Seznam vědeckých a publikačních aktivit, vyžádaných … · 2016-11-24 · Seznam vědeckých a publikačních aktivit, vyžádaných přednášek a grantů a další aktivity

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Seznam vědeckých a publikačních aktivit, vyžádaných přednášek a grantů

a další aktivity dokládající osobnost uchazeče

ABA Studie charakteru vědecké monografie v časopisech a sbornících vydané v zahraničních

vydavatelstvích

ABA01 Jampílek, Josef [UKOEXAF] (50% [2,18 AH]) - Kráľová, Katarína [UKOPRCUS] (50% [2,18 AH]):

Application of Nanotechnology in Agriculture and Food Industry, Its Prospects and Risks

Lit.: 432 zázn.

In: Ecological Chemistry and Engineering S. - Vol. 22, No. 3 (2015), s. 321-361 [4,36 AH]

Registrované v: wos, scopus

Indikátor časopisu:

IF (JCR) 2015= [2014-0,553]

ABA02 Kráľová, Katarína [UKOPRCUS] (70% [2,67 AH]) - Jampílek, Josef [UKOEXAF] (30% [1,14 AH]):

Impact of environmental contaminants on breast cancer

Lit.: 304 zázn.

In: Ecological Chemistry and Engineering S. - Vol. 22, No. 1 (2015), s. 9-44 [3,81 AH]



IF (JCR) 2015= [2014-0,553]

ABC Kapitoly ve vědeckých monografiích vydané v zahraničních vydavatelstvích

ABC01 Doležal, Martin (40%) - Zitko, Jan (25%) - Jampílek, Josef [UKOEXAF] (35%): Pyrazinecarboxylic

acid derivatives with antimycobacterial activity

Lit. 108 zázn.

In: Ed.: Cardona, P.J. : Understanding Tuberculosis : New approaches to fighting against drug resistance. -

Rijeka : InTech, 2012. - S. 233-262 [2,35 AH]. - ISBN 978-953-307-948-6

ABC02 Jampílek, Josef [UKOEXAF] (80%) - Dohnal, Jiří (20%): Investigation of carbohydrates and their

derivatives as crystallization modifiers

Lit. 126 zázn.

In: Ed.: Chang, Ch.F. : Carbohydrates : Comprehensive studies on glycobiology and glycotechnology. -

Rijeka : InTech, 2012. - S. 81-116 [2,74 AH]. - ISBN 978-953-51-0864-1

ABC03 Jampílek, Josef [UKOEXAF] (80%) - Dohnal, Jiří (20%): Alaptide as transdermal permeation modifier

Lit. 69 zázn.

In: Eds.: Nina Dragicevic, Howard I. Maibach : Percutaneous Penetration Enhancers Chemical Methods in

Penetration Enhancement : Modification of the Stratum Corneum. - Berlin : Springer, 2015. - S. 115-132

[1,38 AH]. - ISBN 978-3-662-47038-1

ABC04 Jampílek, Josef [UKOEXAF] (100%) : Azone(R) and its analogues as penetration enhancers

Lit. 114 zázn.

In: Eds.: Nina Dragicevic, Howard I. Maibach : Percutaneous Penetration Enhancers Chemical Methods in

Penetration Enhancement : Modification of the Stratum Corneum. - Berlin : Springer, 2015. - S. 69-105

[3,21 AH]. - ISBN 978-3-662-47038-1

ACB Vysokoškolské učebnice vydané v domácích vydavatelstvích

ACB01 Brusová, Hana (8%) - Dohnal, Jiří (8%) - Grafnetterová, Taťjana (4%) - Grünwaldová, Veronika (12%)

- Havlíček, Jaroslav (7%) - Jampílek, Josef [UKOEXAF] (20%) - Král, Vladimír (1%) - Opatřilová, Radka

(2%) - Pekárek, Tomáš (4%) - Plaček, Lukáš (7%)- Krumbholcová, Lucie (3%) - Řezáčová, Anna (6%) -

Setnička, Vladimír (9%) - Urbanová, Marie (9%): Moderní přístupy k farmaceutické analýze. - 1. vyd. -

Praha : Veterinární a farmaceutická univerzita Brno, 2010. - 500 s. [17,45 AH]

Jampílek, J.: 3,48 AH

Lit. 36 zázn.

ISBN 978-80-7305-085-6

2

ADC Vědecké práce v zahraničních karentovaných časopisech

ADC01 Jampílek, Josef [UKOEXAF] (80%) - Doležal, Martin (10%) - Dvořák, Bohumír (10%): Bis(4-

methoxyphenyl)disulfide formation through copper catalysts

Lit. 17 zázn.

In: Chemical papers. - Vol. 56, No. 3 (2002), s. 147-149

Registrované v: wos


IF (JCR) 2002=0,336

ADC02 Jampílek, Josef [UKOEXAF] (45%) - Doležal, Martin (10%) - Kuneš, Jiří (10%) - Víchová, Petra (10%)

- Jun, Daniel (10%) - Hanika, Jiří (5%) - O'Connor, Robert (5%) - Clynes, Martin (5%): Synthesis of(2E)-

2-methyl-3-(4-[4-(quinolin-2-ylmethoxy)phenyl]sulfanylphenyl)prop-2-enoic acid (VUFB 20609) and 2-

methyl-3-(4-[4-(quinolin-2-ylmethoxy)phenyl]sulfanylphenyl)propanoic acid (VUFB 20584) as potential

antileukotrienic agents

Lit. 30 zázn.

In: Journal of Pharmacy and Pharmacology. - Vol. 56, No. 6 (2004), s. 783-794



IF (JCR) 2004=1,348

Ohlasy (3):

[o1] 2007 Malecki, J.G. - Kruszynski, R. - Tabak, D. - Kusz, J.: Polyhedron, Vol. 26, No. 17, 2007, s. 5130

- SCI

[o1] 2008 Malecki, J.G. - Kusz, J. - Kruszynski, R. - Tabak, D. - Mazurak, Z.: Structural Chemistry, Vol.

19, No. 2, 2008, s. 263 - SCI

[o1] 2009 Brychtova, K. - Farsa, O. - Csollei, J.: Letters in Organic Chemistry, Vol. 6, No. 1, 2009, s. 28 -

SCI

ADC03 Jampílek, Josef [UKOEXAF] (45%) - Doležal, Martin (10%) - Kuneš, Jiří (10%) - Víchová, Petra (10%)

- Raich, Ivan (5%) - Jun, Daniel (10%) - O'Connor, Robert (5%) - Clynes, Martin (5%): Preparation of2-

(4-[4-(Quinolin-2-ylmethoxy)phenyl]sulfanylphenyl) propionic acid (VUFB 20615) and 2-methyl-2-(4-[4-

(quinolin-2- ylmethoxy)phenyl]sulfanylphenyl)propionic acid (VUFB 20623) as potential antileukotrienic

agents

Lit. 27 zázn.

In: Current Organic Chemistry. - Vol. 8, No. 13 (2004), s. 1235-1243



IF (JCR) 2004=2,775

Ohlasy (3):


- SCI


19, No. 2, 2008, s. 263 - SCI


SCI

ADC04 Jampílek, Josef [UKOEXAF] (60%) - Doležal, Martin (10%) - Kuneš, Jiří (10%) - Raich, Ivan (10%) -

Liška, František (10%): 4-substituted aryl bromides coupling with 4-methoxybenzene-1-thiol by means of

copper catalysts

Lit. 38 zázn.




IF (JCR) 2005=0,409

Ohlasy (3):


SCI

[o1] 2010 Del Rosso, P.G. - Almassio, M.F. - Bruno, M. - Garay, R.O.: Tetrahedron Letters, Vol. 51, No.

51, 2010, s. 6733 - SCI

[o1] 2012 Moosun, S. - Joule, J.A. - Bhowon, M.G. - Jhaumeer-Laulloo, S.: Phosphorus Sulfur and Silicon

and the Related Elements, Vol. 187, No. 11, 2012, s. 1400 - SCI

3

ADC05 Jampílek, Josef [UKOEXAF] (60%) - Doležal, Martin (10%) - Kuneš, Jiří (10%) - Šatínsky, Dalibor

(10%) - Raich, Ivan (10%): Novel regioselective preparation of 5-chloropyrazine-2-carbonitrile from

pyrazine-2-carboxamide and coupling study of substituted phenylsulfanylpyrazine- 2-carboxylic acid

derivatives

Lit. 41 zázn.




IF (JCR) 2005=3,102

Ohlasy (2):


SCI

[o1] 2009 Hu, L.X. - Arafa, R.K. - Ismail, M.A. - Patel, A. - Munde, M. - Wilson, W.D. - Wenzler, T. -

Brun, R. - Boykin, D.W.: Bioorganic & Medicinal Chemistry, Vol. 17, No. 18, 2009, s. 6658 - SCI

ADC06 Doležal, Martin (20%) - Pálek, Lukáš (15%) - Vinšová, Jarmila (5%) - Buchta, Vladimír (20%) -

Jampílek, Josef [UKOEXAF] (20%) - Kráľová, Katarína [UKOPRCUS] (20%): Substituted

Pyrazinecarboxamides: Synthesis and Biological Evaluation

Lit.: 27 zázn.

In: Molecules. - Vol. 11, No. 4 (2006), s. 242-256



IF (JCR) 2006=0,841

Ohlasy (20):

[o3] 2008 Martin, S. - Revathi, C. - Dayalan, A. - Mathivanan, N. - Shanmugaiya, V.: Rasayan Journal of

Chemistry, Vol. 1, No. 2, 2008, s. 378-389

[o1] 2009 Ukrainets, L.V. - Grinevich, L.A. - Tkach, A.A. - Bevz, O.V. - Slobodzian, S.V.: Khimiya

Geterotsiklicheskikh Soedinenii, No. 9, 2009, s. 1324-1337 - SCOPUS

[o1] 2009 Ukrainets, L.V. - Grinevich, L.A. - Tkach, A.A. - Bevz, O.V. - Slobodzian, S.V.: Chemistry of

Heterocyclic Compouds, Vol. 45, No. 9, 2009, s. 1058-1068 - SCI

[o1] 2010 Lee, J.H. - Myung, P.K. - Kim, S.J. - Sung, N.D.: Journal of Applied Biological Chemistry, Vol.

53, No. 4, 2010, s. 440-445 - SCOPUS

[o3] 2010 Meenakshi, S. – Malhotra, R.: Agricultural and Biological Research, Vol. 26, No. 2, 2010, s.

123-135

[o3] 2010 Tewatia, N. - Namdeo, K.P. - Jain, S.K. - Prajapati, S.K. - Singh, O. - Jain, V. - Kumar, P.:

Journal of the Institution of Chemists (India), Vol. 82, No. 5, 2010, s. 148-153

[o3] 2011 Lima, C.H.S. - Bispo, M.L.F. - de Souza, M.V.N.: Pirazinamida: Um Fármaco Essencial no

Tratamento da Tuberculose. In: Revista Virtual de Química, Vol. 3, No. 3, 2011, s. 159-180

[o3] 2011 Prasad, R. - Sharma, R.: 2D QSAR Analysis of pyrazinecarboxamides derivatives as an

herbicidal agent. In: Journal of Computational Methods in Molecular Design, Vol. 1, No. 1, 2011, s. 7-13

[o1] 2012 Patel, N. B. - Patel, H. R.: Arabian Journal of Chemistry, Vol. 5, Iss. 1, 2012, s. 81-91 - SCI ;

SCOPUS

[o3] 2011 Khalil, A. - Mohamed, S. I. - Eyada, H. A. - abdel Alaziz, T. A. - Ali, G. A. M. - Mohamed El-

Hag: Journal of Materials Science and Engineering A, Vol. 1, Iss. 2, 2011, s. 228-235

[o1] 2012 Lo Monte, F. - Kramer, T. - Gu, J. - Anumala, U.R. - Marinelli, L. - La Pietra, V. - Novellino, E.

- Franco, B. - Demedts, D. - Van Leuven, F. - Fuertes, A. - Dominguez, J.M. - Plotkin, B. - Eldar-

Finkelman, H. - Schmidt, B.: Journalof Medicinal Chemistry, Vol. 55, No. 9, 2012, s. 4407-4424 - SCI ;

SCOPUS

[o1] 2012 Tewatia, N. - Abidab, Namdeo, K.P.: Journal of Chemical and Pharmaceutical Research, Vol. 4,

No. 3, 2012, s. 1794-1798 - SCOPUS

[o3] 2012 Vikramjeet J. - Balasubramanian N. - Munish A.: A Review of Biological potential of

Pyrazinamide derivatives. In: Hygeia. Journal for drugs and medicines, Vol. 4, No. 1, 2012, s. 6

[o3] 2011 Sato, N.: Pyrazines. In: Science of Synthesis, Knowledge Updates, No. 4, 2011, s. 235-343

[o1] 2013 Zhang, R.Z. - Zhang, X.Z.: Indian Journal of Pure and Applied Physics, Vol. 51, No. 3, 2013, s.

164-173 - SCI ; SCOPUS

[o1] 2013 Helal, M.H. - Abbas, S.Y. - Salem, M.A. - Farag, A.A. - Ammar, Y.A.: Medicinal Chemistry

Research, Vol. 22, No. 11, 2013, s. 5598-5609 - SCOPUS ; SCI

[o3] 2014 Parimala Vaijayanthi, S. - Mathiyalagan, N.: Antibacterial, antifungal, anti-oxidant, anti-

inflammatory and anti-hypertensive activities of N-chloropyrazinamide. In: International Letters of

Chemistry, Physics and Astronomy, Vol. 7, 2014, s. 1-8

4

[o1] 2014 Nayak, P.S. - Narayana, B. - Anthal, S. - Gupta, V.K. - Kant, R.: Molecular Crystals and Liquid

Crystals, Vol. 592, No. 1, 2014, s. 199-208 - SCI ; SCOPUS

[o1] 2015 Verbitskiy, E.V. - Slepukhin, P.A. - Kravchenko, M.A. - Skornyakov, S.N. - Evstigneeva, N.P. -

Kungurov, N.V. - Zil'Berberg, N.V. - Rusinov, G.L. - Chupakhin, O.N. - Charushin, V.N.: Bioorganic and

Medicinal Chemistry Letters, Vol. 25, No. 3, 2015, s. 524-528 - SCI ; SCOPUS

[o1] 2016 Chylewska, A. - Sikorski, A. - Ogryzek, M. - Makowski, M.: Journal of Molecular Structure,

Vol. 1105, 2016, s. 104 - SCI; SCOPUS

ADC07 Jampílek, Josef [UKOEXAF] (75%) - Doležal, Martin (10%) - Opletalová, Veronika (10%) - Hart, Jiří

(5%): 5-lipoxygenase, leukotrienes biosynthesis and potential antileukotrienic agents

Lit. 102 zázn.

In: Current Medicinal Chemistry. - Vol. 13, No.2 (2006), s. 117-129



IF (JCR) 2006=5,207

Ohlasy (18):

[o1] 2006 Ward, W.O. - Delker, D.A. - Hester, S.D. - Thai, S.F. - Wolf, D.C. - Allen, J.W. - Nesnow, S.:

Toxicologic Pathology, Vol. 34, No. 7, 2006, s. 878 - SCI

[o1] 2006 Chen, X.X. - Sood, S. - Yang, C.S. - Li, N. - Sun, Z.: Current Cancer Drug Targets, Vol. 6, No.

7, 2006, s. 622 - SCI

[o1] 2007 Di Mari, J.F. - Saada, J.I. - Mifflin, R.C. - Valentich, J.D. - Powell, D.W.: American Journal of

Physiology-Gastrointestinal and Liver Physiology, Vol. 239, No. 4, 2007, s. G728 - SCI


- SCI

[o1] 2007 Lin, D. - Zhang, J.Y. - Sayre, L.M.: Journal of Organic Chemistry, Vol. 72, No. 25, 2007, s.

9480 - SCI


19, No. 2, 2008, s. 263 - SCI

[o1] 2008 Fiorucci, S. - Golebiowski, J. - Cabrol-Bass, D. - Antonczak, S.: Proteins-Structure Function and

Bioinformatics, Vol. 73, No. 2, 2008, s. 298 - SCI

[o1] 2009 Hoffmann, E.K. - Lambert, I.H - Pedersen, S.F.: Physiological Reviews, Vol. 89, No. 1, 2009, s.

277 - SCI

[o1] 2009 Gomes, A. - Fernandes, E. - Silva, A.M.S. - Pinto, D.C.G.A. - Santos, C.M.M. - Cavaleiro,

J.A.S. - Lima, J.L.F.C.: Biochemical Pharmacology, Vol. 78, No. 2, 2009, s. 177 - SCI

[o1] 2010 Adcock, I.M. - Marwick, J. - Casolari, P. - Contoli, M. - Chung, K.F. - Kirkham, P. - Papi, A. -

Caramori, G.: Current Pharmaceutical Design, Vol. 16, No. 32, 2010, s. 3573 - SCI

[o1] 2011 Pontiki, E. - Hadjipavlou-Litina, D. - Litinas, K. - Nicolotti, O. - Carotti, A.: European Journal

of Medicinal Chemistry, Vol. 46, No. 1, 2011, s. 200 - SCI

[o1] 2011 Li, Y. - Chen, S.H. - Ou, T.M. - Tan, J.H. - Li, D. - Gu, L.Q. - Huang, Z.S.: Bioorganic &

Medicinal Chemistry, Vol. 19, No. 6, 2011, s. 2083 - SCI

[o1] 2011 Tan, C.M. - Chen, G.S. - Chen, C.S. - Chang, P.T. - Chern, J.W.: Bioorganic & Medicinal

Chemistry, Vol. 19, No. 21, 2011, s. 6328 - SCI

[o1] 2012 Gomes, A. - Couto, D. - Alves, A. - Dias, I. - Freitas, M. - Porto, G. - Duarte, J.A. - Fernandes,

E.: Biofactors, Vol. 38, No. 5, 2012, s. 386 - SCI

[o1] 2013 Mathew, G. - Jacob, A. - Durgashivaprasad, E. - Reddy, N.D. - Unnikrishnan, M.K.:

International Immunopharmacology, Vol. 15, No. 1, 2013, s. 189 - SCI

[o1] 2013 Joshi, N. - Hoobler, E.K. - Perry, S. - Diaz, G. - Fox, B. - Holman, T.R.: Biochemistry, Vol. 52,

No. 45, 2013, s. 8035 - SCI

[o1] 2014 Meyers, D.A. - Bleecker, E.R. - Holloway, J.W. - Holgate, S.T.: Lancet Respiratory Medicine,

Vol. 2, No. 5, 2014, s. 415 - SCI

[o1] 2014 Sudha, A. - Srinivasan, P.: Pharmacognosy Magazine, Vol. 10, No. 39, 2014, s. 605 - SCI

ADC08 Musiol, Robert (20%) - Jampílek, Josef [UKOEXAF] (20%) - Buchta, Vladimír (5%) - Silva, Luis

(10%) - Niedbala, Halina (10%) - Podeszwa, Barbara (10%) - Palka, Anna (5%) - Majerz-Maniecka,

Katarzyna (5%) - Oleksyn, Barbara (5%) - Polanski, Jaroslaw(10%): Antifungal properties of new series of

quinoline derivatives

Lit. 20 zázn.

In: Bioorganic and Medicinal Chemistry. - Vol. 14, No. 10 (2006), s. 3592-3598



IF (JCR) 2006=2,624

5

Ohlasy (60):

[o1] 2006 Metwally, K.A. - Abdel-Aziz, L.M. - Lashine, E.S.M. - Hussemy, M.I. - Badawy, R.H.:

Bioorganic & Medicinal Chemistry, Vol. 14, No. 24, 2006, s. 8682 - SCI

[o1] 2007 Kamal, A. - Reddy, K.S. - Khan, M.N.A. - Shetty, R.V.C.R.N.C. - Ahmed, S.K. - Kumar, K.P. -

Murty, U.S.N.: Letters in Drug Design & Discovery, Vol. 4, No. 8, 2007, s. 586 - SCI

[o1] 2007 Bouraiou, A. - Belfaitah, A. - Bouacida, S. - Benard-Rocherulle, P. - Carboni, B.: Acta

Crystallographica Section E-Structure Reports Online, Vol. 63, 2007, s. O2135 - SCI


- SCI

[o1] 2008 Kaplancikli, Z.A. - Turan-Zitouni, G. - Ozdemir, A. - Revial, G.: Journal of Enzyme Inhibition

and Medicinal Chemistry, Vol. 23, No. 6, 2008, s. 870 - SCI

[o1] 2008 Ali, I.A.I. - Fathalla, W. - El Rayes, S.M.: Arkivoc, Part 13, 2008, s. 188 - SCI

[o1] 2008 Prasad, A.K. - Kumar, P. - Dhawan, A. - Chhillar, A.K. - Sharma, D. - Yadav, V. - Kumar, M. -

Jha, H.N. - Olsen, C.E. - Sharma, G.L. - Parmar, V.S.: Bioorganic & Medicinal Chemistry Letters, Vol. 18,

No. 6, 2008, s. 2161 - SCI


19, No. 2, 2008, s. 263 - SCI

[o1] 2008 Abdel-Hafez, S.H. - Hussein, M.A.: Archiv der Pharmazie, Vol. 341, No. 4, 2008, s. 246 - SCI

[o1] 2008 Gomez, C.M.M. - Kouznetsov, V.V. - Sortino, M.A. - Alvarez, S.L. - Zacchino, S.A.:


[o1] 2009 Kaiser, C.R. - Pais, K.C. - de Souza, M.V.N. - Wardell, J.L. - Wardell, S.M.S.V. - Tiekink,

E.R.T.: Crystengcomm, Vol. 11, No. 6, 2009, s. 1140 - SCI

[o1] 2009 de Souza, M.V.N. - Pais, K.C. - Kaiser, C.R. - Peralta, M.A. - Ferreira, M.D. - Lourenco,

M.C.S.: Bioorganic & Medicinal Chemistry, Vol. 17, No. 4, 2008, s. 1480 - SCI

[o1] 2009 da Silva, M.A.V.R. - da Silva, M.D.M.C.R. - Ferreira, A.I.M.C.L. - Santos, A.F.L.O.M. - Galvo,

T.L.P.: Journal of Chemical Thermodynamics, Vol. 41, No. 10, 2009, s. 1080 - SCI

[o1] 2010 Howie, R.A. - de Souza, M.V.N. - Ferreira, M.D. - Kaiser, C.R. - Wardell, J.L. - Wardell,

S.M.S.V.: Zeitschrift fur Kristallographie, Vol. 225, No. 10, 2010, s. 447 - SCI

[o1] 2010 Chang, F.S. - Chen, W.C. - Wang, C.H. - Tzeng, C.C. - Chen, Y.L.: Bioorganic & Medicinal


[o1] 2010 Avetisyan, A.A. - Aleksanyan, I.L. - Ambartsumyan, L.P.: Russian Journal of Organic


[o1] 2010 Murugesan, S. - Ganguly, S. - Maga, G.: Journal of Chemical Sciences, Vol. 122, No. 2, 2010, s.

176 - SCI

[o1] 2010 Fun, H.K. - Chanawanno, K. - Kobkeatthawin, T. - Chantrapromma, S.: Acta Crystallographica

Section E-Structure Reports Online, Vol. 66, 2010, s. U3214 - SCI

[o1] 2010 Ganguly, S. - Murugesan, S.: Journal of the Indian Chemical Society, Vol. 87, No. 7, 2010, s.

885 - SCI

[o1] 2010 Gao, W.T. - Cheng, X.P. - Li, Y.: Heterocycles, Vol. 81, No. 8, 2010, s. 1930 - SCI

[o1] 2010 Prabha, K. - Vennila, K.N. - Prasad, K.J.R. - Velmurugan, D.: Acta Crystallographica Section E-

Structure Reports Online, Vol. 66, 2010, s. U1222 - SCI

[o1] 2010 Kumar, S. - Bawa, S. - Drabu, S. - Kumar, R. - Panda, B.P.: Latin American Journal of

Pharmacy, Vol. 29, No. 6, 2010, s. 975 - SCI

[o1] 2011 El-Agrody, A.M. - Al-Ghamdi, A.M.: Arkivoc, Part 11, 2011, s. 146 - SCI

[o1] 2011 Djamel, D. - Tahar, D. - Djahida, H. - Hanane, H. - Salah, C.: Acta Crystallographica Section E-

Structure Reports Online, Vol. 67, 2011, s. U377 - SCI

[o1] 2011 Kumar, S. - Bawa, S. - Kaushik, D. - Panda, B.P.: Archiv der Pharmazie, Vol. 344, No. 7, 2011,

s. 480 - SCI

[o1] 2011 Thakre, W.B. - Meshram, J.S.: Indian Journal of Heterocyclic Chemistry, Vol. 21, No. 1, 2011,

s. 68 - SCI

[o1] 2011 Ziemons, E. - Bourichi, H. - Mantanus, J. - Rozet, E. - Lebrun, P. - Essassi, E. - Cherrah, Y. -

Bouklouze, A. - Hubert, P.: Journal of Pharmaceutical and Biomedical Analysis, Vol. 55, No. 5, 2011, s.

1212 - SCI

[o1] 2011 Yang, G.H. - Li, Y.X. - Yan, S.H. - Dai, L. - Zhao, B.: Acta Chimica Sinica, Vol. 69, No. 15,

2011, s. 1750 - SCI

[o1] 2011 Kumar, A. - Rao, V.K.: Synlett, No. 15, 2011, s. 2162 - SCI

[o1] 2011 Haggag, S.M.S. - Farag, A.A.M. - Mahmoud, M.E.: Polyhedron, Vol. 30, No. 16, 2011, s. 2732

- SCI

[o1] 2011 Robak, W. - Apostoluk, W. - Ochromowicz, K.: Journal of Chemical and Engineering Data,

Vol. 56, No. 11, 2011, s. 3983 - SCI

6

[o1] 2011 Alshahateet, S.F. - Al-Zereini, W.A. - Alghezawi, N.M.: Journal of Chemical Crystallography,

Vol. 41, No. 12, 2011, s. 1811 - SCI

[o1] 2012 Thapa, P. - Lee, E.S.: Bulletin of the Korean Chemical Society, Vol. 33, No. 5, 2012, s. 1772 -

SCI

[o1] 2012 Li, V.M. - Gavrishova, T.N. - Budyka, M.F.: Russian Journal of Organic Chemistry, Vol. 48,

No. 6, 2012, s. 828 - SCI

[o1] 2012 Kouznetsov, V.V. - Gomez, C.M.M. - Derita, M.G. - Svetaz, L. - del Olmo, E. - Zacchino, S.A.:


[o1] 2012 Tukulula, M. - Little, S. - Gut, J. - Rosenthal, P.J. - Wan, B.J. - Franzblau, S.G. - Chibale, K.:

European Journal of Medicinal Chemistry, Vol. 57, 2012, s. 267 - SCI

[o1] 2012 El-Agrody, A.M. - Khattab, E.S.A.E.H. - Fouda, A.M. - Al-Ghamdi, A.M.: Medicinal

Chemistry Research, Vol. 21, No. 12, 2012, s. 4213 - SCI

[o1] 2013 Goncalves, R.S.B. - de Souza, M.V.N. - Wardell, J.L. - Wardell, S.M.S.V.: Zeitschrift fur

Kristallographie, Vol. 228, No. 12, 2013, s. 668 - SCI

[o1] 2013 Savegnago, L. - Vieira, A.I. - Seus, N. - Goldani, B.S. - Castro, M.R. - Lenardao, E.J. - Alves,

D.: Tetrahedron Letters, Vol. 54, No. 1, 2013, s. 44 - SCI

[o1] 2013 Derita, M. - Montenegro, I. - Garibotto, F. - Enriz, R.D. - Fritis, M.C. - Zacchino, S.A.:

Molecules, Vol. 18, No. 2, 2013, s. 2051 - SCI

[o1] 2013 Serrao, E. - Debnath, B. - Otake, H. - Kuang, Y.T. - Christ, F. - Debyser, Z. - Neamati, N.:

Journal of Medicinal Chemistry, Vol. 56, No. 6, 2013, s. 2322 - SCI

[o1] 2013 Sun, W.Q. - Yuan, G.Z. - Liu, J.X. - Ma, L. - Liu, C.B.: Spectrochimica Acta Part A-Molecular

and Biomolecular Spectroscopy, Vol. 106, 2013, s. 283 - SCI

[o1] 2013 Patel, R.V. - Kumari, P. - Chikhalia, K.H.: Medicinal Chemistry, Vol. 9, No. 4, 2013, s. 607 -

SCI

[o1] 2013 De Leon, F. - Kalagara, S. - Navarro, A.A. - Mito, S.: Tetrahedron Letters, Vol. 54, No. 24,

2013, s. 3149 - SCI

[o1] 2013 Vandekerckhove, S. - Tran, H.G. - Desmet, T. - D'hooghe, M.: Bioorganic & Medicinal

Chemistry, Letters, Vol. 23, No. 16, 2013, s. 4643 - SCI

[o1] 2013 Boechat, N. - Bastos, M.M.: Current Topics in Medicinal Chemistry, Vol. 13, No. 22, 2013, s.

2904 - SCI

[o1] 2014 Gok, D. - Kasimogullari, R. - Cengiz, M. - Mert, S.: Journal of Heterocyclic Chemistry, Vol. 51,

No. 1, 2014, s. 232 - SCI

[o1] 2014 Yernale, N.G. - Mathada, M.B.H.: Bioinorganic Chemistry and Applications, 2014, Article No.

314963 - SCI

[o1] 2014 Ahmed, A. - Dhara, S. - Singha, R. - Nuree, Y. - Sarkar, P. - Ray, J.K.: RSC Advances, Vol. 4,

No. 95, 2014, s. 53141 - SCI

[o1] 2014 Peng, H.K. - Lin, I.L. - Lee, C.C. - Wang, L.Y. -Tzeng, C.C. - Chang, J.G. - Yang, S.C.:

Medicinal Chemistry Research, Vol. 23, No. 3, 2014, s. 1446 - SCI

[o1] 2014 Patel, A.B. - Kumari, P. - Chikhalia, K.H.: Catalysis Letters, Vol. 144, No. 7, 2014, s. 1338 -

SCI

[o1] 2014 Gavrishova, T.N. - Li, V.M. - Karpov, O.N. - Budyka, M.F.: Russian Journal of Organic


[o1] 2014 Haggag, S.M.S. - Farag, A.A.M. - Refea, M.A.: Thin Solid Films, Vol. 566, 2014, s. 44 - SCI

[o1] 2014 Vairavelu, L. - Prasad, K.J.R.: Journal of Chemical Sciences, Vol. 126, No. 6, 2014, s. 1902 -

SCI

[o1] 2015 Yadav, T. - Kishore, D. - Singh, B.: British Journal of Pharmaceutical Research, Vol. 8, No. 3,

2015, Article No. 19615 - SCI

[o1] 2015 Akhter, M. - Saha, R. - Tanwar, O. - Alam, M.M. - Zaman, M.S.: Medicinal Chemistry

Research, Vol. 24, No. 2, 2015, s. 890 - SCI

[o1] 2015 Li, Y.Q. - Chibale, K. - Smith, G.S.: Journal of Chemical Crystallography, Vol. 45, No. 4, 2015,

s. 206 - SCI

[o1] 2015 Tummatorn, J. - Poonsilp, P. - Nimnual, P. - Janprasit, J. - Thongsornkleeb, C. - Ruchirawat, S.:

Journal of Organic Chemistry, Vol. 80, No. 9, 2015, s. 4525 - SCI

[o1] 2015 Yaragorla, S. - Singh, G. - Dada, R.: Tetrahedron Letters, Vol. 56, No. 43, 2015, s. 5929 - SCI

[o1] 2015 Cho, S.K. - Song, J.H. - Lee, E.J. - Lee, D.H. - Hahn, J.T. - Jung, D.I.: Bulletin of the Korean

Chemical Society, Vol. 36, No. 11, 2015, s. 2749 - SCI

ADC09 Vinšová, Jarmila (20%) - Čermáková, Kateřina (10%) - Tomečková, Alexandra (10%) - Jampílek, Josef

[UKOEXAF] (10%) - Čermák, Pavel (10%) - Kuneš, Jiří (10%) - Doležal, Martin (10%) - Štaud, František

(10%) - Čečková, Martina (10%): Synthesis andantimicrobial evaluation of new 2-substituted 5,7-di-tert-

butylbenzoxazoles

7

Lit. 31 zázn.




IF (JCR) 2006=2,624

Ohlasy (51):

[o1] 2007 Janin, Y.L.: Bioorganic & Medicinal Chemistry, Vol. 15, No. 7, 2007, s. 2513 - SCI

[o1] 2007 Hioki, H. - Matsushita, K. - Kubo, M. - Harada, K. - Kodama, M. - Fukuyama, Y.: Tetrahedron,

Vol. 63, No. 46, 2007, s. 11324 - SCI

[o1] 2008 Soni, K. - Samota, M.K. - Jhajharia, P. - Seth, G.: Phosphorus Sulfur and Silicon and the Related

Elements, Vol. 183, No. 11, 2008, s. 2853 - SCI

[o1] 2008 Kumar, D. - Rudrawar, S. - Chakraborti, A.K.: Australian Journal of Chemistry, Vol. 61, No. 11,

2008, s. 887 - SCI

[o1] 2008 Gottumukkala, A.L. - Derridj, F. - Djebbar, S. - Doucet, H.: Tetrahedron Letters, Vol. 49, No.

18, 2008, s. 2930 - SCI

[o1] 2008 Evangelio, E. - Saiz-Poseu, J. - Maspoch, D. - Wurst, K. - Busque, F. - Ruiz-Molina, D.:

European Journal of Inorganic Chemistry, No. 14, 2008, s. 2285 - SCI

[o1] 2008 Salcedo, A. - Neuville, L. - Zhu, J.P.: Journal of Organic Chemistry, Vol. 73, No. 9, 2008, s.

3603 - SCI

[o1] 2008 Siddiqui, N. - Sarafroz, M. - Alam, M.M. - Ahsan, W.: Acta Poloniae Pharmaceutica, Vol. 65,

No. 4, 2008, s. 455 - SCI

[o1] 2008 Costa, S.P.G. - Oliveira, E. - Lodeiro, C. - Raposo, M.M.M.: Tetrahedron Letters, Vol. 49, No.

36, 2008, s. 5261 - SCI

[o1] 2009 Heravi, M.M. - Baghernejad, B. - Oskooie, H.A.: Chinese Journal of Chemistry, Vol. 27, No. 2,

2009, s. 383 - SCI

[o1] 2009 Kumar, A. - Maurya, R.A. - Ahmad, P.: Journal of Combinatorial Chemistry, Vol. 11, No. 2,

2009, s. 201 - SCI

[o1] 2009 Horvati, K. - Mezo, G. - Szabo, N. - Hudecz, F. - Bosze, S.: Journal of Peptide Science, Vol. 15,

No. 5, 2009, s. 391 - SCI

[o1] 2009 Klimesova, V. - Koci, J. - Waisser, K. - Kaustova, J. - Mollmann, U.: European Journal of


[o1] 2009 Husain, A. - Akhter, M.S.A. - Khatoon, Y.: Indian Journal of Heterocyclic Chemistry, Vol. 19,

No. 1, 2009, s. 94 - SCI

[o1] 2009 Chen, W.H. - Pang, Y.: Tetrahedron Letters, Vol. 50, No. 48, 2009, s. 6683 - SCI

[o1] 2010 Kumar, A. - Maurya, R.A. - Saxena, D.: Molecular Diversity, Vol. 15, No. 2, 2010, s. 341

[o1] 2010 Chauhan, P.M.S. - Sunduru, N. - Sharma, M.: Future Medicinal Chemistry, Vol. 2, No. 9, 2010,

s. 1500 - SCI

[o1] 2010 Kumar, A. - Sharma, S. - Maurya, R.A.: Tetrahedron Letters, Vol. 51, No. 48, 2010, s. 6226 -

SCI

[o1] 2010 Rossi, R. - Bellina, F. - Lessi, M.: Synthesis-Stuttgart, No. 24, 2010, s. 4153 - SCI

[o1] 2011 Sun, Q. - Wu, R.Z. - Cai, S.T. - Lin, Y.A. - Sellers, L. - Sakamoto, K. - He, B.A. - Peterson,

B.R.: Journal of Medicinal Chemistry, Vol. 54, No. 5, 2011, s. 1139 - SCI

[o1] 2011 Chari, M.A. - Shobha, D. - Sasaki, T.: Tetrahedron Letters, Vol. 52, No. 43, 2011, s. 5580 - SCI

[o1] 2012 Vaillard, V.A. - Guastavino, J.F. - Buden, M.E. - Bardagi, J.I. - Barolo, S.M. - Rossi, R.A.:

Journal of Organic Chemistry, Vol. 77, No. 3, 2012, s. 1519 - SCI

[o1] 2012 Horvati, K. - Bacsa, B. - Szabo, N. - David, S. - Mezo, G. - Grolmusz, V. - Vertessy, B. -

Hudecz, F. - Bosze, S.: Bioconjugate Chemistry, Vol. 223, No. 5, 2012, s. 907 - SCI

[o1] 2012 Aparaschivei, R. - Holban, M. - Sunel, V. - Popa, M. - Desbrieres, J.: Cellulose Chemistry and

Technology, Vol. 46, No. 5-6, 2012, s. 306 - SCI

[o1] 2012 Li, Y. - Tao, X.Y. - Lin, G.H. - Gao, W.T.: Heterocyclic Communications, Vol. 18, No. 4, 2012,

s. 210 - SCI

[o1] 2012 Gao, W.T. - Lin, G.H. - Li, Y. -Tao, X.Y. - Liu, R. - Sun, L.J.: Beilstein Journal of Organic

Chemistry, Vol. 8, 2012, s. 1857 - SCI

[o1] 2012 Abdou, W.M. - Barghash, R.F. - Sediek, A.A.: European Journal of Medicinal Chemistry, Vol.

57, 2012, s. 372 - SCI

[o1] 2013 Salehzadeh, H. - Nematollahi, D. - Hesari, H.: Green Chemistry, Vol. 15, No. 9, 2013, s. 2446 -

SCI

[o1] 2013 Nieddu, G. - Giacomelli, G.: Tetrahedron, Vol. 69, No. 2, 2013, s. 795 - SCI

[o1] 2013 Protasenko, N.A. - Poddel'sky, A.I. - Bogomyakov, A.S. - Somov, N.V. - Abakumov, G.A. -

Cherkasov, V.K.: Polyhedron, Vol. 49, No. 1, 2013, s. 243 - SCI

8

[o1] 2013 Park, H.J. - Park, M.S. - Lee, T.H. - Park, K.H.: Journal of Heterocyclic Chemistry, Vol. 50, No.

3, 2013, s. 667 - SCI

[o1] 2013 Abdou, W.M. - Barghash, R.F. - Khidre, R.E.: Monatshefte fur Chemie, Vol. 144, No. 8, 2013,

s. 1242 - SCI

[o1] 2013 Arisoy, M. - Temiz-Arpaci, O. - Kaynak-Onurdag, F. - Ozgen, S.: Zeitschrift fur Naturforschung

Section C-A Journal of Biosciences, Vol. 68, No. 11-12, 2013, s. 460 - SCI

[o1] 2013 Li, A.K. - Ma, H.Y. - Huang, J.L.: Organometallics, Vol. 32, No. 24, 2013, s. 7469 - SCI

[o1] 2014 Rana, D.N. - Chhabria, M.T. - Shah, N.K. - Brahmkshatriya, P.S.: Medicinal Chemistry

Research, Vol. 23, No. 1, 2014, s. 381 - SCI

[o1] 2014 Abdou, W.M. - Ganoub, N.A. - Barghash, R.F.: Synthetic Communications, Vol. 44, No. 18,

2014, s. 2678 - SCI

[o1] 2014 Ashfaq, M. - Shah, S.S.A. - Najam, T. - Ahmad, M.M. - Tabassum, R. - Rivera, G.: Current


[o1] 2014 Pardeshi, S.D. - Sonar, J.P. - Pawar, S.S. - Dekhane, D. - Gupta, S. - Zine, A.M. - Thore, S.N.:

Journal of the Chilean Chemical Society, Vol. 59, No. 1, 2014, s. 2340 - SCI

[o1] 2014 Rana, D.N. - Chhabria, M.T. - Shah, N.K. - Brahmkshatriya, P.S.: Medicinal Chemistr Research,

Vol. 23, No. 5, 2014, s. 2228 - SCI

[o1] 2014 Haider, S. - Alam, M.S. - Hamid, H. - Shafi, S. - Dhulap, A. - Hussain, F. - Alam, P. - Umar, S. -

Pasha, M.A.Q. - Bano, S. - Nazreen, S. - Ali, Y. - Kharbanda, C.: European Journal of Medicinal

Chemistry, Vol. 81, 2014, s. 217 - SCI

[o1] 2014 Aparaschivei, R. - Sunel, V. - Popa, M. - Desbrieres, J.: Journal of Heterocyclic Chemistry, Vol

51, No. 4, 2014, s. 1132 - SCI

[o1] 2014 Abdou, W.M. - Ganoub, N.A. - Sabry, E.: Acta Pharmaceutica, Vol. 64, No. 3, 2014, s. 284 -

SCI

[o1] 2014 Barghash, R.F. - Ganoub, N.A. - Abdou, W.M.: Monatshefte fur Chemie, Vol. 145, No. 10,

2014, s. 1630 - SCI

[o1] 2014 Horvati, K. - Bacsa, B. - Kiss, E. - Gyulai, G. - Fodor, K. - Balka, G. - Rusvai, M. - Szabo, E. -

Hudecz, F. - Bosze, S.: Bioconjugate Chemistry, Vol. 25, No. 12, 2014, s. 2268 - SCI

[o1] 2015 Zhang, X.X. - Lin, Y.Y. - Zhang, J. - Cao, S.: RSC Advances, Vol. 5, No. 11, 2014, s. 7908 -

SCI

[o1] 2015 Kochem, A. - Gellon, G. - Jarjayes, O. - Philouze, C. - d'Hardemare, A.D. - van Gastel, M. -

Thomas, F.: Dalton Transactions, Vol. 44, No. 28, 2015, s. 12756 - SCI

[o1] 2015 VenkatRamani, S. - Ghiviriga, I. - Abboud, K.A. - Veige, A.S.: Dalton Transactions, Vol. 44,

No. 42, 2015, s. 18486 - SCI

[o1] 2015 Khandan-Barani, K. - Maghsoodlou, M.T. - Hassanabadi, A. - Hosseini-Tabatabaei, M.R. -

Saffari, J. - Kangani, M.: Research on Chemical Intermediates, Vol. 41, No. 5, 2015, s. 3016 - SCI

[o1] 2015 Lv, M.Y. - Zheng, H.M. - Li, Y. - Gao, W.T.: Research on Chemical Intermediates, Vol. 41, No.

