V. V. Sureshbabu,

Org. Biomol. Chem., 2018, 16, 3524.

Amino acid fluorides: viable tools for the synthesis of peptides, peptidomimetics and

enantiopure heterocycles, Girish prabhu, N. Narendra, Basavaprabhu, V. Panduranga

and V. V. Sureshbabu, RSC Advances, 2015, 5, 48331.

Amino acid chlorides: a journey from instability and racemization toward broader utility

in organic synthesis including peptides and their mimetics, Girish prabhu, Basavaprabhu,

N. Narendra, T. M. Vishwanatha and V. V. Sureshbabu, Tetrahedron, 2015, 71, 2785.

Propanephonic acid anhydride (T3P) – A benign reagent for diverse applications inclusive

of large-scale syntheis, Basavaprabhu, T. M. Vishwanatha, Nageswara Rao Panguluri and

V. V. Sureshbabu, Synthesis, 2013, 45, 1569.

Total chemical synthesis of polypeptides and proteins: Chemistry of ligation techniques

and beyond, H. P. Hemantha., N. Narendra, and V. V. Sureshbabu, Tetrahedron, 2012, 68,

9491. General articles

Ø V. V. Sureshbabu and M. N. Palgunachari, 25years of peptide research in Central

College, Bangalore University, Bangalore, in Peptides: Design, Synthesis and Biological

Acitivity, (Ed. Chenna Basava and G. M. Anantharamaiah), Birkhauser, Boston, 1994, 1-

10. Ø V. V. Sureshbabu, One hundred years of peptide chemistry, Resonance,

Vol.16, No.7, p.640, 2011 [Reprinted (with modifications from Resonance, Vol.6, No.10,

p.68, 2001] Ø V. V. Sureshbabu and H. P. Hemantha, Native Chemical Ligation: An ultimate tool for

chemical synthesis of proteins, Jupiter Group Silver Jubilee report, 2010, 44-52.

Ø V. V. Sureshbabu, N. Narendra and G. Chennakrishnareddy, Peptide drugs : Current

scenario and future prospects, Dr. G. Narayan Felicitation volume, published by

Karnataka Association for the Advancement of Science, Bangalore, 2008.

Research papers: 215 published

216 Santhosh. L, Shekarappa,

Roopesh Kumar. L and V.

V. Sureshbabu

Synthesis of Carbodiimides from

1, 3-Disubstituted Selenoureas by

Iodine-Mediated Deselenization

Indian J. Chem. Sect. B

(in press)

215 U. Vathsala, Roopesh

Kumar. L, Sagar N. R, M.

Mahesh, P.

Venkataramana and V. V.

Sureshbabu

Peptide Bond Formation via Nα-

Protected Diacyldiselenides Int J Pept Res Ther.,

2018, DOI:

10.1007/s10989-018-

9711-z

214 Santhosh L, Shekarappa,

Krishnamurthy M, V V.

Sureshbabu

A convenient synthesis of

enantiomerically pure α-

isocyanato esters & Nβ-fmoc –

amino alkyl isonitriles derived

from α-amino acids employing

PPh3/I2

Indian J Chem. Sect. B

accepted in 2018

213 Santhosh. L, Durgamma. S,

Shekharappa and V. V.

Sureshbabu

Staudinger/aza-Wittig reaction to

access Nβ-protected amino alkyl

isothiocyanate

Org. Biomol. Chem.,

2018, 16, 4874

212 Santhosh. L, Srinivasulu.

C, Durgamma. S, Girish

Prabhu, V. V. Sureshbabu

Facile one-pot synthesis of 2-

amino-1,3,4-oxadiazole tethered

peptidomimetics by molecular-

iodine-mediated

cyclodeselenization

New J. Chem., 2017, 41,

11225-11229

211 Girish prabhu,

Krishnamurthy M,

Samarasimha Reddy M,

Narendra N, V V.

Sureshbabu

Design and synthesis of a novel N-

(1H-tetrazol-5-yl)methyl cyclic

peptoid using Nosyl-protected N-

(1-trityl-1H-tetrazol-5-yl)methyl

substituted glycine

Int J Pept Res Ther.,

2017, 23, 493

210 Roopesh Kumar, Sagar N.

R, Shekharappa,

Montmorillonite K-10-Supported

Palladium Nanoparticles for Chemistry Select

http://pubs.rsc.org/en/content/articlelanding/2018/ob/c8ob01061g



http://pubs.rsc.org/en/content/articlelanding/2017/nj/c7nj02278f



V V. Sureshbabu Copper-Free Acyl Sonogashira

Reaction 2017, 2, 8059-8062

209 L. Santhosh, Sagar N R, T

M. Vishwanatha, V V.

Sureshbabu

Synthesis of 1, 5- Disubstituted

Tetrazole via Ugi Azide Reaction:

An Asymetric Induction

Approach

Chemistry Select

2017, 2, 5497-5500

208 Girish prabhu, L.

Santhosh, G. Nagendra,

Veladi Panduranga, V V.

Sureshbabu

Molecular-iodine-mediated,

efficient one-pot synthesis of 2-

iminohydantoins and 2-amino-1H-

imidazol-4(5H)-ones by

cyclodeselenization of selenourea-

tethered amides/peptides

Chemistry Select

2017, 2, 1202-1206

207 Sherin Joy, V.V.

Sureshbabu, Ganga

Periyasamy

DFT studies on the terminal

dependent reversible switching of

selenoxo peptides induced by

cationization

Chemistry Select

2017, 2, 4261–4266


Sureshbabu, Ganga

Periyasamy

Density functional theoretical

studies on photoswitching and

charge migration dynamics of thio

and selenoureidopeptides

J Phys Org Chem 2017

DOI 10.1002/poc.3693

205 I. S, Vijayashree, P.

Niranjan, G. Prabhu, V

V. Sureshbabu, J.

Manjanna

Conjugation of Au nanoparticles

with chloambucil for improved

anticancer activity

J Clust Sci

2017, 28, 133–148

204 Veladi Panduranga,

Girish prabhu, Roopesh

kumar L, M.

Krishnamurthy, V V.

Sureshbabu

Thionation of di and tripeptides

employing thiourea as a sulfur

transfer reagent

RSC Advances

2016, 06, 98141-98146

203 Girish Prabhu, Nagendra

G, Sagar N R, Rumpa pal,

Guru Row N Tayur, V. V

Sureshbabu.

A facile synthesis of 1,5-

disubstituted tetrazole

peptidomimetics by

desulfurization/electrocyclization

of thiopeptides

Asian J Org Chem

2016, 5,127-137


Sureshbabu, Ganga

Periyasamy

Computational studies on

structural, Excitation, and Charge

transfer properties of

Ureidopeptidomimetics

J. Phys. Chem B

2016, 120, 6469-6479

201 M. Krishnamurthy, Sagar,

N. R, V V. Sureshbabu

One-pot synthesis of Nα-protected

amino/peptide O-benzyl

Int J Pept Res Ther

http://onlinelibrary.wiley.com/doi/10.1002/ajoc.201500384/abstract





hydroximates and acylaminoxy

dipeptides employing hydroxamic

acid

2017, 23:191–197

200 Sharnabai. K. M,

Krishnamurthy. M, Sagar,

N. R, Santhosh. L, V. V.

Sureshbabu

N-Chlorosuccinimide-mediated

oxidative chlorination of thiols to

Nα-protected amino alkyl sulfonyl

azides and their utility in the

synthesis of sulfonyl triazole acids

Protein and peptide

letters

2017, 24, 53-63

199 Uday Das, Basab

Chattopadhyay, Dipak K.

Hazara, V V. Sureshbabu,

Alok K. Mukkherjee,

Two carbamatederivatives with

Z’=2 and 3: An interplay of strong

and weak hydrogen bonds

Journal of Molecular

Structure

1112, 2016, 293-298

198 Paramita Chatterjee,

Tanusri Dey, Uday Das, V.

V. Sureshbabu, Alok

Kumar Mukherjee

Arylsulfonamide Derivative:

Synthesis, Sturctural Study,

Supramolecular Architecture and

Analysis of Molecular surface

Electrostatic Potential

Zeitschrift fur

Kristallographie 2016

197 Krishnamurthy, M

Vishwanatha, T. M.;

Panguluri, Nageswara

Rao; Panduranga, V.; V.

V Sureshbabu.

Iodine-Mediated Oxidative

Coupling of Hydroxamic Acids

with Amines towards a New

Peptide-Bond Formation

Synlett

2015, 26 (18): 2565-1569

196 Panduranga V, Girish

Prabhu, Roopesh Kumar,

Basavaprabhu, V V.

Sureshbabu

A facile one pot route for the

synthesis of imide tethered

peptidomimetics

Org. Biomol. Chem.

2016, 14, 556-563

195 Basavaprabhu,

Krishnamurthy M,

Nageswara Rao P,

Panduranga V, V. V.

Sureshbabu

A simple and greener approach

for the amide bond formation

employing FeCl3 as a catalyst

New J. Chem.

2015, 39, 7746-7749

194 N. Rao P., V.

Panduranga, Girish

Prabhu, T. M.

