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Endocrinology
Found in most species of the animal kingdom, the endocrine systemconsists of glands that secrete hormones, and receptors that detectand react to the hormones. In response to environmental stimuli, theendocrine system secretes hormones and uses them as chemicalmessengers to orchestrate physiological, developmental andreproductive changes that affect the entire body for a long period oftime. In order to maintain the proper functioning of the body throughits entire life cycle, the endocrine system utilizes a complex feedbackmechanism to fine-tune the balance of hormones in the bloodstream.Even a slight disruption to endocrine system’s function can throw offthe delicate balance of hormones in the human body and lead to an
endocrine disorder, or endocrine disease, such as diabetes, adrenal insufficiency, hyper- or hypothyroidism, andpolycystic ovary syndrome (PCOS).
Purity: 99.81%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
10 mg, 50 mg
Purity: 98.93%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
1 mg, 5 mg, 10 mg
Purity: 99.61%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
10 mg, 50 mg, 100 mg
Purity: 98.65%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg
Purity: >98%Clinical Data: No Development ReportedSize:
Purity: 98.16%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
100 mg, 500 mg
Purity: 98.75%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
100 mg, 500 mg
Purity: 99.0%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
1 g, 5 g
Purity: >98%Clinical Data: No Development ReportedSize: 250 mg, 500 mg
Purity: >98%Clinical Data: No Development ReportedSize: 250 mg, 500 mg
Endocrinology Inhibitors & Modulators
Bioactivity: Posiphen is a novel selective noncompetitivecholinesteraseinhibitor with an of 45.3 μM.IC50
Bioactivity: (9Z,11E)-Tetradecadien-1-yl acetate is the main component ofthe sex pheromone of female .Spodoptera littoralis
Bioactivity: 2-Thiouracil is a thiolated uracil derivative that is a knownantihyperthyroid agent.
Bioactivity: 3,3',5-Triiodo-L-thyronine is a potent agonist of thyroidhormone receptors and with s of 2.3 nM.TRα TRβ Ki
Bioactivity: 3,3',5-Triiodo-L-thyronine sodium is an active form of thyroidhormone, which binds to (β1 thyroid hormone receptor
), and activates its activity.TRβ1
Bioactivity: 5a-Pregnane-3,20-dione is the endogenous progesteronemetabolite.
Bioactivity: AL 082D06 is a selective, nonsteroidal glucocorticoid receptor( ) antagonist with of 210 nM.GR Ki
Bioactivity: Alarelin acetate is a synthetic agonist.GnRH
Bioactivity: Alexamorelin is a new synthetic heptapeptide which inhibits binding in vitro. Sequence:GHS
Ala-His-{Me-Trp}-Ala-Trp-Phe-Lys-NH2.
Bioactivity: Alfuzosin is an α1 adrenergic receptor antagonist used totreat benign prostatic hyperplasia (BPH).
2 Tel: 609-228-6898 Fax: 609-228-5909 Email: [email protected]
(+)-PHENSERINE Cat. No.: HY-16009
(9Z,11E)-Tetradecadien-1-yl acetate (Ferodin SL; Litlure A; Prodlure) Cat. No.: HY-101735
2-Thiouracil (Thiouracil) Cat. No.: HY-B0503
3,3',5-Triiodo-L-thyronine (T3; L-3,3',5-Triiodothyronine; Liothyronine; Tresitope) Cat. No.: HY-A0070A
3,3',5-Triiodo-L-thyronine sodium (T3 Sodium salt; Sodium
L-3,3',5-triiodothyronine; Liothyronine sodium) Cat. No.: HY-A0070
5a-Pregnane-3,20-dione Cat. No.: HY-W006492
AL 082D06 (D06; D-06) Cat. No.: HY-15709
Alarelin Acetate (Alarelin) Cat. No.: HY-17405
Alexamorelin Cat. No.: HY-P0166
Alfuzosin (SL 77499) Cat. No.: HY-B0192
www.MedChemExpress.com 3
Purity: 98.0%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg
Purity: 98.70%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg
Purity: 99.20%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
1 mg, 5 mg, 10 mg, 25 mg
Purity: 98.0%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg
Purity: 98.0%Clinical Data: No Development ReportedSize: 10mM x 1mL in Water,
100 mg
Purity: 98.62%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
100 mg, 500 mg
Purity: >98%Clinical Data: No Development ReportedSize: 5 mg, 10 mg, 50 mg
Purity: 99.14%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg
Purity: 99.93%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
100 mg, 200 mg
Purity: >98%Clinical Data: LaunchedSize: 10 mg, 50 mg
Bioactivity: Alfuzosin hydrochloride is an α1 adrenergic receptorantagonist used to treat benign prostatic hyperplasia (BPH).
Bioactivity: Alibendol is an antispasmodic,choleretic, and cholekinetic.