10, 2015, s. 6939 - SCI

[o1] 2015 Abdou, W.M. - Kamel, A.A. - Khidre, M.D.: Journal of Heterocyclic Chemistry, Vol 52, No. 6,

2015, s. 1662 - SCI

[o1] 2015 Qiu, J. - Zhang, Y.D. - Hua, C.W. - Gou, X.F. - Chen, B. - Zhao, J.L.: Heterocycles, Vol. 91,

No. 11, 2015, s. 2162 - SCI

ADC10 Imramovský, Aleš (20%) - Polanc, Slovenko (10%) - Vinšová, Jarmila (20%) - Kočevar, Marijan (10%)

- Jampílek, Josef [UKOEXAF] (15%) - Rečková, Zuzana (15%) - Kaustová, Jarmila (10%): A new

modification of anti-tubercular active molecules

Lit. 25 zázn.




IF (JCR) 2007=2,662

Ohlasy (46):

[o1] 2007 Rollas, S. - Kucukguzel, S.G.: Molecules, Vol. 12, No. 8, 2007, s. 1939 - SCI

[o1] 2008 Fun, H.K. - Chantrapromma, S. - Jana, S. - Hazra, A. - Goswami, S.: Acta Crystallographica

Section E-Structure Reports Online, Vol. 64, 2008, s. U4082 - SCI

[o1] 2008 Turan-Zitouni, G. - Ozdemir, A. - Kaplancikli, Z.A. - Benkli, K. - Chevallet, P. - Akalin, G.:

European Journal of Medicinal Chemistry, Vol. 43, No. 5, 2008, s. 985 - SCI

[o1] 2009 Abdel-Rahman, H.M. - El-Koussi, N.A. - Hassan, H.Y.: Archiv der Pharmazie, Vol. 342, No. 8,

2009, s. 99 - SCI

[o1] 2009 Rogoza, L.N. - Salakhutdinov, N.F. - Tolstikov, G.A.: Mini-Reviews in Organic Chemistry,

Vol. 6, No. 2, 2009, s. 151 - SCI

9

[o1] 2010 Ajani, O.O. - Obafemi, C.A. - Nwinyi, O.C. - Akinpelu, D.A.: Bioorganic & Medicinal


[o1] 2010 Eswaran, S. - Adhikari, A.V. - Pal, N.K. - Chowdhury, I.H.: Bioorganic & Medicinal Letters,

Vol. 20, No. 3, 2010, s. 1044 - SCI

[o1] 2010 Abdel-Aal, W.S. - Hassan, H.Y. - Aboul-Fadl, T. - Youssef, A.F.: European Journal of


[o1] 2010 Turan-Zitouni, G. - Kaplancikli, Z.A. - Ozdemir, A.: European Journal of Medicinal Chemistry,

Vol. 45, No. 5, 2010, s. 2088 - SCI

[o1] 2010 Patel, N.B. - Patel, V.N. - Patel, H.R. - Shaikh, F.M. - Patel, J.C.: Acta Poloniae Pharmaceutica,

Vol. 67, No. 3, 2010, s. 275 - SCI

[o1] 2010 Sharma, P.C. - Jain, A. - Jain, S. - Pahwa, R. - Yar, M.S.: Journal of Enzyme Inhibition and


[o1] 2010 Abdel-Aziz, M. - Abdel-Rahman, H.M.: European Journal of Medicinal Chemistry, Vol. 45, No.

8, 2010, s. 3388 - SCI


s. 1500 - SCI

[o1] 2010 Wiles, J.A. - Bradbury, B.J. - Pucci, M.J.: Expert Opinion on Therapeutic Patents, Vol. 20, No.

10, 2010, s. 1319 - SCI

[o1] 2010 Patel, N.B. - Patel, J.C. - Patel, V.N.: Chinese Journal of Chemistry, Vol. 28, No. 10, 2010, s.

1997 - SCI

[o1] 2010 Mantu, D. - Luca, M.C. - Moldoveanu, C. - Zbancioc, G. - Mangalagiu, I.I.: European Journal of


[o1] 2011 Jiang, X.L. - Cui, Y.B. - Cao, S.H.: Zhongguo Kangshengsu Zazhi, Vol. 36, No. 4, 2011, s. 263

- SCI

[o1] 2011 Joshi, R.S. - Mandhane, P.G. - Badadhe, P.V. - Gill, C.H.: Ultrasonics Sonochemistry, Vol. 18,

No. 3, 2011, s. 738 - SCI

[o1] 2011 Khidre, R.E. - Abu-Hashem, A.A. - El-Shazly, M.: European Journal of Medicinal Chemistry,

Vol. 46, No. 10, 2011, s. 5064 - SCI

[o1] 2012 Shaquiquzzaman, M. - Khan, S.A. - Amir, M. - Alam, M.M.: Saudi Pharmaceutical Journal,

Vol. 20, No. 2, 2012, s. 154 - SCI

[o1] 2012 Gaikwad, N.D. - Patil, S.V. - Bobade, V.D.: Bioorganic & Medicinal Chemistry Letters, Vol.

22, No. 10, 2012, s. 3454 - SCI

[o1] 2012 Malhotra, M. - Sharma, S. - Deep, A.: Medicinal Chemistry Research, Vol. 21, No. 7, 2012, s.

1244 - SCI

[o1] 2012 Malhotra, M. - Sharma, S. - Deep, A.: Acta Poloniae Pharmaceutica, Vol. 69, No. 4, 2012, s.

644 - SCI

[o1] 2012 Gaikwad, N.D. - Patil, S.V. - Bobade, V.D.: European Journal of Medicinal Chemistry, Vol. 54,

2012, s. 302 - SCI

[o1] 2012 Wang, S. - Jia, X.D. - Liu, M.L. - Lu, Y. - Guo, H.Y.: Bioorganic & Medicinal Chemistry

Letters, Vol. 22, No. 18, 2012, s. 5975 - SCI

[o1] 2012 Sarnpitak, P. - Tsirulnikov, S. - Krasavin, M.: Tetrahedron Letters, Vol. 53, No. 48, 2012, s.

6543 - SCI

[o1] 2012 Judge, V. - Narasimhan, B. - Ahuja, M.: Medicinal Chemistry Research, Vol. 21, No. 12, 2012,

s. 3957 - SCI

[o1] 2012 Shaquiquzzaman, M. - Khan, S.A. - Amir, M. - Alam, M.M.: Journal of Enzyme Inhibition and


[o1] 2013 Rudrapal, M. - Satyanandam, R.S. - Swaroopini, T.S. - Lakshmi, T.N. - Jaha, S.K. - Zaheera, S.:


[o1] 2013 Matei, L. - Bleotu, C. - Baciu, I. - Draghici, C. - Ionita, P. - Paun, A. - Chifiriuc, M.C. - Sbarcea,

A. - Zarafu, I.: Bioorganic & Medicinal Chemistry, Vol. 21, No. 17, 2013, s. 5361 - SCI

[o1] 2013 Hagar, M. - Soliman, S.M. - Ibid, F. - El Ashry, E.H.: Journal of Moleular Structure, Vol. 1049,

2013, s. 188 - SCI

[o1] 2013 Anbazhagan, R. - Sankaran, K.R.: Journal of Moleular Structure, Vol. 1050, 2013, s. 80 - SCI

[o1] 2013 Refat, H.M. - Fadda, A.A.: European Journal of Medicinal Chemistry, Vol. 70, 2013, s. 426 -

SCI

[o1] 2014 Refat, H.M. - Fadda, A.A.: Synthetic Communications, Vol. 44, No. 15, 2014, s. 2154 - SCI

[o1] 2014 Bhat, M.A.: Acta Poloniae Pharmaceutica, Vol. 71, No. 5, 2014, s. 770 - SCI

[o1] 2014 Malhotra, M. - Sharma, R. - Rathee, D. - Phogat, P. - Deep, A.: Arabian Journal of Chemistry,

Vol. 7, No. 5, 2014, s. 671 - SCI

10

[o1] 2014 dos Reis, F.D. - Gatti, I.C. - Garcia, H.C. - de Oliveira, V.E. - de Oliveira, L.F.C.: Journal of

Physical Chemistry A, Vol. 118, No. 49, 2014, s. 11528 - SCI

[o1] 2015 Saha, R. - Alam, M.M. - Akhter, M.: RSC Advances, Vol. 5, No. 17, 2015, s. 12820 - SCI

[o1] 2015 Mathew, B. - Suresh, J. - Ahsan, M.J. - Mathew, G.E. - Usman, D. - Subramanyan, P.N.S. -

Safna, K.F. - Maddela, S.: Infectious Disorders - Drug Targets, Vol. 15, No. 2, 2015, s. 88 - SCI

[o1] 2015 Anbazhagan, R. - Sankaran, K.R.: Spectrochimica Acta Part A-Molecular and Biomolecular

Spectroscopy, Vol. 135, 2015, s. 993 - SCI

[o1] 2015 Kamble, R.D. - Hese, S.V. - Meshram, R.J. - Kote, J.R. - Gacche, R.N, - Dawane, B.S.:


[o1] 2015 Casanova, B.B. - Muniz, M.N. - de Oliveira, T. - de Oliveira, L.F. - Machado, M.M. -

Fuentefria, A.M. - Gosmann, G. - Gnoatto, S.C.B.: Molecules, Vol. 20, No. 5, 2015, s. 9241 - SCI

[o1] 2015 Refat, H.M. - Fadda, A.A.: Heterocycles, Vol. 91, No. 6, 2015, s. 1226 - SCI

[o1] 2015 Yurttas, L. - Kaplancikli, Z.A. - Canturk, Z. - Gencer, H.K.: Phosphorus Sulfur and Silicon and

the Related Elements, Vol. 190, No. 7, 2015, s. 1191 - SCI

[o1] 2015 El-Faham, A. - Farooq, M. - Khattab, S.N. - Abutaha, N. - Wadaan, M.A. - Ghabbour, H.A. -

Fun, H.K.: Molecules, Vol. 20, No. 8, 2015, s. 14655 - SCI

[o1] 2015 Dikkar, A.B. - Pethe, G.B. - Aswar, A.S.: Russian Journal of Physical Chemistry A, Vol. 89,

No. 12, 2015, s. 2203 - SCI

ADC11 Musiol, Robert (10%) - Kráľová, Katarína [UKOPRCUS] (10%) - Richardson, Des R. (10%) -

Kalinowski, Danuta (10%) - Podeszwa, Barbara (10%) - Finster, Jacek (10%) - Niedbala, Halina (10%) -

Palka, Anna (10%) - Polański, Jaroslaw (10%) - Jampílek, Josef [UKOEXAF] (10%): Investigating

biological activity spectrum for novel quinoline analogues

Lit.: 32 zázn.

In: Bioorganic & Medicinal Chemistry. - Vol. 15, No. 3 (2007), s. 1280-1288



IF (JCR) 2007=2,662

Ohlasy (74):

[o1] 2007 Malecki, J.G. - Kruszynski, R. - Tabak, D. - Kusz, J.: Polyhedron, Vol. 26, No. 17, 2007, s.

5120-5130 - SCI

[o1] 2008 Gabriele, B. - Mancuso, R. - Salerno, G. - Lupinacci, E. - Ruffulo, G. - Costa, M.: J. Org.

Chem., Vol. 73, No. 13, 2008, s. 4971-4977 - SCI

[o1] 2008 Mendelez-Homez, C.M. - Kouznetsov, V.V. - Sortino, M.A. - Alvarez, S.L. - Zacchino, S.A.:

Bioorg. Med. Chem., Vol. 16, No. 17, 2008, s. 7908-7920 - SCI

[o1] 2008 Madapa, S. - Tusi, Z. - Batra, S.: Current Organic Chemistry, Vol. 12, No. 13, 2008, s. 1116-

1183 - SCI

[o1] 2008 Shindoh, N. - Tokuyama, H. - Takemoto, Y. - Takasu, K.: Journal of Organic Chemistry, Vol.

73, No. 19, 2008, s. 7451-7456 - SCI

[o3] 2008 Batra, M.K. - Batra, C. - Ojha, K.G.: Medicinal Chemistry Research, Vol. 17, No. 9, 2008, s.

604-617

[o1] 2009 Schmidt, F. - Champy, P. - Séon-Méniel, B. - Franck, X. - Raisman-Vozari, R. - Figadere, B.:

PLoS ONE, Vol. 4, No. 7, 2009, S. Article no. e6215 - SCOPUS

[o1] 2009 Lee, C.H. - Lee, H.S.: Journal of the Korean Society for Applied Biological Chemistry, Vol. 52,

No. 4, 2009, s. 331-335 - SCI

[o1] 2010 Garcia-Santos, I. - Sanmartin, J. - Garcia-Deibe, A.M. - Fondo, M. - Gómez, E.: Inorganica

Chimica Acta, Vol. 363, No. 1, 2010, s. 193-198 - SCI

[o1] 2010 Chang, F.S. - Chen, W. - Wang, C. - Tzeng, C.C. - Chen, Y.L.: Bioorganic & Medicinal

Chemistry, Vol. 18, No. 1, 2010, s. 124-133 - SCI

[o1] 2009 Malakyan, M.G. - Badzhinyan, S.A. - Vardevanyan, L.A. - Grigoryan, D.S. - Egiazaryan, D.É. -

Avetisian, A.A. - Aleksanyan, I.L. - Ambartsumyan, L.P. - Sargsyan, K.S.: Pharmaceutical Chemistry

Journal, Vol. 43, No. 1, 2009, . 7-10 -SCI

[o1] 2009 Rajakumar, P. - Raja, R. - Selvam, S. - Rengasamy, R. - Nagaraj, S.: Bioorganic & Medicinal

Chemistry Letters, Vol. 19, No. 13, 2009, s. 3466-3470 - SCI

[o1] 2009 Shen, M.G. - Cai, C. - Yi, W.B.: Journal of Hetecyclic Chemistry Chemistry, Vol. 46, No. 4,

2009, s. 796-799 - SCI

[o1] 2009 Erenler, R. - Uno, M. - Goud, T.V. - Biellmann, J.F.: Journal of Chemical Research-S, No. 7,

2009, s. 459-464 - SCI

[o1] 2009 Barluenga, J. - Rodriguez, F. - Fananas, F.J.: Chemistry - An Asian Journal, Vol. 4, No. 7, 2009,

s. 1036-1048 - SCI

11

[o1] 2010 Broch, S. - Aboab, B. - Anizon, F. - Moreau, P.: European Journal of Medicinal Chemistry, Vol.

45, No. 4, 2010, s. 1657-1662 - SCI

[o1] 2010 Bhatt, H.G. - Agrawal, Y.K.: Medicinal Chemistry Research, Vol. 19, No. 4, 2010, s. 392-402 -

SCI

[o1] 2010 Pinheiro, L.M.V. - Ventura, M.C.M.M. - Moita, M.L.C.J.: Journal of Molecular Liquids, Vol.

154, No. 2-3, 2010, s. 102-110 - SCI

[o1] 2010 Rajakumar, P. - Raja, R.: Tetrahedron Letters, Vol. 51, No. 33, 2010, s. 4365-4370 - SCI

[o3] 2009 Chang, F.S.: Synthesis and Antiproliferative Evaluations of 2-Phenylvinylquinoline (2-

Styrylquinoline) and 2-Furanylvinylquinoline Derivatives. Kaohsiung City : Kaohsiung Medical

University, 2009, S. 151

[o3] 2008 Chao, S.T.: Syntheses of Quinolino-fused Bicyclo [2.2.2] octadienes and Sesquibicyclo [2.2.2]

octadienes from Friedländer Reaction. Taichung : Thunghai University, 2008, S. 156

[o3] 2010 Rachid, O.: Synthese de bromocétones quinoléiques précurseurs de Produits d´intéret

biologique. Batna : Université de Batna, 2010, S. 10, 71

[o1] 2011 Yang, G.H. - Li, Y.X. - Yan, S.H. - Dai, L. - Zhao, B.: Acta Chimica Sinica, Vol. 69, No. 15,

2011, s. 1743-1750 - SCI

[o1] 2011 Saugues, E. - Nauton, L. - Théry, V. - Anizon, F. - Moreau, P.: Bioorganic Chemistry, Vol. 39,

No. 4, 2011, s. 143-150 - SCOPUS

[o1] 2011 Zhang, W.X. - Dai, Y.S. - Wang, X.R. - Zhang, W.: Tetrahedron Letters, Vol. 52, No. 46, 2011,

s. 6122-6126 - SCOPUS

[o3] 2011 Reis, D.C.: Estudo do perfil farmacológico de novas tiossemicarbazonas e novos complexos de

bismuto(III) e antimônio(III). Belo Horizonte : [s.n.], 2011, S. 6

[o1] 2011 Thakre, W. B. - Meshram, J. S.: Indian Journal of Heterocyclic Chemistry, Vol. 21, Iss. 1, 2011,

s. 65-68 - SCI

[o1] 2011 El-Agrody, A. M. - Al-Ghamdi, A. M.: Arkivoc, Part 11, 2011, s. 134-146 - SCI

[o1] 2012 Peng, H.K. - Lin, C.K. - Yang, S.Y. - Tseng, C.K. - Tzeng, C.C. - Lee, J.C. - Yang, S.C.:

Bioorganic and Medicinal Chemistry Letters, Vol. 22, Iss. 2, 2012, s. 1107-1110 - SCI ; SCOPUS

[o1] 2012 Tyagi, R. - Singh, B. - Kishore, D.: Journal of Chemical Sciences, Vol. 124, Iss. 2, 2012, s. 431-

435 - SCI ; SCOPUS

[o1] 2012 Madhu, G. - Jayaveera, K.N. - Ravindra Nath, L.K. - Santosh Kumar, B. - Nagarjuna Reddy, P.:

Journal of Chemical and Pharmaceutical Research, Vol. 4, Iss. 6, 2012, s. 2928-2936 - SCOPUS

[o3] 2011 Li Runlai - Li Shuan - Zhang Zhenming - Ma Xiaobo - Wu Qiong: Study on Synthetic Process

of 5,7-dinitro-8-hydroxy-2-Methylquinoline. In: Chemical Industry Times, Vol. 25, Iss. 9, 2011, s. 1-8

[o3] 2012 Teixeira, R.R. - Pereira, J.L. - Pereira, W.L.: Photosynthetic Inhibitors. In: Applied

Photosynthesis. Rijeka : InTech, 2012, S. 1-22

[o3] 2011 Pandey, H. - Mehta, P. - Pathak, A.K. - Soni, H.: 2D-QSAR study of 4-(4-alkoxylphenyl)-3-

ethyl-4H-1,2,4-triazoles as open-chain analogues of 7-alkoxyl-4,5-dihydro[1,2,4]triazolo[4,3-a] quinolines.

In: Journal of Pharmacy Research,Vol. 4, No. 5, 2011, s. 1349-1352

[o3] 2011 Soto-Lopez, A. F. - Meneses, J. P. - Saez-Vega, J. - Camargo, M.: Cytotoxicity evaluation of

new styrylquinoline analogues in leukemoid jurkat cells. In: Actualidades Biologicas, Vol.33, No. 95,

2011, s. 165-172


Der Pharma Chemica, Vol. 4, No. 3, 2012, s. 1033-1040 - SCOPUS


No. 6, 2012, s. 823-828 - SCOPUS

[o1] 2012 El-Agrody, A.M. - Khattab, E.S.A.E.H. - Fouda, A.M. - Al-Ghamdi, A.M.: Medicinal

Chemistry Research, Vol. 21, No. 12, 2012, s. 4200-4213 - SCI

[o1] 2012 Kouznetsov V.V. - Meléndez Gómez C.M. - Derita M.G. - Svetaz L. - del Olmo E. - Zacchino

S.A.: Bioorganic & Medicinal Chemistry, Vol. 20, No. 21, 2012, s. 6506-6512 - SCI ; SCOPUS

[o3] 2011 Yang Z. - Fang Z. - Wang Z.X.: Synthesis of - 2,5 - dihydro - 3,6 -dimethoxy - 2 -

isopropylpyrazine. In: Chemical Industry Times, Vol. 24, No. 9, 2011, s. 6-8

[o1] 2013 Sun, W. - Yuan, G. - Liu, J. - Ma, L. - Liu, C.: Spectrochimica Acta - Part A: Molecular and

Biomolecular Spectroscopy, Vol. 106, 2013, s. 275-283 - SCOPUS

[o1] 2013 El-Agrody, A.M. - Abd-Rabboh, H.S.M. - Al-Ghamdi, A.M.: Medicinal Chemistry Research,

Vol. 22, Iss. 3, 2013, s. 1339-1355 - SCI ; SCOPUS

[o3] 2013 Kondaiah, S. - Nagarajareddy, G. - Rajesh, D. - Mallikarjuna Rao, R. - Sree Ramulu, J.:

Synthesis, Structural Characterization and Anti-bacterial Activity of some Novel Schiff Base Ligans and

their Vanadium (IV) Metal Complexes. In: IJPI s Journal of Drug Chemistry, Vol 3, No. 12, 2013, Nestr.

http://ijpijournals.com/Articles/PDF/379.pdf

12

[o3] 2013 Sales, E.S. - Schneider, J.M.F.M. – Merlo, A.A.: Síntese Tricomponente de Novos Materiais

Funcionais Quinolínicos. In: XIX Encontro da Quimica de Regiao Sul. Zborník. Tubarao : Universidade

do Sul de Santa Catarina, 2012, Nestr.http://ijpijournals.com/Articles/PDF/379.pdf

[o3] 2011 Shridhar Bhat - Curtis Chong, R. - Jun Liu, O - Sup Joong Shim: Quinoline compounds as

inhibitors of angiogenesis, human methionine aminopeptidase, and sirt1, and methods of treating disorders.

In: Patent EP2350012 A2, 2011, http://www.google.com/patents/EP2350012A2?cl=en

[o3] 2011 Li P. - Wang F. - Lin Z.Y. - Ma, C. - Huang H.H.: Synthesis of 7-Nitro-8-quinolinol. In:

Chinese Journal of Synthetic Chemistry, Vol. 19, No. 5, 2011, s. 656-658

[o1] 2013 Celik, I. - Akkurt, M. - Gezegen, H. - Kazak, C.: Acta Crystallographica Section E: Structure

Reports Online, Vol. 69, No. 6, 2013, s. o956 - SCI; SCOPUS

[o1] 2013 Bompart, D. - Núnez-Durán, J. - Rodríguez, D. - Kouznetsov, V.V. - Meléndez Gómez, C.M. -

Sojo, F. - Arvelo, F. - Visbal, G. - Alvarez, A. - García-Marchán, Y.: Bioorganic and Medicinal Chemistry,

Vol. 21, No. 14, 2013, s. 4426-4431- SCI; SCOPUS

[o1] 2013 Kuroda, Y. - Shindoh, N. - Takemoto, Y. - Takasu, K.: Synthesis (Germany), Vol. 45, No. 16,

2013, s. 2328-2329 - SCI; SCOPUS

[o1] 2013 Fahmy, H.H. - Khalifa, N.M. - Abou El-Ella, D.A. - Ismail, M.A. - Mostafa, N.M. - Hamdy,

A.A.: Life Science Journal, Vol. 10, No. 4, 2013, s. 362-368 - SCI; SCOPUS

[o1] 2013 Devi, K. - Asmat, K. - Agrawal, M. - Sharma, S. - Dwivedi, J.: Journal of Chemical Sciences,

Vol. 125, No. 5, 2013, s. 1093-1101 - SCI

[o1] 2013 Hoda H. - Fahmy, Nagy M. - Khalifa, Dalal A. - Abou El Ella, Mohamed A. - Ismail, Noha M. -

Abdelhamid A. Hamdy: Life Science Journal, Vol. 10, No. 4, 2013, s. 362-368 - SCOPUS

[o1] 2013 Han, J. - Li, L. - Shen, Y. - Chen, J. - Deng, H. - Shao, M. - Lu, X. - Zhang, H. - Cao, W.:

European Journal of Organic Chemistry, No. 36, 2013, s. 8323-8329 - SCI; SCOPUS

[o1] 2014 Lam, K.H. - Gambari, R. - Lee, K.K.H. - Chen, Y.X. - Kok, S.H.L. - Wong, R.S.M. - Lau, F.Y. -

Cheng, C.H. - Wong, W.Y. - Bian, Z.X. - Chan, A.S.C. - Tang, J.C.O. - Chui, C.H.: Bioorganic and

Medicinal Chemistry Letters, Vol. 24, No.1, 2014, s. 367-370 - SCI; SCOPUS

[o3] 2013 Li Shuan, Z.Z. - Qi, J. - Wang, T. - Zhao, H.: Study on synthesis of 8-hydroxyquinoline by

doebnermiller method. In: Speciality Petrochemicals, No. 4, 2013, s. 22-24

[o1] 2014 Rahmati, A. - Eskandari-Vashareh, M.: Journal of Chemical Sciences, Vol. 126, No. 1, 2014, s.

169-176 - SCI; SCOPUS

[o1] 2014 Islam, R. - Hossain, M.I. - Okamoto, Y. - Nagamatsu, T. - Anraku, K. - Okawara, T.:

Heterocycles, Vol. 89, No. 3, 2014, s. 693-708 - SCOPUS

[o1] 2014 Zhang, S. - Wang, Y. - Feng, C. - Yang, T. - Ji, M.ab: Dongnan Daxue Xuebao (Ziran Kexue

Ban)/Journal of Southeast University (Natural Science Edition), Vol. 44, No. 1, 2014, s. 129-132 -

SCOPUS

[o1] 2014 Peng, H.K. - Lin, I.L. - Lee, C.C. - Wang, L.Y. - Tzeng, C.C. - Chang, J.G. - Yang, S.C.:

Medicinal Chemistry Research, Vol. 23, No. 3, 2014, s. 1437-1446 - SCI; SCOPUS

[o3] 2014 Liu, J.O. - Shim, J.S. - Chong, C.R. - Bhat, S.: Quinoline compounds as inhibitors of

angiogenesis, human methionine aminopeptidase, and SIRT1, and methods of treating disorders. United

States Patent No. US 8,729,097 B2. [s.l.] : TheUnited States Patent and Trademark Office, 2014, S. 1

[o3] 2014 Desai, N.C. - Dodiya, A.M.: Microwave-Induced Synthesis of Various Quinoline Derivatives:

Green Methodologies in Organic Synthesis. In: Green Chemistry: Synthesis of Bioactive Heterocycles.

New Delhi : Springer, 2014, S. 163-200

[o1] 2014 Gao, Q. - Liu, S. - Wu, X. - Wu, A.: Organic Letters, Vol. 16, No. 17, 2014, s. 4582-4585 - SCI;

SCOPUS

[o1] 2014 Ahmed, A. - Dhara, S. - Singha, R. - Nuree, Y. - Sarkar, P.: RSC Advances, Vol. 4, No. 95,

2014, s. 53137-53141 - SCOPUS

[o1] 2015 Qi, J.J. - Li, S.A. - Zhang, Z.M. - Wang, T. - Zhao, H.B. - Wang, X. - Yin, F.J.: Asian Journal of

Chemistry, Vol. 27, No. 2, 2015, s. 435-440 - SCI; SCOPUS

[o1] 2015 Shah, A. - Raj, D.: Journal of Saudi Chemical Society, Vol. 19, No. 1, 2015, s. 73-82 - SCI

[o1] 2015 Zayed, M.E.M. - El-Shishtawy, R.M. - Elroby, S.A. - Obaid, A.Y. - Al-Amshany, Z.M.:

International Journal of Molecular Sciences, Vol. 16, No. 2, 2015, s. 3804-3819 - SCOPUS

[o1] 2015 Shadrikova, V.A. - Golovin, E.V. - Zatonskii, G.V. - Klimochkin, Yu.N.: Russian Journal of

Organic Chemistry, Vol. 51, No. 1, 2015, s. 130-131 - SCI; SCOPUS

[o3] 2015 Baluja, S.: Dissociation Constants of Some Quinoline Derivatives in Mixed Solvent mixture. In:

International Letters of Chemistry, Physics and Astronomy, International Letters of Chemistry, Physics

and Astronomy, Vol. 9, No. 1, 2015,s. 32-36

[o3] 2015 Alias, M. - Ismael, S. - Mousa, S.A.: Synthesis, Characterization and Theoretical Study of Some

Mixed-ligand Complexes of 2-Quinoline Carboxylic Acid and 4,4/-dimethyl,2,2/-Bipyridyl with Some

Transition Metal Ions. In: Journal of Al-Nahrain University, Vol. 18, No. 1, 2015, s. 28-38

13

[o1] 2014 Khalifa, N.M. - Eweas, A. - Al-Omar, M.A. - Hozzein, W.: Journal of Pure and Applied

Microbiology, Vol. 8, 2014, s. 629-637 - SCI; SCOPUS

[o1] 2014 Yan, X. - Yu, Y. - Ji, P. - He, H. - Qiao, C.: European Journal of Medicinal Chemistry, Vol. 102,

Art. No. 8024, 2015, s. 180-187 - SCOPUS

[o1] 2015 Gao, Q. - Liu, S. - Wu, X. - Zhang, J. - Wu, A.: Journal of Organic Chemistry, Vol. 80, No. 11,

2015, s. 5984-5991 - SCI; SCOPUS

[o1] 2015 Chung, P.Y. - Bian, Z.X. - Pun, H.Y. - Chan, D. - Chan, A.S.C. - Chui, C.H. - Tang, J.C.O. -

Lam, K.H.: Future Medicinal Chemistry, Vol. 7, No. 7, 2015, s. 947-967 - SCOPUS

[o1] 2015 Yaragorla, S. - Singh, G. - Dada, R.: Tetrahedron Letters, Vol. 56, No. 43, 2015, s. 5929 - SCI;

SCOPUS

ADC12 Podeszwa, Barbara (10%) - Niedbala, Halina (10%) - Polanski, Jaroslaw (10%) - Musiol, Robert (10%)

- Tabak, Dominik (5%) - Finster, Jacek (5%) - Serafin, Karol (5%) - Wietrzyk, Joanna (5%) - Boryczkka,

Stanislaw (5%) - Mól, Wojciech (5%) - Jampílek, Josef [UKOEXAF] (10%) - Dohnal, Jiří (5%) -

Kalinowski, Danuta S. (10%) - Richardson, Des Robert (5%): Investigating the antiproliferative activity of

quinoline-5,8-diones and styrylquinolinecarboxylic acids on tumor cell lines

Lit. 35 zázn.

In: Bioorganic & Medicinal Chemistry Letters. - Vol. 17, No. 22 (2007), s. 6138-6141



IF (JCR) 2007=2,604

Ohlasy (17):

[o1] 2009 Li, Y.Q. - Zheng, D. - Li, J. - Han, L. - Cui, X.L. - Lang, L. - Li, M.G. - Wang, Z.Y. - Zhao, J.Y.

- Huang, X.S.: Journal of Antibiotics, Vol. 62, No. 11, 2009, s. 648 - SCI

[o1] 2010 Sliman, F. - Blairvacq, M. - Durieu, E. - Meijer, L. - Rodrigo, J. - Desmaele, D.: Bioorganic &

Medicinal Chemistry Letters, Vol. 20, No. 9, 2010, s. 2805 - SCI

[o1] 2011 Paretzki, A. - Das, H.S. - Weisser, F. - Scherer, T. - Bubrin, D. - Fiedler, J. - Nycz, J.E. - Sarkar,

B.: European Journal of Inorganic Chemistry, No. 15, 2011, s. 2421 - SCI

[o1] 2011 Khodairy, A. - Abass, M.: Chemistry of Heterocyclic Compounds, Vol. 47, No. 5, 2011, s. 621 -

SCI


No. 6, 2012, s. 828 - SCI

[o1] 2012 Al-Ghamdi, A.M. - Abd El-Wahab, A.H.F. - Mohamed, H.M. - El-Agrody, A.M.: Letters in

Drug Design & Discovery, Vol. 9, No. 5, 2012, s. 470 - SCI

[o1] 2012 Stein, A.L. - Bilheri, F.N. - da Rocha, J.T. - Back, D.F. - Zeni, G.: Chemistry-A European

Journal, Vol. 18, No. 34, 2012, s. 10608 - SCI

[o1] 2013 Keyari, C.M. - Kearns, A.K. - Duncan, N.S. - Eickholt, E.A. - Abbott, G. - Beall, H.D. - Diaz,

P.: Journal of Medicinal Chemistry, Vol. 56, No. 10, 2013, s. 3806-3819 - SCI

[o1] 2014 Keshipour, S. - Shaabani, A. - Pedarpour, M. - Sarvary, A.: Research on Chemical

Intermediates, Vol. 40, No. 1, Spec. Iss., 2014, s. 156 - SCI

[o1] 2014 Bassyouni, F.A. - Abu-Baker, S.M. - Mahmoud, K. - Moharam, M. - El-Nakkady, S.S. - Rehim,

M.A.: RSC Advances, Vol. 4, No. 46, 2014, s. 24141 - SCI

[o1] 2014 Mantovani, A.C. - Pesarico, A.P. - Sampaio, T.B. - Nogueira, C.W. - Zeni, G.: European Journal

of Pharmaceutical Sciences, Vol. 51, 2014, s. 203 - SCI

[o1] 2014 Gavrishova, T.N. - Li, V.M. - Karpov, O.N. - Budyka, M.F.: Russian Journal of Organic


[o1] 2015 Yadav, T. - Kishore, D. - Singh, B.: British Journal of Pharmaceutical Research, Vol. 8, No. 3,

2015, Article No. 19615 - SCI

[o1] 2015 Zayed, M.E.M. - El-Shishtawy, R.M. - Elroby, S.A. - Obaid, A.Y. - Al-amshany, Z.M.:

International Journal of Molecular Sciences, Vol. 16, No. 2, 2015, s. 3819 - SCI

[o1] 2015 Gavrishova, T.N. - Budyka, M.F. - Potashova, N.I. - Karpov, O.N.: Russian Journal of Organic


[o1] 2015 Kumar, N.S. - Rao, L.C. - JagadeeshBabu, N. - Kumar, V.D. - Murthy, U.S.N. - Meshram,

H.M.: Synlett, Vol. 26, No. 13, 2015, s. 1814 - SCI

[o1] 2015 Yaragorla, S. - Singh, G. - Dada, R.: Tetrahedron Letters, Vol. 56, No. 43, 2015, s. 5929 - SCI

ADC13 Vinšová, Jarmila (20%) - Imramovský, Aleš (20%) - Buchta, Vladimír (10%) - Čečková, Martina (10%)

- Doležal, Martin (10%) - Štaud, František (10%) - Jampílek, Josef [UKOEXAF] (10%) - Kaustová,

Jarmila (10%): Salicylanilide acetates: synthesis and antibacterial evaluation

Lit. 14 zázn.


14



IF (JCR) 2007=0,940

Ohlasy (6):

[o1] 2008 Pyka, A.: Journal of Liquid Chromatography & Related Technologies, Vol. 31, No. 13, 2008, s.

1958 - SCI

[o1] 2009 Skala, P. - Machacek, M. - Vejsova, M. - Kubicova, L. - Kunes, J. - Waisser, K.: Journal of

Heterocyclic Chemistry, Vol. 46, No. 5 , 2009, s. 880 - SCI

[o1] 2013 Kang, S. - Min, H.J. - Kang, M.S. - Jung, M.G. - Kim, S.: Bioorganic & Medicinal Chemistry

Letters, Vol. 23, No. 6, 2013, s. 1751 - SCI

[o1] 2013 Nuta, D.C. - Chifiriuc, M.C. - Draghici, C. - Limban, C. - Missir, A.V. - Morusciag, L.:

Farmacia, Vol. 61, No. 5, 2013, s. 974 - SCI

[o1] 2015 Dank, C. - Kirchknopf, B. - Mastalir, M. - Kahlig, H. - Felsinger, S. - Roller, A. - Arion, V.B. -

Gstach, H.: Molecules, Vol. 20, No. 1, 2015, s. 1711 - SCI

[o1] 2015 Diller, D.J. - Connell, N.D. - Welsh, W.J.: Journal of Computer-Aided Molecular Design, Vol.

29, No. 11, 2015, s. 1024 - SCI

ADC14 Doležal, Martin (20%) - Čmedlová, Pavlína (15%) - Pálek, Lukáš (15%) - Vinšová, Jarmila (5%) -

Kuneš, Jiří (5%) - Buchta, Vladimír (10%) - Kráľová, Katarína [UKOPRCUS] (15%) - Jampílek, Josef

[UKOEXAF] (15%): Synthesis and antimycobacterialevaluation of substituted pyrazinecarboxamides

Lit.: 27 zázn., 1 obr., 3 tab.

In: European Journal of Medicinal Chemistry. - Vol. 43, No. 5 (2008), s. 1105-1113



IF (JCR) 2008=2,882

Ohlasy (31):

[o3] 2008 Haruaki, T.: Expert Opinion on Drug Discovery, Vol. 3, No. 1, 2008, s. 21-49

[o3] 2009 Hopper, D.W. - Clemens, J.J. - Kwon, S.: Chapter 6.1 Six-membered ring systems: pyridine and

benzo derivatives. In: Progress in Heterocyclic Chemistry, Volume 21. Amsterdam : Elsevier, 2009, S.

330-414

[o1] 2009 Manlove, A. - Groziak, M.P.: Progress in Heterocyclic Chemistry, Vol. 21, 2009, s. 375-414 -

SCOPUS

[o1] 2010 Dunklevy, J.D. - Soole, K.L. - Perkins, M.V. - Dennis, E.G. - Keyzers, R.A. - Kalua, C.M. -

Boss, P.K.: Plant Molecular Biology, Vol. 74, No. 1-2, 2010, s. 77-89 - SCI


8, 2010, s. 3384-3388 - SCI

[o1] 2010 Yesilel, O.Z. - Mutlu, A. - Darcan, C. - Buyukgungor, O.: Journal of Molecular Structure, Vol.

964, No. 1-3, 2010, s. 39-46 - SCOPUS


s. 1469-1500 - SCOPUS

[o1] 2010 Lee, J.H. - Myung, P.K. - Kim, S.J. - Sung, N.D.: Journal of Applied Biological Chemistry, Vol.

53, No. 4, 2010, s. 440-445 - SCOPUS

[o3] 2010 Yafei, L.I. - Liqun, J.I.N. - Zhiqiang, L.I.U. - Yuguo, Z.: Chinese Journal of Modern Applied

Pharmacy, Vol. 27, No. 4, 2010, s. 307-312

[o3] 2010 Tewatia, N. - Namdeo, K.P. - Jain, S.K. - Prajapati, S.K. - Singh, O. - Jain, V. - Kumar, P.:

Journal of the Institution of Chemists (India), Vol. 82, No. 5, 2010, s. 148-153

[o3] 2011 Lima, C.H.S. - Bispo, M.L.F. - de Souza, M.V.N.: Pirazinamida: Um Fármaco Essencial no

Tratamento da Tuberculose. In: Revista Virtual de Química, Vol. 3, No. 3, 2011, s. 159-180

[o3] 2011 Prasad, R. - Sharma, R.: 2D QSAR Analysis of Pyrazinecarboxamides derivatives as an

herbicidal agent. In: Journal of Computational Methods in Molecular Design, Vol. 1, No. 1, 2011, s. 7-13

[o1] 2011 Dib-Bellahouel, S. - Fortas, Z.: African Journal of Biotechnology, Vol. 10, No. 47, 2011, s.