Vishwanatha and V. V.

Sureshbabu

Synthesis of chiral Nβ-protected

amino diselenides from the

corresponding amino alkyl iodides

using NaBH2Se3 as a selenating

reagent and their conversion to

seleninic acids

RSC Adv.

2015, 5, 51807-51811

193 Krishnamurthy, M.

Basavaprabhu, V. V.

One-Pot Synthesis of New Class of

Dithiocarbonate-Tethered

Int J Pept Res Ther

https://www.thieme-connect.com/products/ejournals/abstract/10.1055/s-0035-1560266




http://pubs.rsc.org/en/content/articlelanding/2016/ob/c5ob01708d



http://pubs.rsc.org/en/content/articlelanding/2015/nj/c5nj01047k



http://pubs.rsc.org/en/journals/journal/nj

http://pubs.rsc.org/en/content/articlelanding/2015/ra/c5ra06147d






http://link.springer.com/10.1007/s10989-014-9448-2


Sureshbabu Peptidomimetics 2015, 21, (2), 195-203

192 Basavaprabhu, Girish

Prabhu, Krishnamurthy,

M. Sureshbabu V. V.

“Thioureidopeptide”: Novel

Synthon for the Synthesis of N, N′,

N″-Trisubstituted

Guanidinopeptide Mimics

Int J Pept Res Ther

2016, 22, (2), 179–185

191 Rumpa Pal, Nagendra G,

M. S. Reddy, V. V.

Sureshbabu T. N. Guru

Row

Observation of a reversible

isomorphous phase transition and

an interplay of “σ-holes” and “π-

holes” in Fmoc-Leu-ψ[CH2-NCS]

Chem. Commun

2015,51,933-936

190 Basavaprabhu, K. M.

Sharanabai, Girish

Prabhu, V. Panduranga V.

V. Sureshbabu

A facile one pot synthesis of

selenoureidopeptides employing

LiAlHSeH through Staudinger

aza-Wittig type reaction

Synthesis

2015, 47(06), 801-806

189 P. Nageswara Rao, N.

Narendra, Vommina V

Sureshbabu

Iodine-accelerated synthesis of Nα-

urethane protected amino/peptide

hydroxamic acids from

amino/peptide thioacids

Indian J Chemistry

2014, 53B,11, 1430

188 Basavaprabhu H

N. Narendra,

Girish Prabhu

V. V. Sureshbabu

Synthesis of N-urethane protected

amino alkyl (S- methyl)-

isothiouronium compounds and

carbodiimide tethered

peptidomimetics: An application

to guanidino and substituted

guanidino peptidomimetics

synthesis

RSC Advances

2014, 4, 48920-48930

187 C. Madhu, P.

Nageswara Rao, N.

Narendra, V. V.

Sureshbabu

An efficient and racemization free

synthesis of C-terminal

arylamides derived from α-amino

acids and peptide acids via T3P

activation

Int J Protein Research &

Therapeutics, 2014, 20,

353-363

186 P. Nageswara Rao, M.

Samarasimhareddy, C.

Madhu, V. V. Sureshbabu

3,3-Dichloro-1,2-

diphenylcyclopropene (CPI-Cl)

mediated synthesis of Nα-

protected amino acid azides and

α-ureidopeptide

Synlett

(2014, 25,

1001-1005)

185 M.Krishnamurthy,

Basavaprabhu, K. M.

Sharanabai, V. V.

Sureshbabu

A facile route for the synthesis of

novel S-linked 1, 3, 5-triazine

tethered peptidomimetics

Tetrahedron Letters

2014,55,5609-5612

184 C Madhu, P Nageswara

Rao, N. Narendra, V.

One pot synthesis of orthogonally

protected dipeptide selenazoles

Tetrahedron Letters

2014,55,6831-6835


http://link.springer.com/journal/10989/21/2/page/1

http://pubs.rsc.org/en/content/articlelanding/2015/cc/c4cc08751h




Panduranga, V. V.

Sureshbabu

employing N-amino

selenocaboxamides and α-

bromomethyl ketones

183 Vikas Kumar, Akshay

Kumar, Vommina V.

Sureshbabu, Swapandeep

S. Chimni

Synthesis and stereochemistry-

activity relationship of chiral

thiourea derivatives as potential

anticancer agents

Anti-Cancer Agents in

Medicinal Chemistry

(2014, 14(6),

910-920)

182 Basavaprabhu, M.

Samarasimhareddy,

Girish Prabhu, V. V

Sureshbabu reactions in

water

A simple and greener approach

for the synthesis of PVC

supported Pd(0): Application to

Heck and Sonogashira

Tetrahedron Letters

2014, 55, 2556-2560*¥

* Highlighted in Synfacts 2014, 10(7), 0776 highlighted by Uozumi, Y.; Tazawa, A

¥ Elsevier article usage dashboard confirms total views of the paper as 629

180 V. V. Sureshbabu*, B.

Vasantha, C. Madhu

A facile synthesis of N/C-terminal

selenourea tethered glycosylated

amino acids

Indian J. Chem.

179 Chilakapati Madhu , H. P.

Hemantha, T. M.

Vishwanatha V. V.

Sureshbabu*

Simple Preparation of N-

Protected Chiral β-Amino Alkyl

Thiols from Corresponding

Iodides Employing Sodium

Trithiocarbonate

Synth. Commun.

43, 228–235, 2013

178 M. Samarasimhareddy,

Girish Prabhu, V. V.

Sureshbabu*

PVC-supported palladium

nanoparticles: An efficient

catalyst for Suzuki cross- coupling

reactions at room temperature

Synthesis

2013, 45, 1201-1206*

* Synfacts 2013, 9(7), 0800, Highlighted by Uozumi, Y.; Tsuji, H

177 V. Panduranga,

Basavaprabhu, V. V.

Sureshbabu*

An efficient transformation of

ethers to N,N′- disubstituted ureas

in a Ritter type reaction

Tetrahedron Letters

2013, 54, 975–979

176 M.K.Sharanabai,

G.Nagendra,

V. V. Sureshbabu*

Synthesis of N-urethane protected

α-amonoalkyl- α’-cyanomethyl

ketones ; Application to the

synthesis of 3-substituted 5-

amino-1H-pyrazole tethered

peptidomimetics

Synlett

2012, 23, 1913-1918

175 Girish Prabhu,

V. V. Sureshbabu*

Hypervalent iodine(V) mediated

mild and convenient synthesis of

substituted

2-amino-1,3,4-oxadiazoles

Tetrahedron Letters

2012, 53, 4232–4234

http://www.sciencedirect.com/science/article/pii/S0040403912021570




Hosahalli P. Hemantha, V.

V. Sureshbabu*

A simple protocol for the synthesis

of triazole-linked cyclic

glycopeptidomimetics: a

sequential Ugi-MCR and azide–

alkyne cycloaddition

approach

Tetrahedron Letters

2012, 53, 3104–3107

173 T. M. Vishwanatha, N.

Narendra, Basab

Chattopadhyay, Monika

Mukherjee,and V. V.

Sureshbabu*

Synthesis of selenoxo peptides and

oligoselenoxo peptides employing

LiAlHSeH

J .org.chem

2012, 77, 2689-2702

172 N. Narendra, T. M.

Vishwanatha, G.

Nagendra, V. V.

Sureshbabu*

Chiral Nβ-Fmoc-amino alkyl

isonitriles in Ugi-4CR: an

assembly of novel 1,1’-

iminodicarboxylated

peptidomimetics

Tetrahedron

2012, 68,1992-2000

171 V. V. Sureshbabu, *

B.Vasantha,G. Nagendra

A facile one-pot synthesis of Na-

Z/Boc-protected S-linked 1,3,4-

oxadiazole tethered

peptidomimetics

Tetrahedron Letters

2012, 53, 1332–1336.

170 Chilakapati Madhu,

Basavaprabhu,T.M.

Vishwanatha, V. V.

Sureshbabu*

T3P (propylphosphonic anhydride)

mediated conversion of Na-protected

amino/peptide acids into thioacids

Tetrahedron Letters

2012, 53, 1406–1409.

169 Hosamani Basavaprabhu

and V. V. Sureshbabu*

Iron(III) catalysed synthesis of

unsymmetrical di and

trisubstituted ureas – a variation

of classical Ritter reaction

Org. Biomol. Chem.,

2012, 10, 2528


Hosahalli P. Hemantha,

Kuppanna Ananda and V.

V. Sureshbabu*

Epimerization Free Synthesis of

O-Acyl Isodipeptides Employing

COMU

Protein Pept. Lett.

2012, 19, 1281-1287

167 T. M. Vishwanatha,

Samarasimhareddy, V. V.

Sureshbabu*

Facile N-Urethane protected α-

amino/peptide thioacid

preparation using EDC/Na2S

Synlett

2012, 23, 89-92

166 T. M. Vishwanatha, N.

Narendra, V. V.

Sureshbabu*

Synthesis of β-lactum

peptidomimetic through Ugi

MCR: First application of chiral

Nβ- Fmoc amino alkyl isonitrile in

MCRs

Tetrahedron Letters

2011, 52, 5620-5624

165 V. V. Sureshbabu,* G.

Chennakrishnareddy, B.

