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Anthelmintik

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Anthelmintik. SIFAT OBAT ANTHELMINTIK UMUMNYA LONG ACTING. “ PULSED – RELEASED “. MORANTEL / PIRANTEL TARTRAT 90 HARI OXFENDAZOL 130 HARI. FORMULASI : ERADIBLE MATRICES DEGRADABLE POLIMER Controlled-Release Glasses (CRG). MEKANISME KERJA. CELLS INTEGRITY EFFECT : - PowerPoint PPT Presentation

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Acronym Class DrugsCommon trade

names

1 BZD Benzimidazoles

ThiabendazoleFenbendazoleAlbendazoleOxfendazole

TBZ®1

Panacur®, Safeguard®2

Valbazen®1

Synanthic®

2IMIDTETR

Nicotinic agonists   Imidazothiaoles   Tetrahydropyrimidines

LevamisoleMorantelPytrantel

Prohibit®1, Levasol1, Tramisol®1

Rumatel®2, Nematel®Strongid®

3 ML

Macrolytic Lactones   Avermectins   Milbemycins

IvermectinEprinomectin DoramectinMoxidectin

Ivomec®1, Primectin™1 Eprinex® Dectomax®Cydectin®1, Quest®

1FDA-approved for use in sheep.       2FDA-approved for use in goats.

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SIFAT OBAT ANTHELMINTIK UMUMNYA LONG ACTING

MORANTEL / PIRANTEL TARTRAT 90 HARI

OXFENDAZOL 130 HARI

“ PULSED – RELEASED “

FORMULASI :

ERADIBLE MATRICESDEGRADABLE POLIMERControlled-Release Glasses (CRG)

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MEKANISME KERJA

CELLS INTEGRITY EFFECT :

Inhibitor Tubulin Polimerase : Benzimidazol melalui Reseptor Tubulin

Uncoupler Oxidative Phosphorilation : Diklorofen, Niklosamid, Nitroxinil, Bithionol

Inhibitor Enzym in Glycolitic Pathway : Mebendazol, Befenium Hidroksinaftoat

NEUROMUSCULAR COORDINATION : Cholinesterase Inhibitor : Albendazol, Mebendazol, Organofosfat

Cholinergic Agonis : Pirantel

Muscle Hyperpolarisation : Piperazin

Potensiation of Inhibitory Transmiter : Ivermectin

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Albendazole Suspesion Solution

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NITROXINIL

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Ivermectin 1 % w/v sc

Ekto/endo parasit

Pada sapi, kambing dan babi