9694-9699 - SCOPUS

[o3] 2011 Vikramjeet J. - Balasubramanian N. - Munish A.: A Review of Biological potential of

Pyrazinamide derivatives. In: Hygeia : Journal for Drugs and Medicines, Vol. 4, Iss. 1, 2012, s. 1-6

[o3] 2012 Ghetiya: Pyrazine derivatives. In: Studies on heterocyclic compounds, Pp. 17, 2012,

http://ir.inflibnet.ac.in:8080/bitstream/10603/3890/7/07_part%20a.pdf

[o1] 2012 Bispo, M.D.L.F. - Gonçalves, R.S.B. - Lima, C.H.D.S. - Cardoso, L.N.D.F. - Lourenço, M.C.S.

- De Souza, M.V.N.: Journal of Heterocyclic Chemistry , Vol. 49, Iss. 6, 2012, s. 1317-1322 - SCOPUS

[o3] 2010 Li, Y. - Kinley L.J.L. - Liu Z. - Yu-Guo Z.: Pyrazinamide research progress. In: Chinese Journal

of Modern Applied Pharmacy, Vol. 27, Iss. 4, 2010, s. 307-312

15

[o1] 2013 Nayak, P.S. - Narayana, B. - Samshuddin, S. - Sarojini, B.K.: MolBank, Vol. 2013, Iss. 2, 2013,

Nestr. - SCOPUS

[o3] 2012 Asif, M.: Recent Efforts for the Development of Antitubercular Drug Containing Diazine Ring.

In: Medicinal Chemistry, Vol. 2, Iss. 7, 2012, s. 151-167

[o3] 2013 Blochin I.V. - Ageev, A.V. - Artošenko J.M. - Chlytin, N.V. - Tormozov, V.A.: Sintez 2-

metoksi-3-T-pirazinov v ionnoj židkosti. In: Izvestja Tulskogo Gosudarstvennoho Universiteta,

Jestestvennye Nauki, 2013, s. 163

[o1] 2013 Achelle, S. - Baudequin, C. - Plé, N.: Dyes and Pigments, Vol. 98, No. 3, 2013, s. 575-600 - SCI

; SCOPUS

[o1] 2013 Miniyar, P.B. - Murumkar, P.R. - Patil, P.S. - Barmade, M.A. - Bothara, K.G.: Reviews in

Medicinal Chemistry, Vol. 13, No. 11, 2013, s. 1607-1625 - SCI

[o1] 2014 Ma, W.J. - Gao, Z.Y. - Zhu, S. - Wu, B.L.: Polyhedron, Vol. 73, May 2014, s. 59-66 - SCOPUS

[o1] 2013 Darcan, C. - Kaygusuz, Ö. - Korkmaz, T.: Journal of Pure and Applied Microbiology, Vol. 7,

No. 4, 2013, s. 2747-2756 - SCOPUS

[o1] 2014 Konar, S. - Saha, U. - Dolai, M. - Chatterjee, S.: Journal of Molecular Structure, Vol. 1075,

2014, s. 286-291 - SCOPUS



Medicinal Chemistry Letters, Vol.25, No. 3, 2015, s. 524-528 - SCI ; SCOPUS

[o1] 2015 Benzon, K.B. - Varghese, H.T. - Panicker, C.Y. - Pradhan, K. - Tiwary, B.K. - Nanda, A.K. -

Alsenoy, C.V.: Spectrochimica Acta - Part A: Molecular and Biomolecular Spectroscopy, Vol. 151, July,

2015, s. 965-979 - SCOPUS

[o3] 2015 Mohammad Asif: Anti-tubercular activity of some six membered heterocycle compounds. In:

Chemistry International, Vol. 1, No. 3, 2015, s. 134-163

[o3] 2015 Elidrissi, B. - Ousaa, A. - Ghamali, M. - Chtita,S. - Ajana, M.A. - Bouachrine - Lakhlifi, T.: The

biological activity of pyrazinecarboxamides derivatives as an herbicidal agent: combining DFT and QSAR

studies. In: Journal of Computational Methods in Molecular Design, Vol. 5, No. 2, 2015, s. 83-91

[o3] 2015 Shaikh, A.R. - Gonsalves, S.I. - Nikam, A. - Kshirsagar, S.J. - Thombare, Y.: Predicting

Pyrazinecarboxamides Derivatives as an Herbicidal Agent: 3d Qsar by kNN-MFA and Multiple linear

regression Approach. In: World Applied Sciences Journal, Vol. 33, No. 6, 2015, s. 980-989


Vol. 1105, 2016, s. 104 - SCI; SCOPUS

ADC15 Jampílek, Josef [UKOEXAF] (50%) - Brojerová, Eliška (25%) - Doležal, Martin (10%) - Kuneš, Jiří

(10%) - Jun, Daniel (5%): Preparation and antiplatelet activity of glycidic acid derivatives

Lit. 30 zázn.




IF (JCR) 2008=0,758

ADC16 Jampílek, Josef [UKOEXAF] (25%) - Rečková, Zuzana (20%) - Imramovský, Aleš (20%) - Raich, Ivan

(20%) - Vinšová, Jarmila (10%) - Dohnal, Jiří (5%): Study of stability of new mutual prodrugs with

antimycobacterial activity

Lit. 45 zázn.




IF (JCR) 2008=3,184

ADC17 Musilek, Kamil (30%) - Jampílek, Josef [UKOEXAF] (30%) - Dohnal, Jiří (5%) - Jun, Daniel (10%) -

Gunn-Moore, Frank (5%) - Doležal, Martin (5%) - Kuča, Kamil (15%): RP-HPLC determination of the

lipophilicity of bispyridinium reactivators of acetylcholinesterase bearing a but-2-ene connecting linker

Lit. 39 zázn.

In: Analytical and Bioanalytical Chemistry. - Vol. 391, No. 1 (2008), s. 367-372



IF (JCR) 2008=3,328

ADC18 Musiol, Robert (20%) - Tabak, Dominik (10%) - Niedbala, Halina (5%) - Podeszwa, Barbara (5%) -

Kráľová, Katarína [UKOPRCUS] (15%) - Dohnal, Jiří (5%) - Finster, Jacek (10%) - Mencel, Agnieszka

(5%) - Polanski, Jaroslaw (10%) - Jampílek, Josef [UKOEXAF] (15%): Investigating biological activity

16

spectrum for novel quinoline analogues 2: Hydroxyquinolinecarboxamides with photosynthesis-inhibiting

activity

Lit.: 44 zázn., 4 obr., 2 tab., 1 schéma




IF (JCR) 2008=3,075

Ohlasy (20):

[o1] 2009 Qui, C.M. - Zheng, Q.W. - Hua, R.M.: Tetrahedron, Vol. 65, No. 7, 2009, s. 1316-1320 -

SCOPUS; SCI

[o1] 2010 Achrem-Achremowicz, J. - Kepczynska, E. - Zylewski, M. - Janeczko, Z.: Biomedical

Chromatography, Vol. 24, No. 3, 2010, s. 261-267 - SCI

[o1] 2010 Rahimizadeh, M. - Pordel, M. - Bakavoli, M. - Eshghi, H.: Dyes and Pigments, Vol. 86, No. 3,

2010, s. 266-270 - SCI

[o1] 2011 Khodairy, A. - Abass, M.: Khimiya Geterotsiklicheskikh Soedinenii, No. 5, 2011, s. 736-749 -

SCOPUS

[o3] 2011 Pan, S.M.: The Synthesis and Characterization of Quinoline-Metallic Complexes and Study

Material for Military Sensor. [S.l.] : National Defense University, 2011, S. 150

[o3] 2011 Gagliardi, S. - Del Sordo, S. - Mailland, F. - Legora, M.A.: Secondary 8 hydroxyquinoline 7

carboxamide derivatives for use as antifungal agents. Patent WO 2011080265, S. 51

[o1] 2011 Khodairy, A. - Abass, M.: Chemistry of Heterocyclic Compounds, Vol. 47, No. 5, 2011, s. 611-

621 - SCI




Journal of Chemical and Pharmaceutical Research, Vol. 4, No. 6, 2012, s. 2928-2936 - SCOPUS



[o1] 2013 Nycz J.E. - Malecki G.J.: Journal of Molecular Structure, Vol. 1032, 2013, s. 159-168 -

SCOPUS


Vol. 22, No. 3, 2013, s. 1339-1355 - SCI; SCOPUS

[o3] 2013 Shet Prakash, M. - Vaidya, V. P. - Mahadevan, K.M. - Shivananda, M.K. - Suchetan, P.A. -

Sunitha, M.: Synthesis characterization and antimicrobial activities of some novel carboxamides derived

from napthofurans and 1,2,4-triazoles.In: National Conference on Challenges and Opportunities of

Chemical Sciences in 21st Century. [S.l.] : [s.n.], 2013, Nestr.

[o1] 2014 Lam, K.H. - Gambari, R. - Lee, K.K.H. - Chen, Y.X. - Kok, S.H.L. - Wong, R.S.M. - Lau, F.Y. -

Cheng, C.H. - Wong, W.Y. - Bian, Z.X., Chan, A.S.C. - Tang, J.C.O. - Chui, C.H.: Bioorganic and

Medicinal Chemistry Letters, Vol. 24, No.1, 2014, s. 367-370 - SCI; SCOPUS

[o1] 2014 El-Agrody, A.M. - Afifi, T.H.: Heterocycles, Vol. 89, No. 7, 2014, s. 1557-1584 - SCOPUS

[o1] 2014 Ariyasu, S. - Mizuseda, Y. - Hanaya, K. - Aoki, S.: Chemical and Pharmaceutical Bulletin, Vol.

62, No. 7, 2014, s. 642-648 - SCI; SCOPUS


Microbiology, Vol. 8, 2014, s. 629-637 - SCOPUS



[o1] 2015 Chung, P.Y. - Bian, Z.X. - Pun, H.Y. - Chan, D. - Chan, A.S.C. - Chui, C.H. - Tang, J.C.O. -

Lam, K.H.: Future Medicinal Chemistry, Vol. 7, No. 7, 2015, s. 947-967 - SCOPUS

[o1] 2015 Fang, F.Q. - Guo, H.S. - Zhang, J. - Ban, L.Y. - Liu, J.W. - Yu, P.Y.: Molecular Medicine

Reports, Vol. 12, No. 6, 2015, s. 8070 - SCI; SCOPUS

ADC19 Opletalová, Veronika (20%) - Kalinowski, Danuta S. (15%) - Vejsová, Marcela (15%) - Kuneš, Jiří

(10%) - Pour, Milan (10%) - Jampílek, Josef [UKOEXAF] (10%) - Buchta, Vladimír (10%) - Richardson,

Rhonda (10%): Identification and characterization of thiosemicarbazones with antifungal and antitumor

effects: cellular iron chelation mediating cytotoxic activity

Lit. 58 zázn.

In: Chemical Resarch in Toxicology. - Vol. 21, No. 9 (2008), s. 1878-1889



IF (JCR) 2008=3,491

17

ADC20 Palek, Lukáš (25%) - Dvořák, Jaroslav (15%) - Svobodová, Michaela (15%) - Buchta, Vladimír (15%) -

Jampílek, Josef [UKOEXAF] (15%) - Doležal, Martin (15%): Synthesis, antimycobacterial and antifungal

evaluation of3-arylaminopyrazine-2,5-dicarbonitriles

Lit. 16 zázn.

In: Archiv der Pharmazie. - Vol. 341, No. 1 (2008), s. 61-65



IF (JCR) 2008=1,429

Ohlasy (3):

[o1] 2009 Ukrainets, I.V. - Grinevich, L.A. - Tkach, A.A. - Bevz, O.V. - Slobodzian, S.V.: Chemistry of

Heterocyclic Compounds, Vol. 45, No. 9, 2009, s. 1068 - SCI

[o1] 2010 Walkiewcz, R. - Chazan, R. - Grubek-Jaworska, H.: Biocybernetics and Biomedical

Engineering, Vol. 30, No. 2, 2010, s. 14 - SCI


8, 2010, s. 3388 - SCI

ADC21 Brychtová, Kateřina (25%) - Slabá, Barbora (10%) - Plaček, Lukáš (15%) - Jampílek, Josef

[UKOEXAF] (20%) - Raich, Ivan (25%) - Csöllei, Jozef (5%): Coupling reactions of alpha-

bromocarboxylate with non-aromatic N-heterocycles

Lit. 25 zázn.




IF (JCR) 2009=1,738

ADC22 Doležel, Jan (20%) - Hiršová, Petra (15%) - Opletalová, Veronika (20%) - Dohnal, Jiří (5%) - Vejsová,

Marcela (10%) - Kuneš, Jiří (10%) - Jampílek, Josef [UKOEXAF] (20%): Rhodanineacetic Acid

Derivatives as Potential Drugs: Preparation, Hydrophobic Properties and Antifungal Activity of (5-

Arylalkylidene-4-oxo-2-thioxo-1,3-thiazolidin-3-yl)acetic Acids

Lit. 63 zázn.




IF (JCR) 2009=1,738

ADC23 Imramovský, Aleš (20%) - Vinšová, Jarmila (20%) - Ferriz, Juana Monreal (10%) - Doležal, Rafael

(10%) - Jampílek, Josef [UKOEXAF] (20%) - Kaustová, Jarmila (10%) - Kunc, Filip (10%): New

antituberculotics originated from salicylanilides with promising in vitro activity against atypical

mycobacterial strains

Lit. 25 zázn.




IF (JCR) 2009=2,822

ADC24 Imramovský, Aleš (20%) - Vinšová, Jarmila (20%) - Ferriz, Juana Monreal (20%) - Buchta, Vladimír

(20%) - Jampílek, Josef [UKOEXAF] (20%): Salicylanilide esters of N-protected amino acids as novel

antimicrobial agents

Lit. 19 zázn.




IF (JCR) 2009=2,650

ADC25 Jampílek, Josef [UKOEXAF] (15%) - Musiol, Robert (15%) - Finster, Jacek (5%) - Peško, Matúš

[UKOPREEF] (10%) - Carroll, James (10%) - Kráľová, Katarína [UKOPRCUS] (10%) - Vejsová,

Marcela (10%) - O Mahony, Jim (5%) - Coffey, Aidan (5%) - Dohnal, Jiří (5%) - Polanski, Jaroslaw

(10%): Investigating Biological Activity Spectrum for Novel Styrylquinazoline Analogues





IF (JCR) 2009=1,738

18

Ohlasy (18):

[o3] 2011 Vijaychand, A. - Manjula, S.N. - Barath, E.N. - Divya, B.: Medicinal and biological significance

of quinazoline a highly important scaffold for drug discovery: a review. In: International Journal of

Pharma and Bio Sciences, Vol. 2, No. 1, 2011, s. 780-809





[o1] 2012 Stein, A.L. - Bilheri, F.N. - Da Rocha, J.T. - Back, D.F. - Zeni, G.: Chemistry - A European

Journal, Vo. 18, No. 34, 2012, s. 10602-10608 - SCI ; SCOPUS



[o1] 2012 Wang, Y.K. - Jin, J. - Zhu, L.N. - Zhang, Y. - Chen, X.G. - Gao, X.Q. - Xu, B.L.: Yaoxue

Xuebao, Vol. 47, No. 9, 2012, s. 1164-1178 - SCOPUS

[o3] 2012 Samira, I. - Patel, S. - Hasmin, M. - Patel, S.: Biological Profile of Quinazoline. In: International

Journal of Pharmaceutical and Chemical Sciences, Vol. 1, No. 4, 2012, s. 1527

[o3] 2012 Wangy, Y.K. - Jin, J. - Zhu, L.N. - Zhang, Y. - Chen, X.G. - Gao, X.Q. - Xu, B.L.: Synthesis

and antitumor activity of novel 2-(1-substituted-piperidin -4-ylamino)quinazolines as antitumor agents. In:

Acta Pharmaceutica Sinica, Vol.47, No. 9, 2012, s. 1178

[o1] 2013 Li, Y. - De Kock, C. - Smith, P.J. - Guzgay, H. - Hendricks, D.T. - Naran, K. - Mizrahi, V. -

Warner D.F. - Chibale, K. - Smith, G.S.: Organometallics, Vol. 32, No. 1, 2013, s. 141-150 - SCI ;

SCOPUS

[o1] 2014 Mantovani, A.C. - Pesarico, A.P. - Sampaio, T.B. - Nogueira, C.W. - Zeni, G.: Journal of

Pharmaceutical Sciences, Vol. 51, No. 1, 2014, s. 196-203 - SCI ; SCOPUS

[o3] 2014 Indubhushan - Choudhary, A.N. - Kothiyal, P.: Synthesis and evaluation of quinazolinthione

derivatives as antibacterial agents. In: International Journal of Pharmacy, Vol. 4, No. 3, 2014, s. 135

[o1] 2014 Lakshmi, K. - Rama Rao, N. - Basaveswararao, M.V.: Rasayan Journal of Chemistry, Vol. 7,

No. 1, 2014, s. 44-54 - SCOPUS

[o1] 2014 Aly, S.A. - Alganzory, H.H. - Salem, T.A.: Journal of Chemical and Pharmaceutical Research,

Vol. 6, No. 6, 2014, s. 101-109 - SCOPUS


International Journal of Molecular Sciences, Vol. 16, No. 2, 2015, s. 3804-3819 - SCI ; SCOPUS

[o1] 2015 Kumar, D. - Jadhavar, P.S. - Nautiyal, M. - Sharma, H. - Meena, P.K. - Adane, L. - Pancholia, S.

- Chakraborti, A.K.: RSC Advances, Vol. 5, No. 39, 2015, s. 30819-30825 - SCOPUS

[o1] 2015 Lakshmi, K. - Rama Rao, N. - Basaveswara Rao, M.V.: Journal of Environmental Biology, Vol.

36, No. 4, 2015, s. 909-918 - SCI ; SCOPUS

[o3] 2015 Wani, Z.A. - Pathania, A.S. - Mahajan, G. - Behl, A. - Mintoo, M.J. - Guru, S.K. - Viswanath,

V. - Malik, F. - Kamal, A. - Mondhe, D.M.: Anticancer activity of a novel quinazolinone-chalcone

derivative through cell cycle arrest inpancreatic cancer cell line. In: Journal of Solid Tumors, Vol. 5, No. 2,

2015, s. 84

[o3] 2014 Krastina, G. - Ravina, I. - Mierina, I. - Zicane, D. - Turks, M. - Tetere, Z. - Leonciks, A.:

Synthesis of novel quinazolinone-1,2,3-triazole conjugates. In: Journal of Chemical and Pharmaceutical

Research, Vol. 6, No. 12, 2014, s.13

ADC26 Jampílek, Josef [UKOEXAF] (10%) - Musiol, Robert (10%) - Peško, Matúš [UKOPREEF] (10%) -

Kráľová, Katarína [UKOPRCUS] (10%) - Vejsová, Marcela (10%) - Carroll, James (10%) - Coffey, Aidan

(5%) - Finster, Jacek (5%) - Tabak, Dominik (5%) - Niedbala,Halina (5%) - Kozik, Violetta (5%) -

Polanski, Jaroslaw (5%) - Csöllei, Jozef (5%) - Dohnal, Jiří (5%): Ring-substituted 4-Hydroxy-1H-

quinolin-2-ones: Preparation and Biological Activity





IF (JCR) 2009=1,738

Ohlasy (16):

[o3] 2010 Ibrahim, M.A. - Hassanin, H.M. - Gabr, Y.A.A. - Alnamer, Y.A.S.: European Journal of

Chemistry, Vol. 1, No. 3, 2010, s. 195-199

[o1] 2011 Ukrainets, I.V. - Golik, N.Y.U. - Bevz, O.V. - Gorokhova, O.V.: Khimiya Geterotsiklicheskikh

Soedinenii, No. 7, 2011, s. 1018-1023 - SCOPUS

[o1] 2011 Ukrainets, I. V. - Golik, N. Y. - Bevz, O. V. - Gorokhova, O. V.: Chemistry of Heterocyclic

Compounds, Vol. 47, No. 2, 2011, s. 833-837 - SCI

19





[o3] 2012 Teixeira R.R. - Pereira J.L. - Pereira W.L: Photosynthetic inhibitors. In: Applied Photosynthesis.

Rijeka : Intech, 2012, S. 1-22

[o1] 2012 Abass, M. - Mohamed, E.H.A. - Mayas, A.S. - Ibrahim, A.H.: Journal of Chemical Sciences,

Vol. 124, No. 5, 2012, s. 1033-1041 - SCI


Vol. 22, No. 3, 2013, s. 1339-1355 - SCI ; SCOPUS

[o1] 2014 Bhat, S.I. - Trivedi, D.R.: RSC Advances, Vol. 4, No. 22, 2014, s. 11300-11304 - SCI ;

SCOPUS

[o1] 2014 El-Agrody, A.M. - Afifi, T.H.: Heterocycles, Vol. 89, No. 7, 2014, s. 1557-1584 - SCOPUS

[o1] 2014 Prajapati, S.M. - Patel, K.D. - Vekariya, R.H. - Panchal, S.N. - Patel, H.D.: RSC Advances, Vol.

4, No. 47, 2014, s. 24463-24476 - SCI ; SCOPUS


Vol. 6, No. 6, 2014, s. 101-109 - SCOPUS


Microbiology, Vol. 8, No. 1, 2014, s. 629-637 - SCOPUS



[o3] 2015 Ruat, M. - Faure, H. - Gorojankina, T.: Use of quinolinone derivatives as a research tool. US

Patent US8957091, http://www.google.com/patents/US8957091

[o1] 2015 Fang, F.Q. - Guo, H.S. - Zhang, J. - Ban, L.Y. - Liu, J.W. - Yu, P.Y.: Molecular Medicine

Reports, Vol. 12, No. 6, 2015, s. 8070 - SCI; SCOPUS

ADC27 Opatřilová, Radka (5%) - Jampílek, Josef [UKOEXAF] (20%) - Raich, Ivan (20%) - Kačerová, Sandra

(15%) - Pekárek, Tomáš (15%) - Dohnal, Jiří (5%) - Csöllei, Jozef (5%) - Havlíček, Jaroslav (15%):

Synthesis, Characterization and Physico-chemical Properties of New 2-(4-Arylpiperazine-1-yl)-1-(3-

methylbenzofuran-2-yl)ethanoles as Potential Antihypertensive Agents

Lit. 24 zázn.




IF (JCR) 2009=2,879

ADC28 Brychtová, Kateřina (20%) - Opatřilová, Radka (5%) - Raich, Ivan (10%) - Kalinowski, Danuta S.

(10%) - Dvořáková, Lenka (10%) - Plaček, Lukáš (10%) - Csöllei, Jozef (5%) - Richardson, Des R. (10%)

- Jampílek, Josef [UKOEXAF] (20%): Investigating the activity of 2-substituted alkyl-6-(2,5-

dioxopyrrolidin-1-yl)hexanoates as skin penetration enhancers

Lit. 44 zázn.




IF (JCR) 2010=2,978

ADC29 Brychtová, Kateřina (35%) - Jampílek, Josef [UKOEXAF] (20%) - Opatřilová, Radka (10%) - Raich,

Ivan (20%) - Farsa, Oldřich (10%) - Csöllei, Jozef (5%): Synthesis, physico-chemical properties and

penetration activity ofalkyl-6-(2,5-dioxopyrrolidin-1-yl)-2-(2-oxopyrrolidin-1-yl)hexanoates as potential

transdermal penetration enhancers

Lit. 47 zázn.




IF (JCR) 2010=2,978

ADC30 Doležal, Martin (20%) - Zitko, Jan (15%) - Osička, Zdeněk (10%) - Kuneš, Jiří (5%) - Vejsová, Marcela

(10%) - Buchta, Vladimír (5%) - Dohnal, Jiří (5%) - Kráľová, Katarína [UKOPRCUS] (15%) - Jampílek,

Josef [UKOEXAF] (15%): Synthesis,Antimycobacterial, Antifungal and Photosynthesis-Inhibiting

Activity of Chlorinated N-phenylpyrazine-2-carboxamides



20



IF (JCR) 2010=1,988

Ohlasy (8):

[o3] 2012 Tewatia, N. - Abida - Namdeo, K. P.: Synthesis and antimicrobial activity of pyrazine

carboxamide derivatives. In: Journal of Chemical and Pharmaceutical Research, Vol. 4, No. 3, 2012,

s.1794-1798

[o1] 2012 Bentabed-Ababsa G. - Hamza-Reguig S. - Derdour A. - Domingo L.R. - Sáez J.A. - Roisnel T. -

Dorcet V. - Nassar E. - Mongin F.: Organic & Biomoecular Cheistry, Vol. 10, No. 42, 2012, s. 8434-8444

- SCI

[o1] 2013 Chan, J.G.Y. - Chan, H.-K. - Prestidge, C.A. - Denman, J.A.b , Young, P.M. - Traini, D.:

European Journal of Pharmaceutics and Biopharmaceutics, Vol. 83, No. 2, 2013, s. 285-292 - SCI ;

SCOPUS

[o3] 2014 Parimala Vaijayanthi, S. - Mathiyalagan, N.: Antibacterial, antifungal, anti-oxidant, anti-

inflammatory and anti-hypertensive activities of N-chloropyrazinamide. In: International Letters of

Chemistry, Physics and Astronomy, Vol. 7, 2014, s. 1-8

[o1] 2014 Nayak, P.S. - Narayana, B. - Anthal, S. - Gupta, V.K. - Kant, R.: Molecular Crystals and Liquid

Crystals, Vol. 592, No. 1, 2014, s. 199-208 - SCI ; SCOPUS



Medicinal Chemistry Letters, Vol.25, No. 3, 2015, s. 524-528 - SCI ; SCOPUS


Vol. 1105, 2016, s. 104 - SCI; SCOPUS

[o1] 2015 Apostolov, S. - Vastag, G. - Matijevic, B. - Petrovic, S.: Journal of Liquid Chromatography and

Related Technologies, Vol. 38, No. 18, 2015, s. 1698 - SCI; SCOPUS

ADC31 Mrozek-Wilczkiewicz, Anna (10%) - Kalinowski, Danuta S. (10%) - Musiol, Robert (10%) - Finster,

Jacek (5%) - Szurko, Agnieszka (10%) - Serafin, Katarzyna (5%) - Knas, Magdalena (5%) -

Kamalapuram, Sishir K. (5%) - Kovacevic, Zaklina (10%) - Jampílek, Josef [UKOEXAF] (10%) -

Ratuszna, Alicja (5%) - Rzeszowska-Wolny, Joanna (5%) - Richardson, Des R. (5%) - Polanski, Jaroslaw

(5%): Investigating the anti-proliferative activity of styrylazanaphthalenes and azanaphthalenediones

Lit. 25 zázn.




IF (JCR) 2010=2,978

ADC32 Musiol, Robert (15%) - Jampílek, Josef [UKOEXAF] (15%) - Nycz, Jacek E. (5%) - Peško, Matúš

[UKOPREEF] (10%) - Carroll, James (10%) - Kráľová, Katarína [UKOPRCUS] (10%) - Vejsova,

Marcela (10%) - O Mahony, Jim (5%) - Coffey, Aidan (5%) - Mrozek,Anna (5%) - Polanski, Jaroslaw

(10%): Investigating the Activity Spectrum for Ring-Substituted 8-Hydroxyquinolines

Lit.: 48 zázn., 3 tab.




IF (JCR) 2010=1,988

Ohlasy (15):







[o1] 2012 Stein, A.L. - Bilheri, F.N. - Da Rocha, J.T. - Back, D.F. - Zeni, G.: Chemistry - A European

Journal, Vol. 18, No. 34, 2012, s. 10602-10608 - SCOPUS

[o3] 2012 Panda, B.K.: Synthesis, characterization and photophysical properties of quinolin-8-olato

chelated osmium(II) organometallics bearing a pendant imine-phenol motif and electrogeneration of

trivalent analogue. In: Open Journal ofInorganic Chemistry, Vol. 2, No. 3, 2012, s. 49-57

[o1] 2013 Li, Y. - De Kock, C. - Smith, P.J. - Guzgay, H. - Hendricks, D.T. - Naran, K. - Mizrahi, V. -

Warner D.F. - Chibale, K. - Smith, G.S.: Organometallics, Vol. 32, No. 1, 2013, s. 141-150 - SCI

21

[o1] 2013 Novakova, J. - Vlkova, E. - Bonusova, B. - Rada, V. - Kokoska, L.: Anaerobe, Vol. 22, 2013, s.


[o1] 2013 Vandekerckhove, S. - Tran, H.G. - Desmet, T. - D'Hooghe, M.: Bioorganic and Medicinal

Chemistry Letters, Vol. 23, No. 16, 2013, s. 4641-4643 - SCI ; SCOPUS

[o1] 2014 Mantovani, A.C. - Pesarico, A.P. - Sampaio, T.B. - Nogueira, C.W. - Zeni, G.: Journal of

Pharmaceutical Sciences, Vol. 51, No. 1, 2014, s. 196-203 - SCI ; SCOPUS

[o3] 2012 Kaiss, R.I. - Noor, F.A.-A.: Synthesis and study some mixed ligands complexes from folic acid

with 1,10-phenanthroline and 8-hydroxyquinoline. In: Journal of University of Anbar for Pure Science,

Vol. 6, No. 3, 2012, s. 67-74

[o1] 2014 Muscia, G.C. - Hautmann, S. - Buldain, G.Y. - Asís, S.E. - Gütschow, M.: Bioorganic and

Medicinal Chemistry Letters, Vol. 24, No. 6, 2014, s. 1545-1549 - SCI

[o1] 2014 De O Freitas, L.B. - Borgati, T.F. - De Freitas, R.P. - Ruiz, A.L.T.G. - Marchetti, G.M. - De

Carvalho, J.E. - Da Cunha, E.F.F. - Ramalho, T.C. - Alves, R.B: European Journal of Medicinal

Chemistry, Vol. 84, September, 2014, s. 595-604 - SCI ; SCOPUS

[o1] 2014 Ariyasu, S. - Mizuseda, Y. - Hanaya, K. - Aoki, S.: Chemical and Pharmaceutical Bulletin, Vol.

62, No. 7, 2014, s. 642-648 - SCOPUS


Vol. 6, No. 6, 2014, s. 101-109 - SCOPUS

[o3] 2015 Siddiqi, H. - Faizi, S. - Naz, S. - Zahir, E.: Synthesis of Mannich Bases of 8-Hydroxyquinoline.

In: Journal of Basic and Applied Sciences, Vol. 11, 2015, s. 539-543

ADC33 Oktábec, Zbyněk (15%) - Kos, Jiří (10%) - Mandelová, Zuzana (10%) - Havelková, Lenka (5%) -

Pekárek, Tomáš (10%) - Řezáčová, Anna (10%) - Plaček, Lukáš (10%) - Tkadlecová, Marcela (5%) -

Havlíček, Jaroslav (5%) - Dohnal, Jiří (5%) - Jampílek, Josef [UKOEXAF] (15%): Preparation and

properties of new Co-crystals of ibandronate with gluco- or galactopyranoside derivatives

Lit. 25 zázn.




IF (JCR) 2010=1,988

ADC34 Otevřel, Jan (10%) - Mandelová, Zuzana (5%) - Peško, Matúš [UKOPREEF] (10%) - Guo, Jiahui (10%)

- Kráľová, Katarína [UKOPRCUS] (10%) - Šeršeň, František [UKOPRCUS] (10%) - Vejsová, Marcela

(5%) - Kalinowski, Danuta S. (5%) - Kovacevic, Zaklina (5%)- Coffey, Aidan (5%) - Csöllei, Jozef (10%)

- Richardson, Des R. (5%) - Jampílek, Josef [UKOEXAF] (10%): Investigating the Spectrum of Biological

Activity of Ring-Substituted Salicylanilides and Carbamoylphenylcarbamates





IF (JCR) 2010=1,988

Ohlasy (4):



[o1] 2012 Krátky, M. - Vinšová, J.: Molecules, Vol. 17, No. 8, 2012, s. 9426-9442 - SCI ; SCOPUS

[o1] 2013 Kang, S. - Min, H.-J. - Kang, M.-S. - Jung, M.-G. - Kim, S.: Bioorganic and Medicinal

Chemistry Letters, Vol. 23, No. 6, 2013, s. 1748-1751 - SCI ; SCOPUS

[o3] 2013 Madhavan, M.S. - Varghese, H.T. - Panicker, C.Y. - Mathew, S.: Natural Bond Orbital (NBO)

Analysis of Certain Salicylanilide Derivatives. In: Material Science Research India, Vol. 10, 2013, s. 37-50

ADC35 Skórska-Stania, Agnieszka (20%) - Sliwa, Magdalena (20%) - Musilek, Kamil (10%) - Kuča, Kamil

(10%) - Jampílek, Josef [UKOEXAF] (10%) - Musiol, Robert (10%) - Oleksyn, Barbara (10%) - Dohnal,

Jiří (10%): Selected AChE reactivators in different crystalline environment: salts and enzyme

Lit. 24 zázn.

In: Structural Chemistry. - Vol. 21, No. 3 (2010), s. 495-501



IF (JCR) 2010=1,727

ADC36 Imramovský, Aleš (20%) - Peško, Matúš [UKOPREEF] (15%) - Ferriz, Juana Monreal (10%) -

Kráľová, Katarína [UKOPRCUS] (25%) - Vinšová, Jarmila (10%) - Jampílek, Josef [UKOEXAF] (20%):

Photosynthesis-Inhibiting efficiency of 4-chloro-2-(chlorophenylcarbamoyl)phenyl alkylcarbamates

22





IF (JCR) 2011=2,554

Ohlasy (1):

[o3] 2013 Madhavan, M.S. - Varghese, H.T. - Panicker, C.Y. - Mathew, S.: Natural Bond Orbital (NBO)

Analysis of Certain Salicylanilide Derivatives. In: Material Science Research India, Vol. 10, 2013, s. 37-50

ADC37 Imramovský, Aleš (25%) - Peško, Matúš [UKOPREEF] (15%) - Kráľová, Katarína [UKOPRCUS]

(15%) - Vejsova, Marcela (10%) - Stolaříková, Jiřina (10%) - Vinsova, Jarmila (10%) - Jampílek, Josef

[UKOEXAF] (15%): Investigating Spectrum of BiologicalActivity of 4-and 5-Chloro-2-hydroxy-N-[2-

(arylamino)-1-alkyl-2-oxoethyl]benzamides





IF (JCR) 2011=2,386

Ohlasy (3):

[o1] 2012 Balkrishna, S.J. - Kumar, S.: Synthesis, Vol. 44, No. 9, 2012, s. 1417-1426 - SCI ; SCOPUS

[o1] 2014 Güell, I. - Ribas, X.: Journal of Organic Chemistry, Vol. 2014, No. 15, 2014, s. 3188-3195 - SCI

[o1] 2015 Mahesh, B. - Mohan, G. - Kabeer, S.A. - Venkateswarulu, N. - Vijaya, T. - Reddy, C.S.:

Synthetic Communications, Vol. 45, No. 7, 2015, s. 838-846 - SCI ; SCOPUS

ADC38 Kos, Jiří (15%) - Pěntáková, Monika (5%) - Oktábec, Zbyněk (10%) - Krejčík, Lukáš (5%) -

Mandelová, Zuzana (5%) - Haroková, Pavla (5%) - Hrušková, Jana (5%) - Pekárek, Tomáš (5%) -

Dammer, Ondrej (5%) - Tkadlecová, Marcela (5%) - Havlíček, Jaroslav(5%) - Vinšová, Jarmila (5%) -

Král, Vladimír (5%) - Dohnal, Jiří (5%) - Jampílek, Josef [UKOEXAF] (15%): Crystallization products of

risedronate with carbohydrates and their substituted derivatives

Lit. 32 zázn.




IF (JCR) 2011=2,386

ADC39 Mandelová, Zuzana (15%) - Opatřilová, Radka (5%) - Raich, Ivan (15%) - Havlíček, Jaroslav (10%) -

Kačerová, Sandra (10%) - Pekárek, Tomáš (10%) - Tkadlecová, Marcela (10%) - Stašková, Petra (5%) -

Dohnal, Jiří (5%) - Csöllei, Jozef (5%) - Jampílek, Josef [UKOEXAF] (10%): Synthesis, Physico-

Chemical Properties and DFT Calculations of New 2-(4-Arylpiperazine-1-yl)-1-(3-ethylbenzofuran-2-

yl)ethanols As Potential Antihypertensive Agents

Lit. 34 zázn.




IF (JCR) 2011=3,064

ADC40 Mrózek, Lech (15%) - Dvořáková, Lenka (15%) - Mandelová, Zuzana (5%) - Rárová, Lucie (10%) -

Řezáčová, Anna (5%) - Plaček, Lukáš (5%) - Opatřilová, Radka (5%) - Dohnal, Jiří (5%) - Paleta, Oldřich

(5%) - Král, Vladimír (5%) - Drašar, Pavel (10%) - Jampílek, Josef [UKOEXAF] (15%): Investigation of

new acyloxy derivatives of cholic acid and their esters as drug absorption modifiers

Lit. 57 zázn.

In: Steroids. - Vol. 76, No. 10-11 (2011), s. 1082-1097



IF (JCR) 2011=2,892

ADC41 Opletalová, Veronika (15%) - Doležel, Jan (15%) - Kráľová, Katarína [UKOPRCUS] (25%) - Peško,

Matúš [UKOPREEF] (15%) - Kunes, Jiří (15%) - Jampílek, Josef [UKOEXAF] (15%): Synthesis and

Characterization of (Z)-5-Arylmethylidene-rhodanines with Photosynthesis-Inhibiting Properties





23

IF (JCR) 2011=2,386

Ohlasy (7):

[o1] 2011 Jacobine, A.M. - Posner, G.H.: Journal of Organic Chemistry, Vol. 76, No. 19, 2011, s. 8121-

8125 - SCI ; SCOPUS

[o1] 2013 Han, L. - Wu, T. - Zhou, Z.: Scientific World Journal, Vol. 2013, 2013, Art. No. 543768 - SCI ;

SCOPUS

[o1] 2014 Guiheneuf, S. - Paquin, L., - Carreaux, F. - Durieu, E. - Roisnel, T. - Meijer, L. - Bazureau, J.P.:

Molecular Diversity, Vol. 18, No. 2, 2014, s. 375-388 - SCI; SCOPUS

[o1] 2014 Zapol'skii, V.A. - Namyslo, J.C. - Gjikaj, M. - Kaufmann, D.E.: Beilstein Journal of Organic

Chemistry, Vol. 10, Art. No. 170, 2014, s. 1638-1644 - SCI; SCOPUS

[o1] 2014 Ramesh, V. - Ananda Rao, B. - Sharma, P. - Swarna, B. - Thummuri, D. - Srinivas, K. - Naidu,

V.G.M. - Jayathirtha Rao, V.: European Journal of Medicinal Chemistry, Vol. 83, August, 2014, s. 569-

580 - SCI; SCOPUS

[o1] 2014 Jadav, S.S. - Sinha, B.N. - Hilgenfeld, R. - Pastorino, B. - de Lamballerie, X. - Jayaprakash, V.:

European Journal of Medicinal Chemistry, Vol. 89, 2014, s. 172-178 - SCOPUS

[o3] 2014 Guihéneuf, S. - Paquin, L. - Carreaux,F. - Durieu, E. - Bénédetti, H. - Le Guével, R.l. - Corlu,A.

- Meijer, L. - Bazureau J.: Microwave Assisted Organic Synthesis (MAOS) of New Dispacamide A

Derivatives Bearing a Thiazolinone Platform, Biological Assays on Inhibition of Protein Kinases and Cell

Effects. In: Current Microwave Chemistry, Vol. 1, No. 1, 2014, s. 40

ADC42 Pejchal, Vladimír (20%) - Štěpánková, Šárka (20%) - Padělková, Zdeňka (20%) - Imramovský, Aleš

(20%) - Jampílek, Josef [UKOEXAF] (20%): 1,3-substituted imidazolidine-2,4,5-triones: synthesis and

inhibition of cholinergic enzymes

Lit. 49 zázn.




IF (JCR) 2011=2,386

ADC43 Bobáľ, Pavel (20%) - Sujan, Josef (20%) - Otevřel, Jan (20%) - Imramovský, Aleš (10%) - Padělková,

Zdeňka (10%) - Jampílek, Josef [UKOEXAF] (20%): Microwave-assisted synthesis of new substituted

anilides of quinaldic acid

Lit. 44 zázn.