Vasantha

N-Urethane protected 3-amino

peptide alkyl isoxazole-5-

carboxylic acids in

peptidomimetics chemistry: A

facile one pot synthesis

Int. J. Peptide and

protein research

2011,17 185-191

164 B.Vasantha, Viswanatha

T. M., V. V. Sureshbabu*

Carbonyldiimidazole (CDI)

mediated synthesis of Nα –

protected acyl azides: Application

to the one pot preparation of

ureidopeptides

Protein Pept. Lett.

2011, 18, 1093-1098


Vishwanatha, V. V.

Sureshbabu*

Hydantoin-free synthesis of

peptide ester isocyanates,

isothiocyanates and dipeptidyl

ureas: Application of Zn-dust in

carbonylation procedure without

base

Snythesis

2011, 3247-3254

162 H. S. Lalitamba, H. P.

Hemantha, V. V.

Sureshabubu*

Synthesis of oligopeptides

throough O-acyl isopeptide

method

Protein Pept. Lett.

2011, 18, 848-857

161 V. V. Sureshbabu,*

Basavaprabhu

N, N’-Carbonyldiimidazole

mediated DBU catalysed one pot

synthesis of urea-tethered

glycoconjugates

Synlett,

2011, 8, 1160-1164

160 V. V. Sureshbabu,* B.

Vasantha, H. P. Hemantha

Synthesis of N-Fmoc Protected

Amino Alkyl

Thiocyanates/Selenocyanates and

Their Application for the

Preparation of 5-substituted S/Se-

linked Tetrazoles

Synthesis

2011, 9, 1447-1455

159 H. P. Hemantha, V. V.

Sureshbabu*

Poly(vinyl)chloride Supported

Palladium Nanoparticles: Catalyst

for Rapid Hydrogenation

Reactions

Organic & Biomolecular

Chemistry

2011, 9, 2597-2601

158 Shankar A. N.,

Lalithamba H. S., V. V.

Sureshbabu*

Application of 2-(1H-

benzotriazol-1-yl)-1,1,3,3-

tetramethyluronium

tettrafluoroborate (TBTU) for the

synthesis of acid azides

Indian J Chem.

2011, 50B, 103-109.

157 M. Ramesh, B. Raju, R.

Srinivas, V. V.

Sureshbabu,* T. M.

Vishwanatha, H. P.

Hemantha

Characterization of

Nα‐Fmoc‐protected dipeptide

isomers by electrospray ionization

tandem mass spectrometry

(ESI‐MSn): effect of

protecting group on

fragmentation of dipeptides

Rapid Commun. Mass

Spectrom.

2011, 25, 1949–1958

156 B Vasantha, H. P.

Hemantha, V. V.

Sureshbabu*

Propanephosphonic acid cylic

anhydride (T3P) as an efficient

promoter for Lossen

rearrangement: Application to the

synthesis of ureidopeptides and

Synthesis

2010, 2990-2996

active carbamates derived from

amino acids

155 M, Ramesh, B. Raju, R.

Srinivas, V. V.

Sureshbabu,* N.

Narendra, B. Vasantha

Characterization of Nα-Fmoc-

protected ureidopeptides by

electrospray ionization tandem

mass spectrometry (ESI-MS/MS):

differentiation of potential

isomers

J. Mass. Spectrom.

2010, 45, 1461-1472

154 Hemantha H. P., Ravi, S.

L., V. V. Sureshbabu*

Synthesis of hybrid

peptidomimetics and

neoglycoconjugates employing

Click protocol: Dual utility of Poc-

group for inserting carbamate-

triazole units into peptide

backbone

Int. J. Pept. Res. Ther.

2010, 16, 267-275.


Vishwanatha, V. V.

Sureshbabu*

Peptidomimetics through Click

Chemistry: Synthesis of novel β-

keto triazole acids from N-

protected amino acids

Int. J. Pept. Res. Ther.

2010, 16, 283-290.

152 Basab Chattopadhyaya,

Alok K. Mukherjee, N.

Narendra, H. P Hemantha,

V. V. Sureshbabu,*

Madeliene Helliwell,

Monika Mukherjee

Supramolecular architectures in

5,5′-substituted hydantoins:

crystal structures and Hirshfeld

surface analyses

Crystal Growth and

Design

2010, 10, 4476-4484

151 N. Narendra, H. S.

Lalithamba, V. V.

Sureshbabu*

An efficient one-pot access to the

synthesis of trithiocarbamate

linked peptidomimetics

Tetrahedron Letters

2010, 51, 6169-6173


Sureshbabu*

Isoselenocyanates derived from

Amino Acid Esters: An Expedient

Synthesis & Application to the

Assembly of

Selenoureidopeptidomimetics,

Unsymmetrical Selenoureas and

Selenohydantoins

J. Pept. Sci.

2010, 16, 644-651.

149 Nagendra, G., Ravi, S.L.,

Narendra. N, V. V.

Sureshbabu*

Synthesis of orthogonally

protected 1,3,4-oxadiazole and

1,3,4-thiadiazole peptidomimetics

Tetrahedron Letters

2010, 51, 6338-6341

148 Lalithamba H. S.,

Narendra, N., Shankar A.

N., V. V. Sureshbabu*

Ultrasound mediated synthesis of

2-amino-1,3-selenazoles derived

from Fmoc/Boc/Cbz-protected α-

amino acids

ARKIVOC

2010, Xi, 77-90

147 Lalithamba H. S., V. V.

Sureshbabu*

Simple and efficient synthesis of

Fmoc/Boc/Cbz-protected β-amino

Indian J. Chem.

2010, 49B, 1372-1378

alcohols and peptidyl alcohols

employing Boc2O

146 Ravi, S. L., Nagendra G,

V. V. Sureshbabu*

A facile synthesis of N-Z/Boc-

protected 1,3,4-oxadiazole based

peptidomimetics employing

peptidyl thiosemicarbazides

Tetrahedron Letters

2010, 51, 4705-4709

145 S. A. Naik, V. V.

Sureshbabu*

Synthesis of Nα-protected amino

acid derived selenocarbamates

employing isocyanates as key

intermediates

Synthetic

communications

2010, 40, 2676-2685

144 G. Chennakrishnareddy,

G. Nagendra, H. P.

Hemantha, Ushati Das,

Tayur N. Guru Row, V. V.

Sureshbabu*

Isoselenocyanates derived from

Boc/Z-Amino Acids: Synthesis,

Isolation, Characterization and

Application in the Synthesis of

Unsymmetrical Selenoureas and

Selenoureidopeptidomimetics

Tetrahedron

2010, 66, 6718-6724.

143 Basavaprabhu, N.

Narendra, S. L. Ravi, V.

V. Sureshbabu*

T3P (propylphposphonic

anhydride) mediated conversion

of carboxylic acids into acid azides

and one pot synthesis of

ureidopeptides

Tetrahedron Letters

2010, 51, 3002-3005

142 V. V. Sureshbabu,* H. S.

Lalithamba, N. Narendra,

H. P. Hemantha

New and simple synthesis of acid

azides, ureas and carbamates

from carboxylic acids :

Application of peptide coupling

agents EDC and HBTU

Organic & Biomolecular

Chemistry

2010, 8, 835-840.

TOP 10 MOST DOWNLOADED OBC ARTICLE IN JANUARY 2010 (FIFTH ONE IN THE

ORDER)

141 B Vasantha, V. V.

Sureshbabu*

Facile one step synthesis of acyl

azides and N-Fmoc/Boc/Z-protected

amino acid azides employing

benzotriazole-1-yl-oxy-tris-

(dimethylamino)-phosphonium

hexafluorophosphate (BOP)

Indian J Chem.

2010, 49B, 812-815

140 B Chattopadhyay, H P

Hemantha, N. Narendra,

V. V. Sureshbabu, J. E.

Warren, M. Helliwell, a.

K. Mukherjee, M.

Mukherjee*

Polymorphism in a symmetrical

dipeptidyl urea with Z'>1

Crystal Growth &

Design

2010, 10, 2239-2246

139 V. V. Sureshbabu,* N.

Narendra, H. P.

Hemantha, G.

Chennakrishnareddy

Click chemistry aided synthesis of 1,

4- substituted 1,2,3-triazole linked N-

Fmoc protected triazole-amino acids:

Isolation, characterization and

synthesi of novel triazole based amino

free unnatural amino acids

Protein & Peptide

Letters

2010, 17, 499-506.

138 Vishwanahta T. M.,

Hemantha, H. P., V. V.

Sureshbabu*

Cyanogen Bromide as

Dehydrosulfurizing Agent for the

Synthesis of Nβ-Fmoc- Amino Alkyl

Isonitriles from Nβ-Fmoc–Amino

Alkyl Thioformamides

Synlett

2010, 7, 1096-1100.


T. M. Vishvanatha,

B. Vasantha,

A Simple Synthesis of Nβ-Fmoc/Z-

Amino Alkyl Thiols and their utility

for the Synthesis of Nβ-Fmoc/Z-

Amino Alkyl Sulfonic Acids

Synlett

2010, 7, 1037-1042.


