Upload
others
View
17
Download
0
Embed Size (px)
Citation preview
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 227
8. REFERENCES
Aanandhi MV, Mansoori MH, Shanmugapriya S, George S, Shanmugasundaram
P. Synthesis and in-vitro antioxidant activity of substituted pyridinyl 1,3,4-
oxadiazole derivatives. Res J Pharm Biol Chem Sci. 2010;1083-1090.
Abadi AH, Eissa AA, Hassan GS. Synthesis of novel 1,3,4-trisubstituted pyrazole
derivatives and their evaluation as antitumor and angiogenic agents. Chem Pharm
Bull. 2003;51:838-844.
Abdrabbo MK. NSAIDS associated GI-complications. Gastrointestinal
Endoscopy. 2005;3:49-52
Adamczak R, Porollo A, Meller J. Combining prediction of secondary structure
and solvent accessibility in proteins. Proteins. 2005;59:467-475.
Adelstein GW, Yen CH, Dajani EZ, Bianchi RG, 3,3-Diphenyl-3-(2-alkyl-1,3,4-
oxadiazol-5-yl)-propylcycloakylamines, a novel series of anti-diarrheal agents. J
Med Chem. 1976;19:1221-1225.
Ainsworth C. 1,3,4-Oxadiazole. J Am Chem Soc. 1965;87:5800-5801.
Alexandru TB, Padmakar VK, Aziz S. Comparison of topological indices based
on iterated sum versus product operations. Iran J Math Chem. 2010;1:43-67.
Ali MA and Yar MS. Oxadiazole Mannich bases: synthesis and antimycobacterial
activity, Bioorg Med Chem Lett. 2007;17:3314-3316.
Al-Omar MA. Synthesis and antimicrobial activity of new 5-(2-thienyl)-1,2,4-
triazoles and 5-(2-thienyl)-1,3,4-oxadiazoles and related derivatives. Molecules.
2010;15:502-514.
Amero CD, Byerly DW, McElroy CA, Simmons A, Foster MP. Ligand-induced
changes in the structure and dynamics of Escherichia Coli peptide deformylase.
Biochemistry. 2009;48:7595-7607.
Amir M and Kumar S. Synthesis and evaluation of anti-inflammatory, analgesic
and lipid peroxidation properties of ibuprofen derivatives. Acta Pharm.
2007;57:31-45.
Amir M and Shikha K. Synthesis and anti-inflammatory, analgesic, ulcerogenic
and lipid peroxidation activities of some new 2-[(2,6-dichloroanilino)
phenyl]acetic acid derivatives. Eur J Med Chem. 2004;39:535-545.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 228
Amir M, Javed SA and Kumar H. Synthesis of some newer analogues of 4-
hydroxyphenyl acetic acid as potent anti-inflammatory agents. J Chine Chem Soc.
2008;55:201-208.
Amir M, Javed SA, Kumar H. Synthesis of some novel 1,3,4-oxadiazole as
potential anti-inflammatory agents,. Indian J Chem. 2007;46:1014-1019.
Anand N. Burger’s medicinal chemistry, 4th
ed. Wiley-Interscience, New York;
1979.
Ananikov VS, Robert S, Keiji M, Musaev GD. Can steric effects induce the
mechanism switch in the rhodium-catalyzed imine boration reaction. A density
functional and ONIOM study. Organometallics. 2005;24:19-38.
Arumugam M, Muthuswamy U, Kuppusamy A, Thirumalaisamy S, Varadharajan
S. In silico docking studies of cyclooxygenase inhibitory activity of commercially
available flavonoids. Asian J Pharm Life Sci. 2012; 2:174
Atkinson AJ, Darrell RA, Danies CE, Dedrick RL, Markey SP. Principles of
clinical pharmacology, 2nd
ed., Elsevier, Book Aid International Sabre
Foundation, U.K; 2007.
Ausaf A, Husain A, Ajmal M, Ahuja P. Fenbufen based 3-[5-(substituted aryl)-
1,3,4-oxadiazol-2-yl]-1-(biphenyl-4-yl)propan-1-ones as safer anti-inflammatory
and analgesic agents. Eur J Med Chem. 2009;44:3798-3804.
Bakhle YS and Botting RM. Cyclooxygenase-2 and its regulation in
inflammation. Med Inflamm.1996; 5:305-323.
Bali A, Ohri R, Deb PK. Synthesis, evaluation and docking studies on 3-alkoxy-4-
methanesulfonamido acetophenone derivatives as non ulcerogenic anti-
inflammatory agents. Eur J Med Chem. 2012;49:397-405.
Bari SB, Aggarwal AO, Patil UK. Synthesis and pharmacological evaluation of
some novel isatin derivatives foe antimicrobial activity. J Sci Islam Repub Iran.
2008;19:217-221.
Bennett DL, Averill S, Priestley JV, McMahon SB. Postnatal changes in the
expression of TrkA high affinity NGF receptor in primary sensory neurons. Eur J
Neurosci. 1998;8:2204-2208
Bennett PN and Brown MJ. Clinical pharmacology, 10th
ed. Churchill
Livingstone, New York; 2009.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 229
Beydoun A and Backonja MM. Mechanistic stratification of antineuralgic agents.
J Pain Symptom Manage. 2003;25:18-30.
Bhandari SV, Bothara KG, Raut MK, Patil AA, Sarkate AP, Mokale VP. Design,
synthesis and evaluation of anti-inflammatory, analgesic and ulcerogenicity
studies of novel S-substituted phenacyl-1,3,4-oxadiazole-2-thiol and schiff bases
of diclofenac acid as nonulcerogenic derivatives. Bioorg Med Chem.
2008;16:1822-1831.
Bhardwaj N, Saraf SF, Sharma P and Kumar P. Synthesis, evaluation and
characterization of some 1, 3, 4-oxadiazoles as antimicrobial agents. E-J Chem.
2009;6:1133-1138.
Bhat MA, Al-Omar MA, Siddiqui N. Synthesis, anticonvulsant and neurotoxicity
of some novel 1,3,4-oxadiazole derivatives of phthalimide. Der Pharma Chemica.
2010;2:1-10.
Bhat MA, Siddiqui N, Khan SA. Synthesis of novel 3-(4-acetyl-5h/methyl-5-
substituted phenyl-4,5-dihydro-1,3,4-oxadiazol-2-yl)-2H-chromen-2-ones as
potential anticonvulsant agents. Acta Pol Pharm. 2008;65:235-239.
Bhatia NM, Mahadik KR, Bhatia MS. Exploring the influence of steric, electronic
and lipophilic descriptors of 1,3-diarylpropenones on their anti-inflammatory
activity. DARU. 2010;18:230-236.