IF (JCR) 2012=2,428

Ohlasy (3):

[o1] 2013 Ju, L. - Yao, J.Z. - Wu, Z.H. - Liu, Z.X. - Zhang, Y.H.: Journal of Organic Chemistry, Vol. 78,

No. 21, 2013, s. 10831 - SCI

[o1] 2014 Lukasik, N. - Wagner-Wysiecka, E.: Current Organic Synthesis, Vol. 11, No. 4, 2014, s. 604 -

SCI

[o1] 2015 Latimer, D. - Wiebe, M.: Green Chemistry Letters and Reviews, Vol. 8, No. 2, 2015, s. 42 - SCI

ADC44 Brychtová, Kateřina (20%) - Dvořáková, Lenka (10%) - Opatřilová, Radka (5%) - Raich, Ivan (10%) -

Kačerová, Sandra (10%) - Plaček, Lukáš (5%) - Kalinowski, Danuta S. (10%) - Richardson, Des R. (10%)

- Jampílek, Josef [UKOEXAF] (20%): Investigationof substituted 6-aminohexanoates as skin penetration

enhancers

Lit. 55 zázn.




IF (JCR) 2012=2,903

Ohlasy (1):

[o1] 2013 Marepally, S. - Boakye, C.H.A. - Shah, P.P. - Etukala, J.R. - Vemuri, A. - Singh, M.: PLoS

ONE, Vol. 8, No. 12, 2013, Article No. UNSP e82581 - SCI

ADC45 Cieslik, Wioleta (20%) - Jampílek, Josef [UKOEXAF] (15%) - Musiol, Robert (15%) - Nycz, Jacek E.

(10%) - Vejsová, Marcela (10%) - Machura, Barbara (10%) - Wolff, Mariusz (10%) - Polanski, Jaroslaw

(10%): Contribution to investigation of antimicrobial activity of styrylquinolines

Lit. 56 zázn.


24



IF (JCR) 2012=2,903

Ohlasy (5):

[o1] 2013 Radchatawedchakoon, W. - Promthong, N. - Sakee, U.: Letters in Organic Chemistry, Vol. 10,

No. 9, 2013, s. 644 - SCI; SCOPUS

[o1] 2014 Mantovani, A.C. - Pesarico, A.P. - Sampaio, T.B. - Nogueira, C.W. - Zeni, G.: European Journal

of Pharmaceutical Sciences, Vol. 51, 2014, s. 203 - SCI; SCOPUS

[o1] 2014 Muscia, G.C. - Hautmann, S. - Buldain, G.Y. - Asis, S.E. - Gutschow, M.: Bioorganic &

Medicinal Chemistry Letters, Vol. 24, No. 6, 2014, s. 1549 - SCI; SCOPUS

[o1] 2015 Xiao, J.C. - Huang, Y. - Song, Z.L. - Feng, W.H.: RSC Advances, Vol. 5, No. 10, 2015, s.

99098 - SCI; SCOPUS

[o1] 2015 Huang, L. - Fei, T.H. - Hu, K. - Liu, F.M.: Journal of Heterocyclic Chemistry, Vol. 52, No. 3,

2015, s. 906 - SCI; SCOPUS

ADC46 Fajkusová, Dagmar (25%) - Peško, Matúš [UKOPREEF] (10%) - Keltošová, Stanislava (5%) - Guo,

Jiahui (5%) - Oktábec, Zbyněk (5%) - Vejsová, Marcela (5%) - Kollár, Peter (5%) - Coffey, Aidan (10%) -

Csöllei, Jozef (10%) - Kráľová, Katarína [UKOPRCUS] (10%) - Jampílek, Josef [UKOEXAF] (10%):

Anti-infective and herbicidal activity of N-substituted 2-aminobenzothiazoles





IF (JCR) 2012=2,903

Ohlasy (3):

[o1] 2013 Zhao, J.W. - Huang, H.W. - Wu, W.Q. - Chen, H.J. - Jiang, H.F.: Organic Letters, Vol. 15, No.

11, 2013, s. 2604-2607 - SCI

[o1] 2015 Keri, R.S. - Patil, M.R. - Patil, S.A. - Budagupi, S.: European Journal of Medicinal Chemistry,

Vol. 89, January, 2015, s. 207-251 - SCI ; SCOPUS

[o1] 2015 Seddighi, M. - Shirini, F. - Mamaghani, M.: Comptes Rendus Chimie, Vol. 18, No. 5, 2015, s.


ADC47 Goněc, Tomáš (15%) - Bobáľ, Pavel (5%) - Sujan, Josef (5%) - Peško, Matúš [UKOPREEF] (10%) -

Guo, Jiahui (5%) - Kráľová, Katarína [UKOPRCUS] (10%) - Pavlacká, Lenka (5%) - Veselý, Libor (5%) -

Kreckova, Eva (5%) - Kos, Jiří (5%) - Coffey, Aidan (5%) - Kollár, Peter [UKOEXAF] (5%) -

Imramovský, Aleš (5%) - Plaček, Lukaš (5%) - Jampílek, Josef [UKOEXAF] (10%): Investigating the

Spectrum of Biological Activity of Substituted Quinoline-2-Carboxamides and Their Isosteres





IF (JCR) 2012=2,428

Ohlasy (9):

[o1] 2013 Tian, T. - Zhong, W.H. - Meng, S. - Meng, X.B. - Li, Z.J.: Journal of Organic Chemistry, Vol.

78, No. 2, 2013, s. 728-732 - SCI; SCOPUS

[o1] 2013 Mamidi, N. - Manna, D.: Journal of Organic Chemistry, Vol.78, No. 6, 2013, s. 2386-2396 -

SCI; SCOPUS

[o1] 2014 Hassan, W.M.I. - Moustafa, H. - Hamed, M.N.H. - Ali, L.I. - Halim, S.A.: Spectrochimica Acta

Part A: Molecular and Biomolecular Spectroscopy, Vol. 117, 2014, s. 587-597 - SCI; SCOPUS

[o1] 2014 Babjak, M. - Caletková, O. - Ďurišová, D. - Gracza, T.: Synlett, Vol. 25, No. 18, 2014, Art. No.

st-2014-b0535-1, s. 2579-2584 - SCI; SCOPUS

[o1] 2014 Keri, R.S. - Patil, S.A.: Biomedicine and Pharmacotherapy, Vol. 68, No. 8, 2014, s. 1161-1175 -

SCI; SCOPUS

[o1] 2015 Funder, E.D. - Trads, J.B. - Gothelf, K.V.: Organic and Biomolecular Chemistry, Vol. 13, No. 1,

2015, s. 185-198 - SCI ; SCOPUS

[o3] 2015 Baluja, S.: Dissociation Constants of Some Quinoline Derivatives in Mixed Solvent mixture. In:

International Letters of Chemistry, Physics and Astronomy, International Letters of Chemistry, Physics

and Astronomy, Vol. 9, No. 1, 2015, s. 32-36

[o3] 2015 Boyarshinov V.D. - Mikhalev A.I. - Yushkova T.A. - Konshina T.A. - Ukhov S.V.: Synthesis

and biological activity quinoline-2-carboxamides. In: Pharmaceutical Sciences, Fundamental Research,

No. 2, 2015, s. 1715-1719

25

[o1] 2015 Xie, H. - Liao, Y. - Chen, S. - Chen, Y. - Deng, G.-J.: Organic and Biomolecular Chemistry,

Vol. 13, No. 25, 2015, s. 6944-6948 - SCI; SCOPUS

ADC48 Imramovský, Aleš (16%) - Štěpánková, Šárka (14%) - Vančo, Ján [UKOEXAF] (14%) - Pauk, Jozef

(14%) - Monreal-Ferriz, Juana (14%) - Vinšová, Jarmila (14%) - Jampílek, Josef [UKOEXAF] (14%):

Acetylcholinesterase-inhibiting activity of salicylanilide N-alkylcarbamates and their molecular docking

Lit. 50 zázn.




IF (JCR) 2012=2,428

Ohlasy (7):

[o1] 2014 Das, R.N. - Roy, K.: Industrial & Engineering Chemistry Research, Vol. 53, No. 2, 2014, s.

1032 - SCI

[o1] 2014 Lo, R. - Ganguly, B.: Molecular Biosystems, Vol. 10, No. 9, 2013, s. 2383 - SCI

[o1] 2014 Varadaraju, K.R. - Kumar, J.R. - Mallesha, L. - Muruli, A. - Mohana, K.N.S. - Mukunda, C.K. -

Sharanaiah, U.: International Journal of Alzheimer's Disease, Vol. 2013, art.no. 653962 - SCOPUS

[o1] 2015 Gocer, H. - Akincioglu, A. - Goksu, S. - Gulcin, I. - Supuran, C.T.: Journal of Enzyme

Inhibition and Medicinal Chemistry, Vol. 30, No. 2, 2015, s. 320 - SCI

[o1] 2015 Thangnipon, W. - Suwanna, N. - Jantrachotechatchawan, C. - Ngampramuan, S. - Tuchinda, P. -

Nobsathian, S.: Archives of Pharmacal Research, Vol. 38, No. 7, 2015, s. 1388 - SCI

[o1] 2015 Basant, N. - Gupta, S. - Singh, K.P.: Journal of Molecular Liquids, Vol. 209, 2015, s. 412 - SCI

[o1] 2015 Kose, L.P. - Gulcin, I. - Goren, A.C. - Namiesnik, J. - Martinez-Ayala, A.L. - Gorinstein, S.:

Industrial Crops and Products, Vol. 74, 2015, s. 721 - SCI

ADC49 Jampílek, Josef [UKOEXAF] (60%) - Brychtová, Kateřina (40%): Azone analogues: classification,

design, and transdermal penetration principles

Lit. 238 zázn.

In: Medicinal Research Reviews. - Vol. 32, No. 5 (2012), s. 907-947



IF (JCR) 2012=9,583

ADC50 Serda, Maciej (20%) - Mrozek-Wilczkiewicz, Anna (10%) - Peško, Matúš [UKOPREEF] (10%) -

Kráľová, Katarína [UKOPRCUS] (10%) - Vejsova, Marcela (10%) - Musiol, Robert (10%) - Ratuszna,

Alicja (10%) - Polanski, Jaroslaw (10%) - Jampílek, Josef [UKOEXAF] (10%): Investigation of the

Biological Properties of (Hetero)Aromatic Thiosemicarbazones





IF (JCR) 2012=2,428

Ohlasy (4):

[o1] 2014 Pino-Cuevas, A. - Carballo, R. - Vázquez-López, E.M.: Acta Crystallographica Section E:

Structure Reports Online, Vol. 70, No. 9, 2014, s. o926 - SCOPUS

[o1] 2014 Carballo, R. - Pino-Cuevas, A. - Ezequiel, M. - Vazquez-Lopez, E.M.: Acta Crystallographica

Section E: Structure Reports Online, Vol. 70, No. 9, 2014, s. o970 S - SCOPUS

[o1] 2014 Paiva, R.O. - Kneipp, L.F. - Goular, C.M. - Albuquerque, M.A. - Echevarria, A.: Ciencia e

Agrotecnologia, Vol. 38, No. 6, 2014, s. 531-537 - SCOPUS; SCI

[o1] 2015 Cui, J. - Lin, Q. - Gan, C. - Zhan, J. - Su, W. - Zhao, D. - Qi, B. - Huang, Y.: Steroids, Vol. 98,

Art. No. 7766, 2015, s. 138-142 - SCOPUS

ADC51 Vaculiková, Eliška (30%) - Grünwaldová, Veronika (20%) - Král, Vladimír (15%) - Dohnal, Jiří (10%) -

Jampílek, Josef [UKOEXAF] (25%): Primary Investigation of the Preparation of Nanoparticles by

Precipitation

Lit. 30 zázn.




IF (JCR) 2012=2,428

Ohlasy (1):

26

[o1] 2015 Pinjari, D.V. - Prasad, K. - Gogate, P.R. - Mhaske, S.T. - Pandit, A.B.: Ultrasonics

Sonochemistry, Vol. 23, 2015, s. 191 - SCI

ADC52 Vaculiková, Eliška (30%) - Grünwaldová, Veronika (20%) - Král, Vladimír (15%) - Dohnal, Jiří (10%) -

Jampílek, Josef [UKOEXAF] (25%): Preparation of candesartan and atorvastatin nanoparticles by solvent

evaporation

Lit. 46 zázn.




IF (JCR) 2012=2,428

Ohlasy (5):

[o1] 2013 Anarjan, N. - Tan, C.P.: Molecules, Vol. 18, No. 1, 2013, s. 777 - SCI

[o1] 2015 Yeom, D.W. - Song, Y.S. - Kim, S.R. - Lee, S.G. - Kang, M.H. - Lee, S. - Choi, Y.W.:

International Journal of Nanomedicine, Vol. 10, 2015, s. 3878 - SCI

[o1] 2015 Sezgin-Bayindir, Z. - Antep, M.N. - Yuksel, N.: AAPS PharmSciTech, Vol. 16, No. 1, 2015, s.

117 - SCI

[o1] 2015 Agrawal, A.G. - Kumar, A. - Gide, P.S.: Drug Development and Industrial Pharmacy, Vol. 41,

No. 4, 2015, s. 604 - SCI

[o1] 2015 Hennig, R. - Ohlmann, A. - Staffel, J. - Pollinger, K. - Haunberger, A. - Breunig, M. - Schweda,

F. - Tamm, E.R. - Goepferich, A.: Journal of Controlled Release, Vol. 22, 2015, s. 274 - SCI

ADC53 Zitko, Jan (25%) - Jampílek, Josef [UKOEXAF] (20%) - Dobrovolný, Lukáš (25%) - Svobodová,

Michaela (10%) - Kuneš, Jiří (10%) - Doležal, Martin (10%): Synthesis and antimycobacterial evaluation

of N-substituted 3-aminopyrazine-2,5-dicarbonitriles

Lit. 23 zázn.




IF (JCR) 2012=2,338

ADC54 Coufalová, Lenka (10%) - Mrózek, Lech (10%) - Rárová, Lucie (10%) - Plaček, Lukáš (10%) -

Opatřilová, Radka (10%) - Dohnal, Jiří (5%) - Kráľová, Katarína [UKOPRCUS] (10%) - Paleta, Oldřich

(5%) - Král, Vladimír (10%) - Drašar, Pavel (10%) - Jampílek, Josef [UKOEXAF] (10%): New

propanoyloxy derivatives of 5 beta-cholan-24-oic acid as drug absorption modifiers

Lit.: 68 zázn., 4 obr., 5 schém, 2 tab.

In: Steroids. - Vol. 78, No. 5 (2013), s. 435-453



IF (JCR) 2013=2,716

Ohlasy (5):

[o1] 2013 Perrone, D. - Bortolini, O. - Fogagnolo, M. - Marchesi, E. - Mari, L. - Massarenti, C. -

Navacchia, M.L. - Sforza, F. - Varani, K. - Capobianco, M.L.: New Journal of Chemistry, Vol. 37, No. 1,

2013, s. 3559-3567 - SCI

[o1] 2014 Ojewole, E. - Kalhapure, R. - Akamanchi, K. - Govender, T.: Drug Development and Industrial

Pharmacy, Vol. 40, No. 5, 2014, s. 657-668 - SCOPUS

[o1] 2014 Yang, Y.X. - Zheng, L.T. - Shi, J.J. - Gao, B. - Chen, Y.K. - Yang, H.C. - Chen, H.L. - Li, Y.C.

- Zhen, X.C.: Bioorganic and Medicinal Chemistry Letters, Vol. 24, No. 4, 2014, s. 1222-1227 - SCI ;

SCOPUS

[o1] 2015 Poša, M. - Bjedov, S. - Škoric, D. - Sakač, M.: Biochimica et Biophysica Acta - General

Subjects, Vol. 1850, No. 7, 2015, s. 1345-1353 - SCOPUS

[o1] 2015 Moghimipour, E. - Ameri, A. - Handali, S.: Molecules, Vol. 20, No. 8, 2015, s. 14451-14473 -

SCOPUS

ADC55 Čulen, Martin (25%) - Řezáčová, Anna (25%) - Jampílek, Josef [UKOEXAF] (25%) - Dohnal, Jiří

(25%): Designing a Dynamic Dissolution Method: A Review of Instrumental Options and Corresponding

Physiology of Stomach and Small Intestine

Lit. 111 zázn.

In: Journal of Pharmaceutical Sciences. - Vol. 102, No. 9 (2013), s. 2995-3017



IF (JCR) 2013=3,007

27

Ohlasy (6):

[o1] 2014 Zhao, Y. - Bettinger, J. - Caritis, S. - Venicataramanan, R.: American Journal of Health-System

Pharmacy, Vol. 71, No. 13, 2014, s. 1127 - SCI

[o1] 2014 Nokhodchi, A. - Asare-Addo, K.: Expert Opinion on Drug Delivery, Vol. 11, No. 9, 2014, s.

1418 - SCI

[o1] 2014 Hens, B. - Brouwers, J. - Anneveld, B. - Corsetti, M. - Symillides, M. - Vertzoni, M. - Reppas,

C. - Turner, D.B. - Augustijns, P.: European Journal of Pharmaceutical Sciences, Vol. 63, 2014, s. 242 -

SCI

[o1] 2014 Rhee, K.H. - Park, J.S. - Cho, M.J.: Yonsei Medical Journal, Vol. 55, No. 6, 2014, s. 1466 - SCI

[o1] 2014 Wu, P. - Chen, L.D. - Wu, X. - Chen, X.D.: Journal of Food Engineering, Vol. 142, 2014, s. 178

- SCI

[o1] 2015 Wuyts, B. - Riethorst, D. - Brouwers, J. - Tack, J. - Annaert, P. - Augustijns, P.: European

Journal of Pharmaceutical Sciences, Vol. 67, 2015, s. 135 - SCI

ADC56 Goněc, Tomáš (10%) - Kos, Jiří (5%) - Zadražilová, Iveta (10%) - Peško, Matúš [UKOPREEF] (10%) -

Govender, Rodney (5%) - Keltošová, Stanislava (5%) - Chambel, Barbara (5%) - Pereira, Diogo (5%) -

Kollár, Peter (5%) - Imramovský, Aleš (5%) – O´Mahony, Jim (5%) - Coffey, Aidan (5%) - Čížek, Alois

(5%) - Kráľová, Katarína [UKOPRCUS] (10%) - Jampílek, Josef [UKOEXAF] (10%): Antibacterial and

herbicidal activity of ring-substituted 2-hydroxynaphthalene-1-carboxanilides





IF (JCR) 2013=2,095

Ohlasy (1):

[o1] 2015 Kotb, E.R. - Anwar, M.M. - Syam, Y.M. - Bagato, O. - AbdelMoaz, S.: International Journal of

Pharmacy and Technology, Vol. 7, No. 1, 2015, s. 8237-8273 - SCOPUS

ADC57 Goněc, Tomáš (10%) - Kos, Jiří (10%) - Zadražilová, Iveta (10%) - Peško, Matúš [UKOPREEF] (10%)

- Keltošová, Stanislava (10%) - Tengler, Jan (10%) - Bobáľ, Pavel (5%) - Kollár, Peter (5%) - Čížek, Alois

(10%) - Kráľová, Katarína [UKOPRCUS] (10%) - Jampílek, Josef [UKOEXAF] (10%):

Antimycobacterial and herbicidal activity of ring-substituted 1-hydroxynaphthalene-2-carboxanilides

Lit.: 50 zázn., 5 obr., 1 schéma, 1 tab.




IF (JCR) 2013=2,951

Ohlasy (3):

[o1] 2014 Xu, S. - Li, D. - Pei, L. - Yao, H. - Wang, C. - Cai, H. - Yao, H. - Wu, X. - Xu, J.: Bioorganic

and Medicinal Chemistry Letters, Vol. 24, No. 13, 2014, s. 2811-2814 - SCOPUS; SCI

[o1] 2014 Chaaban, I. - El Khawass, E.S.M. - Abd El Razik, H.A. - El Salamouni, N.S. - Redondo-

Horcajo, M. - Barasoain, I. - Díaz, J.F. - Yli-Kauhaluoma, J. - Moreira, V.M.: European Journal of

Medicinal Chemistry, Vol. 87, November, 2014, s.805-813 - SCOPUS; SCI

[o1] 2015 Brahmachari, G.: ACS Sustainable Chemistry and Engineering, Vol. 3, No. 9, 2015, s. 2058-

2066 - SCOPUS; SCI

ADC58 Imramovský, Aleš (10%) - Pejchal, Vladimír (9%) - Štěpánková, Šárka (9%) - Vorčáková, Katarína

(9%) - Vančo, Ján [UKOEXAF] (9%) - Šimůnek, Petr (9%) - Královec, Karel (9%) - Brůčková Lenka

(9%) - Mandíková, Jana (9%) - Trejtnar, František (9%) - Jampílek, Josef [UKOEXAF] (9%): Synthesis

and in vitro evaluation of new derivatives of 2-substituted-6-fluorobenzo[d]thiazoles as cholinesterase

inhibitors

Lit. 60 zázn.




IF (JCR) 2013=2,095

Ohlasy (4):

[o1] 2014 Du, X.J. - Bian, Q. - Wang, H.X. - Yu, S.J. - Kou, J.J. - Wang, Z.P. - Li, Z.M. - Zhao, W.G.:

Organic & Biomolecular Chemistry, Vol. 12, No. 29, 2014, s. 5434 - SCI

[o1] 2014 Gundogdu-Karaburun, N.: Letters in Drug Design & Discovery, Vol. 11, No.6, 2014, s. 823 -

SCI

28

[o1] 2015 Keri, R.S. - Patil, M.R. - Patil, S.A. - Budagupi, S.: European Journal of Medicinal Chemistry,

Vol. 89, 2015, s. 251 - SCOPUS

[o1] 2015 Hroch, L. - Aitken, L. - Benek, O. - Dolezal, M. - Kuca, K. - Gunn-Moore, F. - Musilek, K.:

Current Medicinal Chemistry, Vol. 22, No. 6, 2015, s. 747 - SCI

ADC59 Kos, Jiří (20%) - Zadražilová, Iveta (10%) - Peško, Matúš [UKOPREEF] (10%) - Keltošová, Stanislava

(5%) - Tengler, Jan (5%) - Goněc, Tomáš (5%) - Bobáľ, Pavel (5%) - Kauerová, Tereza (5%) - Oravec,

Michal (5%) - Kollár, Peter (5%) - Čížek, Alois (5%) - Kráľová, Katarína [UKOPRCUS] (10%) -

Jampílek, Josef [UKOEXAF] (10%): Antibacterial and herbicidal activity of ring-substituted 3-

hydroxynaphthalene-2-carboxanilides





IF (JCR) 2013=2,095

ADC60 Mrózek, Lech (20%) - Coufalová, Lenka (10%) - Rárová, Lucie (10%) - Plaček, Lukáš (5%) -

Opatřilová, Radka (10%) - Dohnal, Jiří (5%) - Kráľová, Katarína [UKOPRCUS] (10%) - Paleta, Oldřich

(10%) - Král, Vladimír (5%) - Drašar, Pavel (5%) - Jampílek, Josef [UKOEXAF] (10%): New

polyfluorothiopropanoyloxy derivatives of 5 beta-cholan-24-oic acid designed as drug absorption

modifiers

Lit.: 67 zázn., 4 obr., 2 schémy, 1 tab.

In: Steroids. - Vol. 78, No. 9 (2013), s. 832-844



IF (JCR) 2013=2,716

Ohlasy (2):

[o1] 2014 Ojewole, E. - Kalhapure, R. - Akamanchi, K. - Govender, T.: Drug Development and Industrial

Pharmacy, Vol. 40, No. 5, 2014, s. 657-668 - SCI; SCOPUS

[o1] 2015 Poša, M. - Bjedov, S. - Škoric, D. - Sakač, M.: Biochimica et Biophysica Acta - General

Subjects, Vol. 1850, No. 7, 2015, s. 1345-1353 - SCOPUS; SCI

ADC61 Otevřel, Jan (10%) - Bobáľ, Pavel (5%) - Zadražilová, Iveta (10%) - Govender, Rodney (5%) - Peško,

Matúš [UKOPREEF] (10%) - Keltošová, Stanislava (5%) - Kolečkárová, Petra (5%) - Maršálek, Petr (5%)

- Imramovský, Aleš (5%) - Coffey, Aidan (5%) – O´Mahony, Jim (5%) - Kollár, Peter (5%) - Čížek, Alois

(5%) - Kráľová, Katarína [UKOPRCUS] (10%) - Jampílek, Josef [UKOEXAF] (10%): Antimycobacterial

and photosynthetic electron transport inhibiting activity of ring-substituted4-arylamino-7-

chloroquinolinium chlorides





IF (JCR) 2013=2,095

ADC62 Pauk, Karel (25%) - Zadražilová, Iveta (20%) - Imramovský, Aleš (10%) - Vinšová, Jarmila (5%) -

Pokorná, Michaela (10%) - Masaříková, Martina (5%) - Čížek, Alois (5%) - Jampílek, Josef [UKOEXAF]

(20%): New derivatives of salicylamides: Preparationand antimicrobial activity against various bacterial

species

Lit. 44 zázn.




IF (JCR) 2013=2,951

Ohlasy (1):

[o1] 2015 Rajamuthiah, R. - Fuchs, B.B. - Conery, A.L. - Kim, W. - Jayamani, E. - Kwon, B. - Ausubel,

F.M. - Mylonakis, E.: PLoS ONE, Vol. 10, No. 4, Article No. UNSP e0124595 - SCI

ADC63 Tengler, Jan (20%) - Kapustíková, Iva (20%) - Stropnický, Ondřej (20%) - Mokrý, Petr (10%) - Oravec,

Michal (5%) - Csöllei, Jozef (5%) - Jampílek, Josef [UKOEXAF] (20%): Synthesis of new

(arylcarbonyloxy)aminopropanol derivatives and the determination of their physico-chemical properties

Lit. 36 zázn.

In: Central European Journal of Chemistry. - Vol. 11, No. 11 (2013), s. 1757-1767


29


IF (JCR) [2013-1,329]

ADC64 Goněc, Tomáš (15%) - Kos, Jiří (5%) - Nevin, Eoghan (5%) - Govender, Rodney (5%) - Peško, Matúš

[UKOPREEF] (10%) - Tengler, Jan (5%) - Kushkevych, Ivan (5%) - Šťastná, Vendula (5%) - Oravec,

Michal (10%) - Kollár, Peter (5%) – O´Mahony, Jim (5%) - Kráľová, Katarína [UKOPRCUS] (10%) -

Coffey, Aidan (5%) - Jampílek, Josef [UKOEXAF] (10%): Preparation and Biological Properties of Ring-

Substituted Naphthalene-1-Carboxanilides





IF (JCR) 2014=2,416

ADC65 Imramovský, Aleš (25%) - Peško, Matúš [UKOPREEF] (25%) - Kráľová, Katarína [UKOPRCUS]

(25%) - Jampílek, Josef [UKOEXAF] (25%): Synthesis and photosynthetic electron transport inhibition of

2-substituted 6-fluorobenzothiazoles


In: Monatshefte für Chemie. - Vol. 145, No. 11 (2014), s. 1817-1824



IF (JCR) 2014=1,222

ADC66 Jampílek, Josef [UKOEXAF] (100%) : Recent advances in design of potential quinoxaline anti-

infectives

Lit. 267 zázn.

In: Current Medicinal Chemistry. - Vol. 21, No. 38 (2014), s. 4347-4373



IF (JCR) 2014=3,853

ADC67 Krompiec, Stanislav (10%) - Malarz, Joanna (10%) - Pietraszuk, Cezary (10%) - Powala, Beata (5%) -

Rogalski, Szymon (5%) - Malecki, Jan G. (5%) - Penkala, Mateusz (5%) - Filapek, Michal (5%) - Musiol,

Robert (5%) - Jampílek, Josef [UKOEXAF] (5%) - Vejsova, Marcela (5%) - Polanski, Jaroslaw (5%) -

Paluch, Marian (5%) - Pawlus, Sebastian (5%) - Danikiewicz, Witold (5%) - Kania, Magdalena (5%) -

Marcol, Beata (5%): New strategy for the synthesis of 3,4,5-trisubstituted isoxazolines from

allylcompounds

Lit. 78 zázn.




IF (JCR) 2014=2,157

ADC68 Ulahannan, Rajeev T. (20%) - Panicker, C. Yohannan (20%) - Varghese, Hema Tresa (20%) - Musiol,

Robert (10%) - Jampílek, Josef [UKOEXAF] (10%) - Anto, P. L. (10%) - Van Alsenoy, Christian (10%):

Spectroscopic (FT-IR, FT-Raman) investigations and quantum chemical calculations of 4-hydroxy-2-oxo-

1,2-dihydroquinoline-7-carboxylic acid

Lit. 61 zázn.

In: Spectrochimica Acta, Part A-Molecular and Biomolecular Spectroscopy. - Vol. 121 (2014), s. 404-414



IF (JCR) 2014=2,353


Robert (10%) - Jampílek, Josef [UKOEXAF] (10%) - Anto, P. L. (10%) - Van Alsenoy, Christian (10%):

Vibrational spectroscopic, H-1 NMR and quantum chemical computational study of 4-hydroxy-2-oxo-1, 2-

dihydroquinoline-8-carboxylic acid

Lit. 70 zázn.




IF (JCR) 2014=2,353

Ohlasy (1):

30

[o1] 2015 Al-Otaibi, J.S. - Ai-Wabli, R.I.: Spectrochimica Acta Part A-Molecular and Biomolecular

Spectroscopy, Vol. 137, 2015, s. 15 - SCI

ADC70 Vaculiková, Eliška (14%) - Plachá, Daniela (14%) - Pisárčik, Martin [UKOFACH] (15%) - Peikertová,

Pavlína (14%) - Dedková, Kateřina (14%) - Devínsky, Ferdinand [UKOFACH] (15%) - Jampílek, Josef

[UKOEXAF] (14%): Preparation of Risedronate Nanoparticles by Solvent Evaporation Technique

Lit. 30 zázn.




IF (JCR) 2014=2,416

SJR (SCOPUS) [2014-0,650]

SNIP (SCOPUS) [2014-1,220]

Ohlasy (2):

[o1] 2015 Rawat, P. - Manglani, K. - Gupta, S. - Kalam, A. - Vohora, D. - Ahmad, F.J. - Talegaonkar, S.:

Pharmaceutical Research, Vol. 32, No. 10, 2015, s. 3158 - SCOPUS; SCI

[o1] 2015 Sun, D.Q. - Xue, A.Y. - Zhang, B. - Lou, H.Y. - Shi, H.Y. - Zhang, X.M.: Journal of Pharmacy

and Pharmacology, Vol. 67, No. 12, 2015, s. 1662 - SCI

ADC71 Goněc, Tomáš (20%) - Zadražilová, Iveta (5%) - Nevin, Eoghan (5%) - Krauerová, Tereza (5%) -

Peško, Matúš [UKOPREEF] (10%) - Kos, Jiří (5%) - Oravec, Michal (5%) - Kollár, Peter (5%) - Coffey,

Aidan (10%) - O Mahony, Jim (5%) - Cizek, Alois (5%) - Kráľová, Katarína [UKOPRCUS] (10%) -

Jampílek, Josef [UKOEXAF] (10%): Synthesis and Biological Evaluation of N-Alkoxyphenyl-3-






IF (JCR) 2015= [2014-2,416]

ADC72 Kos, Jiří (10%) - Nevin, Eoghan (10%) - Šoral, Michal (10%) - Kushkevych, Ivan (10%) - Goněc,

Tomáš (5%) - Bobáľ, Pavel (10%) - Kollár, Peter (5%) - Coffey, Aidan (5%) – O´Mahony, Jim (10%) -

Liptaj, Tibor (10%) - Kráľová, Katarína [UKOPRCUS] (5%)- Jampílek, Josef [UKOEXAF] (10%):

Synthesis and antimycobacterial properties of ring-substituted 6-hydroxynaphthalene-2-carboxanilides





IF (JCR) 2015= [2014-2,793]

Ohlasy (1):

[o1] 2015 Xiao, Z.P. - Wei, W. - Wang, P.F. - Shi, W.K. - Zhu, N. - Xie, M.Q. - Sun, Y.W. - Li, L.X. -

Xie, Y.X. - Zhu, L.S. - Tang, N. - Ouyang, H. - Li, X.H. - Wang, G.C. - Zhu, H.L.: European Journal of

Medicinal Chemistry, Vol. 102, Art.No. 8061, 2015, s. 631-638 - SCOPUS

ADC73 Kos, Jiří (20%) - Zadražilová, Iveta (5%) - Nevin, Eoghan (10%) - Šoral, Michal (10%) - Goněc, Tomáš

(5%) - Kollár, Peter (5%) - Oravec, Michal (5%) - Coffey, Aidan (5%) - O Mahony, Jim (5%) - Liptaj,

Tibor (10%) - Kráľová, Katarína [UKOPRCUS] (10%) - Jampílek, Josef [UKOEXAF] (10%): Ring-

substituted 8-hydroxyquinoline-2-carboxanilides as potential antimycobacterial agents

Lit.: 50 zázn.,3 obr., 1 tab.

In: Bioorganic and Medicinal Chemistry. - Vol 23, No. 15 (2015), s. 4188-4196



IF (JCR) 2015= [2014-2,793]

ADC74 Peško, Matúš [UKOPREEF] (40%) - Kos, Jiří (20%) - Kráľová, Katarína [UKOPRCUS] (20%) -

Jampílek, Josef [UKOEXAF] (20%): Inhibition of photosynthetic electron transport by 6-


Lit. 48 zázn., 2 obr., 1 tab.

In: Indian Journal of Chemistry Section B-Organic Chemistry Including Medicinal Chemistry. - Vol. 54,

No. 12 (2015), s. 1511-1517



IF (JCR) 2015= [2014-0,387]

31


Robert (10%) - Jampílek, Josef [UKOEXAF] (10%) - Van Alsenoy, Christian (10%) - War, Javeed Ahmad

(10%) - Manojkumar, T. K. (10%): Vibrational spectroscopic studies and molecular docking study of 2-

[(E)-2-phenylethenyl]quinoline-5-carboxylic acid

Lit. 47 zázn.




IF (JCR) [2014-2,353]



(10%) - Al-Saadi, Abdulaziz A. (10%): Vibrational spectroscopic and molecular docking study of (2E)-N-

(4-chloro-2-oxo-1,2-dihydroquinolin-3-yl)-3-phenylprop-2-enamide

Lit. 65 zázn.




IF (JCR) [2014-2,353]



(10%) - Srivastava, S. K. (10%): Molecular structure,FT-IR, FT-Raman, NBO, HOMO and LUMO, MEP,

NLO and molecular docking study of 2-[(E)-2-(2-bromophenyl)ethenyl]quinoline-6-carboxylic acid

Lit. 65 zázn.




IF (JCR) [2014-2,353]

ADC78 Zdražilová, Iveta (25%) - Pospíšilová, Šárka (25%) - Masariková, Martina (5%) - Imramovský, Aleš

(5%) - Ferriz, Juana Monreal (5%) - Vinšová, Jarmila (5%) - Čížek, Alois (10%) - Jampílek, Josef

[UKOEXAF] (20%): Salicylanilide carbamates: Promising antibacterial agents with high in vitro activity

against methicillin-resistant Staphylococcus aureus (MRSA)

Lit. 70 zázn.

In: European Journal of Pharmaceutical Sciences. - Vol. 77 (2015), s. 197-207



IF (JCR) [2014-3,350]

ADC79 Jampílek, Josef [UKOEXAF] (100%) : Potential of agricultural fungicides for antifungal drug discovery

Lit. 45 zázn.

In: Expert Opinion on Drug Discovery. - Vol. 11, No. 1 (2016), s. 1-9


IF (JCR) [2014-3,539]

ADD Vědecké práce v domácích karentovaných časopisech

ADD01 Kučerová-Chlupáčová, Marta (20%) - Opletalová, Veronika (20%) - Jampílek, Josef [UKOEXAF]

(20%) - Doležel, Jan (20%) - Dohnal, Jiří (5%) - Pour, Milan (5%) - Kuneš, Jiří (5%) - Vořišek, Viktor

(5%): New hydrophobicity constants of substituents in pyrazine rings derived from RP-HPLC study

Lit. 29 zázn.

In: Collection of Czechoslovak Chemical Communications. - Vol. 73, No. 1 (2008), s. 1-18



IF (JCR) [2008-0,784]

ADD02 Oktábec, Zbyněk (50%) - Jampílek, Josef [UKOEXAF] (50%): Stručná historie chemoterapie = Brief

history of chemotherapy

Lit. 77 zázn.

In: Chemické listy. - Roč. 107, č. 2 (2013), s. 150-158



IF (JCR) [2013-0,196]

32

ADD03 Černíková, Aneta (50%) - Jampílek, Josef [UKOEXAF] (50%): Strukturní modifikace léčiv ovlivňující

biodostupnost a terapeutický účinek = Structure modification of drugs or prodrugs influencing their

bioavailability and therapeutic effect

Lit. 70 zázn.




IF (JCR) [2014-0,272]

ADD04 Pěntáková, Monika (50%) - Jampílek, Josef [UKOEXAF] (50%): Patentová historie přípravku

Viagra(R) = Patent history of Viagra(R) preparation

Lit. 14 zázn.




IF (JCR) [2014-0,272]

ADD05 Vaculiková, Eliška (50%) - Plachá, Daniela (25%) - Jampílek, Josef [UKOEXAF] (25%): Toxikologie

nanoforem nosičů léčiv = Toxicology of drug nanocarriers

Lit. 74 zázn.




IF (JCR) [2014-0,272]

ADE Vědecké práce v zahraničních nekarentovaných časopisech

ADE01 Doležal, Martin (30%) - Jampílek, Josef [UKOEXAF] (30%) - Osička, Zdeněk (5%) - Kuneš, Jiří (10%)

- Buchta, Vladimír (20%) - Víchová, Petra (5%): Substituted 5-aroylpyrazine-2-carboxylic acid

derivatives: synthesis and biological activity

Lit. 21 zázn.

In: Il Farmaco. - Vol. 58, No. 11 (2003), s. 1105-1111

ADE02 Jampílek, Josef [UKOEXAF] (25%) - Doležal, Martin (15%) - Kuneš, Jiří (10%) - Buchta, Vladimír

(10%) - Silva, Luis (20%) - Kráľová, Katarína [UKOPRCUS] (20%): Quinaldine Derivatives: Preparation

and Biological Activity

Lit.: 35 zázn.

In: Medicinal Chemistry. - Vol. 1, No. 6 (2005), s. 591-599

Ohlasy (25):

[o1] 2007 Malecki, J.G. - Kruszynski, R. - Tabak, D. - Kusz, J.: Polyhedron, Vol. 26, No. 17, 2007, s.

5120-5130 - SCI

[o1] 2008 Prasad, A.K. - Kumar, P. - Dhawan, A. - Chillar, A.K. - Sharma, D. - Parmar, V.S.: Bioorganic

and Medicinal Chemistry Letters, Vol. 18, No. 6, 2008, s. 2156-2161 - SCI


19, 2008, s. 257-263 - SCI

[o1] 2009 Sahidhara, K.V. - Kumar, A. - Bhatia, G. - Khan, M.M. - Khanna, A.K. - Saxena, J.K.:

European Journal of Medicinal Chemistry, Vol. 44, No. 4, 2009, s. 1813-1818 - SCI

[o1] 2010 Ramli, Y. - Slimani, R. - Zouihri, H. - Lazar, S. - Essassi, E.M.: Acta Crystalographica Section

E-Structure Reports Online, Vol. 66, Part. 4, 2010, s. O992-U3649 - SCI

[o1] 2010 Musiol, R. - Serda, M. - Hensel-Bielówska, S. - Polanski, J.: Current Medicinal Chemistry, Vol.

17, No. 18, 2010, s. 1960-1973 - SCI

[o1] 2010 Ramli, Y. - Slimani, R. - Zouihri, H. - Lazar, S. - Essassi, E.M.: Acta Crystalographica Section

E-Structure Reports Online, Vol. 66, Part. 7, 2010, s. O1767-U268 - SCI

[o1] 2010 Tang, W.J. - Sun, Y.W. - Xu, L.J. - Wang, T.L. - Fan, Q.H. - Lam, K.H. - Chan, A.S.C.: Organic

and Biomolecular Chemistry, Vol. 8, No. 15, 2010, s. 3464-3471 - SCI

[o1] 2010 Ramli, Y. - Moussaif, A. - Zouihri, H. - Lazar, S. - Essassi, E.M.: Acta Crystallographica,

Section E- Structure Reports Online, Vol. E66, No. 8, 2010, s. o1922-U379 - SCI

[o1] 2010 Zhong, Q-D. - Xue, Y-Z. - Yan, H. - Song, X-Q. - Zhong, R-G.: Bioorganic & Medicinal

Chemistry Letters, Vol. 20, No. 18, 2010, s. 5532-5535 - SCI

[o1] 2011 Ramli, Y. - Moussaif, A. - Zouihri, H. - Bourichi, H. - Essassi, E.M.: Acta Crystallographica

Section E: Structure Reports Online, Vol. 67, Part. 6, 2011, s. O1374-NIL_362 - SCI

[o1] 2011 Loh, W.S. - Fun, H.K. - Kayarmar, R. - Viveka, S. - Nagaraja, G.K.: Acta Crystallographica

Section E: Structure Reports Online, Vol. 67, Part. 2, 2011, s. O405-NIL_990 - SCI

33

[o1] 2012 Štefane, B. - Požgan, F. - Sosič, I. - Gobec, S.: Tetrahedron Letters, Vol. 53, Iss. 15, 2012, s.