Chennakrishnareddy,

Hemantha H. P.

Synthesis of thioureido-linked

Peptidomimetics, Glycosylated amino

acids and neoglyconjugates using

Bis(benzotriazolyl)methanethione as

thioacylating agent

Synlett

2010, 5, 715-720.


Chennakrishnareddy, S.

A. Naik, Kantharaju

An efficient concomitant synthesis of

O-succinimidyl-(9H-fluoren-9-

ylmethoxy carbonylamino)peptidyl

carbamates and their application in

the synthesis of oligo-α-peptidyl urea

Indian J. Chem.

2010, 49B, 69-76.


Vishwanatha,, N. S.

Sudarshan, V. V.

Sureshbabu*

Fmoc protected halomethylketone

mediated efficient one pot synthesis of

thiazole derivatives of amino acids

and orthogonally protected dipeptide

mimetics

Protein & Peptide

Letters,

2009, 16, 1029-1035.


Sureshbabu*

A simple approach for the synthesis

of new classes of dithiocarbamate-

linked peptidomimetics

Tetrahedron Letters

2009, 50, 7062-7066.


Chennakrishnareddy

HOAt.DCHA as a co-coupling agent

in the synthesis of peptides employing

Fmoc-amino acid chlorides as

coupling agents: Application to the

synthesis of β-casomorphin

Indian J. Chem.

2009, 48B, 981-988.


Shankar A. Naik, H. P.

Hemantha., Narendra, N.,

Das, U, Guru Row, T. N.

N-Urethane Protected Amino Alkyl

Isothiocyanates: Synthesis, Isolation,

Characterization, and Application to

the Synthesis of Thioureidopeptides

J. Org. Chem.

2009, 74, 5260-5266.

130 V. V. Sureshbabu,* N. S.

Sudarshan, G.

Chennakrishnaredd

Simple and rapid synthesis of Nα-

Urethane protected β-amino alcohols

and peptide alcohols employing

HATU

Indian J. Chem.

2009, 48B, 574-579.

129 N. Narendra, G.

Chennakrishnareddy,

V. V. Sureshbabu*

Application of Carbodiimide

Mediated Lossen Rearrangement to

the Synthesis of α-Ureidopeptides and

Peptidyl Ureas employing N-

Urethane α-Amino/Peptidyl

Organic &

Biomolecular

Chemistry

2009, 7, 3520-3526.

Hydroxamic Acids


H. P. Hemantha

Efficient synthesis of Fmoc-

aminoalkoxy pentafluorophenyl

carbonates: Application for the

synthesis of oligopeptidyl carbamates

Synthetic

Communications

2009, 39, 3555-3566.


Narendra, G. Nagendra

Chiral N-Fmoc-β-amino alkyl

isonitriles derived from amino acids:

Synthesis and application in 1-

substituted tetrazoles synthesis

J. Org. Chem.

2009, 74, 153-157.

126 H. P. Hemantha, G.

Chennakrishnareddy, T.

M. Vishwanatha, V. V.

Sureshbabu*

A one pot synthesis of ureidopeptides

and urea tethered glycosylated amino

acids employing DeoxoFluor/TMS-N3

Synlett

2009, 3, 407-410.

125 G. Chennakrishnareddy,

S. J. Tantry, S. A. Naik, V.

V. Sureshbabu*

Synthesis of 1,1-

dioxobenzo[b]thiophene-2-

ylmethyloxycarbonyl (Bsmoc)

protected n-methyl amino acis by

reductin of Bsmoc-5-oxazolidinones

and their use in peptide synthesis

Protein & Peptide

Letters

2009, 16, 105-111.

124 V. V. Sureshbabu,* S. A.

Naik, G. Nagendra

Synthesis of Boc-amino tetrazoles

derived from α-amino acids

Synth. Commun.

2009, 39, 395-406.


Nagendra, H. P.

Hemantha

Synthesis of urea tethered

glycosylated amino acids mediated by

DPPA employing Fmoc-Asp/Glu-5-

oxazolidinones

Indian J. Chem.

2009, 48B, 397-407

122 V. V. Sureshbabu,* S. J.

Tantry, G.

Chennakrishnareddy, G.

Nagendra

Total synthesis of cyclosporine O:

Exploring the utility of Bsmoc-nMe-

amino acid fluorides and KOAt

Protein & Peptide

Letters

2009, 16(3), 312-319

121 B. Chattopadhyay, M.

Mukherjee,* Kantharaju,

V. V. Sureshbabu* and A.

K. Mukherjee

Solvent effect in cyclohexanespiro-5'-

hydantoin- a combined use of X-ray

powder diffraction and solid state

DFT study

Zet Fur Krist

2008, 223, 591-597.

120 Channabasaveshwar, V.

Y,* Shankar, V. S, R. V.

Ramana Rao, D. S.

Shankar Rao S. K. Prasad,

V. V. Sureshbabu*

Supramolecular helical fluid columns

from self assembly of homomeric

dipeptides

Chemistry - A

European Journal

2008, 14, 10462-

10471

119 V. V. Sureshbabu,* H. P.

Hemantha, Shankar A.

Naik

Synthesis of 1,2,4-oxadiazole-linked

orthogonally urethane protected

dipeptide mimetics

Tetrahedron Letters

2008, 49, 5133-5136.

118 K, Srinivasa Sarma, V. V.

Sureshbabu*, S. J. Tantry,

G. Chennakrishnareddy,

N. Sudarshan

Total synthesis of cyclosporine-O Proc. 4th

International Peptide

Symposium -7th

Australian Peptide

Conference – 2nd

Asia-Pacific


Symposium, Jackie

Wilce (Ed),

Australian Peptide

Association, (2008),

pp. 355-357.


Nagendra, R.

Venkataramanarao

Ultrasound accelerated conversion of

N-urethane protected peptide esters

to their thiopeptides using P2S5

Ultrasonics

Sonochemistry

2008, 15, 927-929.


Narendra, Kantharaju

Pentafluorophenyl-(tert-

butoxycarbonylamino)methyl

carbamates: Synthesis, isolation and

application to the synthesis of

ureidopeptides

Ind. J. Chem.

2008, 47B, 920-926.

115 V. V. Sureshbabu,* N

Narendra

Synthesis of N-Z, N'-formyl-α-amino

acid derived gem-diamines

Int. J. of Pep. Res &

Therapeutics

2008, 14, 201-207.


Sudarshan, Kantharaju

Efficient synthesis of O-succinimidyl-

(tert-butoxycarbonylamino)methyl

carbamates derived from α-amino

acids accelerated by ultrasound

Application to the synthesis of

ureidodipeptides

Synth. Commun.

2008, 38, 2168-2184.


Sudarshan, Gundala

chennakrishna

HOBt.DCHA mediated synthesis of

peptides employing Fmoc-amino acid

chlorides in both solution phase and

solid phase methods

Synth. Commun.

2008, 38, 2625- 2637.

112 V. V. Sureshbabu,* Rao

Venkataramanarao, N.

Narendra

Synthesis of ureido linked

glycosylated amino acids from N-

Fmoc-Asp/Glu-5- oxazolidinones and

their application to neoglycopeptides

synthesis

Synth. Commun.

2008, 38, 3640-3654.


Sudarshan, R.

Venkataramanarao

Peptidyl carbamates: Efficient

synthes using N-Fmoc-β-amino

alkoxy carbonyl chlorides/active

pentachlorophenyl carbonates as

monomeric building blocks

Int. J. Peptide Res &

Therapeutics

2008, 14, 149-156.


Sudarshan, Shankar A.

Naik

Synthesis of ureidopeptides and

peptidyl ureas employing Bsmoc

chemistry


Therapeutics

2008, 14, 105-112.

109 V. V. Sureshbabu* R.

Venkataramanarao, H. P.

Hementha

A facile synthesis of C-terminal

neoglycopeptides: Incorporation of

urea moiety between sugar and

peptides employing Curtius

rearrangement


Therapeutics

2008, 14, 34-40


Sureshbabu*

New approach for the efficient

synthesis of carbamate tethered

glycosylated amino acids and their

insertion into peptides

Synlett

2008, 4, 496-500.

107 V. V. Sureshbabu,* G

Chennakrishnareddy, N

Narendra

A facile and one-pot synthesis of Nα

Fmoc/Bsmoc/Boc/Z- protected

ureidopeptides and peptidyl ureas

employing diphenylphosphoryl azide

[DPPA]

Tetrahedron Letters

2008, 49, 1408-1412.

106 V. V. Sureshbabu,* H. P.

Hemantha

A facile synthesis of N-Fmoc

protected amino/ peptidyl weinreb

amides employing acid chlorides as

key intermediates

ARKIVOC

2008, ii, 243-249.

105 V. V. Sureshbabu,* R.

Venkataramanarao

Synthesis of ureidopeptides using

pentafluorophenyl carbamates from

Fmoc-peptide acids

Indian J. Chem.

2008, 47B, 910-919.

104 K. Srinivasa Sarma, V. V.

Sureshbabu,* R

Venkataramanarao, H. P.