Black JG. Growth and culturing the bacteria. Microbiology principle and
exploration. 4th
ed. New Jersey: Prentice Hall; 1999.
Bokoch GM. Chemoattractant signaling and leukocyte activation. Blood.
1995;86:1649-1660.
Borkotoky S. Docking studies on HIV integrase inhibitors based on potential
ligand binding sites. Int J Bioinformatics Biosciences.2012;2:21-29.
Bostrom J, Hogner A, Llins, Wellner E, Plowright AT, Oxadiazoles in medicinal
chemistry. J Med Chem. 2012;55:1817-1830.
Bray MA, Ford-Hutchinson AW, Smith MJ. In: SRA-A and Leukotrienes. Ed. P J
Piper. Research Studies Press, Chichester; 1981.
Bridges D, Thompson SW, Rice AS. Mechanisms of neuropathic pain. Brit J
Anaesth. 2001:87:12-26.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 230
Buttgereit F, Burmester G, Simon S. Gastrointestestinal toxic side effects of non-
steroidal anti-inflammatory drugs and cyclooxygenase-2-specific inhibitors. Am J
Med. 2001;110:135-195
Carlos TM and Harlan JM. Leukocyte-endothelial adhesion molecules. Blood.
1994;84:2068-2101.
Carol P. Essentials of pathophysiology: concepts of altered health states,
Hagerstown, Lippincott Williams & Wilkins; 2007.
Carrieri-Kohlman V, Lindsey AM, West CM. Pathophysiological phenomena in
nursing, 3rd
ed. St. Louis, MO: Saunders; 2003
Carter SJ. Basics of Microbiology, Cooper and Gunn’s Tutorial Pharmacy. 6th
ed.
CBS Publishers and Distributors; 2005.
Casimir CM and Teahan CG, The respiratory burst of neutrophils and its
deficiency. Immunopharmacology of neutrophils. Academic Press Limited,
London; 1994.
Chawla P, Maheshwari R, Saraf SA. Synthesis and evaluation of anti-
inflammatory and antimicrobial activity of 2,5-disubstituted-1,3,4-oxadiazoles.
Der Pharma Chemica. 2010;2:38-45.
Christopher JS, Yan Z, Carol M, Muhammad J, Isakson PC. Pharmacological
analysis of cyclooxygenase-1 in inflammation. Proc Natl Acad. Sci.
1998;95:13313-13318.
Chu CH, Sun XW, Zhang ZY, Li ZC, Liao RA. Synthesis and biological activities
of -heterocyclyl--(1H-1,2,4-triazol-1-yl)acetophenones. Chinese Chem Lett.
1999; 10:361-364.
Cioli V, Putzolu S, Rossi V, Barcellona PS, Corradino C. The role of direct tissue
contact in the production of gastrointestinal ulcers by anti-inflammatory drugs in
rats. Toxicol Appl Pharmacol. 1979;50:283-289.
Connolly ML. Solvent-accessible surface of proteins and nucleic acids. Science.
1983;221:709-713.
Cotran K and Collins R. Pathologic basis of disease. Philadelphia: W.B Saunders
Company, USA; 1998.
Dabiri M, Salehi P, Baghbanzadeh M, Bahramnejad M. A facile procedure for the
one-pot synthesis of unsymmetrical 2,5-disubstituted 1,3,4-oxadiazoles.
Tetrahedron Lett. 2006;47:6983-6986.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 231
Delves PJ, Roitt IM. The immune system. Engl J Med.2000;343:37-49.
Denmark SE, Weber T, David W, Piotrowski. Organocerium addition to SAMP-
Hydrazones: General synthesis of chiral amines. J Chem Soc. 1987;109:2224-
2225.
Deruiter J. Non-steroidal anti-inflammatory drugs (NSAIDS)-principles of drug
action. Fall; 2002;2:1–25.
Desai NC, Bhavsar AM, Shah MD, Saxena A. Synthesis and QSAR studies of
thiosemicarbazide,1,2,4-triazole, 1,3,4-thiadiazole derivatives as potential
antibacterial agents, Indian J Chem. 2008;47:579-589.
Doherty NS and Janusz MJ. Neutrophil proteases: their physiological and
pathological roles. Immunopharmacology of neutrophils. Academic Press
Limited, London; 1994.
Dormandy T. The worst of evils: man's fight against pain. New Haven, Conn:
Yale University Press; 2006.
Dravyakar BR. Kawade DP, Khedekar PB, Bhusari KP. Design and synthesis of
some new diphenylaminoisooxazolines as potent anti-inflammatory agent. Indian
J Chem. 2008;47:1559-1567.
Dworkin RH, Backonja M, Rowbotham MC, Allen RR, Argoff CR, Bennett.
Advances in neuropathic pain-diagnosis, mechanisms and treatment
recommendations. Arch Neuro. 2003;60:1524-1534.
Elkaim L, Grimaud, Jana LN, Tirla C, Nitrohydrazones: Versatile intermediates
for phosphonate derivatives formation from primary nitro compounds, Tetrahed
Lett. 2002;43:2037-2038.
El-Sayed WA, Ali OM, Hendy HA, Abdel-Rahman AA. Synthesis and
antimicrobial activity of new 2,5-disubstituted 1,3,4-oxadiazoles and 1,2,4
triazoles and their sugar derivatives. Chin J Chem. 2012;30:77-83.
El-Sayeda WA, El-Essawyb FA, Alib OM, Nasrb BS, Abdallac MM, Abdel-
Rahmanb A, Anti-HIV activity of new substituted 1,3,4-oxadiazole derivatives
and their acyclic nucleoside analogues. Z Naturforsch. 2009;64:773-778.
Ericsson H and Sherris JC. Antibiotic sensitivity testing report of an international
collaborative study. Acta Pathol Microbiol Scand. 1971;217:1-90.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 232
European commission health & consumer protection directorate-general
Directorate E-Food Safety: plant health, animal health and welfare, international
questions E1-Plant health, Oxadiargyl; 2002.
Ferwanah AR. Synthesis and x-ray crystal structure analysis of substituted-2,3-
dihydro-1,3,4-oxadiazoles via reaction of acetone- and cycloalkanone
benzoylhydrazones with phenylisocyanate. J Islam Univ Gaza. 2005;13:35-45.
Fine PG and Ashburn MA. Functional neuroanatomy and nociception. The
management of pain. Churchill Livingstone. New York; 1998.
Ford-Hutchinson AW, Bray MA, Doig MV, Shipley ME, Smith MJ. Leukotriene
B, a potent chemokinetic and aggregating substance released from
polymorphonuclear leukocytes. Nature. 1980;17:264-265.