1964-1967 - SCOPUS

[o1] 2012 Ramli, Y. - Zouihri, H. - Azougagh, M. - Moussaif, A. - Essassi, E.M.: Acta Crystallographica

Section E: Structure Reports Online, Vol. 68, No. 2, 2012, s. o396 - SCI ; SCOPUS



[o3] 2010 Serda, M. - Musiol, R. - Polanski, J.: New thiosemicarbazones based on quinoline scaffold as

anticancer iron chelators. In: International Electronic Conference on Synthetic Organic Chemistry,

2010,http://www.sciforum.net/presentation/441



[o1] 2012 Armitage M. - Bret G. - Choudary B.M. - Kingswood M. - Loft M. - Moore S. - Smith S. -

Urquhart M.W.: Organic Process Research & Development, Vol. 16, No. 10, 2012, s. 1626-1634 - SCI ;

SCOPUS

[o3] 2011 Wang, L.X. - Sheng, J. - Wang, X.H.: Synthesis and crystal structure of 4- (4-bromophenyl)-9-

)4-chlorophenyl) -2,3,6,7 tetrahydro-6, 6-dimethyl-4H-cyclopenta[b]quinoline-1,8 (5H, 9H)-dione. In:

Journal of Xuzhou Normal University(Natural Science Edition), Vol. 29, No. 4, 2011, s. 58-62

[o3] 2011 Chen, G.M. - Wu, Z.B. - Hu, D.Y. - Yang, S. - Bao, W.Y.: Research Progress on Synthesis and

Bioactivity of Quinoline and Its Derivative Fine Chemical Intermediates. In: Fine Chemical Intermediates,

Vol. 41, No. 2, 2011, s. 6-10

[o1] 2014 Moustafa, A.H. - Said, S.A. - Haikal, A.E.F.Z. - Abu-El-Halawa, R. - Abd-El Kader, R.T.:

Nucleosides, Nucleotides and Nucleic Acids, Vol. 33, No. 3, 2014, s. 111-128 - SCOPUS

[o1] 2014 Bassyouni, F.A. - Abu-Baker, S.M. - Mahmoud, K. - Moharam, M. - El-Nakkady, S.S. - Rehim,

M.A.: RSC Advances, Vol. 4, No. 46, 2014, s. 24131-24141 - SCOPUS

[o1] 2014 Vairavelu, L. - Rajendra Prasad, K.J.: Journal of Chemical Sciences, Vol. 126, No. 6, 2014, s.

1893-1902 - SCOPUS



[o1] 2015 Liu, Y.A. - Zhang, J.A. - Zhang, L.J. - Zou, X.Z. - Li, N. - Li, Y.: Inorganic Chemistry

Communications, Vol. 57, Art. No. 5970, 2015, s. 40-43 - SCOPUS

ADE03 Jampílek, Josef [UKOEXAF] (60%) - Doležal, Martin (20%) - Buchta, Vladimír (20%): Antimicrobial

evaluation of some arylsulfanylpyrazinecarboxylic acid derivatives

Lit. 25 zázn.


ADE04 Vinšová, Jarmila (30%) - Imramovský, Aleš (20%) - Jampílek, Josef [UKOEXAF] (30%) - Monreal-

Ferriz, Juana (10%) - Doležal, Martin (10%): Recent advances on isoniazide derivatives

Lit. 85 zázn.

In: Anti-Infective Agents in Medicinal Chemistry. - Vol. 7, No. 1 (2008), s. 12-31

ADE05 Musiol, Robert (25%) - Jampílek, Josef [UKOEXAF] (25%) - Podeszwa, Barbara (10%) - Finster, Jacek

(%10) - Tabak, Dominik (10%) - Dohnal, Jiří (10%) - Polanski, Jaroslaw (10%): RP-HPLC determination

of lipophilicity in series of quinoline derivatives

Lit. 52 zázn.

In: Central European Journal of Chemistry. - Vol. 7, No. 3 (2009), s. 586-597

ADE06 Kráľová, Katarína [UKOPRCUS] (60%) - Ostrovský, Ivan [UKOPRCUS] (10%) - Jampílek, Josef

[UKOEXAF] (30%): Metabolomics - useful tool for study of plant responses to abiotic stresses =

Metabolomika - uzyteczne narzedzie do oceny wplywu czynników abiotycznych na rosliny

Lit.: 150 zázn.

In: Ecological Chemistry and Engineering S. - Vol. 19, No. 2 (2012), s. 133-161

Ohlasy (6):

[o1] 2013 D'Alessandro, A. - Taamalli, M. - Gevi, F. - Timperio, A.M. - Zolla, L. - Ghnaya, T.: Journal of

Proteome Research, Vol. 12, No. 11, 2013, s. 4979-4997 - SCI ; SCOPUS

[o3] 2013 Zhong G. - Wang, Y.-Z. - Zhang, J. - Jin, H. - Zhang, J.-Y. - Xiao, Y.: Advances in

metabolomics research on genus Panax plants. In: Lishizhen Medicine and Materia Medica Research, Vol.

24, No. 9, 2013, s. 2234-2237

[o1] 2014 Beck, J.J. - Smith, L. - Baig, N.: Phytochemical Analysis, Vol. 25, No. 4, 2014, s. 331-341 - SCI

; SCOPUS

[o1] 2014 Boestfleisch, C. - Wagenseil, N.B. - Buhmann, A.K. - Seal, C.E. - Wade, E.M. - Muscolo, A. -

Papenbrock, J.: AoB Plants, Vol. 13, No. 6, 2014, s. plu046 - SCI

34

[o1] 2015 Mishra, A. - Patel, M.K. - Jha, B.: Journal of Functional Foods, Vol. 13, 2015, s. 21-31 -

SCOPUS

[o1] 2014 Turi, C.E. - Axwik, K.E. - Smith, A. - Jones, A.M.P. - Saxena, P.K. - Murch, S.J.: Plant

Signaling and Behavior, Vol. 9, No. 4, 2014, Art. No. e28645 - SCI ; SCOPUS

ADE07 Černíková, Aneta (25%) - Opatřilová, Radka (25%) - Bobáľ, Pavel (25%) - Jampílek, Josef

[UKOEXAF] (25%): Antimicrobial evaluation of some arylsulfanylpyrazinecarboxylic acid derivatives

Lit. 38 zázn.

In: ADMET & DMPK. - Vol. 2, No. 4 (2014), s. 248-253

ADE08 Malík, Ivan (30%) - Govender, Rodney (10%) - Sedlárová, Eva (10%) - Csöllei, Jozef (10%) - Coffey,

Aidan (10%) - O Mahony, Jim (10%) - Stanzel, Lukáš (10%) - Jampílek, Josef [UKOEXAF] (10%): The

in vitro investigation ofortho-/meta-/para-alkoxyphenylcarbamic acid esters containing substituted N-

phenylpiperazin-1-yl fragment against Mycobacterium tuberculosis H37Ra

Lit. 20 zázn.

In: Journal of Microbiology, Biotechnology and Food Sciences. - Vol. 3, No. 5 (2014), s. 395-397


Aidan (10%) - O Mahony, Jim (10%) - Jampílek, Josef [UKOEXAF] (10%): The in vitro evaluation of

ortho-/meta-/para-alkoxyphenylcarbamic acid esterscontaining 4-(4-fluorophenyl)piperazin-1-yl moiety

against Mycobacterium tuberculosis H37Ra

Lit. 21 zázn.



Aidan (10%) - O Mahony, Jim (10%) - Jampílek, Josef [UKOEXAF] (10%): The in vitro evaluation of

ortho-/meta-/para-alkoxyphenylcarbamic acid estersbearing 4-(2-fluoro-/2-methylphenyl)piperazin-1-yl

moiety against Mycobacterium tuberculosis H37Ra

Lit. 27 zázn.


ADE11 Opatřilová, Radka (50%) - Jampílek, Josef [UKOEXAF] (50%): Rapid Screening of Mupirocin Skin

Permeation Modification by Micronized and Nanonized Alaptide

Lit. 43 zázn.


ADE12 Vaculiková, Eliška (40%) - Plachá, Daniela (20%) - Čech-Barabaszová, Karla (20%) - Jampílek, Josef

[UKOEXAF] (20%): Cimetidine Nanoparticles Study

Lit. 10 zázn.

In: Advanced Science, Engineering and Medicine. - Vol. 6, No. 4 (2014), s. 477-481

ADE13 Černíková, Aneta (60%) - Jampílek, Josef [UKOEXAF] (50%): Permeation of Indomethacin through

Skin Using Nanonized Alaptide

Lit. 43 zázn.


ADF Vědecké práce v domácích nekarentovaných časopisech

ADF01 Kráľová, Katarína (60%) - Jampílek, Josef [UKOEXAF] (30%) - Ostrovský, Ivan (10%): Metabolomika

vo výskume fytoterapeutík = Metabolomics in research of phytotherapeutics

Lit. 43 zázn.

In: Česká a slovenská farmacie. - Roč. 61, č. 1-2 (2012), s. 21-25

ADF02 Černíková, Aneta (34%) - Opatřilová, Radka (33%) - Jampílek, Josef [UKOEXAF] (33%): Rapid

informative screening of nano-alaptide as potential transdermal permeation enhancer of acetylsalicylic acid

and paracetamol

Lit. 29 zázn.

In: Military Medical Science Letters. - Vol. 83, No. 1 (2014), s. 34-39

ADM Vědecké práce v zahraničních časopisech registrovaných v databázích Web of Science nebo

SCOPUS

ADM01 Brezovská, Monika (45%) - Jampílek, Josef [UKOEXAF] (10%) - Opatřilová, Radka (45%): A review

of HPLC methods used for determining the presence of meloxicam

Lit. 44 zázn.

In: Current Pharmaceutical Analysis. - Vol. 9, No. 1 (2013), s. 69-76


35


IF (JCR) [2013-0,771]

SJR (SCOPUS) [2013-0,275]

SNIP (SCOPUS) [2013-0,686]

Ohlasy (2):

[o1] 2015 Yang, W.J. - Li, J. - Gao, J.H. - Huang, Z.Y. - Tang, C.W.: Current Pharmaceutical Analysis,

Vol. 11, No. 3, 2015, s. 172 - SCI

[o1] 2015 Sim, A. - Cho, Y. - Kim, D. - Witt, M. - Birdwell, J.E. - Kim, B.J. - Kim, S.: Fuel, Vol. 140,

2015, s. 723 - SCI

ADM02 Jampílek, Josef [UKOEXAF] (100%) : Transdermal application of drugs and techniques affecting skin

barrier

Lit. 45 zázn.

In: Journal of Bioequivalence and Bioavailability. - Vol. 5, No. 6 (2013), s. 233-235

Registrované v: scopus


SJR (SCOPUS) [2013-0,163]

SNIP (SCOPUS) [2013-0,358]

Ohlasy (1):

[o1] 2015 Han, T. - Das, D.B.: European Journal of Pharmaceutics and Biopharmaceutics, Vol. 89, 2015,

s. 328 - SCOPUS

ADM03 Opatřilová, Radka (20%) - Černíková, Aneta (20%) - Coufalová, Lenka (20%) - Dohnal, Jiří (20%) -

Jampílek, Josef [UKOEXAF] (20%): In Vitro Permeation of Micronized and Nanonized Alaptide from

Semisolid Formulations

Lit. 45 zázn.

In: The Scientific World Journal [elektronický zdroj]. - Vol. 2013, (2013), Art. No. 787283, s. [8 s.]

[online]



IF (JCR) [2013-1,219]

SJR (SCOPUS) [2013-0,407]

SNIP (SCOPUS) [2013-0,578]

ADM04 Tengler, Jan (20%) - Kapustíková, Iva (10%) - Peško, Matúš [UKOPREEF] (10%) - Govender, Rodney

(10%) - Keltošová, Stanislava (10%) - Mokrý, Petr (5%) - Kollár, Peter (5%) - O Mahony, Jim (5%) -

Coffey, Aidan (5%) - Kráľová, Katarína [UKOPRCUS](10%) - Jampílek, Josef [UKOEXAF] (10%):

Synthesis and Biological Evaluation of 2-Hydroxy-3-[(2-aryloxyethyl)amino]propyl4-

[(Alkoxycarbonyl)amino]benzoates


In: The Scientific World Journal [elektronický zdroj]. - Vol. 2013 (2013), Art. No. 274570 [13 s.] [online]

Registrované v: scopus, wos


IF (JCR) [2013-1,219]

SJR (SCOPUS) [2013-0,407]

SNIP (SCOPUS) [2013-0,578]

Ohlasy (2):

[o1] 2014 Bado, O. - Frydrych, M. - Kolmanová, E. - Dlouhá, M.: Ceska a Slovenska Farmacie, Vol. 63,

No. 4, 2014, s. 167-173 - SCOPUS

[o1] 2015 Romano, B. - Plano, D. - Encío, I. - Palop, J.A. - Sanmartín, C.: Bioorganic and Medicinal

Chemistry, Vol. 23, No. 8, 2015, s. 1716-1727 - SCOPUS

ADM05 Bojňanská, Erika (25%) - Kalina, Michal (10%) - Pařízek, Ladislav (5%) - Bartoníčková, Eva (5%) -

Opravil, Tomáš (15%) - Veselý, Michal (10%) - Pekař, Miloslav (5%) - Jampílek, Josef [UKOEXAF]

(25%): Determination of critical parameters of drug substance influencing dissolution: a case study

Lit. 20 zázn.

In: BioMed Research International. - Vol. 2014 (2014), Art. No. 929248, s. [9 s.]



IF (JCR) [2014-1,579]

SJR (SCOPUS) [2014-0,613]

SNIP (SCOPUS) [2014-0,576]

36

ADM06 Imramovský, Aleš (30%) - Kozic, Jan (10%) - Peško, Matúš [UKOPREEF] (15%) - Stoláriková, Jirina

(10%) - Vinšová, Jarmila (10%) - Kráľová, Katarína [UKOPRCUS] (15%) - Jampílek, Josef [UKOEXAF]

(10%): Synthesis and antimycobacterial andphotosynthesis-inhibiting evaluation of 2-[(E)-2-Substituted-

ethenyl]-1,3-benzoxazoles


In: The Scientific World Journal [elektronický zdroj]. - Vol. 2014 (2014), Art. No. 705973 [11 s.] [online]



IF (JCR) [2014-1,219]

SJR (SCOPUS) [2014-0,350]

SNIP (SCOPUS) [2014-0,531]

ADM07 Vaverková, Veronika (20%) - Vrána, Oldřich (10%) - Adam, Vojtěch (10%) - Pekárek, Tomáš (20%) -

Jampílek, Josef [UKOEXAF] (20%) - Babula, Petr (20%): The study of naphthoquinones and their

complexes with DNA by using Raman spectroscopy and surface enhanced Raman spectroscopy: new

insight into interactions of DNA with plant secondary metabolites

Lit. 95 zázn.




IF (JCR) [2014-1,579]

SJR (SCOPUS) [2014-0,613]

SNIP (SCOPUS) [2014-0,576]

Ohlasy (1):

[o1] 2016 Gasior-Glogowska, M. - Malek, K. - Zajac, G. - Baranska, M.: Analyst, Vol. 141, No. 1, 2016, s.

296

ADM08 Cieslik, Wioleta (20%) - Spaczynska, Ewelina (10%) - Jampílek, Josef [UKOEXAF] (15%) - Malarz,

Katarzyna (10%) - Tabak, Dominik (5%) - Nevin, Eoghan (10%) - O Mahony, Jim (5%) - Coffey, Aidan

(5%) - Mrozek-Wilczkiewicz, Anna (5%) - Musiol, Robert(15%): Investigation of the Antimycobacterial

Activity of 8-Hydroxyquinolines

Lit. 47 zázn.


Registrované v: scopus


IF (JCR) [2014-1,363]

SJR (SCOPUS) [2014-0,381]

SNIP (SCOPUS) [2014-0,618]

ADM09 Jampílek, Josef [UKOEXAF] (18%) - Záruba, Kamil (17%) - Oravec, Michal (18%) - Kuneš, Martin

(17%) - Babula, Petr (5%) - Ulbrich, Pavel (5%) - Brezániová, Ingrid (5%) - Opatřilová, Radka (5%) -

Triska, Jan (5%) - Suchý, Pavel (5%): Preparation of silica nanoparticles loaded with nootropics and their

in vivo permeation through blood-brain barrier

Lit. 34 zázn.




IF (JCR) [2014-1,579]

SJR ( [2014-0,613]

SNIP (SCOPUS) [2014-0,576]

ADM10 Kráľová, Katarína [UKOPRCUS] (60%) - Perina, V. (5%) - Waisser, Karel (5%) - Jampílek, Josef

[UKOEXAF] (30%): Structure-Activity Relationships of N-benzylsalicylamides for Inhibition of

Photosynthetic Electron Transport





IF (JCR) [2014-1,363]

SJR (SCOPUS) [2014-0,381]

SNIP (SCOPUS) [2014-0,618]

37

ADM11 Zdražilová, Iveta (25%) - Pospíšilová, Šárka (20%) - Pauk, Karel (10%) - Imramovský, Aleš (10%) -

Vinšová, Jarmila (5%) - Čížek, Alois (10%) - Jampílek, Josef [UKOEXAF] (20%): In vitro bactericidal

activity of 4- and5-chloro-2-hydroxy-N-[1-oxo-1-(phenylamino)alkan-2-yl]benzamides against MRSA

Lit. 40 zázn.

In: BioMed Research International. - Vol. 2015 (2015), s. [8 s.], Art.No. 349534



IF (JCR) [2014-1,579]

SJR ( [2014-0,613]

SNIP (SCOPUS) [2014-0,576]

AED Vědecké práce v domácích recenzovaných vědeckých sbornících

AED01 Jampílek, Josef [UKOEXAF] (50%) - Doležal, Martin (25%) - Deigner, Hans Peter (25%): Optimization

of Sphingosine Synthesis by Tkaczuk-Thornton Method

Lit. 8 zázn.

In: Folia Pharmaceutica Universitatis Carolinae, Roč. 27-28. - Praha : Karolinum, 2002. - S. 69-75

AED02 Jampílek, Josef [UKOEXAF] (50%) - Doležal, Martin (25%) - Kuneš, Jiří (25%): Quinlukast

Azaanalogues Preparation

Lit. 9 zázn.

In: Folia Pharmaceutica Universitatis Carolinae, Roč. 31-32. - Praha : Karolinum, 2004. - S. 27-32

AED03 Doležal, Martin (20%) - Opletalová, Veronika (20%) - Bagi-Krinková, Jana (10%) - Jampílek, Josef

[UKOEXAF] (10%) - Kučerová-Chlupáčová, Marta (10%) - Palek, Lukáš (10%) - Kešetovičová, Diana

(10%) - Zitko, Jan (10%): Development of New Antituberculous Active Pyrazines Evaluated in Co-

operation with TAACF Program within a Perion of 15 years

Lit. 20 zázn.

In: Folia Pharmaceutica Universitatis Carolinae, Roč. 39. - Praha : Karolinum, 2010. - S. 31-40

BCI Skripta a učební texty

BCI01 Jampílek, Josef [UKOEXAF] (80%) - Opatřilová, Radka (10%) - Liška, Ivo (10%): Návody do cvičení z

analytické chemie : Vybrané instrumentální metody. - 1. vyd. - Brno : Veterinární a farmaceutická

univerzita Brno, 2007. - 74 s.

Lit. 13 zázn.

ISBN 978-80-7305-007-8

BCI02 Dohnal, Jiří (10%) - Grafnetterová, Taťjana (10%) - Grünwaldová, Veronika (10%) - Havlíček, Jaroslav

(10%) - Jampílek, Josef [UKOEXAF] (10%) - Opatřilová, Radka (10%) - Pekárek, Tomáš (10%) - Plaček,

Lukáš (10%) - Tisovská, Lucie (10%) - Zerzaňová,Anna (10%): Moderní přístupy k farmaceutické analýze

: 1. Analýza chirálních léčiv. - 1. vyd. - Brno : Veterinární a farmaceutická univerzita Brno, 2008. - 122 s.

Lit. 10 zázn.

ISBN 978-80-7305-056-6

BCI03 Liška, Ivo (80%) - Jampílek, Josef [UKOEXAF] (10%) - Opatřilová, Radka (10%): Návody do cvičení z

analytické chemie : Kvalitativní anorganická analýza. - 1. vyd. - Brno : Veterinární a farmaceutická

univerzita Brno, 2008. - 67 s.

Lit. 43 zázn.

ISBN 978-80-7305-044-3

BCI04 Opatřilová, Radka (80%) - Jampílek, Josef [UKOEXAF] (10%) - Liška, Ivo (10%): Návody do cvičení z

analytické chemie : Kvantitativní analýza. - 1. vyd. - Brno : Veterinární a farmaceutická univerzita Brno,

2008. - 82 s.

Lit. 21 zázn.

ISBN 978-80-7305-027-6



Lukáš (10%) - Tisovská, Lucie (10%) - Zerzaňová,Anna (10%): Moderní přístupy k farmaceutické analýze

: 2. Strukturní analýza léčiv. - 1. vyd. - Brno : Veterinární a farmaceutická univerzita Brno, 2009. - 105 s.

Lit. 12 zázn.

ISBN 978-80-7305-058-0

38



Lukáš (10%) - Tisovská, Lucie (10%) - Zerzaňová,Anna (10%) - Brusová, Hana (10%): Moderní přístupy

k farmaceutické analýze : 3. Farmaceutická analýza v pevné fázi. - 1. vyd. - Brno : Veterinární a

farmaceutická univerzita Brno, 2009. - 159 s.

Lit. 33 zázn.

ISBN 978-80-7305-075-7

Další ukazatele publikační činnosti ve vědeckých časopisech

Publikace s IF >1,000 81

a zároveň z nich jako první nebo korespondující autor 49

Publikace v karentovaných časopisech (ADC, ADD) 84

Součet IF všech vědeckých prací 214

h-index 17 (Web of Science – Core Collection; ke dni 5.2.2016)

19 (Web of Science – All Databases; ke dni 5.2.2016)

Práce, které nebyly zařazené do seznamu kontroly AK UK – na základě kritérii VR FaF

UK ke splnění podmínek získání vědecko-pedagogického titulu „profesor“ se

nevyžadují:

AGJ Patenty a přihlášky patentů

1. MUSIOŁ, Robert and JAMPÍLEK, Josef and KRÁĽOVÁ, Katarína and NIEDBALA, Halina and PAŁKA,

Anna and PODESZWA, Barbara and POLAŃSKI, Jarosław (Uniwersytet Śląski v Katowicach). Pochodne

chinoliny wykazujące aktywność jako herbicydy i algicydy, ich prekursory, sposoby wytwarzania oraz ich

stosowanie. P 375678 A1, 13.06.2005.

2. MUSIOŁ, Robert and JAMPÍLEK, Josef and BUCHTA, Vladimír and NIEDBALA, Halina and PAŁKA,

Anna and PODESZWA, Barbara and POLAŃSKI, Jarosław (Uniwersytet Śląski v Katowicach). Pochodne

chinoliny wykazujące aktywność jako fungicydy oraz ich stosowanie. P 375805, 20.06.2005.

3. SVOBODA, Martin a JAMPÍLEK, Josef a ŠEBEK, Pavel (Zentiva). Farmaceutická kompozice clopidogrel

hydrogenbromidu. CZ 298349 B6, 25.07.2007.

4. SVOBODA, Martin a JAMPÍLEK, Josef a KAČÍRKOVÁ, Martina a TOMÁŠEK, Václav a LEHOCKÝ,

Mikuláš (Zentiva). Farmaceutická kompozice s obsahem tolterodinu. CZ 298448 B6, 24.08.2007.

5. MUSIOŁ, Robert and JAMPÍLEK, Josef and BUCHTA, Vladimír and KRÁĽOVÁ, Katarína

and FINSTER, Jacek and PODESZWA, Barbara and TABAK, Dominik and POLAŃSKI, Jarosław

(Uniwersytet Śląski v Katowicach). Analogi chinazoliny jako fungicydy i herbicydy oraz ich zastosowanie.

P 379252, 21.03.2006.

6. SVOBODA, Martin and JAMPÍLEK, Josef and KAČÍRKOVÁ, Martina and TOMÁŠEK, Václav and

LEHOCKÝ, Mikuláš and HEJTMÁNKOVÁ, Ludmila and VOSÁTKA, Václav (Zentiva). Crystalline

Tolterodine Tartarate and a Pharmaceutical Composition Containing the Same. WO/2008/017278 A3,

28.08.2008.

7. KRÁL, Vladimír a JAMPÍLEK, Josef a HAVLÍČEK, Jaroslav a BRUSOVÁ, Hana a PEKÁREK, Tomáš

(Zentiva). Lékové formy inhibitorů tyrosinových kináz. PV 2009-8, 13.01.2009.

8. KRÁL, Vladimír a BRUSOVÁ, Hana a HAVLÍČEK, Jaroslav a Tkadlecová, Marcela a JAMPÍLEK, Josef

a PEKÁREK, Tomáš (Zentiva). Příprava, stabilizace a využití polymorfů imatinib mesylatu pro vývoj

lékových forem. PV 2009-570, 26.08.2009.

9. KRÁL, Vladimír and JAMPÍLEK, Josef and HAVLÍČEK, Jaroslav and BRUSOVÁ, Hana and PEKÁREK,

Tomáš (Zentiva). Dosage Forms of Tyrosine Kinase Inhibitors. WO/2010/081443 A2, 22.07.2010.

10. KRÁL, Vladimír and BRUSOVÁ, Hana and JAMPÍLEK, Josef and HAVLÍČEK, Jaroslav and PEKÁREK,

Tomáš and TKADLECOVÁ, Marcela (Zentiva). Imatinib Mesylate Polymorphs Generated by

Crystallization in Aqueous Inorganic Salt Solutions. WO/2011/023146 A1, 03.03.2011.

11. MUDRA, Petr a POKORNÝ, Vít a PEŠEK, Václav a PONCAR, Pavel a BÁRTA, Jaroslav a ŘEZÁČOVÁ,

Anna a JAMPÍLEK, Josef a DOHNAL, Jiří a KRÁL, Vladimír (Zentiva & Ústav organické chemie a

biochemie AV ČR). Simulátor trávicího traktu. CZ 302422 B6, 30.03.2011.

39

12. KRÁL, Vladimír a OKTÁBEC, Zbyněk a JAMPÍLEK, Josef a BRUSOVÁ, Hana a PEKÁREK, Tomáš a

ŘEZÁČOVÁ, Anna a DOHNAL, Jiří (Zentiva). Příprava, stabilizace a využití nových polymorfů imatinib

mesylatu pro vývoj lékových forem. PV 2011-228, 19.04.2011.

13. JAMPÍLEK, Josef a OPATŘILOVÁ, Radka a ŘEZÁČOVÁ, Anna a OKTÁBEC, Zbyněk a PÁVEK, Petr a

KRÁL, Vladimír a DOHNAL, Jiří (VFU Brno). Způsob ovlivnění rozpustnosti alaptidu, ovlivnění jeho

prostupu přes membrány a jeho farmaceutické kompozice pro humánní a veterinární aplikace. PV 2011-

232, 20.04.2011.

14. KRÁL, Vladimír and OKTÁBEC, Zbyněk and JAMPÍLEK, Josef and PEKÁREK, Tomáš and PROKSA,

Bohumil and DOHNAL, Jiří and MALOVÍKOVÁ, Anna and EBRINGEROVÁ, Anna and ŘEZÁČOVÁ,

Anna (Zentiva). Pectin Complexes of Steroids and Pharmaceutical Compositions Based Thereon.

WO/2011/063774 A2, 03.06.2011.

15. KRÁL, Vladimír and OKTÁBEC, Zbyněk and JAMPÍLEK, Josef and PEKÁREK, Tomáš and PROKSA,

Bohumil and DOHNAL, Jiří and MALOVÍKOVÁ, Anna and EBRINGEROVÁ, Anna and ŘEZÁČOVÁ,

Anna (Zentiva). Pectin Complexes of Sartans and Pharmaceutical Compositions Based Thereon.

WO/2011/063775 A2, 03.06.2011.

16. KRÁL, Vladimír a RAK, Jakub a ZAGORA, Jiří a GRÜNWALDOVÁ, Veronika a ŘEZÁČOVÁ, Anna a

JAMPÍLEK, Josef a KŮTKOVÁ, Božena (Zentiva). Příprava, stabilizace a využití nanočástic API

pro vývoj moderních lékových forem. PV 2011-353, 13.06.2011.

17. MUDRA, Petr and POKORNÝ, Vít and PEŠEK, Václav and PONCAR, Pavel and BÁRTA, Jaroslav and

ŘEZÁČOVÁ, Anna and JAMPÍLEK, Josef and DOHNAL, Jiří and KRÁL, Vladimír (Zentiva & Institute

of Organic Chemistry and Biochemistry of Academy of Sciences of the Czech Republic). Digestive Tract

Simulator. WO/2011/069472 A1, 16.06. 2011.

18. KRÁL, Vladimír a KRÁLOVÁ, Jarmila a FLIEGER, Miroslav a JAMPÍLEK, Josef a ŘEZÁČOVÁ, Anna

a DOHNAL, Jiří a OKTÁBEC, Zbyněk a ZÁRUBA, Kamil a GRÜNWALDOVÁ, Veronika

a POUČKOVÁ, Pavla a MARTÁSEK, Pavel (Zentiva). Způsob podávání léčiv ve formě nanočástic

umožňující průchod hematoencefalickou bariéru. PV 2011-366, 21.06.2011.

19. KRÁL, Vladimír a OKTÁBEC, Zbyněk a JAMPÍLEK, Josef a PEKÁREK, Tomáš a PROKSA, Bohumil a

DOHNAL, Jiří a MALOVÍKOVÁ, Anna a EBRINGEROVÁ, Anna a ŘEZÁČOVÁ, Anna (Zentiva).

Způsob zvýšení rozpustnosti farmaceuticky aktivních látek a cílený (kontrolovaný) transport do střeva. CZ

302789 B6, 29.09.2011.

20. JAMPÍLEK, Josef a OPATŘILOVÁ, Radka a DVOŘÁKOVÁ, Lenka a DOHNAL, Jiří (VFU Brno).

Využití alaptidu jako modifikátoru transdermální penetrace ve farmaceutických kompozicích pro humánní

a veterinární aplikace obsahující glukokortikoidy. PV 2012-72, 01.02.2012.

21. JAMPÍLEK, Josef a OPATŘILOVÁ, Radka a DVOŘÁKOVÁ, Lenka a ČERNÍKOVÁ, Aneta

a DOHNAL, Jiří (VFU Brno). Využití alaptidu jako modifikátoru transdermální penetrace

ve farmaceutických kompozicích pro humánní a veterinární aplikace obsahující antimikrobiální

chemoterapeutika. PV 2012-511, 26.07.2012.

22. JAMPÍLEK, Josef and OPATŘILOVÁ, Radka and COUFALOVÁ, Lenka and ČERNÍKOVÁ, Aneta and

DOHNAL, Jiří (University of Veterinary and Pharmaceutical Sciences Brno). Utilization of Alaptide as

Transdermal Penetration Modifier in Pharmaceutical Compositions for Human and Veterinary Applications

Containing Anti-Inflammatory Drugs and/or Antimicrobial Chemotherapeutics. WO/2013/020527 A1,

14.02.2013.

23. JAMPÍLEK, Josef a ČERNÍKOVÁ, Aneta a OPATŘILOVÁ, Radka a DOHNAL, Jiří (VFU Brno). Využití

alaptidu jako modifikátoru transdermální penetrace ve farmaceutických kompozicích pro humánní a

veterinární aplikace obsahující léčiva centrálního a/nebo vegetativního nervového systému a/nebo pohlavní

hormony, resp. modulátory genitálního systému. PV 2013-1000, 13.12.2013.

24. JAMPÍLEK, Josef a ČERNÍKOVÁ, Aneta a OPATŘILOVÁ, Radka a DOHNAL, Jiří (VFU Brno). Využití

(R)-alaptidu jako modifikátoru transdermální penetrace léčiv ve farmaceutických kompozicích pro humánní

a veterinární aplikace. PV 2013-1001, 13.12.2013.

25. JAMPÍLEK, Josef and OPATŘILOVÁ, Radka and ŘEZÁČOVÁ, Anna and OKTÁBEC, Zbyněk

and DOHNAL, Jiří (University of Veterinary and Pharmaceutical Sciences Brno). Alaptide: Methods of

Effecting its Solubility, Membrane Permeation and Pharmaceutical Compositions for Human and/or

Veterinary Applications. WO/2014/019556 A1, 06.02.2014.

26. JAMPÍLEK, Josef a ČERNÍKOVÁ, Aneta a OPATŘILOVÁ, Radka a BOBÁĽ, Pavel (VFU Brno). Využití

substituovaných analogů alaptidu jako modifikátorů transdermální penetrace ve farmaceutických

kompozicích pro humánní a veterinární aplikace. PV 2014-416, 17.06.2014.

27. JAMPÍLEK, Josef a OPATŘILOVÁ, Radka a DVOŘÁKOVÁ, Lenka a BRYCHTOVÁ, Kateřina

a DOHNAL, Jiří (VFU Brno). Využití alaptidu jako modifikátoru transdermální penetrace

40

ve farmaceutických kompozicích pro humánní a veterinární aplikace obsahující nesteroidní antiflogistika

a/nebo antipyretika-analgetika. CZ 304915 B6, 10.12.2014.

AEG Abstrakty vědeckých prací v zahraničních karentovaných časopisech

1. JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří and RAICH, Ivan. Preparation of 2-(4-{[4-

(quinolin-2-ylmethoxy)phenyl]sulfanyl}phenyl)propanoic acid (VUFB 20615) and 2-methyl-2-(4-{[4-

(quinolin-2-ylmethoxy)phenyl]sulfanyl}phenyl)propanoic acid (VUFB 20623) as potential antileukotrienic

agents. Book of Abstracts: The XVIIIth

International Symposium on Medicinal Chemistry (ISMC 2004),

Copenhagen, Denmark & Malmö, Sweden, August 15-19, 2004, Drug Future 2004, vol. 29, no. Suppl. A,

399. [ISSN 0377-8282, IF2004 = 0.548]

2. JAMPÍLEK, Josef and DOLEŽAL, Martin and PALEK, Lukáš and VINŠOVÁ, Jarmila. Structure-

lipophilicity Relationships in Series of Phenolic Moiety Ring-substituted Pyrazinecarboxanilides. Book of

Abstracts: The XIXth

International Symposium on Medicinal Chemistry (ISMC 2006), Istanbul, Turkey,

August 29-September 2, 2006, Drug Future 2006, vol. 31, no. Suppl. A, 51. [ISSN 0377-8282, IF2006 =

0.777]

3. DOLEŽAL, Martin and PALEK, Lukáš and VINŠOVÁ, Jarmila and BUCHTA, Vladimír and JAMPÍLEK,

Josef and KRÁĽOVÁ, Katarína. Preparation, Antimycobacterial, Antifungal and Photosynthesis-inhibiting

Evaluation of Some Anilides of Substituted Pyrazinecarboxylic Acid. Book of Abstracts: The XIXth

International Symposium on Medicinal Chemistry (ISMC 2006), Istanbul, Turkey, August 29-September 2,

2006, Drug Future 2006, vol. 31, no. Suppl. A, 53. [ISSN 0377-8282, IF2006 = 0.777]

4. IMRAMOVSKÝ, Aleš and VINŠOVÁ, Jarmila and MONREAL-FÉRRIZ, Juana and DOLEŽAL, Martin

and JAMPÍLEK, Josef. Synthesis, Antituberculotic Activity and Stability of New Hydrazonoformamide

Derivatives of Isoniazide. Book of Abstracts: The XIXth

International Symposium on Medicinal Chemistry

(ISMC 2006), Istanbul, Turkey, August 29-September 2, 2006, Drug Future 2006, vol. 31, no. Suppl. A,

60. [ISSN 0377-8282, IF2006 = 0.777]

5. JAMPÍLEK, Josef and DOLEŽAL, Martin and HOŠŤÁLKOVÁ, Anna and VINŠOVÁ, Jarmila. Structure-

lipophilicity Relationships in Series of New Substituted N-phenylpyrazine-2-carboxamides as Biologically

Active Compounds. Book of Abstracts: The XXth

International Symposium on Medicinal Chemistry (ISMC

2008), Vienna, Austria, August 31-September 4, 2008, Drug Future 2008, vol. 33, no. Suppl. A, 60. [ISSN

0377-8282, IF2008 = 0.468]

6. SKÓRSKA-STANIA, Agnieszka and ŚLIWA, Magdalena and OLEKSYN, Barbara and MUSÍLEK, Kamil

and KUČA, Kamil and JAMPÍLEK, Josef and MUSIOŁ, Robert and DOHNAL, Jiří. Is It Possible to Guess

Potential Drug Activity from Its Crystal Structure? Book of Abstracts: The 25th

European Crystallographic

Meeting (ECM-25), Istanbul, Turkey, August 16-21, 2009, Acta Cryst. A 2009, vol. A65, no. S., s148

(FA1-MS07-P04). [ISSN 2053-2733, IF2009 = 49.93]

7. DOLEŽAL, Martin and JAMPÍLEK, Josef and ZITKO, Jan and OSIČKA, Zdeněk and SERVUSOVÁ,

Barbora. Structure-property Relationships in Series of Chlorine-substituted Pyrazinecarboxanilides as

Biologically Active Compounds. Book of Abstracts: The XXIst International Symposium on Medicinal

Chemistry (ISMC 2010), Brussels, Belgium, September 5-9, 2010, Drug Future 2010, vol. 35, no. Suppl. A,

76 (PO-60). [ISSN 0377-8282, IF2010 = 0.324]

8. JAMPÍLEK, Josef and BRYCHTOVÁ, Kateřina and OPATŘILOVÁ, Radka and RAICH, Ivan.

Preparation and Physico-chemical Properties of Alkyl-6-(2,5-dioxopyrrolidin-1-yl)-2-(2-oxopiperidin-1-

yl)hexanoates. Book of Abstracts: The XXIst International Symposium on Medicinal Chemistry (ISMC

2010), Brussels, Belgium, September 5-9, 2010, Drug Future 2010, vol. 35, no. Suppl. A, 77 (PO-61).

[ISSN 0377-8282, IF2010 = 0.324]

9. KOS, Jiří and GONĚC, Tomáš and BOBÁL, Pavel and JAMPÍLEK, Josef. Synthesis of

Hydroxynaphthalene-2-carboxanilides as Biologically Active Compounds. Book of Abstracts: The XXIInd

International Symposium on Medicinal Chemistry (ISMC 2012), Berlin, Germany, September 2-6, 2012,

ChemMedChem 2012, vol. 7, no. Suppl. A, 194 (P256). [ISSN 1860-7179, IF2012 = 2.835]

10. ZADRAŽILOVÁ, Iveta and POSPÍŠILOVÁ, Šárka and PAUK, Karel and IMRAMOVSKÝ, Aleš and

VINŠOVÁ, Jarmila and ČÍŽEK, Alois and JAMPÍLEK, Josef. Bactericidal Activity of (S)-5-Chloro-2-

hydroxy-N-{3-methyl-1-oxo-1-[4-(trifluoromethyl)phenylamino]butan-2-yl}benzamide against MRSA in

Dependence on Time and Concentration. Book of Abstracts: The XXIIIrd

International Symposium on

Medicinal Chemistry (ISMC 2014), Lisbon, Portugal, September 7-11, 2014, ChemMedChem 2014, vol. 9,

no. Suppl. A, 103 (C017). [ISSN 1860-7179, IF2014 = 2.968]

41

AEH Abstrakty vědeckých prací v domácích karentovaných časopisech

1. DOLEŽAL, Martin and JAMPÍLEK, Josef and KUTILOVÁ, Helena and KRÁĽOVÁ, Katarína. Synthesis

and Biological Evaluation of Anilides Pyrazine-2-carboxylic Acid. Book of Abstracts: The 54th

International Conference of Chemical Societies, Brno, Czech Republic, June 30-July 4, 2002, Chem. Listy

2002, vol. 96, no. 6, 398. [ISSN 0009-2770, IF2002 = 0.336]

2. DOLEŽAL, Martin and KRÁĽOVÁ, Katarína and JAMPÍLEK, Josef. Inhibition of Photosynthetic

Electron Transport in Spinach Chloroplasts by Some Anilides of Pyrazine-2-Carboxylic Acids. Book of

Abstracts: The 54th

International Conference of Chemical Societies, Brno, Czech Republic, June 30-July 4,

2002, Chem. Listy 2002, vol. 96, no. 6, 399. [ISSN 0009-2770, IF2002 = 0.336]

3. JAMPÍLEK, Josef and DOLEŽAL, Martin and DVOŘÁK, Bohumír. Studies of the Influence of

Semiconductor Heterogeneous Catalysts on the Bis(4-methoxyphenyl)disulfide Formation. Book of

Abstracts: The 54th

International Conference of Chemical Societies, Brno, Czech Republic, June 30-July 4,


4. JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří. Aliphatic Iodo Derivatives of

Tetrahydrofuran Formation by means of Titanic Heterogeneous Catalyst as By-Products at the Synthesis of

2-Arylpropanoic Acids from Acetophenone Derivatives. Book of Abstracts: LIBLICE 2002 – The 37th

Conference “Advances in Organic, Bioorganic and Pharmaceutical Chemistry”, Nymburk, Czech

Republic, November 22-24, 2002, Chem. Listy 2002, vol. 96, no. 11, 932. [ISSN 0009-2770, IF2002 = 0.336]

5. JAMPÍLEK, Josef and DOLEŽAL, Martin and OSIČKA, Zdeněk and KUNEŠ, Jiří. Study of Radical

Aroylation of the Pyrazine Nucleus Through Homogeneous Catalysis by Means of Salts of Transition

Metals. Book of Abstracts: LIBLICE 2002 – The 37th

Conference “Advances in Organic, Bioorganic and

Pharmaceutical Chemistry”, Nymburk, Czech Republic, November 22-24, 2002, Chem. Listy 2002, vol.

