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![Page 1: 1,2-azoles - [DePa] Departamento de Programas …depa.fquim.unam.mx/amyd/archivero/AZOLES1,2_31931.pdfsulfonamide aromatic heterocyclic rings Me Me 1-102 1. (MeO)2S02 2. NaOH/H20 pyrazole](https://reader043.dokumen.tips/reader043/viewer/2022030718/5b03002d7f8b9a6561901abc/html5/page/1.jpg)
1,2-azoles
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Antibióticos.Sulfonamidas
sulfametoxazol sulfatiazol sulfafurazol
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antihelmínticos
mebendazol albendazol
tiabendazol fenbendazol
niridazol levamisol
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Two routes for the ringsynthesis of1,2- azoles
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Synthesis of 1,2–azoles from 1,3-dicarbonylcompounds and hydrazines or hydroxylamine
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reactividad
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Reactions with Electrophilic Reagents
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Substitution atCarbon
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Reactions with Bases
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C-Metallation andreactions.Metal–halogenexchange
![Pyrazole-oxadiazole Conjugates: Synthesis, …Pyrazole-oxadiazole Conjugates: Synthesis, Antiproliferative Activity and Inhibition of Tubulin Polymerization Ahmed Kamal, *[a,d] Anver](https://img.dokumen.tips/doc/110x75/5e8c65afba3d737ddc66773e/pyrazole-oxadiazole-conjugates-synthesis-pyrazole-oxadiazole-conjugates-synthesis.jpg)