Ford-Hutchinson AW. Leukotriene B4 and neutrophil function: a review. J R Soc
Med. 1981;74: 831-833.
Frank PV, Girish KS, Kalluraya B. Solvent-free microwave-assisted synthesis of
oxadiazoles containing imidazole moiety. J Chem Sci. 2007;119:41-46.
Franski R. Biological activities of the compounds bearing 1,3,4-oxa(thia)diazole
ring. Asian J Chem. 2005;17:2063-2075.
Fuloria NK, Singh V, Shaharyar M, Ali M. Synthesis and antimicrobial evaluation
of some new oxadiazoles derived from phenylpropionohydrazides. Molecules.
2009:14:1898-1903.
Gaonkar SL, Rai KM, Prabhuswamy B. Synthesis and antimicrobial studies of a
new series of 2-4-[2-(5-ethylpyridin-2-yl)ethoxy]phenyl-5-substituted-1,3,4-
oxadiazoles. Eur J Med Chem. 2006;41:841-846.
Gaud RS and Gupta GD. Practical microbiology. 5th
ed. Nirali Prakashan; 2006.
Gauto DF, Carlos M, Dumas VG, Lucia A, Bustamante JP, Turjanski AG, Marti
MA. Determining free energies of protein-ligand binding and
association/dissociation processes using computer simulations. World Res J
peptide protein. 2012;1:21-32.
Geronikaki AA, Lagunin AA, Hadjipavlou-Litina DI, Eleftheriou PT, Filimonov
DA, Poroikov VV, Alam I, Saxena AK. Computer-aided discovery of anti-
inflammatory thiazolidinones with dual cyclooxygenase/lipoxygenase Inhibition. J
Med Chem. 2008;51:1601-160.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 233
Gilroy DW, Colville-Nash PR, Willis D, Chivers J. Clark MJP, Willoughby DJ.
Inducible cyclooxygenase may have anti-inflammatory properties. Nature Med.
1999;5:698-701.
Giugliano D, Marfella R, Coppola L. Vascular effects of acute hyperglycemia in
humans are reversed by L-arginine. Evidence for reduced availability of nitric
oxide during hyperglycemia.Circulation. 1997;95:783-790.
Goodman and Gillman. Manual of pharmacology and therapeutics. McGraw Hill,
NewDelhi; 2007.
Goodman and Gilman’s. The pharmacological basis of therapeutics, 11th
ed.
McGraw Hill; 2008.
Granger DN and Kubes P. The microcirculation and inflammation: modulation of
leukocyte-endothelial cell adhesions. J Leukoc Biol. 1994;55:662-675.
Gudasi K, Patil M, Vadavi R, Shenoy R, Patil S. Transition metal complexes with
a new tridentate ligand, 5-[6-(5-mercapto- 1,3,4-oxadiazol-2-yl)pyridin-2-yl]-
1,3,4-oxadiazole-2-thiol. J Serb Chem Soc. 2007;72:357–366.
Gupta RR, Kumar M, Gupta V. Five membered heterocycles. Heterocyclic Chem.
1st ed. India: Springer; 2005.
Halperin I, Ma B, Wolfson H, Nussinov R. Principles of docking: an overview of
search algorithms and a guide to scoring functions. Proteins. 2002;4:409-443.
Han WS, Lee JK, Lee JS, Hahn HG, Yoon CN. Study of thiazoline derivatives for
the design of optimal fungicidal compounds using multiple linear regressions
(MLR). Bull Korean Chem Soc. 2012;33:1703-1706.
Hansch LA, Elkins D. Partition coefficients and their uses. Chem Rev.
1971;71:525-616.
Harfenist M, Heuser DJ, Joyner CT, Batchelor JF, White HL. Selective inhibitors
of monoamine oxidase structure activity relationship of tricyclics bearing
imidazoline, oxadiazole or tetrazole groups. J Med. Chem. 1996;39:1857-1863.
Harry WS, Paul JV, John JL. Culturing Microorganism Microbes in action. A
Laboratory manual of Microbiology. 4th
ed. New York: WH Freeman and
Company; 1991.
Haslett C, Savill JS, Meagher L. The neutrophil. Curr Opin Immunol. 1989;2:10-
18.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 234
Haslett. C and Henson P. Resolution of inflammation. The molecular and cellular
biology of wound repair. Plenum Press, New York; 1996.
He D, Zhu Y, Yang Z, Hu A, Cao G. Synthesis, characterization and optical
properties of novel 2,5-bis[4-(2-(arylvinyl)phenyl]-1,3,4-oxadiazoles. Turk J
Chem. 2009;33:393-397.
Higgs GA, Salmon JA, Spayne JA. The inflammatory effects of hydroperoxy and
hydroxy acid products of arachidonate lipoxygenase in rabbit skin. J. Pharmac.
1981;74:429-433.
Howard SS. Arachidonic acid pathway in nociception review. J Supp. Onco.
2006;6:267-276.
http://proteopedia.org/wiki/index.php/1g2a
http://proteopedia.org/wiki/index.php/1jxa
http://www.proteopedia.org/wiki/index.php/1cx2
Husain A and Mohammed A. Synthesis of novel 1,3,4-oxadiazole derivatives and
their biological properties. Acta pharm.2009;59:223-233.
Husain A, Ahmad FJ, Ajmal M and Ahuja P. Synthesis of 1-(4-phenoxyphenyl)-3-
[5-(substituted aryl)-1,3,4-oxadiazol-2-yl]propan-1-ones as safer anti-
inflammatory and analgesic agents. Eur J Med Chem. 2009; 44:3798-3804.
Husain A, Ahuja P, Sarafroj. Synthesis and biological evaluation of β-Aroyl
propionic acid based 1,3,4-oxadiazole. Indian J Pharm Sci. 2009;71:62-66.
Husain A, Sarafroz M, Ahuja P. 2-[3-(4-Chloro/ethyl phenyl)propan-3-one]-5-
(substituted phenyl)-1,3,4-oxadiazoles: synthesis and biological evaluation. Acta
Pol Pharm. 2008;65:527-534.
Husain MI, Kumar A, Srivastava RC. Synthesis of N-(2-naphthyloxyacetyl)-
thiosemicarbazides and 2-arylamino-5-(2-naphthyloxymethyl)-1,3,4-
thiadiazoles/oxadiazoles as oral hypoglycemic agents. Curr Sci. 1986;55:644-646.
Husain, M. S. Y. Khan, S. M. Hasan, M. M. Alam, 2-Arylidene-4-(4-phenoxy-
phenyl)but-3-en-4-olides: synthesis, reactions and biological activity, Eur J Med
Chem. 2005;40:1394-1404.