96, no. 11, 939. [ISSN 0009-2770, IF2002 = 0.336]

6. JAMPÍLEK, Josef and DOLEŽAL, Martin and HANIKA, Jiří. Double Bond Catalytic Hydrogenation on

Palladium Heterogeneous Catalyst in Presence of Sulfanyl Group. Book of Abstracts: The 55th

International Conference of Chemical Societies, Košice, Slovakia, September 8-12, 2003, Chem. Listy

2003, vol. 97, no. 9, 757. [ISSN 0009-2770, IF2003 = 0.345]

7. JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří and RAICH, Ivan. Synthesis of 5- or 6-[(3-

Methoxyphenyl)sulfanyl]pyrazine-2-carboxylic Acid and 5- or 6-[(4-Methoxyphenyl)sulfanyl]pyrazine-2-

carboxylic Acid Derivatives. Book of Abstracts: LIBLICE 2003 – The 38th

Conference “Advances in

Organic, Bioorganic and Pharmaceutical Chemistry”, Nymburk, Czech Republic, November 28-30, 2003,

Chem. Listy 2003, vol. 97, no. 11, 1108. [ISSN 0009-2770, IF2003 = 0.345]

8. JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří and ŠATÍNSKÝ, Dalibor. Novel

Regioselective Preparation of 5-Chloropyrazine-2-carbonitrile from Pyrazine-2-carboxamide. Book of

Abstracts: The 56th

International Conference of Chemical Societies, Ostrava, Czech Republic, September 6-

9, 2004, Chem. Listy 2004, vol. 98, no. 8, 670. [ISSN 0009-2770, IF2004 = 0.348]

9. JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří and JUN, Daniel. Preparation and Antiplatelet

Activity of Glycidic Acid Derivatives. Book of Abstracts: LIBLICE 2004 – The 39th Conference “Advances

in Organic, Bioorganic and Pharmaceutical Chemistry”, Nymburk, Czech Republic, November 26-28,


10. IMRAMOVSKÝ, Aleš and VINŠOVÁ, Jarmila and POLANC, Slovenko and JAMPÍLEK, Josef. New

Derivatives of Isoniazide and Pyrazinamide. Book of Abstracts: LIBLICE 2005 – The 40th

Conference

“Advances in Organic, Bioorganic and Pharmaceutical Chemistry”, Nymburk, Czech Republic, November

18-20, 2005, Chem. Listy 2005, vol. 99, no. 11, 845. [ISSN 0009-2770, IF2005 = 0.445]

11. JAMPÍLEK, Josef and VINŠOVÁ, Jarmila and IMRAMOVSKÝ, Aleš and GRAFNETTEROVÁ, Taťjana,

and DOHNAL, Jiří. Hydrophobic Properties of Some Antimicrobially Active Esters of Salicylanilides.

Book of Abstracts: LIBLICE 2005 – The 40th

Conference “Advances in Organic, Bioorganic and

Pharmaceutical Chemistry”, Nymburk, Czech Republic, November 18-20, 2005, Chem. Listy 2005, vol.

99, no. 11, 846. [ISSN 0009-2770, IF2005 = 0.445]

12. IMRAMOVSKÝ, Aleš and VINŠOVÁ, Jarmila and JAMPÍLEK, Josef. Preparation and Antimycobacterial

Activity of Hydrazonoformamide Derivatives of Isoniazide. Book of Abstracts: The 58th

International

Conference of Chemical Societies, Ústí nad Labem, Czech Republic, September 4-8, 2006, Chem. Listy

2006, vol. 100, no. 8, 659. [ISSN 0009-2770, IF2006 = 0.431]

13. JAMPÍLEK, Josef and IMRAMOVSKÝ, Aleš and VINŠOVÁ, Jarmila and DOHNAL, Jiří. Hydrophobic

Properties of New Hydrazonoformamide Derivatives of Isoniazide. Book of Abstracts: The 58th

International Conference of Chemical Societies, Ústí nad Labem, Czech Republic, September 4-8, 2006,

Chem. Listy 2006, vol. 100, no. 8, 659-660. [ISSN 0009-2770, IF2006 = 0.431]

42

14. JAMPÍLEK, Josef and VINŠOVÁ, Jarmila and IMRAMOVSKÝ, Aleš and MONREAL-FÉRRIZ, Juana

and DOHNAL, Jiří. Hydrophobic Properties of Substituted Salicylanilide Esters of Amino Acids. Book of

Abstracts: LIBLICE 2007 – The 42nd

Conference “Advances in Organic, Bioorganic and Pharmaceutical

Chemistry”, Nymburk, Czech Republic, November 16-18, 2007, Chem. Listy 2007, vol. 101, no. 11, 977.

[ISSN 0009-2770, IF2007 = 0.683]

15. DOHNAL, Jiří and JAMPÍLEK, Josef and IMRAMOVSKÝ, Aleš and MONREAL-FÉRRIZ, Juana and

VINŠOVÁ, Jarmila. Preparation and Hydrophobic Properties of 5-Chloro-N-[1-(3,4-

dichlorophenylcarbamoyl)alkyl]-2-hydroxybenzamides. Book of Abstracts: The XXXVIIth

Conference

“Synthesis and Analysis of Drugs”, Brno, Czech Republic, September 8-10, 2008, Chem. Listy 2008, vol.

102, no. S, s214. [ISSN 0009-2770, IF2008 = 0.593]

16. DOLEŽEL, Jan and HIRŠOVÁ, Petra and OPLETALOVÁ, Veronika and VEJSOVÁ, Marcela and

JAMPÍLEK, Josef. Synthesis and Biological Evaluation of Rhodanine and N-Substituted Rhodanine

Derivatives. Book of Abstracts: The XXXVIIth

Conference “Synthesis and Analysis of Drugs”, Brno, Czech

Republic, September 8-10, 2008, Chem. Listy 2008, vol. 102, no. S, s215. [ISSN 0009-2770, IF2008 = 0.593]

17. JAMPÍLEK, Josef and MUSIOŁ, Robert and BUCHTA, Vladimír and DOHNAL, Jiří and FINSTER, Jacek

and TABAK, Dominik and NIEDBALA, Halina and POLAŃSKI, Jarosław. Preparation and Antifungal

Activity of Ring-Substituted 4-Hydroxy-1H-quinolin-2-ones. Book of Abstracts: The XXXVIIth

Conference

“Synthesis and Analysis of Drugs”, Brno, Czech Republic, September 8-10, 2008, Chem. Listy 2008, vol.

102, no. S, s222. [ISSN 0009-2770, IF2008 = 0.593]

18. IMRAMOVSKÝ, Aleš a VINŠOVÁ, Jarmila a MONREAL-FÉRRIZ, Juana a JAMPÍLEK, Josef.

Decomposition Hydrolytic Study of Hydrazonoformamide Prodrugs of Isoniazide. Book of Abstracts: LIBLICE

2008 – The 43rd

Conference “Advances in Organic, Bioorganic and Pharmaceutical Chemistry”,

Nymburk, Czech Republic, November 14-16, 2008, Chem. Listy 2008, vol. 102, no. 11, 1041. [ISSN 0009-

2770, IF2008 = 0.593]

19. IMRAMOVSKÝ, Aleš and BRITO, Alexandra Maria and PEJCHAL, Vladimír and OKTÁBEC, Zbyněk

and JAMPÍLEK, Josef. Syntesis and Antifungal Properties of New 2-Substituted Benzothiazoles. Book of

Abstracts: LIBLICE 2010 – The 45th Conference “Advances in Organic, Bioorganic and Pharmaceutical

Chemistry”, Nymburk, Czech Republic, November 20-22, 2010, Chem. Listy 2010, vol. 104, no. 11, 1084-

1085. [ISSN 0009-2770, IF2010 = 0.620]

20. RAICH, Ivan and KÁČEROVÁ, Sandra and JAMPÍLEK, Josef and BRYCHTOVÁ, Kateřina.

Conformational Analysis of Substituted Alkyl-6-(2,5-dioxopyrrolidin-1-yl)hexanoates: Calculation study. Book

of Abstracts: LIBLICE 2010 – The 45th

Conference “Advances in Organic, Bioorganic and Pharmaceutical

Chemistry”, Nymburk, Czech Republic, November 20-22, 2010, Chem. Listy 2010, vol. 104, no. 11, 1087-

1088. [ISSN 0009-2770, IF2010 = 0.620]

AFA Publikované vyžádané referáty na zahraničních vědeckých konferencích

1. JAMPÍLEK, Josef and ZADRAŽILOVÁ, Iveta and KOS, Jiří and GONĚC, Tomáš. Design, Synthesis and

Anti-staphylococcus Activity of Hydroxynaphthalenecarboxanilides. Proceedings: International Scientific-

Practical Conference “Pharmaceutical Education, Scientific and Manufacturing as a Reference to the

Strategy Kazakhstan-2020”, South Kazakhstan State Pharmaceutical Academy, Shymkent, Kazakhstan,

October 23-24, 2014, Republican Scientific Journal 2014, vol. 68, no. 3, 3-7. [ISSN 2306-6822]

2. JAMPÍLEK Josef and KRÁĽOVÁ, Katarína. Applications of nanoformulations in Agricultural Production

and Their Potential Impact on Food and Human Health. Proceedings: The 24th

Annual Central European

Conference (ECOpole’15), Opole – Jarnołtówek, Poland, October 14-17, 2015, Proceedings of ECOpole

(PECO-2015), 2015, vol. 9, no. 2, 465-472. [ISSN 1898-617X]

AFC Publikované příspěvky na zahraničních vědeckých konferencích

1. JAMPÍLEK, Josef and DOLEŽAL, Martin and DVOŘÁK, Bohumír. Comparison of Influence of

Conductor, Semiconductor and Insulator Copper Heterogeneous Catalysts on Bis(4-

methoxyphenyl)disulfide Formation. Proceedings: The 6th

International Electronic Conference on Synthetic

Organic Chemistry (ECSOC-6), September 1-30, 2002, http://www.mdpi.net/ec/papers/ecsoc-

6/187/jamp2002.htm. Editors: Shu-Kun Lin and Julio A. Seijas, CD-ROM edition. Published in 2002 by

MDPI, Basel, Switzerland. [ISBN 3-906980-11-1]

2. JAMPÍLEK, Josef and DOLEŽAL, Martin and OSIČKA, Zdeněk and KUNEŠ, Jiří and KRÁĽOVÁ,

Katarína. Substituted Pyrazine-2-carboxamides: Preparation and Their Photosynthesis-inhibiting Activity.

Proceedings: The 7th

International Electronic Conference on Synthetic Organic Chemistry (ECSOC-7),

November 1-30, 2003, http://www.mdpi.net/ec/ec_article.php?id=81&file=papers/ecsoc-7/C001/C001.htm.

Editors: Julio A. Seijas, De-Chun Ji and Shu-Kun Lin, CD-ROM edition. Published in 2003 by MDPI,

Basel, Switzerland. [ISBN 3-906980-13-8]

http://www.mdpi.net/ec/papers/ecsoc-6/187/jamp2002.htm

http://www.mdpi.net/ec/papers/ecsoc-6/187/jamp2002.htm

http://www.mdpi.net/ec/ec_article.php?id=81&file=papers/ecsoc-7/C001/C001.htm

43

3. JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří and BUCHTA, Vladimír. Quinaldine

Derivatives Preparation and Their Antifungal Activity. Proceedings: The 8th

International Electronic

Conference on Synthetic Organic Chemistry (ECSOC-8), November 1-30, 2004, c005,

http://www.usc.es/congresos/ecsoc/8/BOCNP/005/index.htm. Editors: Julio A. Seijas, M. Pilar Vázquez

Tato, CD-ROM edition. Published in 2004 by MDPI, Basel, Switzerland. [ISBN 3-906980-15-4]

4. JAMPÍLEK, Josef and OPLETALOVÁ, Veronika and GRAFNETTEROVÁ, Taťjana and DOHNAL, Jiří.

Thiosemicarbazones of Acetylpyrazines: Preparation and Their Hydrophobic Properties. Proceedings: The

9th

International Electronic Conference on Synthetic Organic Chemistry (ECSOC-9), November 1-30,

2005, http://www.usc.es/congresos/ecsoc/9/GOS/a001/index.htm. Editors: Julio A. Seijas, M. Pilar

Vázquez Tato, CD-ROM edition. Published in 2005 by MDPI, Basel, Switzerland. [ISBN 3-906980-16-2]

5. JAMPÍLEK, Josef and VINŠOVÁ, Jarmila and GRAFNETTEROVÁ, Taťjana and DOHNAL, Jiří.

Synthesis and Hydrophobic Properties of Benzoxazoles. Proceedings: The 9th


Conference on Synthetic Organic Chemistry (ECSOC-9), November 1-30, 2005,

http://www.usc.es/congresos/ecsoc/9/GOS/a008/index.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato,

CD-ROM edition. Published in 2005 by MDPI, Basel, Switzerland. [ISBN 3-906980-16-2]

6. OPLETALOVÁ, Veronika and JAMPÍLEK, Josef and CHLUPÁČOVÁ, Marta and DOLEŽEL, Jan and

GRAFNETTEROVÁ, Taťjana and DOHNAL, Jiří. Chromatographic and Computational study of

Hydrophobic Properties of Ring Substituted Pyrazinecarbonitriles and Acetylpyrazines. Proceedings: The

9th


2005, http://www.usc.es/congresos/ecsoc/9/BOCNP/c004/index.htm. Editors: Julio A. Seijas, M. Pilar


7. MUSIOŁ, Robert and JAMPÍLEK, Josef and KRÁĽOVÁ, Katarína and PODESZWA, Barbara and

FINSTER, Jacek and NIEDBALA, Halina and PAŁKA, Anna and POLAŃSKI, Jarosław. New Quinoline

Derivatives Possessing Herbicidal Activity. Proceedings: The 9th

International Electronic Conference on

Synthetic Organic Chemistry (ECSOC-9), November 1-30, 2005,

http://www.usc.es/congresos/ecsoc/9/BOCNP/c005/index.htm. Editors: Julio A. Seijas, M. Pilar Vázquez


8. DOLEŽAL, Martin and ČMEDLOVÁ, Pavlína and PALEK, Lukáš and KUNEŠ, Jiří and BUCHTA,

Vladimír and JAMPÍLEK, Josef and KRÁĽOVÁ, Katarína. Synthesis and Biological Evaluation of

Pyrazinecarboxamides. Proceedings: The 9th

International Electronic Conference on Synthetic Organic

Chemistry (ECSOC-9), November 1-30, 2005,

http://www.usc.es/congresos/ecsoc/9/BOCNP/c020/index.htm. Editors: Julio A. Seijas, M. Pilar Vázquez


9. JAMPÍLEK, Josef and VINŠOVÁ Jarmila and DOHNAL, Jiří. Synthesis and Hydrophobic Properties of

Substituted 2-Aryl-5,7-di-tert-butylbenzoxazoles. Proceedings: The 10th


Conference on Synthetic Organic Chemistry (ECSOC-10), November 1-30, 2006, a003,

http://www.usc.es/congresos/ecsoc/10/ECSOC10.htm. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-

ROM edition. Published in 2006 by MDPI, Basel, Switzerland. [ISBN 3-906980-18-9]

10. JAMPÍLEK, Josef and OPLETALOVÁ, Veronika and DOHNAL, Jiří. N,N-Dimethylthiosemicarbazones

of Acetylpyrazines: Preparation and Their Hydrophobic Properties. Proceedings: The 10th

International

Electronic Conference on Synthetic Organic Chemistry (ECSOC-10), November 1-30, 2006, a004,



11. JAMPÍLEK, Josef and PALEK, Lukáš and DOLEŽAL, Martin. Synthesis and Hydrophobic Properties of

Some Substituted 3-Arylaminopyrazine-2,5-dicarbonitriles. Proceedings: The 10th





12. MUSIOŁ, Robert and JAMPÍLEK, Josef and KRÁĽOVÁ, Katarína and TABAK, Dominik and

PODESZWA, Barbara and FINSTER, Jacek and POLAŃSKI, Jarosław. Substituted Amides of Quinoline

Derivatives: Preparation and Their Photosynthesis-inhibiting Activity. Proceedings: The 10th

International

Electronic Conference on Synthetic Organic Chemistry (ECSOC-10), November 1-30, 2006, c007,



13. JAMPÍLEK, Josef and VINŠOVÁ, Jarmila and KADEŘÁVKOVÁ, Zuzana and DOHNAL, Jiří. Synthesis

and Hydrophobic Properties of New 2-Aryl-5,7-di-tert-butylbenzoxazoles. Proceedings: The 11th

International Electronic Conference on Synthetic Organic Chemistry (ECSOC-11), November 1-30, 2007,

a009, http://www.usc.es/congresos/ecsoc/11/hall_aGOS/a009/index.htm. Editors: Julio A. Seijas, M. Pilar


http://www.usc.es/congresos/ecsoc/8/BOCNP/005/index.htm

http://www.usc.es/congresos/ecsoc/9/GOS/a001/index.htm

http://www.usc.es/congresos/ecsoc/9/GOS/a008/index.htm

http://www.usc.es/congresos/ecsoc/9/BOCNP/c004/index.htm



http://www.usc.es/congresos/ecsoc/10/ECSOC10.htm




http://www.usc.es/congresos/ecsoc/11/hall_aGOS/a009/index.htm

44

14. MUSIOŁ, Robert and JAMPÍLEK, Josef and KRÁĽOVÁ, Katarína and TABAK, Dominik and FINSTER,

Jacek and PODESZWA, Barbara and KOZIK, Violetta and DOHNAL, Jiří and POLAŃSKI, Jarosław.

Preparation and Herbicidal Activities of Substituted Amides of Quinoline Derivatives. Proceedings: The

11th


2007, a011, http://www.usc.es/congresos/ecsoc/11/hall_aGOS/a011/index.htm. Editors: Julio A. Seijas, M.

Pilar Vázquez Tato, CD-ROM edition. Published in 2007 by MDPI, Basel, Switzerland. [ISBN 3-906980-

19-7]

15. JAMPÍLEK, Josef and OPLETALOVÁ, Veronika and DOLEZEL, Jan and DOHNAL, Jiří. Preparation and

Hydrophobic Properties of 5-Arylalkylidenerhodanines. Proceedings: The 11th



http://www.usc.es/congresos/ecsoc/11/hall_aGOS/a012/index.htm. Editors: Julio A. Seijas, M. Pilar


16. DOLEŽAL, Martin and JAMPÍLEK, Josef and BIELESZ, Stanislav and KUNEŠ, Jiří. Substituted

pyrazine-2,5-dicarboxamides: Synthesis, Hydrophobicity Parameters, and Antimycobacterial Evaluation.



November 1-30, 2007, c005, http://www.usc.es/congresos/ecsoc/11/hall_cBCNP/c005/index.htm. Editors:

Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2007 by MDPI, Basel, Switzerland.

[ISBN 3-906980-19-7]

17. DOLEŽAL, Martin and and LEŠŇANSKÁ, Katarína and PEŠKO, Matúš and JAMPÍLEK, Josef and

KRÁĽOVÁ, Katarína. Pyrazinecarboxamides, Their Synthesis and Evaluation as Potential Herbicides.



November 1-30, 2008, c0004, http://www.usc.es/congresos/ecsoc/12/ECSOC12.htm. Editors: Julio A.

Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2008 by MDPI, Basel, Switzerland. [ISBN

3-906980-20-0]

18. OPLETALOVÁ, Veronika and JAMPÍLEK, Josef and DOLEŽEL, Jan and HIRŠOVÁ, Petra and

DOHNAL, Jiří. Rhodanineacetic Acid Derivatives as Potential Drugs: Preparation and Hydrophobic

Properties of 5-Arylalkylidene-3-carboxymethylrhodanines. Proceedings: The 12th


Conference on Synthetic Organic Chemistry (ECSOC-12), November 1-30, 2008, c0006,



19. MUSIOŁ, Robert and JAMPÍLEK, Josef and KRÁĽOVÁ, Katarína and FINSTER, Jacek and TABAK,

Dominik and NIEDBALA, Halina and CSOLLEI, Jozef and DOHNAL, Jiří and POLAŃSKI, Jarosław.

Ring-substituted 4-Hydroxy-1H-quinolin-2-ones: Preparation and Their Photosynthesis-inhibiting Activity.



November 1-30, 2008, c0012, http://www.usc.es/congresos/ecsoc/12/ECSOC12.htm. Editors: Julio A.

Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2008 by MDPI, Basel, Switzerland. [ISBN

3-906980-20-0]

20. JAMPÍLEK, Josef and OKTÁBEC, Zbyněk and ŘEZÁČOVÁ, Anna and PLAČEK, Lukáš and KOS, Jiří

and HAVELKOVÁ, Lenka and DOHNAL, Jiří and KRÁL Vladimír. Preparation and Properties of New

Co-crystals of Ibandronate. Proceedings: The 13th


Organic Chemistry (ECSOC-13), November 1-30, 2009, c001, http://www.sciforum.net/presentation/201.

Editors: Julio A. Seijas, M. Pilar Vázquez Tato, CD-ROM edition. Published in 2009 by MDPI, Basel,

Switzerland. [ISBN 3-906980-23-5]

21. MUSIOŁ, Robert and JAMPÍLEK, Josef and PEŠKO, Matúš and CARROLL, James and KRÁĽOVÁ,

Katarína and FINSTER, Jacek and O'MAHONY, Jim and COFFEY, Aidan and POLAŃSKI, Jarosław.

Substituted 2-Styrylquinazoline Derivatives: Preparation and Their Biological Activities. Proceedings: The

13th


2009, c004, http://www.sciforum.net/presentation/204. Editors: Julio A. Seijas, M. Pilar Vázquez Tato,


22. BRYCHTOVÁ, Kateřina and DITTRICHOVÁ, Sylva and SLABÁ, Barbora and PLAČEK, Lukáš and

OPATŘILOVÁ, Radka and JAMPÍLEK, Josef and CSÖLLEI, Jozef. Synthesis of Esters of 6-(2,5-

Dioxopyrrolidin-1-yl)-2-(morpholin-4-yl)hexanoic Acid as Potential Transdermal Penetration Enhancers.



November 1-30, 2009, c010, http://www.sciforum.net/presentation/210. Editors: Julio A. Seijas, M. Pilar


23. BRYCHTOVÁ, Kateřina and OPATŘILOVÁ, Radka and PLAČEK, Lukáš and JAMPÍLEK, Josef and

CSÖLLEI, Jozef. Synthesis of Esters of 6-(2,5-Dioxopyrrolidin-1-yl)-2-(2-oxoazepan-1-yl)hexanoic Acid

as Potential Transdermal Penetration Enhancers. Proceedings: The 14th

International Electronic Conference

on Synthetic Organic Chemistry (ECSOC-14), November 1-30, 2010, A417,



http://www.usc.es/congresos/ecsoc/11/hall_cBCNP/c005/index.htm

http://www.usc.es/congresos/ecsoc/11/hall_cBCNP/c005/index.htm




http://www.sciforum.net/presentation/201



45

http://www.sciforum.net/conference/ecsoc-14/paper/417. Editors: Julio A. Seijas, M. Pilar Vázquez Tato,


24. JAMPÍLEK, Josef and KOS, Jiří and OKTÁBEC, Zbyněk and MANDELOVÁ, Zuzana and PEKÁREK,

Tomáš and TKADLECOVÁ, Marcela and HAVLÍČEK, Jaroslav and DOHNAL, Jiří and KRÁL Vladimír..

Co-crystal Screening Study of Risedronate and Unsubstituted Hexoses. Proceedings: The 14th

International

Electronic Conference on Synthetic Organic Chemistry (ECSOC-14), November 1-30, 2010, A421,



25. IMRAMOVSKÝ, Aleš and JAMPÍLEK, Josef and PEŠKO, Matúš and KRÁĽOVÁ, Katarína and

MONREAL-FÉRRIZ, Juana and VINŠOVÁ, Jarmila. Preliminary Study of Photosynthesis-Inhibiting

Activity of Substituted Phenylcarbamoylphenyl N-alkylcarbamates. Proceedings: The 14th

International

Electronic Conference on Synthetic Organic Chemistry (ECSOC-14), November 1-30, 2010, B375,



26. DOLEŽAL, Martin and OSIČKA, Zdeněk and ZITKO, Jan and KUNEŠ, Jiří and JAMPÍLEK, Josef and

VEJSOVÁ, Marcela and BUCHTA Vladimír and KRÁĽOVÁ, Katarína. Substituted N-phenylpyrazine-2-

carboxamides, Their Synthesis, Hydro-lipophilic Properties and Evaluation of Their Antimycobacterial,

Antifungal and Photosynthesis-inhibiting Activity. Proceedings: The 14th


Conference on Synthetic Organic Chemistry (ECSOC-14), November 1-30, 2010, B380,



27. ŽELAZKOVÁ, Jana and JAMPÍLEK, Josef. Total Synthesis of Arctigenin Derivatives as Potential

Anticancer Agents. Proceedings: The 15th

International Electronic Conference on Synthetic Organic

Chemistry (ECSOC-15), November 1-30, 2011, A598, http://www.sciforum.net/conference/ecsoc-

15/paper/598. Editors: Julio A. Seijas, Shu-Kun Lin, M. Pilar Vázquez Tato, CD-ROM edition. Published

in 2011 by MDPI, Basel, Switzerland. [ISBN 3-906980-25-1]

28. MUSIOŁ, Robert and JAMPÍLEK, Josef and PEŠKO, Matúš and KRÁĽOVÁ, Katarína and

KOWALCZYK, Wioleta and FINSTER, Jacek and POLAŃSKI, Jarosław. Preparation and Herbicidal

Properties of Ring-Substituted 4-Chloro-2-styrylquinazolines. Proceedings: The 15th

International


http://www.sciforum.net/conference/ecsoc-15/paper/586. Editors: Julio A. Seijas, Shu-Kun Lin, M. Pilar


29. ŠUJAN, Josef and PEŠKO, Matúš and GONĚC, Tomáš and KOS, Jiří and BOBÁĽ, Pavel and

IMRAMOVSKÝ, Aleš and PLAČEK, Lukáš and KRÁĽOVÁ, Katarína and JAMPÍLEK, Josef.

Preparation and Herbicidal Properties of Substituted Quinoline-2-carboxanilides. Proceedings: The 15th


B588, http://www.sciforum.net/conference/ecsoc-15/paper/588. Editors: Julio A. Seijas, Shu-Kun Lin, M.


25-1]

30. ŠUJAN, Josef and OTEVŘEL, Jan and IMRAMOVSKÝ, Aleš and JAMPÍLEK, Josef and BOBÁĽ, Pavel.

Microwave-assisted synthesis of new substituted anilides of quinaldic acid. Proceedings: The 15th


C681, http://www.sciforum.net/conference/ecsoc-15/paper/681. Editors: Julio A. Seijas, Shu-Kun Lin, M.


25-1]

31. VACULÍKOVÁ, Eliška and GRÜNWALDOVÁ, Veronika and KRÁL, Vladimir and DOHNAL, Jiří and

JAMPÍLEK, Josef. Preparation of Candesartan Cilexetil Nanoparticles by Precipitation. Proceedings: The

16th


2012, B1008, http://www.sciforum.net/conference/ecsoc-16/paper/1008. Editors: Julio A. Seijas, M. Pilar

Vázquez Tato, Shu-Kun Lin, CD-ROM edition. Published in 2013 by MDPI, Basel, Switzerland. [ISBN 3-

906980-26-X]

32. KOS, Jiří and ZADRAŽILOVÁ, Iveta and PEŠKO, Matúš and PAVLICA, Jiří and GONĚC, Tomáš and

BOBÁL, Pavel and ORAVEC, Michal and ČÍŽEK, Alois and KRÁĽOVÁ, Katarína and JAMPÍLEK,

Josef. Preparation and Biological Properties of Ring-Substituted 3-Hydroxynaphthalene-2-carboxanilides.



November 1-30, 2012, B1009, http://www.sciforum.net/conference/ecsoc-16/paper/1009. Editors: Julio A.

Seijas, M. Pilar Vázquez Tato, Shu-Kun Lin, CD-ROM edition. Published in 2013 by MDPI, Basel,

Switzerland. [ISBN 3-906980-26-X]

http://www.sciforum.net/conference/ecsoc-14/paper/417











46

33. ZADRAŽILOVÁ, Iveta and PAUK, Karel and IMRAMOVSKÝ, Aleš and HANUSEK, Jiří and

MASAŘÍKOVÁ, Martina and ČÍŽEK, Alois and JAMPÍLEK, Josef. 2-Hydroxy-N-[1-(2-

hydroxyphenylamino)-1-oxoalkan-2-yl]benzamides – Potential drugs of MRSA infections? Proceedings:

The International Student Scientific Conference of Faculty of Natural Sciences of Comenius University

2013, Faculty of Natural Sciences, Comenius University, Bratislava, Slovakia, April 24, 2013, p. 857-862.

[ISBN 978-80-223-3392-4]

34. KOS, Jiří and GONĚC, Tomáš and TENGLER, Jan and ZADRAŽILOVÁ, Iveta and PEŠKO, Matúš and

ORAVEC, Michal and KRÁĽOVÁ, Katarína and ČÍŽEK, Alois and JAMPÍLEK, Josef: Synthesis of

amides of hydroxynaphthoic acids as biologically active compounds. Proceedings: The International

Student Scientific Conference of Faculty of Natural Sciences of Comenius University 2013, Faculty of

Natural Sciences, Comenius University, Bratislava, Slovakia, April 24, 2013, p. 1044-1047. [ISBN 978-80-

223-3392-4]

35. VACULÍKOVÁ, Eliška and PLACHÁ, Daniela and JAMPÍLEK, Josef. Preparation of atorvastatin

nanoparticles by solvent evaporation method. Proceedings: The International Student Scientific Conference

of Faculty of Natural Sciences of Comenius University 2013, Faculty of Natural Sciences, Comenius

University, Bratislava, Slovakia, April 24, 2013, p. 1199-1204. [ISBN 978-80-223-3392-4]

36. VACULÍKOVÁ, Eliška and PLACHÁ, Daniela and PISÁRČIK Martin and JAMPÍLEK, Josef. Preparation

of Risedronate Nanoparticles Using Selected Polymeric Excipients. Proceedings: The 17th

International


http://sciforum.net/conference/ecsoc-17/paper/2256. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, Shu-

Kun Lin, CD-ROM edition. Published in 2014 by MDPI, Basel, Switzerland. [ISBN 3-906980-46-0]

37. KOS, Jiří and MACHALOVÁ, Petra and PEŠKO, Matúš and GONĚC, Tomáš and BOBÁL, Pavel and

ORAVEC, Michal and LIPTAJ, Tibor and KRÁĽOVÁ, Katarína and JAMPÍLEK, Josef. Preparation and

Herbicidal Activity of Halogenated 8-Hydroxyquinoline-2-carboxanilides. Proceedings: The 17th


B013, http://sciforum.net/conference/ecsoc-17/paper/2261. Editors: Julio A. Seijas, M. Pilar Vázquez Tato,

Shu-Kun Lin, CD-ROM edition. Published in 2014 by MDPI, Basel, Switzerland. [ISBN 3-906980-46-0]

38. GONĚC, Tomáš and KOS, Jiří and ŠORAL, Michal and PEŠKO, Matúš and ORAVEC, Michal and

LIPTAJ, Tibor and KRÁĽOVÁ, Katarína and JAMPÍLEK, Josef. Preparation and Photosynthesis-

Inhibiting Activity of N-(n-Alkoxy)phenylamides of 2-Hydroxynaphthalene-1-carboxylic acid.



November 1-30, 2014, b010, http://www.sciforum.net/conference/ecsoc-18/paper/2538. Editors: Julio A.

Seijas, M. Pilar Vázquez Tato, Shu-Kun Lin, CD-ROM edition. Published in 2015 by MDPI, Basel,

Switzerland. [ISBN 978-3-906980-55-3]


of Glibenclamide Nanoparticles. Proceedings: The 18th


Organic Chemistry (ECSOC-18), November 1-30, 2014, b025, http://www.sciforum.net/conference/ecsoc-

18/paper/2573. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, Shu-Kun Lin, CD-ROM edition. Published

in 2015 by MDPI, Basel, Switzerland. [ISBN 978-3-906980-55-3]

40. GONĚC, Tomáš and STRÁNÍK, Josef and PEŠKO, Matúš and KOS, Jiří and ORAVEC, Michal and

KRÁĽOVÁ, Katarína and JAMPÍLEK, Josef. Preparation and Photosynthesis-Inhibiting Activity of 1-[(2-

Chlorophenyl)carbamoyl]naphthalen-2-yl Alkylcarbamates. Proceedings: The 19th


Conference on Synthetic Organic Chemistry (ECSOC-19), November 1-30, 2015, b006,

http://sciforum.net/conference/80/paper/3079. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, Shu-Kun

Lin, CD-ROM edition. Published in 2016 by MDPI, Basel, Switzerland. [ISBN 978-3-03842-145-0]


of Hydrochlorothiazide Nanoparticles. Proceedings: The 19th

International Electronic Conference on

Synthetic Organic Chemistry (ECSOC-19), November 1-30, 2015, b007,

http://sciforum.net/conference/80/paper/3080. Editors: Julio A. Seijas, M. Pilar Vázquez Tato, Shu-Kun

Lin, CD-ROM edition. Published in 2016 by MDPI, Basel, Switzerland. [ISBN 978-3-03842-145-0]

AFD Publikované příspěvky na domácích vědeckých konferencích

1. ZADRAŽILOVÁ, Iveta and GONĚC, Tomáš and ČÍŽEK, Alois and JAMPÍLEK, Josef. In vitro

Antimicrobial Screening of N-(n-Alkoxy)phenylanilides of 2-Hydroxynaphthalene-1-carboxylic acid.

Proceedings: Inter-University Postgraduate Student Conference, University of Veterinary and

Pharmaceutical Sciences Brno, Brno, Czech Republic, October 2, 2014, p. 85-88. [ISBN 78-80-7305-740-4]

2. ČERNÍKOVÁ, Aneta and OPATŘILOVÁ, Radka and JAMPÍLEK, Josef. Rapid Screening of Rutin Skin

Permeation. Proceedings: Inter-University Postgraduate Student Conference, University of Veterinary and


http://sciforum.net/conference/ecsoc-17/paper/2256

http://sciforum.net/conference/ecsoc-17/paper/2261




http://sciforum.net/conference/80/paper/3079

http://sciforum.net/conference/80/paper/3080

47

3. VACULÍKOVÁ, Eliška and JAMPÍLEK, Josef. Preparation of Glibenclamide Nanoparticles via Solvent

Evaporation. Proceedings: Inter-University Postgraduate Student Conference, University of Veterinary and


AFE Abstrakty vyžádaných referátů ze zahraničních konferencí

1. JAMPÍLEK, Josef. Advances in Investigation of Hydrophilic and Lipophilic Properties of Drugs. Book of

Abstracts: The XXXVth

Symposium 'Chromatographic Methods of Investigating the Organic Compounds',

Katowice – Szczyrk, Poland, May 30 - June 1, 2012, OS-5.

2. JAMPÍLEK, Josef. Pharmaceutical nanoparticles and methods of their characterization. Book of Abstracts:

The XXXVIth

Symposium 'Chromatographic Methods of Investigating the Organic Compounds', Katowice –

Szczyrk, Poland, June 5-7, 2013, OS-19.

3. JAMPÍLEK, Josef and MUSIOŁ, Robert and KOS, Jiří and GONĚC, Tomáš and BOBÁL, Pavel and

POLAŃSKI, Jarosław. Design and Antimicrobial Screening of New Ring-Substituted Quinoline

Analogues. Book of Abstracts: The BIT′s 4th

Annual International Congress of Medichem 2013 (ICM-

2013), Haikou, China, November 13-16, 2013, p. 62.

4. JAMPÍLEK, Josef and COUFALOVÁ, Lenka and MRÓZEK, Lech. Investigation of Cholic Acid

Derivatives as Transdermal Permeation Enhancers. Book of Abstracts: The XXXVIIth

Symposium

'Chromatographic Methods of Investigating the Organic Compounds', Katowice – Szczyrk, Poland, June

11-14, 2014, OS-18.

5. JAMPÍLEK, Josef and KOS, Jiří and ZADRAŽILOVÁ, Iveta and GONĚC, Tomáš and HRUBÁ, Michaela

and MORAVCOVÁ, Marie and ŠTUJBER, Michal and LIPTAJ, Tibor. Synthesis and Antimicrobial

Activity of Hydroxy(aza)naphthalenecarboxamides. Book of Abstracts: The 7th Central European

Conference "Chemistry towards Biology", Katowice, Poland, September 9-12, 2014, p. O5.

6. JAMPÍLEK, Josef and CLEMENTS, Carol and KOS, Jiří and GONĚC, Tomáš and GRAY, Alexander I.

Synthesis and In Vitro Anti-trypanosomal Screening of Hydroxynaphthalene-2-carboxanilides. Book of

Abstracts: The VIth

Conversatory on Medicinal Chemistry, Lublin, Poland, September 18-20, 2014, p. 24

(K5). [ISSN 978-83-63657-38-3]

7. JAMPÍLEK, Josef. Recent Advances in Design of Potential Quinoxaline Anti-Infectives. Book of

Abstracts: The BIT′s 5th

Annual International Congress of Medichem 2014 (ICM-2014), Suzhou, China,

November 18-20, 2014, p. 197.

8. JAMPÍLEK, Josef. Azanaphthalenes as Potential Antimycobacterial Agents. Book of Abstracts: The 13th

Ibn Sina International Conference on Pure and Applied Heterocyclic Chemistry, Hurghada, Egypt,

February 14-17, 2015, p. 8 (PL-06).

9. ORAVEC, Michal and JAMPÍLEK, Josef. Determination of Drugs Loaded to Silica Nanoparticles in Brain

Tissue. Book of Abstracts: The XXXVIIIth

Symposium 'Chromatographic Methods of Investigating the

Organic Compounds', Katowice – Szczyrk, Poland, May 27-29, 2015, OS-27.

10. JAMPÍLEK, Josef and KOS, Jiří and ZADRAŽILOVÁ, Iveta. Advances in Design of Potential Quinoline

Antimycobacterial Agents. Book of Abstracts: The IXth

Joint Meeting in Medicinal Chemistry

(JMMC 2015), Athens, Greece, June 7-10, 2015, O6.

11. JAMPÍLEK, Josef and ČERNÍKOVÁ, Aneta and BOBÁĽ, Pavel. Design, Synthesis and Investigation of

Aryl Derivatives of Alaptide as Potential Transdermal Permeation Enhancers. Book of Abstract: European

Pharma Congress “Pharma Europe-2015”, Valencia, Spain, August 25-27, 2015, J. Pharma. Care Health

Sys. 2015, vol. 2, no. 4, 63. [ISSN 2376-0419]

12. JAMPÍLEK Josef and ČERNÍKOVÁ, Aneta and TABIOVÁ, Katarína and BOBÁĽ, Pavel. In Vitro

Evaluation of 8-Substituted 6,9-diazaspiro[4.5]decan-7,10-diones as Skin Permeation Modifiers. Book of

Abstracts: The 4th

World Conference on Physico-Chemical Methods in Drug Discovery and Development

(PCMDDD-4), Rovinj – Red Island, Croatia, September 21-24, 2015, p. 10 (OP 08).

13. JAMPÍLEK Josef and KOS, Jiří and ZADRAŽILOVÁ, Iveta and GONĚC, Tomáš and BOBÁĽ, Pavel.

Design and Antimicrobial Activity of Ring-Substituted Hydroxynaphthalenecarboxamides and Their Aza-

Analogues. Book of Abstracts: The BIT's 13th

Annual World Congress of International Drug Discovery

Science & Technology 2015 (IDDST 2015), Beijing, China, October 20-22, 2015, p. 109.