Hemantha, N. Narendra

The utility of Fmoc-Asp/Glu derived

5-oxazolidinones for side chain

carboxyl group modifications

Proc. 4th


Symposium -7th

Australian Peptide

Conference – 2nd

Asia-Pacific


Symposium, Jackie

Wilce (Ed),

Australian Peptide

Association, (2008),

pp.259-261.


Sureshbabu,* S. A. Naik,

G. Chennakrishnareddy

Synthesis of tetrazoles analogues of

amino acids: The Fmoc approach

Proc. 4th


Symposium -7th

Australian Peptide

Conference – 2nd

Asia-

Pacific International

Peptide Symposium,

Jackie Wilce (Ed),

Australian Peptide

Association, (2008)

pp.159-160.


Sudarshan, L.

Muralidhar, N. Narendra

Synthesis of N-urethane protected β-

amino alcohols employing N-

protected-α-amino acyl

benzotriazoles

J. Chem. Res.

2007, 683-685.

101 N. S. Sudarshan, N.

Narendra, H. P.

An efficient conversion of carboxylic

group of N-Fmoc-α-amino

J. Org. Chem.

2007, 72, 9804-07.

Hemantha, V. V.

Sureshbabu*

acids/peptide acids into N-

formamides employing isocyanates as

key intermediates

100 Subramanyam J Tantry,

Rao Venkataramanarao,

G. Chennakrishnareddy,

V. V. Sureshbabu*

Total synthesis of cyclosporin O by

convergent approach employing

Fmoc-amino acid chlorides mediated

by Zinc dust

J. Org. Chem.

2007, 72, 9360-9363.

99 Rao Venkarramanarao, V.

V. Sureshbabu*

An efficient synthesis route to N-

glycosylamino acids using Nα-Fmoc-

Asp/Glu-5-oxazolidinone as internal

protection

Synlett

2007, 16, 2492-2496.

98 V. V. Sureshbabu,* Rao

Venkataramanarao,

Shankar A. Naik, G

Chennakrishnareddy

Synthesis of tetrazole analogues of

amino acids using Fmoc-chemistry:

Isolation of

free amino tetrazoles and their

incorporation into peptides

Tetrahedron Letters

2007, 48, 7038-7041.

97 R. Venkataramanarao, N.

S. Sudarshan, V. V.

Sureshbabu*

Microwave assisted alcoholysis of

isocyanates derived from Nα-[(9-

fluorenylmethyl)oxy]carbonyl amino

acids: Synthesis of N-Fmoc-N1-Z-

/Boc-/Alloc- /Bsmoc-gem-diamines

Int. J. of Pep. Res

and Therapeutics

2007, 13, 393-397.


Kantharaju, G.

Chennakrishna

Microwave irradiated accelerated

rapid, efficiency and high yield

esterification of Boc-amino acid to

Merrifield resin mediated by KF

Indian J. Chem.

2007, 46B, 1466-1469.

95 V. V. Sureshbabu,* B. S.

Patil, R. V. Ramanarao

Preparation, isolation, and

characterization of Nα-Fmoc-peptide

isocyanates: Solution synthesis of

oligo-α-peptidyl ureas

J. Org. Chem.

2006, 71, 7697-7705.

94 P. Cano-Sanchez, B.

Severino, V. V.

Sureshbabu, J. Russo, T.

Inui, F.X. Ding, B.

Arshava, J. Becker and F.

Naider*

Effects of N- and C-terminal addition

of oligolysines or native loop residues

on the biophysical properties of

transmembrane domain peptides

from a G-protein coupled

receptor

Journal of Peptide

Science

2006, 12, 808-822.


Sureshbabu,* R.

Venkataramanarao

Nα-Fmoc-Peptide isocyanates and their

utilization in synthesis of ureidopeptides

and retro-inverso peptides

Peptide Science,

T.Wakamiya (Ed)

2005, 29 – 32.

92 K. S. Devaraju, B. S. Patil,

S. J. Tantry, Taranath

Shetty K, V. V.

Sureshbabu*

Synthesis of a modified peptide

fragment analog Val-Tyr (P)-Val-Ala-

Ala-OH of cAMP protein kinase

regulatory sub unit type II employing

Fmoc chemistry

Indian J. Chem.

2006, 45B, 1747 -

1752.

91 R. Venkataramanarao, S.

J. Tantry, V. V.

Sureshbabu*

Practical and efficient synthesis of

orthogonally protected α-2,3-

diaminopropionic acid (2,3-Dap) and

Synth. Commun.

2006, 36, 2901-2912.

2,4-diaminobutanoic acid (2,4-Dab)

and their N-methylated derivatives


Kantharaju, N. S.

Sudarshan

Synthesis of Fmoc-protected β-amino

alcohols and peptidyl alcohols from

Fmoc- amino acid / peptide acid

azides

Indian J. Chem.

2006, 45B, 1880-

1886.

89 R.Venkataramana Rao, V.

V. Sureshbabu*

Synthesis of retro-inverso peptides

employing isocyanates of Nα-Fmoc-

amino acids catalyzed by DMAP

Tetrahedron Letters

2006, 47, 9139-9141.

88 Kantharaju, V. V.

Sureshbabu*

Ultrasound accelerated synthesis of

proteinogenic and α,α-dialkylamino

acid ester salts

Indian J. Chem.

2006, 45B, 1942-1944.


Sudarshan

Synthesis of peptidyl ureas employing

O-succinimidyl-(9H-fluoren-9-

ylmethoxy

carbonylamino)methylcarbamate

derivatives as activated monomers

Protein and Peptide

Lett.

2006, 493-498.

86 Subramanyam J. Tantry,

R.enkataramanarao, V. V.

Sureshbabu*

Rapid and efficient synthesis of the

penta-peptide of elastin protein and

peptides containing highly

hindered α,α-dialkyl amino acids

employing Fmoc-amino acid chlorides

under microwave irradiation in

solution phase

ARKIVOC

2006, 21-30.

85 V. V. Sureshbabu,* R.

Venkataramana Rao

Microwave irradiated high-speed

solution synthesis of peptide acids

employing pentafluorophenyl esters

as coupling agents

Indian J. Chem.

2005, 44B, 2328-2332.

84 P. Cano-Sanchez, T.

Inui, B. Severino, V. V.

Sureshbabu,* B. Arshava,

J. M. Becker, F. Naider*

Influence of natural loop residues or

oligolysines on the biophysical

properties of transmembrane

domains of a G Protein-Coupled

Receptor

Understanding

Biology using

Peptides

2005, S. Blondelle

(Eds), o49-o51.

83 N. Sudarshan, V. V.

Sureshbabu*

Microwave accelerated high speed

solution synthesis of peptides

employing HATU/HOAt

Indian J. Chem.

2005, 44B, 1509-1511.

82 S. S. Chimni,* D.

Mahajan, V. V.

Sureshbabu

Protonated chiral prolinamide

catalyzed enantioselective direct aldol

reaction in water

Tetrahedron Letters

2005, 46, 5617-5619.


Kantharaju

2,4,5-Trichlorophenyl-(9H-fluoren-9-

ylmethoxycarbonylamino)methyl

carbamates ;Synthesis, isolation,

characterization and utility in the

synthesis of dipeptidyl ureas

Indian J. Chem.

2005, 44B, 1046-1053

80 V. V. Sureshbabu,* B. S.

Patil, G. R.

MW enhanced high speed

deprotection of Boc-group using p-

Synth. Commun.

2005, 35, 1795-1802.

Vasanthakumar TsOH and concomitant formation of

NMe-Amino Acid benzyl ester p-

TsOH salts

79 Kantharaju, B. S. Patil,

V. V. Sureshbabu*

Wolff rearrangement of Nα-Boc-/Z-

protected aminodiazoketones to the

corresponding β-amino acids under

microwave irradiation

Indian J Chem.

2005, 2611-2613.


Kantharaju, S. J. Tantry

Curtius rearrangement using

ultrasonication: Isolation of

isocyanates of Fmoc-amino acids and

their utility for the synthesis of

dipeptidyl ureas

Int. J. of Peptide Res.

& Therapeutics

2005 11, 131-137.

77 V. V. Sureshbabu,* G-R

Vasanthakumar, B. S.

Patil

Nα-Fmoc-peptide azides : Synthesis,

isolation, characterization and utility

in the extension of peptide chains

Indian J. Chem.

2002, 44B, 1853-1858.

76 D. Gayathri, D.

Velmurugan,*

Kantharaju, V. V.

Sureshbabu*

tert-Butyl 4,4-dimethyl-5-oxo-1,3-

oxazolidine-3-carboxylate

Acta Cryst

2005, E61, 4088–

4090.

75 V. V. Sureshbabu,* G. R.

Vasanthakumar, S. J.

Tantry,

N-Silylation of amines and amino acid

esters under neutral conditions

employing TMS-Cl in the presence of

zinc dust

Tetrahedron Letters

2005, 46 4099-4102.

74 S. J. Tantry, V. V.

Sureshbabu*

Synthesis of Nα-protected peptide

acids by the N-C chain extension

employing O, N-bis-trimethylsilyl-

amino acids using the mixed

anhydride method

Indian J. Chem.