Hwang JY, Choi H, Lee D, Gong Y. Solid-phase synthesis of 1,3,4-oxadiazole
and 1,3,4-thiadiazole derivatives via selective, reagent-based cyclization of
acyldithiocarbazate resins. J Comb Chem. 2005;7:816-819.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 235
Inderba Indian drugs (Indian Drugs manufacturing association 102B Poonam
chambers, Dr. A. B. Rd., Worli, Bombay, India). 1982;19:301.
Indian Pharmacopoeia. Cotroller of publication, Govt. of India. Vol-I, Ghaziabad;
2007.
Jain N, Pathak DP, Mishra P, Jain S. Syntheses and antibacterial studies of some
2-[5-(aryl)-[1,3,4]oxadiazole-2-ylsulfanyl]alkanoic acids. J Iran Chem Soc.
2009;6:77-81.
Jakubkiene V, Burbuliene MM, Mekuskiene G, Udrenaite E, Gaidelis P,
Vainilavicius P. Synthesis and anti-inflammatory activity of 5-(6-methyl-2-
substituted-4-pyrimidyloxymethyl)-1,3,4-oxadiazole-2-thiones and their 3-
morpholinomethyl derivatives. Farmaco. 2003;58:323-328.
Jeffrey and George A. An introduction to hydrogen bonding, Oxford University
Press; 1997.
Jha KK, Samad A, Kumar Y, Shaharya M, Khosa RL, Jain J, Bansal S. 3D QSAR
studies of 1,3,4-oxadiazole derivatives as antimycobacterial agents. Iran J Pharm
Res. 2009;8:163-167.
Jin L, Chen J, Song B, Chen Z, Yang S, Li Q, Hu D, Xu R.Synyhesis, structure,
and bioactivity of N’-substituted benzylidene-3,4,5-trimethoxybenzohydrazide
and 3-acetyl-2-substituted phenyl-5-(3,4,5-trimethoxyphenyl)-2,3-dihydro-1,3,4-
oxadiazole derivatives. Bioorg Med Chem Lett. 2006;16:5036-5040.
Joyashis B, Kuldeep P, Prafull T, Karthikeyan C. Design, synthesis and
characterization of novel 1,3,4-oxadiazole dimers from benzoic acids. Int J Chem
Tech Res. 2010;2:2055-2062.
Kadi AA, El-Brollosy NR, Al-Deeb OA, Habib EE, Ibrahim TM, El-Emam AA.
Synthesis, antimicrobial, and anti-inflammatory activities of novel 2-(1-
adamantyl)-5-substituted-1,3,4-oxadiazoles and 2-(1-adamantylamino)-5-
substituted-1,3,4-thiadiazoles. Eur J Med Chem. 2007;42:235-242.
Kalemba D and Kunicka A. Antibacterial and antifungal properties of essential
oils. Curr Med Chem. 2003;10:813-829.
Kalgutkar AS, Crews BC, Rowlinson SW, Garner C, Seibert K, Marnett LJ.
Aspirin-like molecules that covalently inactive cyclooxygenase-2. Science.
1998;280:1268-1270.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 236
Kalgutkar AS, Marnett AB, Crews BC, Remmel RP. Ester and amide derivatives
of non-steroidal anti-inflammatory drug, indomethacin as selective COX-2
inhibitors. J Med Chem. 2000;43:2860-2870.
Kamble RR and Sudha BS. Synthesis and pharmacological screening 5-methyl-3-
[p-(6'-aryl-2'-thioxo-1',2',5',6'-tetrahydropyrimidin-4'-yl)-phenyl]-3h-2-oxo-δ4-
1,3,4-oxadiazole, Indian J Pharm Sci. 2006;68:249-253.
Katzung GB. Basic and clinical pharmacology. International 9th
ed., Mc Graw
Hill, New York; 2004.
Kaur H, Kumar S, Singh I and Kumar A. Synthesis, characterization and
antibacterial activity of various substituted oxadiazolylpyrazolinyl/isoxazolinyl
coumarin derivatives. Int J Pharm Sci Res. 2010;1:58-65.
Kaur H, Kumar S, Singh I, Saxena KK, Kumar A. Synthesis, characterization and
biological activity of various substituted benzothiazole derivatives. Digest journal
of Nanomaterial Biostructures. 2010;5:67-76.
Kawade DP, Khedekar PB, Bhusari KP. QSAR studies of 6-aminopyrimidin-4-
one derivatives as anti-inflammatory agent. Int J Pharm Biomed Res. 2011;2:13-
16.
Kay AB. Overview of allergy and allergic diseases: with a view to the future. Br
Med Bull. 2000;56:843-864.
Khan KM, Ullah Z, Rani M,. Perveen S, Haider SM, Choudhary MI, Rahman A,
Voelter W. Microwave-assisted synthesis of 2,5-disubstituted1,3,oxadiazoles. Lett
Org Chem. 2004;1:50-52.
Khan MS and Husain A. Syntheses and reactions of some new 2-arylidene-4-
(biphenyl-4-yl)-but-3-en-4-olides with a study of their biological activity.
Pharmazie. 2002;57:448-452.
Konstantinos A. Testing for tuberculosis. Australian Prescriber. 2010;33:12-18.
Koparır M, Cetin A, Cansiz A. 5-Furan-2yl[1,3,4]oxadiazole-2-thiol, 5-furan-2yl-
4H-[1,2,4]triazole-3-thiol and their thiol-thione tautomerism. Molecules.
2005;10:475-480.
Kramer VI and Schunack W. Synthesis and H2-antagonistic activity of N,N-
substituted 1,3,4-oxadiazole-2,5-diamines. Arzneim-Forsch. 1986;36:1564-1567.
Kubinyi H. Similarity and dissimilarity: a medicinal chemist’s view, in 3D QSAR
in Drug Design. Kluwer Academic Publishers, Dordrecht; 1998.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 237
Kudelko A and Zieliǹski W. Microwave-assisted synthesis of 2-styryl-1,3,4-
oxadiazoles from cinnamic acid hydrazide and triethyl orthoesters. Tetrahedron
Lett. 2012;53:76-77.
Kuhns DB, Priel DA, Gallin JI. Loss of L-selectin (CD62L) on human neutrophils
following exudation in vivo. Cell Immunol. 1995;164:306-310.
Kumar RS, Pradeepchandran RV, Jayaveera KN. Computer aided discovery of
benzimidazole derivatives on peptide deformylase as antimicrobial agent using
HEX. Eur J Chem. 2011;2:558‐560.