Bioactivity: Alrestatin is an inhibitor of aldose reductase, an enzymeinvolved in the pathogenesis of complications of diabetesmellitus, including diabetic neuropathy.
Bioactivity: Alrestatin sodium is an inhibitor of aldose reductase, anenzyme involved in the pathogenesis of complications ofdiabetes mellitus, including diabetic neuropathy.
Bioactivity: Altrenogest(A35957; RU2267) is a progestogen structurallyrelated to veterinary steroid trenbolone.
Bioactivity: Aminoguanidine hydrochloride is a diamine oxidase and NOsynthase inhibitor, reduces levels of advanced glycation endproducts (AGEs) through interacting with 3-deoxyglucosone, isan investigational drug for the treatment of diabeticnephropathy.
Bioactivity: Azoramide is a small-molecule modulator of the unfoldedprotein response with antidiabetic activity.
Bioactivity: BI 689648 is a novel, highly selective aldosterone synthaseinhibitor which can inhibit and with sCYP11B1 CYP11B2 IC50of 310 and 2.1 nM, respectively.
Bioactivity: BMS-564929 is an (AR) agonist, binds toandrogen receptorandrogen receptor (AR) with a of 2.11±0.16 nM.Ki
Bioactivity: BRD7552 is an inducer of transcription factor PDX1, whichincreases insulin expression.
Alfuzosin hydrochloride (SL 77499-10) Cat. No.: HY-B0192A
Alibendol Cat. No.: HY-B0326
Alrestatin (AY-22284) Cat. No.: HY-B1202
Alrestatin sodium (AY-22284A) Cat. No.: HY-B1202A
Altrenogest (A35957; Allyltrenbolone; R2267; RU2267) Cat. No.: HY-B0521
Aminoguanidine hydrochloride (Pimagedine hydrochloride;
GER-11; Aminoguanidinium chloride) Cat. No.: HY-B1041
Azoramide Cat. No.: HY-18705
BI 689648 Cat. No.: HY-101217
BMS-564929 Cat. No.: HY-12111
BRD7552 Cat. No.: HY-19694
Purity: 98.76%Clinical Data: Phase 3Size: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg
Purity: 98.0%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
1 g, 5 g
Purity: 99.24%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
100 mg
Purity: 95.0%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
100 mg
Purity: >98%Clinical Data: No Development ReportedSize: 1 mg, 5 mg, 10 mg, 20 mg
Purity: 99.93%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
100 mg, 500 mg
Purity: 98.0%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
1 g, 5 g
Purity: >98%Clinical Data: No Development ReportedSize: 1 mg, 5 mg, 10 mg, 20 mg
Purity: 99.47%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg
Purity: 98.18%Clinical Data: Phase 3Size: 10mM x 1mL in DMSO,
10 mg, 50 mg
Bioactivity: Bremelanotide Acetate is a melanocortin agonist. IC50 value:Target: melanocortin in vivo: Bremelanotide is a novel drugcandidate for the treatment of male and female sexualdysfunction. Bremelanotide has shown promise in effectivelytreating erectile dysfunction (ED) without the cardiovascular…
Bioactivity: Cabergoline is an ergot derived-dopamine D -like receptor2agonist that has high affinity for , , and D2 D3 5-HT2Breceptors ( =0.7, 1.5, and 1.2, respectively).Ki
Bioactivity: Carbazole derivative 1 is a carbazole derivative which can beused to reduce androgen or oestrogen levels in mammals,including humans.
Bioactivity: Carbimazole is an imidazole antithyroid agent.
Bioactivity: Carvedilol(BM14190) is a non-selective beta blocker/alpha-1blocker with an IC50 of 3.8 μM for inhibition of LDLoxidation. IC50 Value: 3.8 μM ( inhibition of LDL oxidation)Target: beta Adrenergic Receptor Carvedilol is anonselective-blocking agent and is used in the treatment of…
Bioactivity: CGP-53153 is a steroidal inhibitor of with5 alpha reductases of 36 and 262 nM in rat and human prostatic tissue,IC50
respectively.
Bioactivity: Chlormadinone acetate is a steroidal progestin, withantiandrogen and antiestrogenic effects.
Bioactivity: Chlorpropamide is an oral antihyperglycemic agent used for thetreatment of non-insulin-dependent diabetes mellitus (NIDDM).
Bioactivity: Clomifene Citrate is a selective estrogen receptor modulator. Bioactivity: Cortexolone 17 alpha-propionate(CB-03-01) is a new topical andperipherally selective androgen antagonist.