2004, 43B 1282-1287.

73 B. S. Patil, G. R.

Vasanthakumar, V. V.

Sureshbabu*

Synthesis of peptidyl ureas using p-

nitrophenyl-(9-fluorenylmethoxy

carbonyl amino) methyl carbamate

derivatives

Synth. Commun.

2004, 34, 2313-2321.

72 B. S. Patil, V. V.

Sureshbabu*

A rapid synthesis of dipeptidyl urea

acids employing p-nitrophenyl-(9-

fluorenyl

methoxycarbonylamino)ethyl

carbamates

Indian J. Chem.

2004, 43B, 1721-1728.

71 B.S. Patil, V. V. Suresh

babu*

A rapid and convenient synthesis of α

and β forms of acetylated derivatives

of sugars under microwave

irradiation

Indian J. Chem.

2004, 43B, 1288-1291.

70 Kantharaju, V. V.

Sureshbabu*

Homologation of α-amino acids to β-

amino acids: 9-fluorenylmethyl

chloroformate as a carboxyl group

activating agent for the synthesis of

Nα-protected

Indian J. Chem.

2004, 43B, 2152-2158.

aminoacyldiazomethanes

69 F. Naider,* R. Estepphan,

J. Englander, V. V.

Sureshbabu, E. Arevalo,

K. Samples, J. M. Becker

Sexual conjugation in yeast : A

paradigm to study G Protein-Coupled

Receptor Domain Structure

Biopolymers (Peptide

Science)

2004, 76 (2), 119-128.

68 V. V. Sureshbabu,* S. J.

Tantry

A rapid and efficient synthesis of β-

casomorphin employing Boc-amino

acids and 9-fluorenylmethyl

chloroformate as a coupling agent

Indian J. Chem.

2004, 43B, 2708-2712.

67 G. R. Vasanthakumar, V.

V. Sureshbabu*

Simple and stereospecific

homologation of urethane protected

-amino acids to their higher

homologues using HBTU

J. Peptide Research

2003, 61, 230-236.

66 S. J. Tantry, R. I.

Mathad, V. V.

Sureshbabu*

Synthesis of -casomorphin

employing Fmoc – amino acid

chlorides and t-butyl

dimethylsiloxybenzotriazole

(TBDMS-OBt)

Indian J. Chem,

2003, 42B, 2104-2108.



Sureshbabu*

Isocyanates of Nα-[(9-

fluorenylmethyl)oxy]carbonyl (Fmoc)

amino acids :Synthesis, isolation,

characterization and application to

the efficient synthesis of urea

peptidomimetics

J. Org. Chem.

2003, 68, 7274-7280.


V. Sureshbabu*

Direct synthesis of Fmoc-protected

amino acid hydroxamates from acid

chlorides mediated by magnesium

oxide

Tetrahedron Letters

2003, 44, 4099-4101.



Sureshbabu*

Synthesis of β-amino acids : 2-(1H-

Benzotriazol-1-yl)-1,1,3,3

tetramethyluronium

tetrafluoroborate (TBTU) for

activation of Fmoc-/Boc-/Z-α-amino

acids

Synth. Commun.

2003, 33, 3089-3096.


V. Sureshbabu*

Synthesis of Fmoc-/Boc-/Z-β-amino

acids via Arndt-Eistert homologation

of Fmoc-/Boc-/Z- α-amino acids

employing BOP & PyBOP,

Indian J. Chem.

2003, 42B, 1691-1695.


Sureshbabu*

Synthesis of peptides employing

Fmoc-Cl as coupling agent

Letters in Peptide

Science

2003, 10, 51-55.

60 B. S. Patil, V. V.

Sureshbabu*

Synthesis of peptidylureas employing

O-pentafluorophenyl-(9-

fluorenylmethoxycarbonylamino)met

hylcarbamate derivatives

Letters in Peptides

Science

2003, 10, 93-97.

59 V. V. Sureshbabu, J. M. Native Chemical Ligation of Peptide Revolution:

Becker, F. Naider* transmembrane receptor fragments

of Step2

Genomics,

Proteomics &

Therapeutics Kluwer

Academic Pub, M.

Chorev & T. K.

Sawyer (Eds.), (2003)

630-631.


Sureshbabu*

9-Fluorenylmethyl chloroformate

(Fmoc-Cl) as a useful reagent for the

synthesis of pentafluorophenyl, 2,4,5-

trichlorophenyl, pentachlorophenyl,

p-nitrophenyl, o-nitro phenyl and

succinimidyl esters of Nα-urethane

protected amino acids

Letters in Peptide

Science

2003, 10, 655-662.

57 Kantharaju, B. S. Patil, V.

V. Sureshbabu*

Synthesis of Fmoc-amino acid

chlorides assisted by ultra sonication,

a rapid approach

Letters in Peptide

Science

2002, 9, 227-229.


V. Sureshbabu*

A convenient method for the synthesis

of -amino acids via the Arndt-Eistert

approach using p-toluene sulphonyl

chloride as a carboxylic group

activating agent

Synth. Commun.

2002, 32, 651-657.

55 G. R. Vasanthakumar, K.

Ananda, V. V.

Sureshbabu*

Fmoc-amino acid azides in peptide

synthesis

Indian. J. Chem.

2002, 41B, 1733-1735.

54 V. V. Sureshbabu,* K.

Ananda, G. R.

Vasanthakumar

A convenient method for the synthesis

of C–protected esters of Boc-/Z-,-

dialkylamino acids by the mixed

carboxylic–carbonic anhydride

method

Protein and Peptide

Letters

2002, 9, 345.

53 S. J. Tantry, K. Ananda,

V. V. Sureshbabu*

Coupling in the absence of tertiary

base: A method for the

deprotonation of hydrochloride salts

of peptide esters to amino free peptide

esters

Indian J. Chem.

2002, 41B, 1028-1031.

52 G. R. Vasanthakumar, H.

N. Gopi, V. V.

Sureshbabu*

Synthesis of alkyl and aryl esters of

N-protected -homoamino acids from

N-protected -aminodiazoketones

Protein and Peptide

Letters

2002, 9, 529.

51 L. K. Henry, S. Khare, C.

Son, V. V. Sureshbabu, F.

Naider,* J. M. Becker

Identification of a contact region

between the tridecapeptide -factor

mating pheromone of Saccharomyces

cerevisiae and its G Protein Coupled

Receptor by photoaffinity labeling,

Biochemistry

2002, 41,

6128-6139.

50 G. R.Vasanthakumar, B.

S. Patil, V. V.

Sureshbabu*

Homologation of -amino acids to -

amino acids using Boc2O

J. Chem. Soc, Perkin

Trans 1

2002, 2087-2089.

49 S. J. Tantry, Kantharaju,

V. V. Sureshbabu*

Microwave accelerated efficient

synthesis of N-

fluorenylmethoxycarbonyl / benzyl

oxycarbonyl –5-oxazolidinones

Tetrahedron Letters

2002, 43, 9461-9462.


Sureshbabu*

1-(t-

Butyldimethylsilyloxy)benzotriazole

[TBDMS-OBt] : A new and novel

reagent for the synthesis of peptides

Letters in Peptide

Science

2002, 9, 35-41.

47 G. R. Vasanthakumar, B.

S. Patil, V. V. Suresh

babu*

Microwave assisted facile synthesis of

amino acid benzyl ester p-

toluenesulphonate and hydrochloride

salts

Letters in Peptide

Science

2002, 9, 207-209.



Sureshbabu*

Microwave assisted Wolff

rearrangement: A facile method for

the synthesis of Fmoc--amino acids

Letters in Peptide

Science

2002, 9, 231-233.

45 K. Ananda, H. N. Gopi, V.

V. Sureshbabu*

Convenient and simple homologation

of N-urethane protected -amino

acids to their -homologues with

concomitant o-nitrophenyl esters

formation

Indian J. Chem.

2001, 40B, 790–795.

44 K. Ananda, V. V.

Sureshbabu*

Deprotonation of hydrochloride salts

of amino acid esters and peptide

esters using commercial zinc dust

J. Peptide Research

2001, 57, 223-226.


Ananda

Zinc promoted rapid and efficient

synthesis of Fmoc- and Z-,-

dialkylamino acids under neutral

conditions

Indian J. Chem.

2001, 40B, 70-74.


Ananda, R. I. Mathad

Synthesis of pentafluorophenyl, 2,4,5–

trichlorophenyl and

pentachlorophenyl esters of Fmoc-

amino acids using Fmoc-amino acid

chlorides as intermediates

Letters in Peptide

Science

2001, 7, 239–242.

41 K. Ananda, G. R.


Sureshbabu*

Simple and efficient method for the

synthesis of Z-/Boc-amino acid

amides using p-toluenesulphonyl

chloride

Protein and Peptide

Letters

2001, 8, 45-48.

40 V. V. Sureshbabu,* H. N.

Gopi, K. Ananda

Synthesis of Boc- & Z-protected

amino acid fluorides employing

DAST as a fluorinating agent

Indian J. Chem.

2000, 39B, 384-386.