Kumar RS, Pradeepchandran RV, Jayaveera KN. Docking studies of
benzimidazole derivatives on peptide deformylase and heptosyltransferase waac
as antibacterial agent. Int J Pharma Res Innovation. 2011;4:1-5.
Kumar V, Abbas AK, Fausto N, Mitchell RN. Robbins Basic Pathology. 8th
ed.
Saunders Elsevier; 2007.
Lanza FL. A guideline for the treatment and prevention of NSAID- induced
ulcers. Am J Gastroenterol. 1998;93:2037-2046.
Lee B and Richards FM. The interpretation of protein structures, estimation of
static accessibility. J Mol Bio. 1971;55:379-400.
Lee CH and Cho HI. Synthesis of 1,3,4-oxadiazoles having phenol or thiophenol
group. Bull Korean Chem Soc. 2001;22:1153-1155.
Lennette EH, Balows A, Hausler WJ, Shadowmy HJ. Manual of clinical
microbiology. 4th
ed. American Society for Microbiology: Washington, D. C. 995;
1985
Levine JD and Taiwo YO. Involvement of the mu-opiate receptor in peripheral
analgesia. Neuroscience. 1984;32:571-575.
Levine JD, Taiwo TO, Collins SD, Tam JK. Noradrenaline hyperalgesia is
mediated through interaction with sympathetic postganglionic neurone terminals
rather than activation of primary afferent nociceptors. Nature. 1986;323:158-l60.
Lindner M, Sippl W, Radwan AA. Pharmacophore elucidation and molecular
docking studies on 5-phenyl-1-(3-pyridyl)-1h-1,2,4-triazole-3-carboxylic acid
derivatives as COX-2 inhibitors. Sci Pharm. 2010;78:195-214.
Ma W and Eisenach JC. Morphological and pharmacological evidence for the role
of peripheral prostaglandins in the pathogenesis of neuropathic pain. Eur J
Neurosci. 2003;15:1037-47.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 238
Macaev F, Rusu G, Pogrebnoi S, Gudima A, Stingaci E, Vlad L, Shvets N,
Kandemirli F, Dimoglo A, Reynolds R. Synthesis of novel 5-aryl-2-thio-1,3,4-
oxadiazoles and the study of their structure anti-mycobacterial activities, Bioorg
Med Chem. 2005;13:4842-4850.
Malmberg AB and Yaksh TL. Antinociceptive actions of spinal nonsteroidal anti-
inflammatory agents on the formalin test in the rat. J Pharmacol Exp Ther.
1992;263:136-146.
Martin YC, Kofron JL, Traphagen LM. Do structurally similar molecules have
similar biological activity?. J Med Chem; 2002; 45:4350-4358.
Masferrer JL, Seibert K, Zweifel B, Needleman P. Proc Natl Acad Sci. USA;
1992.
Max B and Wolf B. Principles of optics: electromagnetic theory of propagation,
interference and diffraction of light. 7th
ed. Cambridge University Press; 1999.
Mayekar AN. Synthesis and antimicrobial studies on new substituted 1,3,4-
oxadiazole derivatives bearing 6-bromonaphthalene moiety. Int J Chem.
2010;2:38-54.
Mazouz F, Guiddari S, Burstein C, Mansuy D, Milcent R. 5-[4-
(Benzyloxy)phenyl]-1,3,4-oxadiazol-2(3H)-one derivatives and related analogues:
New reversible, highly potent and selective monoamine oxidase type B inhibitors.
J Med Chem. 1993;36:1157–1167.
Mazouz F, Lebreton L, Milcent R, Burskin C. 5-Aryl-1,3,4-oxadiazol-2-(3H)-one
derivatives and sulfur analogues as new selective and competitive monoamine
oxidase type B inhibitors. Eur Med Chem. 1990;25:659-671.
Melo SJ, Sobral SD, Lopes HL, Srivastav RM. Synthesis of some 3-aryl-1,2,4-
oxadiazoles carrying a protected L-alanine side chain. J Braz Chem Soc.
1989;9:465-468.
Milewski S. Glucosamine-6-phosphate synthase-the multi-facets enzyme.
Biochimica Biophysica Acta. 2002;1597:173-192.
Misra U, Hitkari A, Saxena AK, Gurtu S, Shanker K. Biologically active
indolylmethyl-1,3,4-oxadiazoles, 1,3,4-thiadiazoles, 4H-1,3,4-triazoles and 1,2,4-
triazines. Eur J Med Chem. 1996;31:629-634.
Mohammed IA, Subrahmanyam EV, Hareesh AR, Kowti R. Synthesis,
antimicrobial studies of some Schiff bases and novel 5- aryl (8-
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 239
quinolinoxymethyl)-1,3,4-oxadiazoles derivatives. Int. J Pharm Sci Bio.
2010;2:80-85.
Mohan H. Textbook of pathology, 5th
ed., Jaypee Brothers Medical Publishers,
New Delhi, India; 2005.
Momen-Roknabadi A, Sadeghi M, Pezeshk H, Marashi SA. Impact of residue
accessible surface area on the prediction of protein secondary structures.
Bioinform. 2008;9:357.
Mullican MD, Wilson MW, Connor DT, Kostlan CR, Schrier DJ, Dyer RJ. Design
of 5-(3,5-di-tert-butyl-4-hydroxyphenyl)-1,3,4-thiadiazoles, -1,3,4-oxadiazoles
and -1,2,4-triazoles as orally-active, nonulcerogenic anti-inflammatory agents. J
Med Chem. 1993;36:1090-1099.
Musser G, Amori G, Hutterer R, Kryštufek B, Yigit N, Mitsain G. Mus Musculus.
In: IUCN Red List of Threatened Species; 2008.
Muthumani P, Meera R, Agarwal SB, Devi P, Kameswari B, Muthuppandi R.
Synthesis of some derivatives of pyrimidine, oxadiazole and indole in
combination by conventional and microwave method. Der Pharma Chemica.
2009;1:167-177.
Nagalakshmi G. Synthesis, antimicrobial and anti-inflammatory activity of 2,5-
disubstituted-1,3,4-oxadiazoles, Indian J Pharm Sci. 2008;70:49-55.
Naik TA and Chikhalia KH. Studies on synthesis of pyrimidine derivatives and
their pharmacological evaluation. E-J Chem. 2007;4:60-66.
Narayana B, Vijayaraj KK, Ashlatha B, Kumari NS. Synthesis of some new 2-(6-
methoxy-2-naphthyl)-5-aryl-1,3,4- oxadiazoles as possible non-steroidal anti-
inflammatory and analgesic agents. Arch Pharm. 2005;338:373-377.
Nathan C. Points of control in inflammation. Nature. 2002;420:846-852.
Nicholson B. Gabapentin use in neuropathic pain syndromes. Acta Neurol Scand.
