Multi-membered N-heterocyclesR 0690 DOI: 10.1002/chin.201123164

Efficient and Novel One-Pot Synthesis of Antifungal Active 1-Substituted-8-aryl--3-alkyl/aryl-4H-pyrazolo[4,5-f][1,2,4]triazolo[4,3-b][1,2,4]triazepines Using Solid Support. — A simple, efficient and environmentally friendly procedure for the synthesis of title compounds (III) (10 examples) is developed. Compounds (IIIb)—(IIIe) show excellent efficacy against A. niger and Penicillium species. — (GUPTA*, M.; PAUL, S.; GUPTA, R.; Eur. J. Med. Chem. 46 (2011) 2, 631-635, http://dx.doi.org/10.1016/j.ejmech.2010.11.043 ; Dep. Chem., Univ. Jammu, Jammu 180 006, India; Eng.) — H. Haber

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