39 H. N. Gopi, K. Ananda, V.

V. Sureshbabu*

Wolff rearrangement of N-protected

-aminodiazoketones in presence of

substituted phenol as a method for

the synthesis of 2,4,5-trichlorophenyl

esters of Fmoc-/Boc-/Z--homoamino

acids

Protein and Peptide

Letters

2000, 7, 33-36.

38 V. V. Sureshbabu,* K. Synthesis of peptides employing Letters in Peptide

Ananda Fmoc/Boc/Z-amino acid fluorides and

activated commercial zinc dust

Science

2000, 7, 41-46.


V. Sureshbabu*

Convenient and efficient synthesis of

Boc-/Z-/Fmoc--amino acids

employing N- protected -amino acid

fluorides

J. Peptide Research

2000, 55, 289-294.

36 H. N. Gopi, V. V.

Sureshbabu*

Zinc promoted simple synthesis of

oligomer free N-Fmoc-amino acids

using Fmoc- Cl as an cylating

agent under neutral conditions

J. Peptide Research

2000, 55, 295-299.


Ananda, G. R.

Vasanthakumar

(9-Fluorenylmethyloxy)carbonyl

(Fmoc) amino acid azides : Synthesis,

isolation,characterization, stability

and application to synthesis of

peptide

J. Chem. Soc, Perkin

Trans 1

2000, 4328-4331.


Sureshbabu*

Convenient and simple homologation

of N-urethane protected -amino

acids to their - homologues with

concomitant pentafluorophenyl ester

formation

Letters in Peptide

Science

2000, 7, 165-169.

33 V. V. Sureshbabu,* H.N.

Gopi Synthesis of -amino acids using Boc-

/Z-amino acid pentafluorophenyl

esters

Letters in Peptide

Science

1999, 6, 173-178.


Gayathri, H.N. Gopi

Fmoc-peptide acid chlorides in

fragment coupling : Synthesis of -

casmorphin by 3+2 divergent

approach

Synth. Commun.

1999, 29, 79-91.

31 K. Ananda, V. V.

Sureshbabu*

Convenient and simple synthesis of N-

{[(9H-fluoren-9-

yl)methoxy]carbonyl}– (Fmoc)

protected -amino acids (homo--

amino acids) employing Fmoc--

amino acids and

dicyclohexylcarbodiimide (DCC)

mixtures

Indian J. Chem.

1999, 38B, 418-423.

30 H. N. Gopi, K. Ananda,

V. V. Sureshbabu*

Zinc promoted simple synthesis of Z-

amino acids under neutral conditions

Protein and Peptide

Letters

1999, 6, 233-236.


Gopi, K. Ananda, Homologation of -amino acids to -

amino acids using Fmoc-amino acid

pentafluorophenyl esters

J. Peptide Research

1999, 53, 308-313.

28 K M. Sivanandaiah,* V.

V. Sureshbabu, S. C.

Shankaramma

Solid phase synthesis of O-

glycoopioid peptides related to

dermorphin

Indian J. Chem,

1998, 37B, 760-767.

27 H. N. Gopi, V. V. Suresh Synthesis of peptides mediated by Indian J. Chem,

babu* potassium salt of 1-hydroxy-7-

azabenzotriazole

1998, 37B, 394-396.


Gopi

. Rapid and efficient synthesis of

peptide fragments containing Aib

using Fmoc-amino acid chlorides /

KOBt

Tetrahedron Letters

1998, 39, 1049-1050.

25 K. Gayathri, H. N. Gopi,

V. V. Sureshbabu*

Fmoc-Peptide acid chlorides :

preparation, characterization and

utility in peptide synthesis

Indian J. Chem.

1998, 37B, 151-154.


V. Sureshbabu*

Rapid and efficient synthesis of

peptides containing ,-dialkylamino

acids employing KOBt

Letters in Peptide

Science

1998, 5, 277-283.


Sureshbabu*

Synthesis of [Leu5]enkephalin using

Fmoc-amino acid chlorides/KOAt

J. Indian Chem.

Society

1998, 75, 511-513.


Gayathri

Synthesis of peptides mediated by

AgCN

Indian J. Chem.

1998, 37B, 1109-1113.


Sureshbabu*

Synthesis of peptides employing

Fmoc-amino acid chlorides and

commercial zinc dust

Tetrahedron Letters

1998, 39, 9769-9772.

20 K. M. Sivanandaiah,* V.


Shankaramma, M.

Lakshmana

Pharmacological activities of some

synthetic peptides related to

dermorphin

Indian J. Pharm

1997, 29, 92-98.



Shnkaramma, M.

Lakshmana, M. A. Arif &

M. Kumar

Synthetic peptides related to laminin

pentapeptide (YIGSR) fragment

Indian J. Expt.

Biology

1996, 34, 658-662.


V. Sureshbabu, B. P.

Gangadhar

Silicon tetrachloride and phenol as N-

t-Butyloxycarbonyl group

deprotecting agent in solid phase

peptide synthesis

Tetrahedron Letters

1996, 37, 5689-5990.



Shankaramma, M.

Lakshmana, M. A. Arif

Synthetic peptides related to -

receptor agonist, dermorphin gene

associated peptide

Indian J. Pharm,

1996, 28, 155-160.



Shankaramma

Solid phase synthesis of oxytocin

using iodotrichlorosilane as Boc

deprotecting agent

Int. J. Peptide and

Protein Research

1995, 45, 377-379.


V. Sureshbabu, H. C.

Renukeshwar, B. P.

Gangadhar

Iodotrichlorosilane as N-Z cleaving

agent in solid phase synthesis of

dermorphin and oxytocin

Indian J. Chem.

1995, 34B, 487-491.


V. Sureshbabu, H. C. Synthetic peptides related to -

receptor agonist, dermorphin gene

Indian J. Bio Chem.

And Bio. Phys.

Renukeshwar, M.

Lakshmana, Rachu babu

associated peptid 1995, 32, 196-199.

13 K. M. Sivanandaiah*, V.


Renukeshwar, B. P.

Gangadhar,

N-Benzyloxycarbonylamino acids in

solid phase peptide synthesis

Indian J. Chem.

1994, 33B, 618-619.


V. Sureshbabu, B. P.

Gangadhar

Fmoc-amino acid chlorides-KOBt in

solid phase peptide synthesis

Indian J. Chem.

1994, 33B, 620-62.



Renukeshwar, M.

Lakshmana, M. A. Asif &

S. Chiplunkar

Synthesis of peptides related to the -

receptor agonist, dermorphin

Indian J. Pharm.

1994, 26, 204-208.



Shankaramma

Synthesis of peptides mediated by

KOBt

Int. J. Peptide and

Protein Research

1994, 44, 24-30.



Renukeshwar, B. P.

Gangadhar

A rapid and efficient synthesis of the

opioid agonist, deltorphin

Indian J. Chem.

1993, 32B, 465-467.

8 K. M. Sivanandaiah,* S.

Gurusiddappa, D. Channe

Gowda, V. V. Suresh babu

Solid phase synthesis of leuteinizing

hormone-releasing hormone

Vignana Bharathi

1993, 13, 1-7.



Renukeshwar

Fmoc-amino acid chlorides in solid

phase synthesis of opioid peptides

Int. J. Peptide and

Protein Research

1992, 39, 201-206.



Shankaramma

Acid chloride / KOBt as a coupling

agent in peptide synthesis

Indian J. Chem.

1992, 31B, 379-380.


Gurusiddappa, V. V.

Sureshbabu

Solid phase synthesis of acyl carrier

protein 65-74 decapeptide sequence

India J. Chem.

1991, 30B, 302-305.


Gurusiddappa, V. V.

Sureshbabu

Synthesis and biological activities of

new analogues of dermorphin

substituted at position 2

Indian J. Chem.

1989, 28B, 338-341.


Gurusiddappa, V. V.

Sureshbabu

Synthesis and biological studies of

dermorphin and its analogues

substituted at position 5 and 7

Int. J. Peptide and

Protein Research

1989, 33, 463-467.


Gurusiddappa, D. Channe

Gowda, V. V. Suresh babu

Improved solid phase synthesis of

LHRH analogues using Fmoc-amino

acid active esters and catalytic

transfer hydrogenation with minimal

side-chain protection and their

biological activities

J. of Biosciences

1989, 14, 311-317.


Gurusiddappa, V. V.

Sureshbabu

Peptides related to

Leucine/Methionine-enkephalinamide

: synthesis & biological activities

Indian J. Chem.

1988, 27B, 645-468.

Seminars and conferences attended and papers presented:

a Seminars, Symposia, Workshops, attended 23

b Poster presentations 23

c Oral and Invited presentations 12

d Conferences attended in U.S.A. Japan and Australia 06

e Details of talks delivered in Japan 02

f Lectures delivered related to research work 08

g Participation in Refresher Courses as Resource person 08

h Popular lectures delivered for UG students and faculty 07

i Conferences, workshops, Lectures organized 11

Invited Lectures Delivered in national symposia:

1. National conference on chemical sciences for industry and society emerging trends for the

third millennium, Dept. of Industrial Chemistry, Kuvempu University, Shankaraghatta, Jan 6-8,

2006, Studies on chemical synthesis of ureidopeptides.