2000;101:359-371.
Nigam R, Swarup S, Saxena VK, Singh HK, Synthesis and pharmacological
screening of some new 2-thio-3-(substituted-aminomethyl)-5-(3,5-dinitrophenyl)-
1,3,4-oxadiazoles. J Indian Chem Soc. 1992;69:692-693.
Nikolova N and Jaworska J. Approaches to measure chemical similarity-a review.
QSAR Comb Sci. 2003;22:1006-1026.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 240
Omar FA, Mahfouz NM, Rahman MA. Design, synthesis and anti-inflammatory
activity of some 1,3,4-oxadiazole derivatives. Eur J Med Chem. 1996;31:819-825.
Palomer A, Cabre F, Pascual J, Campos J. Identification of novel cyclooxygenase-
2 selective inhibitors using pharmacophore models. J Med Chem. 2002;45:1402-
1411.
Parakrama C and Taylor CR. General pathology, section II. The host response to
Injury, 3rd
ed. McGraw Hill, New York; 2005.
Parameswaran M, Thengungal KR, Gopalakrishnan S. Synthesis of coumarin
heterocyclic derivatives with antioxidant activity and in vitro cytotoxic activity
against tumour cells. Acta Pharm. 2009;59:159-170.
Parekh. J and Chanda S. In vitro antimicrobial activity of Trapa natans L. fruit
rind extracted in different solvents. Afr J Biotechnol. 2007;6:766-770.
Pasero C, Paice J, McCaffery M. Basic mechanisms underlying the causes and
effects of pain. 2nd
ed. St. Louis, MO: Mosby; 1999.
Patel NB and Patel JC. Synthesis and antimicrobial activity of 3-(1,3,4-oxadiazol-
2-yl)quinazolin-4(3H)-ones. Sci Pharm. 2010;78:171-193.
Patil UD, Nikum AP, Nagle PS, Mahulikar PP. Synthesis, antimicrobial and
antifungal activity evaluation of 2,6-diaryl-4-sec-aminonicotinonitrilesand 4-sec-
amino-6-aryl-2-(pyridin-yl)pyridine-3-carbonitriles i.e. bipyridines and their
docking study. J Pharm Res. 2012;5:1383-1386.
Pattan SR, Rabara PA, Pattan JS, Bukitagar AA, Wakale VS, Musmade DS.
Synthesis and evaluation of some novel substituted 1,3,4-oxadiazole and pyrazole
derivatives for antitubercular activity. Indian J Chem. 2009;48:1453-1456.
Portenoy RK and Kanner RM. Definition and assessment of pain. Pain
management: theory and practice. FA Davis Co. Philadelphia; 1996.
Pramanik SS and Mukherjee A. Synthesis and in-vitro serotonin-3-antagonist
activities of some new 1,3,4-oxadiazole-2-thiones. J Indian Chem Soc.
1998;75:53-54.
Prasanna S, Daga PR, Xie A, Doerksen RJ. Glycogen synthase kinase-3 inhibition
by 3-anilino-4-phenylmaleimides: insights from 3D-QSAR and docking. J
Comput Aided Mol Des. 2009;23:113-127.
Prescott LM, Harley JP, Klein DA. Microbial growth and metabolism.
Microbiology. 2nd
ed. England: Wm C Brown Publisher; 1990.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 241
Rajak H, Kharya DM, Mishra P. Synthesis of some novel oxadiazole and
oxadiazoline analogues for their anti-inflammatory activity, Yakuga Zasshi.
2007;127:1757-1764.
Rajasekaran S, Rao GK, Pai SP, Vedavathy J. Microwave assisted synthesis of
some 5-pyridyl-2-[(N-substituted phenyl) thioacetamido]-1,3,4-oxadiazoles as
antibacterial and antioxidant agents. J Chem Pharm Res. 2010;2:101-106.
Rakesh R, Somani A, Prabhakar Y, Shirodkar B. Oxadiazole: a biologically
important heterocycle. Der Pharma Chemica. 2009;1:130-140.
Ramalingam T, Deshmukh AA, Sattur PB. Synthesis and pharmacology of 2,5-
disubstituted-1,3,4-oxadiazoles. J Indian Chem Soc. 1981;58:269-271.
Ramazani A, Karimi Z, Souldozi A, Ahmadi Y. Four-component synthesis of
1,3,4-oxadiazole derivatives from N-isocyaniminotriphenylphosphorane, aromatic
carboxylic acids, aromatic bis-aldehydes, and secondary amines. Turk J Chem.
2012;36:81-91.
Ramazani A, Souldozib A. Iminophosphorane-mediated one-pot synthesis of
1,3,4-oxadiazole derivatives. Arkivoc. 2008;xvi:235-242.
Ramlingam T, Sattur PB. Synthesis and biological evaluation of α-(3-
pentadecylaryloxy)-propionic acids, their hydrazides and cyclic derivatives:
oxadiazoles and pyrroles. Indian Drugs. 1987;24:514–517.
Ravindra KC, Vagdevi HM, Vaidya VP, Basavaraj P. Synthesis, antimicrobial and
anti-inflammatory activities of 1,3,4-oxadiazole linked to naptho[2,1-b]furan.
Indian J Chem. 2006;45:2506-2511.
Red R, Homes D, Wayer J, Jone A. Sterile technique and microbial culture pour
plate technique. Practical skill in microbial culture pours plate technique. Practical
skill in biomolecular sciences. England:Addison Wesley Longman Limited; 1998.
Regina GL, Romano S, Valerio G, Antonio L, Ettore N, Olivia B, Paola T, Enzo
A. Synthesis, structure-activity relationships and molecular modeling studies of
new indole inhibitors of monoamine oxidases A and B. Bioorg Med Chem.
2008;22:9729-9740.
Regoli D, Drapeau G, Rovero P, Dion S, Orleans-Juste PD. The actions of
bradykinin antagonists on B1 and B2 receptor systems. Eur J Pharmacol.
1986;123:61-67.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 242
Rivera NR, Balsells J, Hansen KB. Synthesis of 2-amino-5-substituted-1,3,4-
oxadiazoles using 1,3-dibromo-5,5-dimethylhydantoin as oxidant. Tetrahedron
Lett. 2006;46:4889-4891.
Robins KC. Basic pathology. 6th
ed. Harcoure, Asia; 2001.
Saini R, Rai AK, Kesari A, Yar MS. Synthesis and biological evaluation of 2,5 di-
substituted 1,3,4-oxadiazoles. Asian j Research Chem. 2009;2:34-36.
Samuelsson B. Leukotrienes: mediators of immediate hypersensitivity reactions
and inflammation. Science. 1983;220:568-575.