14. JAMPÍLEK Josef and ČERNÍKOVÁ, Aneta and BOBÁĽ, Pavel and DOHNAL, Jiří. Investigation of Alkyl

Derivatives of Alaptide as Transdermal Permeation Modifier. Book of Abstracts: The BIT's 5th

Annual

World Symposium of Drug Delivery System 2015 (SDDS-2015), Beijing, China, October 20-22, 2015, p.

387.

48

AFF Abstrakty vyžádaných referátů z domácích konferencí

1. JAMPÍLEK, Josef. Perspectives of nanoparticles in pharmacy. Book of Abstracts: The 1st International

Symposium and Workshop on Environment and Health (ISEH 2012), Ostrava, Czech Republic, November

22-23, 2012, p. 44. [ISBN 978-80-248-2882-4]

2. JAMPÍLEK, Josef. Polymorphism and Its Influence to Biovailability. Book of Abstracts: The 2nd

International Symposium and Workshop on Environment and Health (ISEH 2013), Ostrava, Czech

Republic, November 6-8, 2013, p. 20-21. [ISBN 978-80-248-3240-1]

3. JAMPÍLEK, Josef. Overcoming Blood-Brain Barrier Using Nanoparticles. Book of Abstracts:

The 4th

Nanomaterials and Nanotechnology Meeting (NanoOstrava 2015), Ostrava, Czech Republic, May

18-21, 2015, p. 63. [ISBN 978-80-248-3745-1]

4. JAMPÍLEK, Josef. Nanoformulations of Antimicrobial Chemotherapeutics. Book of Abstracts: The

International Conference on Nanomedicine, Drug Delivery, and Tissue Engineering (NDDTE'16), Prague,

Czech Republic, April 1-2, 2016, Keynote-2, http://nddte.com/paper/Keynote%20-

%20Dr.%20Jampilek.pdf.

AFG Abstrakty příspěvků ze zahraničních konferencí

1. JAMPÍLEK, Josef and DOLEŽAL, Martin. Preparation and Biological Evaluation of 5-Aroylpyrazine-2-

carboxylic Acid Derivatives. Book of Abstracts: The 1st International Student Scientific Conference of

Faculty of Natural Sciences, Comenius University, Bratislava, Slovakia, April 25-26, 2001, p. Po-2.

2. JAMPÍLEK, Josef and DOLEŽAL, Martin and DVOŘÁK, Bohumír. Bis(4-methoxyphenyl)disulfide

Preparation by Means of Copper Catalysts. Book of Abstracts: The 53th

International Conference of

Chemical Societies, Banská Bystrica, Slovakia, September 3-6, 2001, p. 268-269.

3. JAMPÍLEK, Josef and DOLEŽAL, Martin and DVOŘÁK, Bohumír. Comparison of Effect of

Semiconductor and Insulator Copper Heterogeneous Catalysts on Bis(4-methoxyphenyl)disulfide

Formation. Book of Abstracts: The International Conference on Organic Synthesis “Balticum Organicum

Syntheticum” (BOS 2002), Vilnius, Lithuania, June 23-27, 2002, p. 79. [ISBN 9986-19-485-7]

4. JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří and OSIČKA, Zdeněk. Preparation of Thiazol-

2-ylamide, or Pyrid-2-ylamide Pyrazine-2-carboxylic Acid Derivatives. Book of Abstracts: The XXXIst

Conference “Synthesis and Analysis of Drugs”, Bratislava, Slovakia, September 11-13, 2002, p. 60.

5. JAMPÍLEK, Josef and DOLEŽAL, Martin and KUCHAŘ, Miroslav. Synthesis of 2-Methyl-3-(4-{[4-

(quinolin-2-ylmethoxy)phenyl]sulfanyl}phenyl)propionic Acid (VUFB 20584) as a Potential

Antileukotrienic. Book of Abstracts: The 1st International SPECS and BioSPECS Symposium on The New

Chemistries, Delft, the Netherlands, September 18-21, 2002, p. 98.

6. JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří. Synthesis of (2E)-2-methyl-3-(4-{[4-

(quinolin-2-ylmethoxy)phenyl]sulphanyl}phenyl)acrylic Acid (VUFB 20609) as a Potential

Antileukotrienic Agent. Book of Abstracts: The 9th

European Symposium on Organic Reactivity (ESOR IX),

Oslo, Norway, July 12-17, 2003, p.153.

7. JAMPÍLEK, Josef and DOLEŽAL, Martin and RAICH, Ivan and LIŠKA, František. 4-Substituted Aryl-

and 6-Substituted Heteroarylhalides Coupling with 4-Methoxybenzenethiol by Means of Copper

Heterogeneous Catalysts. Book of Abstracts: The 9th

European Symposium on Organic Reactivity (ESOR

IX), Oslo, Norway, July 12-17, 2003, p. 169.

8. JAMPÍLEK, Josef and CHLUPÁČOVÁ, Marta and DOLEŽAL, Martin and KRÁĽOVÁ, Katarína:

Quinaldine Derivatives and Their Herbicidal Activities. Book of Abstracts: The International Conference

“Jahrestagung – Joint Meeting 2004”, Faculty of Chemistry and Pharmacy, University of Regensburg,

Regensburg, Germany, October 6-9, 2004, p. 111 (P-C63). [ISBN 3-00-014723-3]

9. JAMPÍLEK, Josef and DOLEŽAL, Martin and BROJEROVÁ Eliška and OPLETAL, Lubomír and JUN,

Daniel. Substituted Diarylsulfides and Their Antiplatelet Activity. Book of Abstracts: The International

Conference “The 4th

Joint Meeting on Medicinal Chemistry 2005” (JMMC 2005), Vienna, Austria, June 20-

23, 2005, Sci. Pharm. 2005, vol. 73, no. 2 Suppl. 1, 83. [ISSN 0036-8709]

10. VINŠOVÁ, Jarmila and IMRAMOVSKÝ, Aleš and BUCHTA, Vladimír and DOLEŽAL, Martin and

JAMPÍLEK, Josef. Biodegradable Esters of Salicylanilides with Significant Antimicrobial Activity. Book

of Abstracts: The 14th

European Symposium on Organic Chemistry (ESOC 14), Helsinki, Finland, July 4-8,

2005, p. 258. [ISBN 952-10-2553-0]

11. JAMPÍLEK, Josef and DOLEŽAL, Martin and PALEK, Lukáš. Radical Aroylation of Pyrazine-2-

carboxylic Acid Derivatives. Book of Abstracts: The 14th

European Symposium on Organic Chemistry

(ESOC 14), Helsinki, Finland, July 4-8, 2005, p. 272. [ISBN 952-10-2553-0]

12. IMRAMOVSKÝ, Aleš and VINŠOVÁ, Jarmila and POLANC, Slovenko and JAMPÍLEK, Josef and

DOLEŽAL, Martin. New Hydrazonoformamide Derivatives of Isoniazide. Book of Abstracts: The 14th

http://nddte.com/paper/Keynote%20-%20Dr.%20Jampilek.pdf


49

European Symposium on Organic Chemistry (ESOC 14), Helsinki, Finland, July 4-8, 2005, p. 295. [ISBN

952-10-2553-0]

13. DOLEŽAL, Martin and PALEK, Lukáš and VINŠOVÁ, Jarmila and BUCHTA, Vladimír and JAMPÍLEK,

Josef and KRÁĽOVÁ, Katarína. Substituted Amides of Pyrazinoic Acid, Synthesis and Biological

Evaluation. Book of Abstracts: The 14th

European Symposium on Organic Chemistry (ESOC 14), Helsinki,

Finland, July 4-8, 2005, p. 350. [ISBN 952-10-2553-0]

14. DOLEŽAL, Martin and BRUNER, Rudolf and BUCHTA, Vladimír and JAMPÍLEK, Josef and

KRÁĽOVÁ, Katarína: Amides of Pyrazin-2-carboxylic acid: Synthesis, Antifungal Evaluation and Their

Photosynthesis Inhibition. Book of Abstracts: The 57th

International Conference of Chemical Societies,

Tatranské Matliare, Slovakia, September 4-8, 2005, ChemZi 2005, vol. 1, no. 1, 206. [ISSN 1336-7242]

15. JAMPÍLEK, Josef and DOLEŽAL, Martin and PALEK, Lukáš. Preparation and Antimycobacterial

Activity of Pyrazine-2-carboxylic Acid Thiazol-2-ylamide Derivatives. Book of Abstracts: The

International Conference “Frontiers in Medicinal Chemistry”, Frankfurt am Main, Germany, March 12-15,

2006, p. 90.

16. JAMPÍLEK, Josef and VINŠOVÁ, Jarmila and IMRAMOVSKÝ, Aleš and DOLEŽAL, Martin and

DOHNAL, Jiří. RP-HPLC Method for Determination of Isoniazide Prodrugs. Book of Abstracts: The

International Conference “Drug Analysis 2006”, Namur, Belgium, May 16-19, 2006, PE-09.

17. PALEK, Lukáš and JAMPÍLEK, Josef and DOLEŽAL, Martin. RP-HPLC Assay and Hydrophobic

Properties of Novel Pyrazinamide Derivatives. Book of Abstracts: The International Conference “Drug

Analysis 2006”, Namur, Belgium, May 16-19, 2006, PK-28.

18. MUSIOŁ, Robert and JAMPÍLEK, Josef and PODESZWA, Barbara and FINSTER, Jacek and TABAK,

Dominik and POLAŃSKI, Jarosław. Structure-lipophilicity Relationships in Series of Quinoline

Derivatives. Book of Abstracts: The 18th

International Conference on Physical Organic Chemistry

(ICPOC-18), Warsaw, Poland, August 20-25, 2006, p. 76. [ISBN 83-89585-11-1]

19. JAMPÍLEK, Josef and OPLETALOVÁ, Veronika, and POUR, Milan and KUNEŠ, Jiří and SILVA, Luís

and BUCHTA, Vladimír and RICHARDSON, Des Robert and KALINOWSKI, Danuta and AL-HALLAK,

Linda and HONCOVÁ, Dana. N,N-Dimethylthiosemicarbazones of Acetylpyrazines as Potential Drugs.

Book of Abstracts: The International Conference “Joint Meeting of the Czech, German and Hungarian

Pharmaceutical Societies”, Marburg, Germany, October 4-7, 2006, p. 122 (C076). [ISBN 3-89703-685-1]

20. DOLEŽAL, Martin and MONKS, Kathryn and PLAŠOVÁ, Petra and VINŠOVÁ, Jarmila and JAMPÍLEK,

Josef and SVOBODOVÁ, Michaela and BUCHTA, Vladimír. Synthesis, Antifungal and Antimycobacterial

Properties of Pyrazine Analogues. Book of Abstracts: The International Conference “The 5th

Joint Meeting

on Medicinal Chemistry 2007” (JMMC 2007), Portorož, Slovenia, June 17-21, 2007, Farmacevtski vestnik

2007, vol. 58, no. Suppl. 1, 85 (PO031). [ISSN 0014-8229]

21. JAMPÍLEK, Josef and DOLEŽAL, Martin and VINŠOVÁ, Jarmila. Structure-lipophilicity Relationships in

Series of Methyl Moiety Ring-substituted Pyrazinecarboxanilides as New Antituberculotics. Book of

Abstracts: The International Conference “The 5th

Joint Meeting on Medicinal Chemistry 2007” (JMMC 2007),

Portorož, Slovenia, June 17-21, 2007, Farmacevtski vestnik 2007, vol. 58, no. Suppl. 1, 112 (PO059).

[ISSN 0014-8229]

22. JAMPÍLEK, Josef and MUSIOŁ, Robert and BUCHTA, Vladimír and PODESZWA, Barbara and

FINSTER, Jacek and NIEDBALA, Halina and PAŁKA, Anna and POLAŃSKI, Jarosław. Preparation and

Antifungal Activity of 8-Hydroxyquinoline Derivatives. Book of Abstracts: The 8th Tetrahedron Symposium

“50th Anniversary Meeting – Challenges in Organic Chemistry”, Berlin, Germany, June 27-29, 2007, P2.1.

23. JAMPÍLEK, Josef and VINŠOVÁ, Jarmila and IMRAMOVSKÝ, Aleš and MONREAL-FÉRRIZ, Juana

and DOHNAL, Jiří. Hydrophobic Properties of Some Novel Esters of Salicylanilides. Book of Abstracts:

The 59th

International Conference of Chemical Societies, Tatranské Matliare, Slovakia, September 2-6,

2007, ChemZi 2007, vol. 3, no. 1, 212. [ISSN 1336-7242]

24. PETRIK, Pavel and VEJSOVÁ, Marcela and KUNEŠ, Jiří and JAMPÍLEK, Josef and ŠPANINGEROVÁ,

Eliška and KEŠETOVIČOVÁ, Diana and VLČKOVÁ, Martina and MAJD, Morid and KALAFUTOVÁ,

Stanislava and OPLETALOVÁ, Veronika. Antifungal and Antimycobacterial Properties of 5-

Arylmethylidenerhodanines and Their N3-Substituted Analogues. Book of Abstracts: The 5

th International

Postgraduate Research Symposium on Pharmaceutics (IPORSIP-2007), Istanbul, Turkey, September 13-

15, 2007, Acta Pharm. Sci. 2007, 49 (Suppl.), 77. [ISSN 1300-638X]

25. JAMPÍLEK, Josef and DOLEŽAL, Martin and BIELESZ, Stanislav and VINŠOVÁ, Jarmila. RP-HPLC

Determination of Hydrophobic Properties of New Pyrazindicarboxamide Derivatives. Book of Abstracts:

The 12th International Meeting on Recent Developments in Pharmaceutical Analysis (RDPA 2007), Island

of Elba, Italy, September 23-26, p. 96.

50

26. DOHNAL, Jiří and JAMPÍLEK, Josef and IMRAMOVSKÝ, Aleš and REČKOVÁ, Zuzana and VINŠOVÁ,

Jarmila. Stability Study of Pyrazinamide Prodrugs as New Effective Antituberculotics. Book of Abstracts:

The 12th International Meeting on Recent Developments in Pharmaceutical Analysis (RDPA 2007), Island

of Elba, Italy, September 23-26, p. 97.

27. REČKOVÁ, Zuzana and JAMPÍLEK, Josef and IMRAMOVSKÝ, Aleš and VINŠOVÁ, Jarmila and

DOHNAL, Jiří. Stability Study of Isoniazid Prodrugs as New Effective Antituberculotics. Book of

Abstracts: The 12th International Meeting on Recent Developments in Pharmaceutical Analysis (RDPA

2007), Island of Elba, Italy, September 23-26, p. 98.

28. JAMPÍLEK, Josef and PEKÁREK, Tomáš and ZERZAŇOVÁ, Anna and MATĚJKA, Pavel and

HAVLÍČEK, Jaroslav and BRUSOVÁ, Hana and DOHNAL, Jiří and KRÁL, Vladimír. Application of NIR

for Characterization of Polymorph Purity and API-Excipient Cocrystals. Book of Abstracts: The XIXth

Slovak - Czech Spectroscopic Conference, Častá-Papiernička, Slovakia, October 12-16, 2008, p. 96 (P-21).

[ISBN 978-80-223-2557-8]

29. JAMPÍLEK, Josef and BRYCHTOVÁ, Kateřina and OPATŘILOVÁ, Radka and RAICH, Ivan.

Preparation and Physico-chemical Properties of Alkyl-6-(2,5-dioxopyrrolidin-1-yl)-2-(2-oxopyrrolidin-1-

yl)hexanoates. Book of Abstracts: The International Conference “Frontiers in Medicinal Chemistry”,

Heidelberg, Germany, March 15-18, 2009, p. 84.

30. JAMPÍLEK, Josef and OKTÁBEC, Zbyněk and PEKÁREK, Tomáš and HAVLÍČEK, Jaroslav and

DOHNAL, Jiří and KRÁL, Vladimír. Characterization of Polymorphs and API-Excipient Cocrystals Using

Vibration Spectroscopy and Solid-state NMR. Book of Abstracts: The 11th

International Workshop on

Physical Characterization of Pharmaceutical Solids (IWPCPS®

11), Stamford, Connecticut, USA, June 14-

19, 2009.

31. JAMPÍLEK, Josef and MUSIOŁ, Robert and CARROLL, James and O'MAHONY, Jim and COFFEY,

Aidan and FINSTER, Jacek and TABAK, Dominik and NIEDBALA, Halina and DOHNAL, Jiří and

POLAŃSKI, Jarosław. Synthesis and Antimycobacterial Activity of Styrylquinazolinone Derivatives. Book

of Abstracts: The International Conference “The 6th

Joint Meeting on Medicinal Chemistry 2009” (JMMC

2009), Budapest, Hungary, June 24-27, 2009, p. 73 (P-11). [ISBN 978-963-9319-95-0]

32. DOHNAL, Jiří and JAMPÍLEK, Josef and OKTÁBEC, Zbyněk and ZERZAŇOVÁ, Anna and KRÁL,

Vladimír. Utilization of NIR Spectroscopy in Candesartan Cilexetil Stability Study. Book of Abstracts: The

34th

International Conference on Infrared, Millimeter, and Terahertz Waves (IRMMW-THz 2009), Busan,

South Korea, September 21-25, 2009, p.59 (T5E25.0194). [ISBN 978-1-4244-5417-4]

33. OKTÁBEC, Zbyněk and JAMPÍLEK, Josef and ZERZAŇOVÁ, Anna and DOHNAL, Jiří and KRÁL,

Vladimír. Study of Interactions between API and Excipients in Solid Drug Formulation via NIR. Book of

Abstracts: The 1st World Conference on Physico-Chemical Methods in Drug Discovery and Development,

Rovinj, Croatia, September 27-October 1, 2009, p. 33 (OP-05).

34. ZERZAŇOVÁ, Anna and OKTÁBEC, Zbyněk and JAMPÍLEK, Josef and DOHNAL, Jiří and KRÁL,

Vladimír. Absorption Study of Binary Mixtures. Book of Abstracts: The 1st World Conference on Physico-

Chemical Methods in Drug Discovery and Development, Rovinj, Croatia, September 27-October 1, 2009,

p. 48 (PP-06).

35. PAZOUREK, Jiří and DOHNAL, Jiří and JAMPÍLEK, Josef. Chiral Purity Determination of Z-alanine

Using Capillary Electrophoresis. Book of Abstracts: The XXXIXth

Conference “Synthesis and Analysis of

Drugs”, Modra, Slovakia, September 2-4, 2010, p. 105 (P-58). [ISBN 978-80-7399-986-5]

36. OKTÁBEC, Zbyněk and IMRAMOVSKÝ, Aleš and PEJCHAL, Vladimír and JAMPÍLEK, Josef. RP-

HPLC Determination of Hydrophobic Properties of Novel Substituted Benzothiazole Derivatives. Book of

Abstracts: The 28th

International Symposium on Chromatography (ISC 2010), Valencia, Spain, September

12-16, 2010, p. 285 (P03-017).

37. IMRAMOVSKÝ, Aleš and ŠTĚPÁNKOVÁ, Šárka and PEJCHAL, Vladimír and JAMPÍLEK, Josef.

Benzothiazole Derivates as Potent Acetylcholinesterase Inhibitors. Book of Abstracts: The International

Conference “The 7th

Joint Meeting on Medicinal Chemistry 2011” (JMMC 2011), Catania, Sicily, Italy, June

30-July 2, 2011.

38. JAMPÍLEK, Josef and OPATŘILOVÁ, Radka and ŘEZÁČOVÁ, Anna and OKTÁBEC, Zbyněk and

ČULEN, Martin and DOHNAL, Jiří. Approaches to Alaptide Water-Solubilization and Improvement of its

Permeation Across Membranes. Book of Abstracts: The International Symposium on Advances in Synthetic

and Medicinal Chemistry (ASMC 2011), St. Petersburg, Russia, August 21-25, 2011, p. 195 (P082).

39. JAMPÍLEK, Josef and MUSIOŁ, Robert and PÁVEK, Petr and KOWALCZYK, Wioleta and MAZUR,

Paweł and POLAŃSKI, Jarosław. Investigation of Ring-substituted 3-(Benzylideneamino)-2-methyl-

quinazolin-4(3H)-ones. Book of Abstracts: The International Symposium on Advances in Synthetic and

Medicinal Chemistry (ASMC 2011), St. Petersburg, Russia, August 21-25, 2011, p. 196 (P083).

51

40. IMRAMOVSKÝ, Aleš and ŠTĚPÁNKOVÁ, Šárka and MONREAL-FÉRRIZ, Juana and VINŠOVÁ,

Jarmila and VANČO, Ján and JAMPÍLEK, Josef. New Carbamates of Salicylanilides as Potential

Acetylcholinesterase Inhibitors and Their Molecular Docking. Book of Abstracts: The 63rd

International

Conference of Chemical Societies, Tatranské Matliare, Slovakia, September 5-9, 2011, ChemZi 2011, vol.

7, no. 13, 218. [ISSN 1336-7242]

41. ČULEN, Martin and DOHNAL, Jiří and JAMPÍLEK, Josef and ŘEZÁČOVÁ, Anna. Dynamic Dissolution

Testing in R&D. Book of Abstracts: The 2nd

World Conference on Physico-Chemical Methods in Drug

Discovery and Development, Zadar, Croatia, September 18-22, 2011, p. 7 (OP-05).

42. BRYCHTOVÁ, Kateřina and JAMPÍLEK, Josef and DVOŘÁKOVÁ, Lenka and OPATŘILOVÁ, Radka

and DOHNAL, Jiří. Investigating Alkyl-6-(2,5-dioxopyrrolidin-1-yl)-2-(2-oxoazepan-1-yl)hexanoates as

Potential Transdermal Penetration Enhancers. Book of Abstracts: The 2nd

World Conference on Physico-

Chemical Methods in Drug Discovery and Development, Zadar, Croatia, September 18-22, 2011, p. 42 (PP-

02).

43. OKTÁBEC, Zbyněk and JAMPÍLEK, Josef and DOHNAL, Jiří and ČULEN, Martin and KRÁL, Vladimír.

Increasing of Drugs Water Solubility Using Pectines and Their Derivatives. Book of Abstracts: The 2nd

World Conference on Physico-Chemical Methods in Drug Discovery and Development, Zadar, Croatia,

September 18-22, 2011, p. 50 (PP-10).

44. JAMPÍLEK, Josef and VACULÍKOVÁ, Eliška and GRÜNWALDOVÁ, Veronika and KRÁL, Vladimír

and DOHNAL, Jiří. Pilot Investigation of Nanoparticles Preparation by Precipitation. Book of Abstracts:

The 48th

International Conference on Medicinal Chemistry (RICT 2012), Poitiers, France, July 4-6, 2012, p.

103 (NA-03).

45. ČULEN, Martin and ŘEZÁČOVÁ, Anna and JAMPÍLEK, Josef and DOHNAL, Jiří. Dynamic dissolution

using Golem apparatus – prediction of bioequivalence. Book of Abstracts: The XLIst Conference “Synthesis

and Analysis of Drugs”, Bratislava, Slovakia, September 10-12, 2012, Farm. Obzor 2012, vol. 81, no. 5-6,

79. [ISSN 0014-8172]

46. TENGLER, Jan and KAPUSTÍKOVÁ, Iva and BAĎO, Ondřej and RAČANSKÁ, Eva and JAMPÍLEK,

Josef and MOKRÝ, Petr and CSÖLLEI, Jozef Preparation and study of physico-chemical and biological

properties of new aryloxyaminopropanole derivatives. Book of Abstracts: The XLIst Conference “Synthesis

and Analysis of Drugs”, Bratislava, Slovakia, September 10-12, 2012, Farm. Obzor 2012, vol. 81, no. 5-6,

81-82. [ISSN 0014-8172]

47. GONĚC, Tomáš and CSÖLLEI, Jozef and MALÍK, Ivan and STOLAŘÍKOVÁ, Jiřina and COFFEY,

Aidan and JAMPÍLEK, Josef and WAISSER, Karel. Phenylcarbamate derivatives with arylpiperazine

fragment as antimycobacterial compounds. Book of Abstracts: The XLIst Conference “Synthesis and

Analysis of Drugs”, Bratislava, Slovakia, September 10-12, 2012, Farm. Obzor 2012, vol. 81, no. 5-6, 87.

[ISSN 0014-8172]

48. KOS, Jiří and GONĚC, Tomáš and PEREIRA, Diogo and CHAMBEL, Bárbara and NĚMČÍKOVÁ, Ivana

and MIKLASOVÁ, Hana and JAMPÍLEK, Josef. Synthesis of amides of hydroxynaphthalene acids as

biologically active compounds. Book of Abstracts: The XLIst Conference “Synthesis and Analysis of

Drugs”, Bratislava, Slovakia, September 10-12, 2012, Farm. Obzor 2012, vol. 81, no. 5-6, 88. [ISSN 0014-

8172]

49. DVOŘÁKOVÁ, Lenka and COUFAL, Libor and OPATŘILOVÁ, Radka and JAMPÍLEK, Josef.

Influencing penetration of corticoids through membranes using substance ALA. Book of Abstracts: The

XLIst Conference “Synthesis and Analysis of Drugs”, Bratislava, Slovakia, September 10-12, 2012, Farm.

Obzor 2012, vol. 81, no. 5-6, 99. [ISSN 0014-8172]

50. FAJKUSOVÁ, Dagmar and PEŠKO, Matúš and KRÁĽOVÁ, Katarína and VEJSOVÁ, Marcela and

KELTOŠOVÁ, Stanislava and GUO, Jiahui and OKTÁBEC, Zbyněk and KOLLÁR, Peter and COFFEY,

Aidan and CSÖLLEI, Jozef and JAMPÍLEK, Josef. Herbicidal and anti-infective activity of substituted 2-

aminobenzothiazoles. Book of Abstracts: The XLIst Conference “Synthesis and Analysis of Drugs”,

Bratislava, Slovakia, September 10-12, 2012, Farm. Obzor 2012, vol. 81, no. 5-6, 100. [ISSN 0014-8172]

51. ZITKO, Jan and DUFKOVÁ, Ida and PATEROVÁ, Pavla and JAMPÍLEK, Josef and KUBÍČEK,

Vladimír and DOLEŽAL, Martin. Preparation, antimycobacterial and other biological effects of

benzylamino derivatives of pyrazinamide. Book of Abstracts: The XLIst Conference “Synthesis and

Analysis of Drugs”, Bratislava, Slovakia, September 10-12, 2012, Farm. Obzor 2012, vol. 81, no. 5-6, 127.

[ISSN 0014-8172]

52. ZADRAŽILOVÁ, Iveta and PAUK, Karel and MASAŘÍKOVÁ, Martina and IMRAMOVSKÝ, Aleš and

ČÍŽEK, Alois and JAMPÍLEK, Josef. Antibacterial activity of salicylanilide esters against methicillin-

resistant Staphylococcus aureus (MRSA). Book of Abstracts: The IInd

International Conference on

Antimicrobial Research (ICAR 2012), Lisbon, Portugal, November 21-23, 2012, p. 481.

52

53. ZADRAŽILOVÁ, Iveta and KOS, Jiří and POKORNÁ, Michaela and GONĚC, Tomáš and BOBÁL, Pavel

and ČÍŽEK, Alois and JAMPÍLEK, Josef. In vitro antimycobacterial activity of ring-substituted 3-

hydroxynaphthalene-2-carboxanilides. Book of Abstracts: The IInd

International Conference on

Antimicrobial Research (ICAR 2012), Lisbon, Portugal, November 21-23, 2012, p. 510.

54. ŽEMLIČKA, Milan and OPATŘILOVÁ, Radka and DOHNAL, Jiří and JAMPÍLEK, Josef. Internal

differentiation of study, profiling of student according to choice of compulsory optional courses. Book of

Abstracts: The 19th

Annual Conference of the European Association of Faculties of Pharmacy (EAFP

2013), Ankara, Turkey, May 16-18, 2013, p. 106 (P-33).


MASAŘÍKOVÁ, Martina and ČÍŽEK, Alois and JAMPÍLEK, Josef. In vitro anti-MRSA activity of 2-

hydroxy-N-[1-(2-hydroxyphenylamino)-1-oxoalkan-2-yl]benzamides? Book of Abstracts: Antimicrobial

Drug Conference, STARS EC FP7 Initial Training Network & TRAIN-ASAP ITN, Madrid, Spain, June

10-12, 2013, p. 70 (PO 19).

56. KOS, Jiří and GONĚC, Tomáš and JAMPÍLEK, Josef. Investigating the Spectrum of Biological Activity of

Ring-Substituted 3-Hydroxynaphthalene-2-carboxanilides. Book of Abstracts: The 49th

International

Conference on Medicinal Chemistry (RICT 2013), Nice, France, July 3-5, 2013, p. 229 (HT-053).

57. ORAVEC, Michal and JAMPÍLEK, Josef and ZÁRUBA, Kamil and OPATŘILOVÁ, Radka and SUCHÝ,

Pavel. Determination of Drugs in Silica Gel-Based Nanocarriers in Tissues. Book of Abstracts: The XVIIth

euroANALYSIS, Warsaw, Poland, August 25–29, 2013, p. 183. [ISBN 978-83-7798-089-7]

58. ČERNÍKOVÁ, Aneta and COUFALOVÁ, Lenka and OPATŘILOVÁ, Radka and DOHNAL, Jiří and

JAMPÍLEK, Josef. Evaluation of Alaptide as a Potential Modifier of Transdermal Penetration of

Antimicrobial Agents. Book of Abstracts: The 9th

Balaton Symposium on High-Performance Separation

Methods, Siófok, Hungary, September 4-6, 2013, p. 15 (L-13).

59. JAMPÍLEK, Josef and OPATŘILOVÁ, Radka and ČERNÍKOVÁ, Aneta and COUFALOVÁ, Lenka and

DOHNAL, Jiří. In vitro evaluation of penetration of nanonized alaptide from semi-solid formulations. Book

of Abstracts: The 3rd

World Conference on Physico-Chemical Methods in Drug Discovery and

Development, Dubrovnik, Croatia, September 22-26, 2013, p. 48 (PP-10).

60. PĚNTÁKOVÁ, Monika and MUSIOŁ, Robert and POLAŃSKI, Jarosław and JAMPÍLEK, Josef.

Molecular Dynamics of the Newly Designed Inhibitors EGRF. Book of Abstracts: The BIT′s 4th

Annual

International Congress of Medichem 2013 (ICM-2013), Haikou, China, November 13-16, 2013, p. 94.

61. DOHNAL, Jiří and COUFALOVÁ, Lenka and ČERNÍKOVÁ, Aneta and OPATŘILOVÁ, Radka and

JAMPÍLEK, Josef. Alaptide as Transdermal Penetration Modifier. Book of Abstracts: The BIT′s 3rd

Annual

Symposium of Drug Delivery Systems 2013 (SDDS-2013), Haikou, China, November 13-16, 2013, p. 244.

62. FAJKUSOVÁ, Dagmar and PEŠKO, Matúš and KELTOŠOVÁ, Stanislava and GUO, Jiahui and

OKTÁBEC, Zbyněk and VEJSOVÁ, Marcela and KOLLÁR, Peter and COFFEY, Aidan and CSÖLLEI,

Jozef and KRÁĽOVÁ, Katarína and JAMPÍLEK, Josef. Synthesis and Biological Activities of Substituted

2-Aminobenzothiazoles. Book of Abstracts: The 16th

JCF-Frühjahrssymposium 2014, Friedrich-Schiller-

Universität Jena, Jena, Germany, March 26-29, p. 70 (P-4).

63. KELTOŠOVÁ, Stanislava and JAMPÍLEK, Josef and KOLLÁR, Peter. In Vitro Biological Evaluation of

New Potential Anticancer Drugs. Book of Abstracts: The 64th

Pharmacological days and the 24th Martin

Respiration Days, Martin, Slovakia, June 25-27, 2014, p. 40. [ISBN 978-80-89544-70-7]

64. GONĚC, Tomáš and ZADRAŽILOVÁ, Iveta and NEVIN, Eoghan and KOS, Jiří and COFFEY, Aidan and

JAMPÍLEK, Josef. Synthesis and Biological Activity of N-(alkoxyphenyl)-2-hydroxynaphthalene-1-

carboxamides. Book of Abstracts: The XLIIIrd

Conference “Synthesis and Analysis of Drugs”, Bratislava,

Slovakia, September 4-6, 2014, Farm. Obzor 2014, vol. 83, no. 8-9, 182. [ISSN 0014-8172]

65. ČERNÍKOVÁ, Aneta and JAMPÍLEK, Josef. Modification of Transdermal Penetration of Different Drugs

with Alaptide as Potential Enhancer. Book of Abstracts: The 7th Central European Conference "Chemistry

towards Biology", Katowice, Poland, September 9-12, 2014, p. P19.

66. JAMPÍLEK, Josef and ORAVEC, Michal and ZÁRUBA, Kamil and ULBRICH, Pavel and BABULA, Petr

and KUNEŠ, Martin and SUCHÝ, Pavel. Preparation and In Vivo Permeation of Drugs in Silica Gel-Based

Nanocarriers through Blood–Brain Barrier. Book of Abstracts: The 7th Central European Conference

"Chemistry towards Biology", Katowice, Poland, September 9-12, 2014, p. P21.

67. MALARZ, Joanna and KROMPIEC, Stanisław and PIETRASZUK, Cezary and JAMPÍLEK, Josef and

VEJSOVÁ, Marcela. Synthesis of trisubstituted isoxazoles and their biological properties. Book of

Abstracts: The 57th

Meeting of the Polish Chemical Society and the Society of Engineers and Technicians of

Chemical Industry, Częstochowa, Poland, September 14-18, 2014, p. 115 (S01-P121). [ISSN 978-83-

931072-6-1]

53


VINŠOVÁ, Jarmila and ČÍŽEK, Alois and JAMPÍLEK, Josef. Time-kill curve kinetics of 4-chloro-N-

{(2S)-1-[(3,4-dichlorophenyl)amino]-3-methyl-1-oxobutan-2-yl}-2-hydroxybenzamide against multidrug-

resistant clinical isolates of methicillin-resistant Staphylococcus aureus (MRSA). Book of Abstracts: The

3rd

International Conference on Antimicrobial Research (ICAR 2014), Madrid, Spain, October 1-3, 2014, p.

327 (T71).

69. DOHNAL, Jiří and ČERNÍKOVÁ, Aneta and OPATŘILOVÁ, Radka and JAMPÍLEK, Josef. Advances in

Investigation of Alaptide as Transdermal Permeation Modifier. Book of Abstracts: The BIT′s 4th

Annual

Symposium of Drug Delivery Systems 2014 (SDDS-2014), Suzhou, China, November 18-20, 2014, p. 66.


ČÍŽEK, Alois and JAMPÍLEK, Josef. Antibacterial Activity of Novel Salicylanildes Against Vancomycin-

resistant Enterococcus faecalis (VRE). Book of Abstracts: The 25th

European Congress of Clinical

Microbiology and Infectious Diseases (ECCMID 2015), Copenhagen, Denmark, April 25-28, 2015,

EV0211.

71. GONĚC, Tomáš and STRÁNÍK, Josef and KOS, Jiří and ORAVEC, Michal and JAMPÍLEK Josef.

Synthesis of Substituted 1-(Phenylcarbamoyl)naphthalen-2-yl Alkylcarbamates with Potential

Antimycobacterial Activity. Book of Abstracts: The 67th

International Conference of Chemical Societies,

Horný Smokovec, Slovakia, September 7-11, 2015, ChemZi 2015, vol. 11, no. 1, 144-145 (3Po09). [ISSN

1336-7242]

72. KOS, Jiří and GONĚC, Tomáš and NEVIN, Eoghan and COFFEY, Aidan and JAMPÍLEK Josef. Ring-

Substituted 8-Hydroxyquinoline-2-carboxanilides as Potential Antitubercular Agents. Book of Abstracts:

The 67th

International Conference of Chemical Societies, Horný Smokovec, Slovakia, September 7-11,

2015, ChemZi 2015, vol. 11, no. 1, 152 (3Po22). [ISSN 1336-7242]

AFH Abstrakty příspěvků z domácích vědeckých konferencí

1. DOLEŽAL, Martin and JAMPÍLEK, Josef and BUCHTA, Vladimír. Synthesis and Biological Evaluation

of 5-Aroylpyrazine-2-carboxylic Acid Derivatives. Book of Abstracts: The XXVIIIth

Conference "Synthesis

and Analysis of Drugs", Hradec Králové, Czech Republic, September 15-17, 1999, p. 40.

2. JAMPÍLEK, Josef and DOLEŽAL, Martin and DEIGNER, Hans-Peter. Sphingosine Preparation as

Potential Antineoplastics by Optimized Tkaczuk-Thornton Method. Book of Abstracts: The XXXth

Conference “Synthesis and Analysis of Drugs”, Brno, Czech Republic, September 17-19, 2001, p. 73.

[ISBN 80-7305-416-7]

3. JAMPÍLEK, Josef and DOLEŽAL, Martin and OSIČKA, Zdeněk and KUNEŠ, Jiří and BUCHTA,

Vladimír. Preparation and Antimycotic Activity of Thiazol-2-ylamide pyrazine-2-carboxylic acid

Derivatives. Book of Abstracts: The XXXIInd

Conference “Synthesis and Analysis of Drugs”, Velké

Karlovice, Czech Republic, September 16-19, 2003, p. 134. [ISBN 80-900306-5-3]

4. JUN, Daniel and JAMPÍLEK, Josef and DOLEŽAL, Martin and KUNEŠ, Jiří and HRDINA, Radomír and

OPLETAL, Lubomír. Antiplatelet Activity of Arylalkanoic Acid. Book of Abstracts: The XXXIInd

Conference “Synthesis and Analysis of Drugs”, Velké Karlovice, Czech Republic, September 16-19, 2003,

p. 135. [ISBN 80-900306-5-3]

5. OPLETALOVÁ, Veronika and POUR, Milan and KUNEŠ, Jiří and SILVA, Luís and BUCHTA, Vladimír

and JAMPÍLEK, Josef and RICHARDSON, Des Robert and KALINOWSKI, Danuta. Thiosemicarbazones

of Acetylpyrazines as Potential Drugs. Book of Abstracts: The 11th

Blue Danube Symposium on

Heterocyclic Chemistry, Brno, Czech Republic, August 28-September 1, 2005, PO-70. [ISBN 80-210-

3763-6]

6. IMRAMOVSKÝ, Aleš and VINŠOVÁ, Jarmila and POLANC, Slovenko and JAMPÍLEK Josef.

Hydrazone Derivatives of Some Antituberculotics. Book of Abstracts: The XXXIVth

Conference “Synthesis

and Analysis of Drugs”, Brno, Czech Republic, September 12-14, 2005, p. 68. [ISBN 80-7305-533-3]

7. DOLEŽEL, Jan and OPLETALOVÁ, Veronika and BUCHTA, Vladimír and SILVA, Luís and

JAMPÍLEK, Josef and DOHNAL, Jiří and RICHARDSON, Des Robert and KALINOWSKI, Danuta and

KRÁĽOVÁ, Katarína. Synthesis and Biological Evaluation of Thiazole Derivatives. Book of Abstracts:

The XXXVth

Conference “Synthesis and Analysis of Drugs”, Velké Karlovice, Czech Republic, September

12-15, 2006, p. 85. [ISBN 80-7305-566-X]

8. OPLETALOVÁ, Veronika and DOLEŽEL, Jan and KUNEŠ, Jiří and JAMPÍLEK, Josef and SILVA, Luís

and BUCHTA, Vladimír and ŠPANINGEROVÁ, Eliška and KEŠETOVIČOVÁ, Diana and VLČKOVÁ,

Martina. Antifungal Activity of Benzylidenerhodanines. Book of Abstracts: The XXXVth

Conference

“Synthesis and Analysis of Drugs”, Velké Karlovice, Czech Republic, September 12-15, 2006, p. 120.

[ISBN 80-7305-566-X]

54

9. DOHNAL, Jiří and HAVLÍČEK, Jaroslav and JAMPÍLEK, Josef and BRUSOVÁ, Hana. Pharmaceutical

Analysis in Solid State. Book of Abstracts: The XXXVIIIth

Conference “Synthesis and Analysis of Drugs”,

Hradec Králové, Czech Republic, September 14-16, 2009, p. 25-26 (L-2). [ISBN 978-80-7305-078-8]

10. JAMPÍLEK, Josef and DOLEŽAL, Martin and KEŠETOVIČOVÁ, Diana. Structure-lipophilicity

Relationships in Series of Methoxy Moiety Ring-substituted Pyrazinecarboxanilides. Book of Abstracts:

The XXXVIIIth

Conference “Synthesis and Analysis of Drugs”, Hradec Králové, Czech Republic,

September 14-16, 2009, p. 90 (P-28). [ISBN 978-80-7305-078-8]

11. SLABÁ, Barbora and PLAČEK, Lukáš and RIDVAN, Luděk and JAMPÍLEK, Josef. Identification of

Almotriptan Impurity Using HPLC-MS/MS and HR-MS. Book of Abstracts: The XXXVIIIth

Conference

“Synthesis and Analysis of Drugs”, Hradec Králové, Czech Republic, September 14-16, 2009, p. 141 (P-

79). [ISBN 978-80-7305-078-8]

12. DOHNAL, Jiří and HAVLÍČEK, Jaroslav and JAMPÍLEK, Josef and BRUSOVÁ, Hana and KREJČÍK,

Lukáš. Position of Thermal Methods in Pharmaceutical Analysis of Solid State. Book of Abstracts: The

32nd

International Czech and Slovak Calorimetric Meeting (Kalsem 2010), Lísek u Bystřice pod

Pernštejnem, Czech Republic, May 24-28, 2010, p. 77-78. [ISBN 978-80-7395-259-4]

13. JAMPÍLEK, Josef and OKTÁBEC, Zbyněk and DOHNAL, Jiří. NIR and its Application in Pharmacy.

Proceedings of lifelong learning lectures „Properties and Analysis of Solid Pharmaceutical Substances

2011“. Department of Solid State Chemistry, Faculty of Chemical Technology, Institute of Chemical

Technology Prague, Czech Republic, April 28-29, 2011.