2. First Indian Peptide Symposium organized by Indian Peptide Society at Hyderabad, Feb 22,

2007, Application of Nα-Fmoc amino acid derived isocyanates in peptidomimetics and peptidyl

conjugate synthesis.

3. National seminar on Modern Trends in Analytical methods of analysis, Dept. of Chemistry,

Sri Krishnadevaraya University, Anantapur, Feb. 25-27, 2008, Nα-Fmoc amino acid derived

isocyanates: Stable and Versatile intermediates for the synthesis of peptides and glycopeptide

mimics.

4. Symposium on Current trends in organic chemistry at Department of Organic Chemistry,

Indian Institute of Science, Bangalore, Nov. 20-22, 2008, Peptides and peptidomimetics

synthesis with Fmoc group: Novel Methods and Intermediates.

5. New vistas in Chemistry during 21st centure at Department of Chemistry, Pingle Govt.

College for women, Warangal, Sept. 11th & 12, 2009, Recent developments in the synthesis of

ureido and thioureido peptidomimetics.

6. National Conference on RECENT TRENDS IN ORGANIC SYNTHESIS–2011 (RTOS-

2011)School of Chemistry Bharathidasan University Tiruchirappalli Feb24-26, 2011, New

protocols and strategies for the synthesis of peptidomimetics.

Oral and Invited presentations:

1) 4th National Symposium on Bio-Organic Chemistry, Bhabha Atomic Research Center,

Bombay, Jan. 27-29, 1992, Solid phase synthesis of deltorphin using Fmo -amino acid chlorides

and Merrifield Resin.

2) XII Conference of Indian Council of Chemists, Kakatiya University, Warangal, Dec.28-30,

1993, Glycosylated Asp derivative for solid phase glycoopioid peptide synthesis.

3) 6th National bioorganic symposium, JNCASC and Dept. of Organic Chemistry, I.I.Sc.,

Bangalore, June 5-7, 1997, Synthesis of peptides mediated by acid chlorides of Fmoc-amino

acids in the absence of a base..

4) VI NOST symposium, Lonavala, Pune, April 20-23, 1997, Fmoc-arnino acid

chlorides/KOAt in peptide synthesis.

5) 16th Conference of Indian Council of Chemists, Mangalore University, Mangalore, Dec. 29-

31, 1997, Rapid & efficient synthesis of peptides containing Aib employing Fmoc-amino acid

chlorides/KOBt.

6) National symposium on newer vistas in synthetic protocols and structural elucidation in

chemistry, School of Chemistry, Madurai Kamaraj University, Madurai, April 22-24, 1998,

Synthesis of β-amino acids employing Fmoc-amino acid chlorides.

7) 35th Annual convention of chemists, Department of Chemistry, Karnatak University,

Dharwad, Nov. 4-7 1998, Synthesis of β-amino acids.

8) National Symposium in Chemistry, Department of Organic Chemistry, I.I.Sc., Bangalore,

Jan. 27-30. 1999, Synthesis of β-amino acids employing Fmoc-/Boc-Z-amino acid

pentafluorophenyl esters.

9) International conference on chemistry and 36th annual convention of chemists, Department

of Chemistry, University of Calcutta, Calcutta, Dec. 11-16. 1999. Synthesis of peptides

employing Fmoc-/Boc-/Z-a -amino acid fluorides and zinc dust.

10) SIF User’s one day symposium, I.I.Sc., Bangalore, May 2, 2002, Studies on synthesis of

oligoureas peptidomimetics employing the Fmoc-protection strategy.

11) National Symposium in Bio-organic and Medicinal Chemistry (NSBM), Mysore

University, Mysore, Oct.5-7, 2005, Practical and efficient synthesis of orthogonally

protected α-2,3-diaminopropionic acid (2,3-Dap) and 2,4- diaminobutanoic acid (2,4-Dab) and

their N-methylated derivatives.

12) 44th Annual Convention of Chemists 2007 organized by Indian Chemical Society at

Mahatma Gandhi Institute of Applied Sciences, Jaipur, Dec 23-27, 2007. Application of N-

Fmoc-Asp/Glu derived Oxazolidin-5-one for the synthesis of neoglycopeptides.

Lectures delivered related to research work:

Title of the topic Place & Date

1. Solid phase synthesis of deltorphin using Bhaba Atomic Research Centre

Fmoc-amino acid chlorides & Merrifield Bombay, Jan. 27, 1992.

Resin

2. Glycosilated Asp derivatives for solid phase XII conference of Indian Council of

glycoopioid peptide synthesis Chemists, Warangal, Dec. 29. 1993.

3. Chemical synthesis of peptides Chemical Society, Dept. of

Chemistry, Central College Campus,

Bangalore University, Bangalore,

Feb. 1, 1995.

4. Recent studies on chemical synthesis of National Chemical Laboratory

peptides Pune, April 1995.

5. Rapid and efficient synthesis of XIV conference of Indian Council

α-methylalanine containing peptide of Chemists, Institute of Science,

antibiotics Bombay, Dec. 29, 1995.

6. Why do we live in the world of α-peptides Chemical Society, PG Dept. of

but not in β-peptides Chemistry, St. Joseph’s College,

Bangalore, Dec. 9, 2002.

7. Studies on the use of acid chlorides as coupling Dept. of Organic Chemistry, I.I.Sc.,

agents in the synthesis of α- and β-peptides Bangalore 560 012, March 26, 2001.

8. Studies on chemical synthesis of Dept. of Chemistry, University

peptidomimetics of Calicut, Calicut, March 23, 2005.

Popular lectures delivered in refresher courses as a resource person:

Sl. No. Title of course University Period No. of Title of lectures

lectures

1 15th Refresher Kerala, Sept. 9th & Four 1) Synthesis of

course in Trivandrum 10th 2004 peptidomimetics

Chemistry 2) Microwave irradiation in

Nov. 6th

organic synthesis

2 Refresher Cochin Two 1) Green chemistry

course in University of 2004 2) Recent trends in peptide

Chemistry Science and chemistry

Technology,

Kochi

3 5th Refresher Karnatak, Feb. 2nd & Four 1) Green Chemistry

course in Dharwad 3rd 2005 2) Solid phase peptide

Chemistry synthesis

3) Studies on chemical

Feb.14th

synthesis of peptidomimetics

4 Refresher Bangalore One Peptidomimetics

course in 2005

Chemistry

5 13th Refresher Mysore Feb.22nd Two 1) Green chemistry

course in 2005 2) Synthesis of

Chemistry

Jan. 3rd

peptidomimetics

6 1st Refresher Karnatak Two 1) Green /Sustainable

course in

Environmental

Sciences

Inter Karnatak

2006

16/1/2007

Chemistry

2) Microwave irradiation in

peptide synthesis

Two Green Chemistry-I

Disciplinary Green Chemistry- II

Refresher

Course in

Environmenta

l

Sciences

7 Refresher Bangalore 22/9/2008 Two Aspects of Green Chemistry Course in

Chemistry

Popular lectures delivered to UG students and faculty: 7

Sl. No. Date College Title of topic 1 18-12-2004 PES Degree College Peptides as drug candidates 2 8-8-2005 Sri Bhagavan Mahaveer Jain Microwave synthesis :

College Chemistry at the speed of light

3 1-9-2005 MES College of Science Green Chemistry

4 12-9-2005 Sri Bhagavan Mahaveer Jain Green Chemistry College

5 27-11-2005 MVJ College of Engineering Green Chemistry : An introduction

6 31-1-2006 Jyoti Nivas Degree College Green Chemistry

7 2-2-2006 Maharani’s Science College Green Chemistry

for Women

Research Collaborations :

Sl Name of Institution Area of interest

No. Scholar

1 Prof. D Dept. of Crystallography and Biophysics, Crystal structure of peptides

Velumurugan Univ. of Madras, Chennai. and peptidomemitics

2 Dr. C V Centre for Liquid Crystal Research, Exploration of peptides as

Yelamaggad Bangalore liquid crystals 3 Dr. S S Chimni Dept. of Chemistry, Guru Nanak Dev Development of peptide

Univ., Amritsar. catalysts in asymmetric

synthesis 4 Prof. Monika Indian Association for cultivation of X-ray crystallographic

Mukherjee Science, Kolkata studies of some amino acid

derivatives

5 Prof. T. N.

Guru Row Dept. of Solid State and Structural Chemistry Unit, Indian Institute of

Science, Bangalore

X-ray crystallographic studies of peptidomimetics

6 Prof. R. Srinivas

National Centre for Mass Spectrometry, Indian Institute of Chemical Technology,

Hyderabad 500 607, Andhra Pradesh,

India

Mass spectroscopic analysis of peptidomimetics

7 Dr. Nitish R Mahapatra

Indian Institute of Technology, Madras Studies on biological activity of human catestatin and its

analogues

Documents

CURRICULUM VITAE VOMMIMA V. SURESHBABU Bangalore … · 2018-09-14 · including native chemical ligation; Development of new synthetic methods Academic assignment : Served as sectional