Satoshkar RS, Bhandarkar SD, Rege NN. Pharmacology and
Pharmacotherapeutics, 20th
ed. Popular Prakashan, India; 2007.
Satyajit S and Lutfun N. Chemistry for pharmacy students: general, organic and
natural product chemistry. John Wiley & Sons; 2007
Sauers, Ronald R. Steric attraction: the far side. J Chem Edu. 1996;73:114.
Savariz FC, Formagio AS, Barbosa VA, Foglio MA, Carvalho JED, Duarte
MC, Filhoc BP, Sarragiotto MH. Synthesis, antitumor and antimicrobial activity
of novel 1-substituted phenyl-3-[3-alkylamino(methyl)-2-thioxo-1,3,4-oxadiazol-
5-yl]β-carboline derivatives. J Braz Chem Soc. 2010;21:288-298.
Selassie CD. History of quantitative structure activity relationships. Burger’s
Medicinal Chemistry and Drug Discovery. 6th
ed. John Wiley and Sons; 2003
Sengupta P, Mal M, Mandal S, Singh J, Maity TK. Evaluation of antibacterial and
antifungal activity of some 1,3,4-oxadiazoles. Iranian Journal of Pharmacology
and Therapeutics. 2008;7:165-167.
Seth SD. Text book of Pharmaology, 2nd
ed. Elsevier: A division of Reed Elsevier,
India; 2005.
Shaban MA, Nasr AZ, El-Badry SM. Synthesis and biological activities of some
1,3,4-oxadiazoles and bis(1,3,4-oxadiazoles). J Islam Acad Sci. 1991;4:184-191.
Shabani H, Ashrafi AR, Didea MV. Balaban index of an infinite class of
dendrimers, Croat Chem Acta. 2010; 83:439-442.
Shapiro R and Vallee BL. Interaction of human placental ribonuclease with
placental ribonuclease inhibitor. Biochem. 1991;30:2246–55.
Sharma MC, Kohli DV, Sahu NK, Sharma S, Chaturvedi SC. 2D-QSAR studies
of some 1,3,4-thiadiazole-2-yl azetidine-2-one as antimicrobial activity. Dig J
Nanomater Bios. 2009;4:339-347.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 243
Sharma S, Sharma PK, Kumar N, Dudhe R. A review: oxadiazole their chemistry
and pharmacological potentials. Der Pharma Chemica. 2010;2:253-263.
Shi W, Qian X, Song G, Zhang R, Li R. Synthesis and insecticidal activities of
novel 2-fluorophenyl-5-aryl/cyclopropyl-1,3,4-oxadiazoles. J Fluorine Chem.
2000;106:173-179.
Siddall PJ and Cousins MJ. Spine update: Spinal pain mechanisms. Spine.
1997;22:98-104.
Siddiqui AA, Islam M, Kumar S. Synthesis and antituberculostic activity of 5-{3’-
oxo-6’-(substituted phenyl)-2’,3’,4’,5’-tetrahydropyridazin-2’-yl}methyl-2-
substituted 1,3,4-oxadiazole. Der Pharmacia Lettre. 2010;2:319-327.
Silva CH and Taft CA. Molecular dynamics database screening, density functional
and docking studies of novel RAR ligand in cancer chemotherapy. Biophysical
Chem. 2005;117:73-77.
Singh IP, Saxena AK, Shankar K. Synthesis and anti-inflammatory activity of
oxadiazolines thione hydrochlorides. Eur J Med Chem. 1986;21:267–269.
Sivaraj S, Muthumani P, Venkataraman S, Raamamurthy J, Kumar RS. Design,
molecular docking, synthesis and evaluation of some novel heterocyclic analogues
of diclofenac as potent analgesic and anti-inflammatory agents with less
ulcerogenicity. Der Pharma Chemica. 2011;3:443-455.
Smeyers YG, Senen ML, Villa M, Theoretical structural & QSAR studies of some
arylpropionic acids as anti-inflammatory agents: an overview. Bio Appl Quantum
Chem Theory, 2002:1-15.
Smith WC, Neutrophils. In: Rich RR, Fleisher TA, Kotzin BL & Schroeder HW
(eds) Clinical Immunology. Principles and practice. Mosby International Limited,
London; 2001.
Smith WL and Willis AL. Aspirin selectively inhibits prostaglandin production in human
platelets. Nature. 1971;231:235-239.
Soni N, Barthwal JP, Saxena AK, Bhargava KP, Parmar SS. Monoamine oxidase
and succinate dehydrogenase inhibitory properties of substituted 1,3,4-oxadiazole-
2-thiones. J Heterocyclic Chem. 1982;19:29-32.
Srinivas K and Kumar KP. Synthesis, antimicrobial and anthelmintic activity of 1-
[(5-sustituted-1,3,4-oxadiazol-2-yl)methyl]-4-propylpiperazines. Int J Biopharm.
2010;1:14-19.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 244
Taiwo YO and Levine JD. Prostaglandin effects after elimination of indirect
hyperalgesic mechanisms in the skin of the rat, Brain Res. 1989;492:397-399.
Tan TM, Chen Y, Kong KH, J. Bai, Li Y, Lim SG, Ang TH, Lam Y. Synthesis
and the biological evaluation of 2-benzenesulfonylalkyl-5-substituted-sulfanyl-
(1,3,4)-oxadiazoles as potential anti-hepatitis B virus agents. Antiviral Res.
2006;71:7-14.
Teplyakov A, Obmolova G, Badet M, Badet M. The mechanism of sugar
phosphate isomerization by glucosamine 6-phosphate synthase, Protein Sci.
1999;8:596-602.
Testa B and Jenner P. Drug metabolism, chemical and biochemical aspect, Marcel
Dekker inc., New York; 1976.
Thakur A, Thakur M, Kakani N, Joshi A, Thakur S, Gupta A. Application of
topological and physicochemical descriptors: QSAR study of phenylamino-
acridine derivatives. Arkivoc. 2004;xiv:36-43.
Thomas W. Shattuck, Colby college molecular mechanics tutorial. Introduction.
Chemical Computing Group, Canada; 2008
Thomsen R, Christensen MH. MolDock: A new technique for high-accuracy
molecular docking. J Med Chem. 2006;49:3315-3321.
Timothy JR. Solvent accessible surface area and excluded volume in proteins:
analytical equations for overlapping spheres and implications for the hydrophobic
effects. J Mol Bio. 1984;178:63-89.
Toliwal SD, Jadav K, Gupte A, Banu A. Synthesis and biological evaluation of
phenyl hydrazides and their derivatives from rice bran oil. Der Pharma Chemica.