14. IMRAMOVSKÝ, Aleš and ŠTĚPÁNKOVÁ, Šárka and MONREAL-FÉRRIZ, Juana and VINŠOVÁ,

Jarmila and VANČO, Ján and JAMPÍLEK, Josef. Salicylanilide Carbamates as Acetylcholinesterase

Inhibitors and Their Molecular Docking. Book of Abstracts: The 2nd

French-Czech Vltava Chemistry

Meeting, Pardubice, Czech Republic, August 30-31, 2011, p. 31. [ISBN 978-80-7395-412-3]

15. GONĚC, Tomáš and KRÁĽOVÁ, Katarína and JAMPÍLEK, Josef and PAVLACKÁ, Lenka. Synthesis of

Substituted 2-Naphthoylanilides as Potential Photosynthesis Inhibitors. Book of Abstracts: The XLth

International Conference “Synthesis and Analysis of Drugs”, Brno, Czech Republic, September 12-14,

2011, S-6. [ISBN 978-80-7305-593-6]

16. ČULEN, Martin and DOHNAL, Jiří and JAMPÍLEK, Josef and ŘEZÁČOVÁ, Anna. Example of Dynamic

Dissolution Testing Results Obtained with Golem Apparatus. Book of Abstracts: The XLth

International

Conference “ Synthesis and Analysis of Drugs ”, Brno, Czech Republic, September 12-14, 2011, P-11.

[ISBN 978-80-7305-593-6]

17. JAMPÍLEK, Josef and IMRAMOVSKÝ, Aleš and PEJCHAL, Vladimír and OKTÁBEC, Zbyněk.

RP-HPLC Determination of Hydrophobic Properties of Substituted Fluorobenzothiazole Derivatives. Book

of Abstracts: The XLth

International Conference “Synthesis and Analysis of Drugs”, Brno, Czech Republic,

September 12-14, 2011, P-32. [ISBN 978-80-7305-593-6]

18. KOS, Jiří and JAMPÍLEK, Josef and GONĚC, Tomáš and BOBÁL, Pavel. Synthesis of N-

Arylquinoxaline-2-carboxamides as Potential Antimicrobial Compounds. Book of Abstracts: The XLth

International Conference “ Synthesis and Analysis of Drugs ”, Brno, Czech Republic, September 12-14,

2011, P-42. [ISBN 978-80-7305-593-6]

19. OPATŘILOVÁ, Radka and BREZOVSKÁ, Monika, JAMPÍLEK, Josef. Study of Drug Penetration

through a Barier. Book of Abstracts: The XLth

International Conference “Synthesis and Analysis of Drugs”,

Brno, Czech Republic, September 12-14, 2011, P-61. [ISBN 978-80-7305-593-6]

20. ČULEN, Martin and DOHNAL, Jiří and ŘEZÁČOVÁ, Anna and JAMPÍLEK, Josef. Artificial Digestive

Tract – Golem. Book of Abstracts: Science and Research for Innovations (Part of net NINET realized with

financial support of the program EUPRO-OK08003 of the Ministry of Education of the Czech Republic),

Brno, Czech Republic, September 5, 2012, p. 12.

21. VACULÍKOVÁ, Eliška and PLACHÁ, Daniela and ČECH-BARABASZOVÁ, Karla and JAMPÍLEK,

Josef. Nanotechnologies in field of pharmacy. Book of Abstracts: The 3rd

International Nanomaterials and

Nanotechnology Meeting “NANO-Ostrava 2013”, Ostrava, Czech Republic, June 17-20, 2013, p. 61

(OP 12). [ISBN 978-80-7329-361-1]


POKORNÁ, Michaela and ČÍŽEK, Alois and JAMPÍLEK, Josef. In vitro antimycobacterial activity of new

synthesized salicylanilide esters. Book of Abstracts: The 26th

Congress of the Czechoslovak Society for

Microbiology, Brno, Czech Republic, June 24-26, 2013, p. 128. [ISBN 978-80-260-4507-6]

23. VACULÍKOVÁ, Eliška and PLACHÁ, Daniela and JAMPÍLEK, Josef. Permeation/Penetration of Drug

Nanoparticles through Skin and Their Potential Toxicity. Book of Abstracts: The 2nd

International

Symposium and Workshop on Environment and Health (ISEH 2013), Ostrava, Czech Republic, November

6-8, 2013, p. 19. [ISBN 978-80-248-3240-1]

55

24. ZADRAŽILOVÁ, Iveta and POSPÍŠILOVÁ, Šárka and PAUK, Karel and MASAŘÍKOVÁ, Martina and

IMRAMOVSKÝ, Aleš and HANUSEK, Jiří and ČÍŽEK, Alois and JAMPÍLEK, Josef. Analysis of

Bactericidal Effect of 4-Chloro-2-(4-chlorophenylcarbamoyl)phenyl Decylcarbamate against MRSA in

Dependence on Time and Concentration under Conditions in Vitro. Book of Abstracts: The XXIIIrd

Tomášek Days of Young Microbiologists 2014, Brno, Czech Republic, June 5-6, 2014, p. 39. [ISBN 978-

80-210-6508-6]

25. ČERNÍKOVÁ, Aneta and JAMPÍLEK, Josef. Evaluation of Alaptide as Potential Permeation Enhancer for

Transdermal Delivery of Model Drug Theophylline. Book of Abstracts: The 4th

Meeting of the Paul Ehrlich

MedChem Euro-PhD Network, Hradec Králové, Czech Republic, June 20-22, 2014, p. 40 (O-21).

26. VACULÍKOVÁ, Eliška and PLACHÁ, Daniela and JAMPÍLEK, Josef. Preparation of Risedronate

Nanoparticles for Permeability Improvement. Book of Abstracts: The 4th

Meeting of the Paul Ehrlich

MedChem Euro-PhD Network, Hradec Králové, Czech Republic, June 20-22, 2014, p. 41 (O-22).

27. VACULÍKOVÁ, Eliška and PLACHÁ, Daniela and PISARČÍK, Martin and PEIKERTOVÁ, Pavlína and

DĚDKOVÁ, Kateřina and JAMPÍLEK, Josef. Characterization of cimetidine nanoparticles for solubility

test. Book of Abstracts: The 4th

Nanomaterials and Nanotechnology Meeting (NanoOstrava 2015), Ostrava,

Czech Republic, May 18-21, 2015, p. 79. [ISBN 978-80-248-3745-1]

28. BÁBKOVÁ, Zuzana and POLÁŠKOVÁ, Alena and ADÁMIK, Matej and HELMA, Robert and KOS, Jiří

and GONĚC Tomáš and JAMPÍLEK, Josef and BRÁZDOVÁ, Marie. Study of Biological Activity of

Hydroxynaphthalene Carboxanilide Derivatives on Tumor Cell Lines. Book of Abstracts:

The 20th

Interdisciplinary Czech-Slovak Toxicology Conference (TOXCON 2015), Brno, Czech Republic,

May 27-29, 2015, p. 26. [ISBN 978-80-263-0933-8]

29. KELTOŠOVÁ, Stanislava and JAMPÍLEK, Josef and KOLLÁR, Peter. Evaluation of Effect of Newly

Synthesized Quinazolines on Proliferation and Cell Cycle of Human Tumor Cell Lines. Book of Abstracts:

The 20th

Interdisciplinary Czech-Slovak Toxicology Conference (TOXCON 2015), Brno, Czech Republic,

May 27-29, 2015, p. 74. [ISBN 978-80-263-0933-8]

30. ČERNÍKOVÁ, Aneta and BOBÁĽ, Pavel and JAMPÍLEK, Josef. Analogues of Alaptide and Their Effect

on the Penetration of Drugs. Book of Abstract: The XLIVth

Conference “Synthesis and Analysis of Drugs”,

Brno, Czech Republic, September 2-4, 2015, p. 46 (P07). [ISBN 978-80-7305-760-2]

31. GONĚC, Tomáš and KMEŤKO, Juraj and KOS, Jiří and POSPÍŠILOVÁ, Šárka and ZADRAŽILOVÁ,

Iveta and JAMPÍLEK Josef. Synthesis and Antimicrobial Activity of N-(halogenphenyl)-1-

hydroxynaphthalene-2-carboxamides. Book of Abstract: The XLIVth

Conference “Synthesis and Analysis of

Drugs”, Brno, Czech Republic, September 2-4, 2015, p. 57 (P16). [ISBN 978-80-7305-760-2]

32. JĘDRZEJOWSKA, Agnieszka and MATUSSEK, Marek and KOZIK, Violetta and BĄK, Andrzej and

ZADRAŽILOVÁ, Iveta and JAMPÍLEK Josef. Synthesis and Biological Properties of Chosen Symmetrical

Amides and Thioamides of Terephthalic Acid. Book of Abstract: The XLIVth

Conference “Synthesis and

Analysis of Drugs”, Brno, Czech Republic, September 2-4, 2015, p. 63 (P20). [ISBN 978-80-7305-760-2]

33. KOS, Jiří and GONĚC, Tomáš and ZADRAŽILOVÁ, Iveta and VALEŠOVÁ, Miroslava and

POSPÍŠILOVÁ, Šárka and SPACZYŃSKA, Ewelina and JAMPÍLEK Josef. Ring-Substituted 1-

Hydroxynaphthalene-2-Carboxanilides as Potential Antibacterial Agents. Book of Abstract: The XLIVth

Conference “Synthesis and Analysis of Drugs”, Brno, Czech Republic, September 2-4, 2015, p. 72 (P27).

[ISBN 978-80-7305-760-2]

34. KAUEROVÁ, Tereza and GONĚC, Tomáš and KOS, Jiří and JAMPÍLEK Josef and KOLLÁR, Peter. In

Vitro Analysis of Antiproliferative Effects of Newly Synthesized Nitro-substituted Hydroxynaphthanilides

with Focus on Cell Cycle of Tumor Cell Lines. Book of Abstracts: The 65th

Pharmacological Days, Prague,

Czech Republic, September 16-18, 2015, p. 31. [ISBN 978-80-260-8027-5]

35. GONĚC, Tomáš and KOS, Jiří and ZADRAŽILOVÁ, Iveta and POSPÍŠILOVÁ, Šárka and ŠORAL,

Michal and LIPTAJ, Tibor and JAMPÍLEK Josef. Synthesis and Antibacterial Activity of N-(substituted

phenyl)-1-hydroxynaphthalene-2-carboxamides. Book of Abstracts: LIBLICE 2015 – The 50th

Conference:

“Advances in Organic, Bioorganic and Pharmaceutical Chemistry”, Olomouc, Czech Republic, November

6-8, 2015, p. 72 (Po20).

Výzkumné projekty obhájené nebo řešené (celkem 15 projektů)

1. Člen řešitelského kolektivu. HARTL, Jiří. „Biologicky aktivní deriváty pyrazinu a pyridinu“. Grantová

agentura Univerzity Karlovy (GAUK 026/1998/B-CH/FaF) v letech 1998–2000.

2. Člen řešitelského kolektivu. KARLÍČEK, Rolf. „Vývoj, příprava a technologie léčiv“. Výzkumné záměry

Ministerstva školství, mládeže a tělovýchovy České republiky (MSM 111600001) v letech 1999–2004.

56

3. Člen řešitelského kolektivu. KVASNIČKOVÁ, Eva. „Centrum pro výzkum struktury a mechanismu účinku

potenciálních léčiv B5“. Ministerstvo školství, mládeže a tělovýchovy České republiky (LN00B125)

v letech 2000–2004.

4. JAMPÍLEK, Josef. „Dokončení přípravy série potenciálních antituberkulotik a antimykotik“. Fond

rozvoje vysokých škol 2002 G4a – Tvůrčí činnost studentů – přírodovědné obory (FRVŠ 2245/G4/2002).

5. JAMPÍLEK, Josef. „Pokračování přípravy potenciálně účinných antituberkulotik a antimykotik“. Fond

rozvoje vysokých škol 2003 G6a – Tvůrčí činnost studentů – přírodovědné obory (FRVŠ 2998/G6/2003).

6. CHLUPÁČOVÁ, Marta a JAMPÍLEK, Josef. „Chalkony a jejich analoga jako potenciální léčiva“. Fond

rozvoje vysokých škol 2003 G3a – Tvůrčí činnost studentů – biomedicínské obory (FRVŠ 2970/G3/2003).

7. JAMPÍLEK, Josef. „Cílený transport léčiva přes biologické membrány“. Grantová agentura České

republiky (GAČR P304/11/2246) v letech 2011–2014.

8. KOS, Jiří a JAMPÍLEK, Josef. „Syntéza amidů kyselin hydroxynaftoových jako biologicky aktivních

látek“. Interní grantová agentura Veterinární a farmaceutické univerzity Brno (IGA VFU Brno

96/2012/FaF) v roce 2012.

9. Člen řešitelského kolektivu. SEDMÍKOVÁ, Markéta a SALAŠOVÁ, Alena a VEČEREK, Vladimír.

Centralizovaný rozvojový projekt Ministerstva školství, mládeže a tělovýchovy České republiky 2014

„Zvyšování kvalifikace studentů doktorských studijních programů a post-doktorandů zemědělských

a veterinárních oborů zapojením do multidisciplinárních meziuniverzitních týmů.“ (MŠMT ČR, projekt

č. C3) v roce 2014.

10. JAMPÍLEK, Josef. „Syntéza amidů kyseliny kynureninové jako biologicky aktivních látek“. Interní

grantová agentura Veterinární a farmaceutické univerzity Brno (IGA VFU Brno 37/2014/FaF) v roce 2014.

11. ZADRAŽILOVÁ, Iveta a JAMPÍLEK, Josef. „Studium antimikrobiálních vlastností nově syntetizovaných

potenciálních chemoterapeutik“. Interní grantová agentura Veterinární a farmaceutické univerzity Brno

(IGA VFU Brno 52/2014/FaF) v roce 2014.

12. Člen řešitelského kolektivu. SOPUCH, Tomáš. „Matricové systémy pro hojení kožních defektů

pro humánní a veterinární použití“. Technologická agentura České republiky (TAČR TA04010065)

v letech 2014–2017.

13. ČERNÍKOVÁ, Aneta a JAMPÍLEK, Josef. „Hodnocení derivátů alaptidu jako potenciálních

modifikátorů transdermální penetrace“. Interní grantová agentura Veterinární a farmaceutické univerzity

Brno (IGA VFU Brno 302/2015/FaF) v roce 2015.

14. JAMPÍLEK, Josef. „Protiinvazivní aktivita nových antimikrobiálních chemoterapeutik“. Interní grantová

agentura Veterinární a farmaceutické univerzity Brno (IGA VFU Brno 304/2015/FaF) v roce 2015.

15. Member of research group. SOBCZAK-KUPIEC, Agnieszka. “Innovative Composite Biomaterials

Contained Bioactive Calcium Phosphates”. The National Centre for Research and Development, Warsaw,

Poland (LIDER/037/481/L-5/13/NCBR) in 2015.

Vyžádané přednášky na konferencích a workshopech (celkem 26 přednášek)

Vyžádané přednášky na vědeckých konferencích konaných v České republice

1. The 1st International Symposium and Workshop on Environment and Health (ISEH 2012), Ostrava, Czech

Republic, November 22-23, 2012. (Invited plenary lecture “Perspectives of Nanoparticles in Pharmacy”,

Book of Abstract: p. 44 [ISBN 978-80-248-2882-4]).

2. The 2nd

International Symposium and Workshop on Environment and Health (ISEH 2013), Ostrava, Czech

Republic, November 6–8, 2013. (Invited plenary lecture “Polymorphism and Its Influence to

Bioavailability”, Book of Abstract: pp. 20-21 [ISBN 978-80-248-3240-1]).

3. The 4th

Nanomaterials and Nanotechnology Meeting (NanoOstrava 2015), Ostrava, Czech Republic, May

18–21, 2015. (Invited lecture “Overcoming Blood-Brain Barrier Using Nanoparticles”, Book of Abstract:

p. 63 [ISBN 978-80-248-3745-1]).

4. The International Conference on Nanomedicine, Drug Delivery, and Tissue Engineering (NDDTE'16),

Prague, Czech Republic, April 1-2, 2016. (Invited keynote lecture “Nanoformulations of Antimicrobial

Chemotherapeutics”, Book of Abstracts: Keynote-2, http://nddte.com/keynote/#Prof.%20Josef%20Jampilek &

http://nddte.com/paper/Keynote%20-%20Dr.%20Jampilek.pdf).

Vyžádané přednášky na zahraničních vědeckých konferencích

1. The XXXV Symposium 'Chromatographic Methods of Investigating the Organic Compounds', Katowice –

Szczyrk, Poland, May 30–June 1, 2012. (Invited plenary lecture “Advances in Investigation of Hydrophilic

and Lipophilic Properties of Drugs”, Book of Abstract: OS-5).

http://nddte.com/keynote/#Prof.%20Josef%20Jampilek


57

2. The XXXVI Symposium 'Chromatographic Methods of Investigating the Organic Compounds', Katowice –

Szczyrk, Poland, June 5–7, 2013. (Invited plenary lecture “Pharmaceutical nanoparticles and methods of

their characterization”, Book of Abstract: OS-19).

3. The BIT′s 4th

Annual International Congress of Medichem 2013 (ICM-2013), Haikou, China, November

13–16, 2013. (Invited lecture “Design and Antimicrobial Screening of New Ring-substituted Quinoline

Analogues”, Book of Abstract: p. 62).

4. The XXXVII Symposium 'Chromatographic Methods of Investigating the Organic Compounds', Katowice –

Szczyrk, Poland, June 11–13, 2014. (Invited plenary lecture “Investigation of Cholic Acid Derivatives as

Transdermal Permeation Enhancers”, Book of Abstract: OS-18).

5. The 7th

Central European Conference 'Chemistry towards Biology, Katowice, Poland, September 9–12,

2014. (Invited lecture “Synthesis and Antimicrobial Activity of Hydroxy(aza)naphthalenecarboxamides”,

Book of Abstract: O5).

6. The VI Conversatory on Medicinal Chemistry, Lublin, Poland, September 18–20, 2014. (Invited lecture

“Synthesis and In Vitro Anti-trypanosomal Screening of Hydroxynaphthalene-2-carboxanilides”, Book of

Abstract: p. 24 (K5) [ISSN 978-83-63657-38-3]).

7. International Scientific-Practical Conference Pharmaceutical Education, Scientific and Manufacturing as a

Reference to the Strategy Kazakhstan-2020, Faculty of Pharmacy, South Kazakhstan State Pharmaceutical

Academy, Shymkent, Kazakhstan, October 23–24, 2014. (Invited opening lecture “Quality by Design: New

Approach to Development of Drugs and Assurance of Their Quality”).

8. International Scientific-Practical Conference Pharmaceutical Education, Scientific and Manufacturing as a

Reference to the Strategy Kazakhstan-2020, Faculty of Pharmacy, South Kazakhstan State Pharmaceutical

Academy, Shymkent, Kazakhstan, October 23–24, 2014. (Invited plenary lecture “Design, Synthesis and

Anti-staphylococcus Activity of Hydroxynaphthalenecarboxanilides”, Book of Abstract: Republican

Scientific Journal 2014, vol. 68, no. 3, 3–7 [ISSN 2306-6822]).

9. The BIT′s 5th

Annual International Congress of Medichem 2014 (ICM-2014), Suzhou, China, November

18–20, 2014. (Invited lecture “Recent Advances in Design of Potential Quinoxaline Anti-Infectives”, Book

of Abstract: p. 197).

10. The 13th

Ibn Sina International Conference on Pure and Applied Heterocyclic Chemistry, Hurghada, Egypt,

February 14–17, 2015. (Invited plenary lecture “Azanaphthalenes as Potential Antimycobacterial Agents”,

Book of Abstract: p. 8 (PL-06)).

11. The XXXVIII Symposium 'Chromatographic Methods of Investigating the Organic Compounds', Katowice –

Szczyrk, Poland, May 27–29, 2015. (Invited plenary lecture “Determination of Drugs Loaded to Silica

Nanoparticles in Brain Tissue”, Book of Abstract: OS-27).

12. The IX Joint Meeting in Medicinal Chemistry (JMMC 2015), Athens, Greece, June 7–10, 2015. (Invited

keynote lecture “Advances in Design of Potential Quinoline Antimycobacterial Agents”, Book of Abstract:

O6).

13. European Pharma Congress “Pharma Europe-2015”, Valencia, Spain, August 25-27, 2015. (Invited

lecture “Design, Synthesis and Investigation of Aryl Derivatives of Alaptide as Potential Transdermal

Permeation Enhancers”, Book of Abstract: J. Pharma. Care Health Sys. 2015, vol. 2, no. 4, 63. [ISSN

2376-0419]).

14. The 4th

World Conference on Physico-Chemical Methods in Drug Discovery and Development (PCMDDD-

4), Rovinj – Red Island, Croatia, September 21-24, 2015. (Invited lecture “In Vitro Evaluation of 8-

Substituted 6,9-diazaspiro[4.5]decan-7,10-diones as Skin Permeation Modifiers”, Book of Abstract: p. 10

(OP-08)).

15. The 24th

Annual Central European Conference (ECOpole’15), Jarnołtówek, Poland, October 14-17, 2015.

(Invited keynote lecture “Applications of nanoformulations in Agricultural Production and Their Potential

Impact on Food and Human Health” (http://ecopole.uni.opole.pl/index.php/invited-presentations).

Proceedings: Proceedings of ECOpole 2015 (PECO-2015), 2015, vol. 9, no. 2, 465-472. [ISSN 1898-

617X]

16. The BIT's 13th

Annual World Congress of International Drug Discovery Science & Technology, Therapy

and EXPO-2015 (IDDST 2015), Beijing, China, October 20-22, 2015. (Invited lecture “Design and

Antimicrobial Activity of Ring-Substituted Hydroxynaphthalenecarboxamides and Their Aza-Analogues”,

Book of Abstract: p. 109).

17. The BIT's 5th

Annual World Symposium of Drug Delivery System 2015 (SDDS-2015), Beijing, China,

October 20-22, 2015. (Invited lecture “Investigation of Alkyl Derivatives of Alaptide as Transdermal

Permeation Modifier”, Book of Abstract: p. 387).

http://ecopole.uni.opole.pl/index.php/invited-presentations

58

Vyžádané odborné přednášky na seminářích a workshopech

1. Zentiva Praha, Česká republika, 28. březen 2008 („Infračervená spektroskopie v blízké oblasti – NIR“,

přednáška v rámci přednáškového cyklu „Science Forum” v délce 2 akademických hodin).

2. Ústav chemie pevných látek, Fakulta chemické technologie, Vysoká škola chemicko-technologická

v Praze, 28.–29. duben 2011. („NIR a jeho využití ve farmacii“, přednáška v rámci kurzu celoživotního

vzdělávání „Vlastnosti a analýza pevných farmaceutických substancí 2011” v délce 3 akademických

hodin).

3. Státní ústav pro kontrolu léčiv (SÚKL), Praha, Česká republika, 19.–20. duben 2012. (“Polymorphism –

What It Say?”, přednáška v rámci vzdělávací akce „EU Assessors Training on Efficient and Effective

Quality Assessment“ v délce 3 akademických hodin).

4. Ústav analytické chemie, Akademie věd České republiky, Brno, 2. květen 2012. („Polymorfie léčiv

a metody jejího stanovení“, přednáška v rámci cyklu „Kulatý stůl“ v délce 3 akademických hodin).

5. Centrum výzkumu globální změny Akademie věd České republiky, Brno, 4. listopad 2014 (“Application of

Nanoparticles in Pharmacy – Overcoming BBB and Methods Analysis of Nanoparticles“, odborný seminář

v délce 3 akademických hodin).

Členství v redakčních radách (celkem 6)

Členství v redakčních radách (tuzemských)

1. Military Medical Science Letters [ISSN 0372-7025], Faculty of Military Health Sciences, University of

Defense, http://www.mmsl.cz/editorial-board (od roku 2011)

Členství v redakčních radách (zahraničních)

1. Journal of Bioequivalence & Bioavailability [ISSN 0975-0851], OMICS Group, http://www.omicsonline.

org/editorialboard-bioequivalence-bioavailability-open-access.php (od roku 2013)

2. ADMET & DMPK [ISSN 1848-7718], IAPC Publishing, http://pub.iapchem.org/ojs/index.php/admet/

about/editorialTeam (od roku 2014)

3. Open Pharmaceutical Sciences Journal [ISSN 1874-8449], Bentham Science Publishers,

http://benthamopen.com/PHARMSCI/editorial-board/ (od roku 2015)

4. ChemistrySelect [ISSN 2365-6549], Wiley-VCH, http://onlinelibrary.wiley.com/journal/10.1002/%28

ISSN%292365-6549/homepage/2766_edbd.html (od roku 2015)

5. Medicinal Chemistry [ISSN 1875-6638, IF2014 = 1.363], Bentham Science Publishers,

http://benthamscience.com/journals/medicinal-chemistry/editorial-board/#top (od roku 2015)

Redaktor speciálních čísel

1. Prodrugs: Pharmaceutical Design and Current Perspectives. Current Pharmaceutical Design 2011, vol. 17,

no. 32, http://benthamscience.com/journal/contents.php?journalID=cpd&issueID=7364. [ISSN 1381-6128,

IF2011 = 3.870]

2. Enhanced skin drug permeability: methodology, assessment and enhancement approaches. ADMET &

DMPK 2014, vol. 2, no. 4, http://pub.iapchem.org/ojs/index.php/admet/issue/view/26. [ISSN 1848-7718]

3. Modern Approaches to Quality Assurance of Drug Formulations. BioMed Research International 2015,

vol. 2015, http://www.hindawi.com/journals/bmri/si/970238/. [ISSN 2314-6133, IF2014 = 1.579]

4. Anti-Infective Drug Discovery Based on Diversified Plant Natural Compounds. Current Organic

Chemistry 2016, http://benthamscience.com/journal-files/special-issue-details/COC-SII20151116-01.pdf.

[ISSN 1875-5348, IF2014 = 2.157]

Členství v komisích výzkumných agentur a vědeckých výborech

1. Člen hodnotícího panelu P207 „Chemické a biochemické přeměny” Grantové agentury České republiky

(2015–2017), http://gacr.cz/poradni-organy/panely/

Členství ve vědeckých a odborných společnostech

1. Česká společnost chemická – sekce Organická, bioorganická a farmaceutická chemie (od roku 2002)

2. Česká farmaceutická společnost – sekce Syntetických léčiv (od roku 2002)

3. International Association of Physical Chemists (od roku 2014)

4. Working Group on New TB Drugs (od roku 2015)

http://www.mmsl.cz/editorial-board

http://pub.iapchem.org/ojs/index.php/admet/%0babout/editorialTeam

http://pub.iapchem.org/ojs/index.php/admet/%0babout/editorialTeam

http://benthamopen.com/PHARMSCI/editorial-board/

http://onlinelibrary.wiley.com/journal/10.1002/%28%0bISSN%292365-6549/homepage/2766_edbd.html

http://onlinelibrary.wiley.com/journal/10.1002/%28%0bISSN%292365-6549/homepage/2766_edbd.html

http://benthamscience.com/journals/medicinal-chemistry/editorial-board/#top

http://benthamscience.com/journal/contents.php?journalID=cpd&issueID=7364

http://pub.iapchem.org/ojs/index.php/admet/issue/view/26

http://www.hindawi.com/journals/bmri/si/970238/

http://benthamscience.com/journal-files/special-issue-details/COC-SII20151116-01.pdf

http://gacr.cz/poradni-organy/panely/

59

Vypracování posudků

Oponentské posudky na vědecké články (celkem 118 posuzovaných rukopisů)

1. Acta Chromatographica [ISSN 1233-2356, IF2014 = 0.577], Institute of Chemistry, University of Silesia,

Katowice, Poland 1×

2. ADMET & DMPK [ISSN 1848-7718], IAPC Publishing 1×

3. African Journal of Pharmacy and Pharmacology [ISSN 1996-0816], Academic Journals 1×

4. Anti-Cancer Agents in Medicinal Chemistry [ISSN 1871-5206, IF2014 = 2.469], Bentham Science Publishers

2×

5. Arabian Journal of Chemistry [ISSN 1878-5352, IF2014 = 2.725], Elsevier 2×

6. ASC Combinatorial Science [ISSN 2156-8952, IF2014 = 3.032], American Chemical Society 1×

7. Biochemistry and Biophysics Reports [ISSN 2405-5808], Elsevier 1×

8. Bioinorganic Chemistry and Applications [ISSN 1565-3633, IF2014 = 2.081], Hindawi Publishing

Corporation 1×

9. BioMed Research International [ISSN 2314-6133, IF2014 = 1.579], Hindawi Publishing Corporation 1×

10. Bioorganic & Medicinal Chemistry [ISSN 0968-0896, IF2014 = 2.793], Elsevier 8×

11. Bioorganic & Medicinal Chemistry Letters [ISSN 0960-894X, IF2014 = 2.420], Elsevier 4×

12. British Journal of Pharmaceutical Research [ISSN 2231-2919], Science Domain International 2×

13. Carbohydrate Polymers [ISSN 0144-8617, IF2014 = 4.074], Elsevier 1×

14. Central European Journal of Chemistry [ISSN 1895-1066, IF2013 = 1.329], Springer 3×

15. Chemical Biology & Drug Design [ISSN 1747-0277, IF2014 = 2.485], Wiley-Blackwell 1×

16. Chemical Engineering Journal [ISSN 1385-8947, IF2014 = 4.321], Elsevier 1×

17. Chemické listy [ISSN 0009-2770, IF2014 = 0.272], Czech Chemical Society 6×

18. ChemMedChem [ISSN 1860-7179, IF2014 = 2.968], Wiley-VCH 8×

19. Chemistry and Biodiversity [ISSN 1612-1880, IF2014 = 1.515], Wiley-VCH 1×

20. Chromatography Research International [ISSN 2090-3502], Hindawi Publishing Corporation 1×

21. Combinatorial Chemistry & High Throughput Screening [ISSN 1386-2073, IF2014 = 1.222], Bentham

Science Publishers 2×

22. Current Pharmaceutical Design [ISSN 1381-6128, IF2014 = 3.452], Bentham Science Publishers 3×

23. Current Organic Synthesis [ISSN 1570-1794, IF2014 = 2.117], Bentham Science Publishers 1×

24. Česká a Slovenská Farmacie [ISSN 1803-6597], Czech Medical Association of J.E. Purkyne 2×

25. European Journal of Medicinal Chemistry [ISSN 0223-5234, IF2014 = 3.447], Elsevier 9×

26. European Journal of Organic Chemistry [ISSN 1434-193X, IF2014 = 3.065], Wiley-VCH 2×

27. Expert Opinion on Drug Discovery [ISSN 1746-0441, IF2014 = 3.539], Informa Healthcare 1×

28. Frontiers in Life Science [ISSN 2155-3769, IF2014 = 0.294], Taylor & Francis 1×

29. International Journal of Medicinal Chemistry [ISSN 2090-2069], Hindawi Publishing Corporation 1×

30. International Journal of Pharmaceutics [ISSN 0378-5173, IF2014 = 3.650], Elsevier 1×

31. Journal of Applied Biomedicine [ISSN 1214-021X, IF2014 = 1.302], Elsevier 3×

32. Journal of Biochemical and Molecular Toxicology [ISSN 1095-6670, IF2014 = 1.925], Wiley-Blackwell

1×

33. Journal of Bioequivalence & Bioavailability [ISSN 0975-0851], OMICS Group 5×

34. Journal of Biomolecular Structure & Dynamics [ISSN 0739-1102, IF2014 = 2.919], Taylor & Francis 1×

35. Journal of the Brazilian Chemical Society [ISSN 0103-5053, IF2014 = 1.129], Sociedade Brasileira de

Química 2×

36. Journal of Microencapsulation [ISSN 0265-2048, IF2014 = 1.585], Informa Healthcare 2×

37. Journal of Molecular Structure [ISSN 0022-2860, IF2014 = 1.602], Elsevier 1×

38. Journal of Nanoscience and Nanotechnology [ISSN 1533-4880, IF2014 = 1.556], American Scientific

Publishers 1×

39. Letters in Drug Design & Discovery [ISSN 1570-1808, IF2014 = 0.770], Bentham Science Publishers 3×

40. Letters in Organic Chemistry [ISSN 1570-1786, IF2014 = 0.664], Bentham Science Publishers 2×

41. Medicinal Chemistry [ISSN 1573-4064, IF2014 = 1.363], Bentham Science Publishers 3×

42. Military Medical Science Letters [ISSN 0372-7025], Faculty of Military Health Sciences, University of

Defence 2×

43. Molecules [ISSN 1420-3049, IF2014 = 2.416], MDPI 7×

60

44. Monatshefte fur Chemie [ISSN 0026-9247, IF2014 = 1.222], Springer 4×

45. Pest Management Science [ISSN 1526-498X, IF2014 = 2.694], Wiley-VCH 1×

46. Pharmaceutical Research [ISSN 0724-8741, IF2014 = 3.420], Springer 2×

47. Steroids [ISSN 0039-128X, IF2014 = 2.639], Elsevier 7×

48. Tuberculosis [ISSN 1472-9792, IF2014 = 2.711], Elsevier 1×

Externí hodnotitel projektů (celkem 65 grantových projektů)

1. Interní grantová agentura Veterinární a farmaceutické univerzity Brno (2010–2011) 6×

2. South African Medical Research Council (2010–2011) 2×

3. Technologická agentura České republiky (2010–2013) 18×

4. Interní grantová agentura Ministrstva zdravotnictví České republiky (2011–2013) 2×

5. Agentúra na podporu výskumu a vývoja Slovenské republiky (2012, 2015, 2016) 5×

6. Fulbright Visiting Scholar Program (2014–2015) 1×

7. Hungarian Scientific Research Fund (2014–2015) 3×

8. Grantová agentura České republiky (2015, 2016) 25×

9. Vedecká grantová agentúra MŠ SR a SAV (2015) 2×

10. Polish National Centre for Research and Development (2015) 1×

Člen hodnotící komise

1. Člen finálové výběrové poroty Ceny za nejlepší výzkumnou práci ve farmaceutických vědách 2010 „Ceny

za farmacii 2010“ udílenou Francouzským velvyslanectvím v České republice a společností Sanofi-

Aventis, 17. červen 2010.

2. Člen finálové výběrové poroty (chemická sekce) „Nadnárodního kola studentské vědecké konference“

Praha, České republika, 12. květen 2015.

Organizování vědeckých konferencí (celkem 15)

Člen organizačního výboru konferencí konaných v České republice

1. The XXXVIIth

conference "Synthesis and Analysis of Drugs", Brno 2008

2. The XLth


3. The 4th

Nanomaterials and Nanotechnology Meeting "NanoOstrava 2015", Ostrava, 2015

4. The XLIVth


Člen vědeckého výboru konferencí konaných v České republice

1. The 1st International Symposium and Workshop on Environment and Health, Ostrava, Czech Republic,

2012

2. The 2nd

International Symposium and Workshop on Environment and Health, Ostrava, Czech Republic,

2013

3. International Conference on Nanomedicine, Drug Delivery, and Tissue Engineering, Prague, Czech

Republic, 2016

4. World Congress on Recent Advances in Nanotechnology (Chair of the Congress,

http://rancongress.com/chair/), Prague, Czech Republic, 2016

Člen vědeckého výboru zahraničních konferencí

1. The XXXV Symposium "Chromatographic Methods of Investigating the Organic Compounds", Katowice

– Szczyrk, Poland, 2012

2. The XXXVI Symposium "Chromatographic Methods of Investigating the Organic Compounds", Katowice

– Szczyrk, Poland, 2013

3. The XXXVII Symposium "Chromatographic Methods of Investigating the Organic Compounds",

Katowice – Szczyrk, Poland, 2014

4. The 7th

Central European Conference "Chemistry towards Biology", Katowice, Poland, 2014

5. The XXXVIII Symposium "Chromatographic Methods of Investigating the Organic Compounds",

Katowice – Szczyrk, Poland, 2015

6. The 4th

World Conference on Physico-Chemical Methods in Drug Discovery and Development, Rovinj –

Red Island, Croatia, 2015

7. The 5th

IAPC Meeting “Emerging Technologies in Drug Discovery and Development”, Macau, China, 2016

(https://www.iapchem.org/page.php?page_id=73)

http://rancongress.com/chair/

https://www.iapchem.org/page.php?page_id=73

61

Ocenění za vědecko-výzkumnou činnost (celkem 5)

Vědecká ocenění

1. „PRIX DE PHARMACIE 2004” – 2. místo v celostátní soutěži „Cena za farmacii 2004” vyhlášené

společností Aventis Pharma s.r.o., Praha, Česká republika. Uděleno: 11. červen 2004.

Téma práce: „Quinlukast Analogues as Potential Antileukotrienic Agents: Synthesis and Study of

Biological Properties”.

2. „MOST CITED PAPER 2006–2009 AWARD“ udělena časopisem Bioorganic & Medicinal Chemistry, Elsevier

BV, Amsterodam, Nizozemí za článek publikovaný v BMC 2006, 14 (10): 3592-3598.

3. „2011 INDUSTRIAL AFFAIRS INNOVATION AWARD – TECHNOLOGY AND PROCESSES“ uděleno 1. místo

v rámci Sanofi-Aventis korporátního „3. ročníku Industrial Innovation Awards 2011“. Uděleno: 22. červen

2011.

Téma práce: „Artificial Digestive System GOLEM” (Reg. No. 2011TI-00082).

Ostatní ocenění

1. „OCENĚNÍ A PODĚKOVÁNÍ ZA DOSAVADNÍ SPOLUPRÁCI“ udělené děkanem Farmaceutické fakulty VFU Brno

formou plakety při příležitosti 20. výročí založení Farmaceutické fakulty v rámci Veterinární

a farmaceutické univerzity Brno. Uděleno: 14. září 2011.

2. „OUTSTANDING REVIEWER 2014–2015 AWARD“ uděleno vydavatelstvím Wiley-VCH dne 17.září 2015.

Spolupráce s praxí – aktivity v rámci aplikovaného výzkumu

V letech 2004–2011 byl pracovníkem R&D divize Zentiva Praha, konkrétně „Centra pro výzkum a metodický

rozvoj“, kde byl zodpovědný mimo jiné za vývoj/troubleshooting/portfolio care přípravků, resp. substancí, např.:

Lozap H, Lindaxa, Coxtral, atorvastatin, Torvacard, tolterodin, Uroflow, risedronát, Risendros, klopidogrel,

Trombex, levocetirizin, Zenaro, tibolon, Ladybon, kandesartan, Carzap, montelukast, Montelar, pregabalin,

topiramát. V rámci aplikovaného výzkumu byly rovněž zkoumány možnosti přípravy, stability a využití

kokrystalů a dalších krystalických, resp. amorfních forem substancí, např. agomelatin, aprepitant, risedronát,

ibandronát, imatinib, gefitinib, erlotinib, sunitinib, dasatinib, sorafenib, lapatinib. Ve spolupráci s Vývojovými

dílnami Ústavu organické chemie a biochemie AV ČR se podílel na vývoji unikátního přístroje pro dynamické

disoluce pojmenovaný „Golem“, který byl posléze patentován a za jehož přínos pro usnadnění vývoje

generických formulací v rámci celého korporátního R&D bylo celému týmu uděleno 1. místo v rámci

korporátního 3. ročníku „Industrial Innovation Awards 2011“ Sanofi-Aventis za projekt „Artificial Digestive

System GOLEM“. Dále se podílel na projektování laboratoří pro analýzu v pevné fázi, zaváděl metodiky NIR

a THz spektroskopie ve vývojových a QC laboratořích v rámci celé společnosti Zentiva. Na základě řešení výše

uvedených problematik je spoluautorem 15 patentů, resp. patentových přihlášek.

Od roku 2012 vykonává externí poradenskou, resp. školící činnost pro různé farmaceutické firmy v České

republice a Slovenské republice.

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Doklady o získaných oceněních

87

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Documents

Seznam vědeckých a publikačních aktivit, vyžádaných … · 2016-11-24 · Seznam vědeckých a publikačních aktivit, vyžádaných přednášek a grantů a další aktivity