2009;1:185-195.
Tramont EC and Hoover DL. Innate (general or nonspesific) host defence
mechanisms. In: Mandell GL, Bennett JE, Dolin R. Principles and practice of
infectious diseases. Churchill Livingstone, Philadelphia; 2000.
Tripathi KD. Essentials of Medicinal Chemistry. 2nd
ed. Jaypee Brothers Medical
Publishers. New Delhi, India; 2003.
Vander D, Tsai WA, Kulmacz AL. The cyclooxygenase reaction mechanism,
Biochem. 2002;41:15451-15458.
Vane JR and Botting RM. New insights into the mode of action of anti-
inflammatory drugs. Inflamm Res.1995;44:1-10.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 245
Vane JR, Prostaglandins as mediators of inflammation, Adv Prostaglandin
Thromboxane Res. 1976;2:791-780.
Vane JR. Inhibition of prostaglandin synthesis as a mechanism of action for
aspirin-like drugs. Nature. 1971;231:232-237.
Vanegas H and Schaible HG. Prostaglandins and cyclooxygenases in the spinal
cord. Prog Neurobiol. 2001;64:327-363.
Veerasamy R, Sivadasan S, Karupiah S, Arumugam DS. QSAR study of
substituted 1,3,4-oxadiazole naphthyridines as HIV-1integrase inhibitors. Eur J
Med Chem. 2010;45:2791-2797.
Venkatapuram P, Sanapalli RN, Konda M. Synthesis, antimicrobial and
antioxidant activities of sulfone linked bis heterocycles-pyrazolyl oxadiazoles and
pyrazolyl thiadiazole. Chem Pharm Bull. 2009; 57:1376-1380.
Vogel HG. Drug discovery and evaluation. Pharmacological assay. 2nd
Edition
Springer, New York; 2002.
Wang H, Kohno T, Nobuko I, Andrew A, Fumimas A, Gary BJ. Bradykinin
produces pain hypersensitivity by potentiating spinal cord glutamatergic synaptic
transmission. J Neuroscience. 2005;25:7986-92.
Warner TD and Giuliano F. Nonsteroid drug selectivities for cyclooxygenase-1
rather than cyclooxygenase-2 are associated with human gastrointestinal toxicity:
A full in vitro analysis. Proc Natl Acad Sci. 1999;96:7563-7568.
Wedmore CV and Williams TJ. Control of vascular permeability by
polymorphonuclear leukocytes in inflammation. Nature. 1981;289:646-650.
Weiser ME. Atomic weights of elements. Pure Appl Chem. 2006;78:2051-2056.
Wiener H. Structural determination of paraffin boiling points. J Am Chem Soc.
1974;69:17-20.
Wilder-Smith CH. Predicting pain and pain responses to opioids. Eur J Pain
Suppl. 2007;1:31-31-37.
Williams JA and Shacter E. Regulation of macrophage cytokine production by
prostaglandin E2. Distinct roles of cyclooxygenase-1 and -2. J Biol Chem.
1997;272:25693-25699.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 246
Winter A, Risley EA, Nuss GW. Carrageenan-induced oedema in hind paws of
the rat as an assay for anti-inflammatory drugs. Proc Soc Exp Biol. 1962;111:544-
547.
Wojciechowski M, Mazerski J, Borowski E. Constrained search of conformational
hyperspace of inactivators of glucosamine-6-phosphate synthase. J Enzyme Inhib.
1996;10:17-26.
Wojciechowski M, Milewski S, Mazerski J, Borowski E, Glucosamine-6-
phosphate synthase, a novel target for antifungal agents-molecular modelling
studies in drug design. Acta Biochim Pol. 2005;52:647-653.
Wu J, Song B, Chen H, Bhadury P, Hu D. Synthesis and antifungal activity of 5-
chloro-6-phenylpyridazin-3(2H)-one derivatives. Molecules. 2009;14:3676-3687.
Wyllie AH, Kerr JFR, Currie AR. Cell death: the significance of apoptosis. Int
Rev Cytol. 1980;68:251-306.
Xu X, Zhu W, Zhang Y. The reductive reaction of substituted 2-chloromethyl-
1,3,4-oxadiazole to aldehydes and ketones promoted by samarium diiodide, Chin
Chem Lett. 2005;16:1566-1568.
Yang YH and Shi M. Halogen effects in Robinson-Gabriel type reaction of
cyclopropanecarboxylic acid N'-substituted-hydrazides with PPh3/CX4.
Tetrahedron Lett. 2005;46:6285-6288.
Yao X, Jericho M, Pink D, Beveridge T. Thickness and elasticity of gram-negative
murein sacculi measured by atomic force microscopy. J Bacterial. 1999;
181:6865-6875.
Yar MS, Siddiqui AA, Ali MA. Synthesis and anti tuberculostatic activity of
novel 1,3,4-oxadiazole derivatives. J Chinese Chem Soc. 2007;54:5-8.
Yasuyuki M, Takahiro N, Kenji S. Studies on pesticides for a rice plant
accumulation of oxadiazon and its metabolites in processed foods. Toxicol
Environ Chem. 1994;45:225- 235.
Yin L,
Xu W,
Wang Z,
Zhang D,
Jia J,
Ge Y, Li Y, Wang J. Synthesis and
antimicrobial activities of novel peptide deformylase inhibitors. Arkivoc.
2010;ix:196-205.
Yokomizo T, Izumi T, Shimizu T. Leukotriene B4: metabolism and signal
transduction. Arch Biochem Biophys. 2001;385:231-241.
Chapter-8 References
Faculty of Pharmaceutical Sciences, M.M. University, Mullana, Ambala, Haryana (India) 247
Zahid M,
Yasin KA, Akhtar T, Rama NH,
Hameed S,
Al-Masoudi NA, Loddo R,
Colla PL. Synthesis and in vitro antiproliferative activity of new
adamantylthiazolyl-1,3,4-oxadiazoles. Arkivoc. 2009;xi:85-93.
Zarghi A, Hamedi S, Tootooni F, Amini B, Sharifi B, Faizi M, Tabatabai SA,
Shafiee A. Synthesis and pharmacological evaluation of new 2-substituted-5-{2-
[(2-halobenzyl)thio)phenyl}-1,3,4-oxadiazoles as anticonvulsant agents. Sci
Pharm. 2008; 76:185-201.
Zarghi A, Tabatabai SA, Faizi M, Ahadian A, Navabi P, Zanganeh V, Shafiee A.
Synthesis and anticonvulsant activity of new 2-substituted-5-(2-
benzyloxyphenyl)-1,3,4-oxadiazole. Bioorg Med Chem Lett. 2005;15:1863-1865.