4 Tel: 609-228-6898 Fax: 609-228-5909 Email: [email protected]
Bremelanotide Acetate (PT-141 Acetate) Cat. No.: HY-18678A
Cabergoline (FCE-21336) Cat. No.: HY-15296
Carbazole derivative 1 (2-Fluoro-7-[(3-pyridinyl)methyl]-9H-carbazole) Cat. No.: HY-U00323
Carbimazole Cat. No.: HY-B0558
Carvedilol (BM 14190) Cat. No.: HY-B0006
CGP-53153 Cat. No.: HY-U00125
Chlormadinone acetate Cat. No.: HY-B1095
Chlorpropamide Cat. No.: HY-B1429
Clomiphene citrate (Clomifene citrate) Cat. No.: HY-B0463
Cortexolone 17 alpha-propionate (Cortexolone 17α-propionate; CB-03-01) Cat. No.: HY-13331
www.MedChemExpress.com 5
Purity: 98.0%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
200 mg, 1 g, 5 g
Purity: 99.12%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
10 mg, 50 mg, 100 mg
Purity: 96.0%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
50 mg
Purity: 98.0%Clinical Data: Phase 4Size: 10mM x 1mL in DMSO,
100 mg, 500 mg
Purity: 98.0%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
100 mg
Purity: 98.0%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
1 g, 5 g
Purity: 97.95%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
1 g
Purity: 98.28%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
100 mg, 250 mg
Purity: 99.66%Clinical Data: Phase 4Size: 10mM x 1mL in DMSO,
500 mg, 1 g, 5 g, 10 g
Purity: 99.71%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
250 mg, 500 mg
Bioactivity: Cyproterone acetate is an androgen receptor (AR) antagonistwith IC50 of 7.1 nM, as well as a weak progesterone receptoragonist with weak pro-gestational and glucocorticoid activity.
Bioactivity: Daidzein is a soy isoflavone, which acts as a activator.PPAR
Bioactivity: Danazol is a derivative of the synthetic steroid ethisterone,that suppresses the production of gonadotrophins, and has someweak androgenic effects.
Bioactivity: Dehydrocholic acid is a synthetic bile acid, manufactured bythe oxidation of cholic acid. Dehydrocholic acid acts as ahydrocholeretic, increasing bile output to clear increasedbile acid load.
Bioactivity: Dehydroepiandrosterone 3-acetate is a testosterone/estrogenprecursor and known modulator of vertebrate aggression.
Bioactivity: Deoxycorticosterone acetate is a steroid hormone produced bythe adrenal gland that possesses mineralocorticoid activityand acts as a precursor to aldosterone.
Bioactivity: DHEA is one of the most abundant steroid hormones. DHEAmediates its action via multiple signaling pathways involvingspecific membrane receptors and via transformation intoandrogen and estrogen derivatives (e.g., androgens, estrogens,7α and 7β DHEA, and 7α and 7β epiandrosterone derivatives)…
Bioactivity: Dienestrol is a synthetic, non-steroidal estrogen, is anestrogen receptor agonist, for the treatment of menopausal andpostmenopausal symptoms.
Bioactivity: Dienogest(STS-557) is a specific progesterone receptor agonistwith potent oral endometrial activity and is used in thetreatment of endometriosis. Target: progesterone receptoragonist Dienogest is an orally active synthetic progesterone(or progestin). It is available for use as an oral…
Bioactivity: Diethylstilbestrol, a synthetic nonsteroidal estrogen used inthe treatment of menopausal and postmenopausal disorders.
Cyproterone acetate Cat. No.: HY-13604
Daidzein (Isoflavone) Cat. No.: HY-N0019
Danazol Cat. No.: HY-B1029
Dehydrocholic acid Cat. No.: HY-B1393
Dehydroisoandrosterone 3-acetate (Dehydroepiandrosterone 3-acetate; DHEA acetate) Cat. No.: HY-B1405
Deoxycorticosterone acetate (11-Deoxycorticosterone acetate;
DOC acetate; Cortexone acetate) Cat. No.: HY-B1472
DHEA (trans-Dehydroandrosterone; Prasterone;
Dehydroisoandrosterone; Dehydroepiandrosterone) Cat. No.: HY-14650
Dienestrol Cat. No.: HY-B1403
Dienogest (STS 557) Cat. No.: HY-B0084
Diethylstilbestrol (DES; Stilbestrol) Cat. No.: HY-14598
Purity: 98.0%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
1 g
Purity: 99.69%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
1 g
Purity: 99.91%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
1 g
Purity: >98%Clinical Data: No Development ReportedSize: 50 mg, 100 mg
Purity: 98.0%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
1 mg
Purity: 98.0%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
1 g, 5 g
Purity: 99.20%Clinical Data: Phase 3Size: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg
Purity: 99.88%Clinical Data: LaunchedSize: 10 mg, 50 mg
Purity: 98.0%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
10 mg, 50 mg, 100 mg
Purity: 99.83%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
10 mg, 50 mg
Bioactivity: Diphemanil methylsulfate is a quaternary ammoniumanticholinergic. It binds muscarinic acetycholine receptorsand thereby decreases secretory excretion of stomach acids aswell as saliva and sweat.
Bioactivity: Drospirenone(Dihydrospirorenone) is a synthetic progestin thatis an analog to spironolactone.
Bioactivity: Dydrogesterone(Duphaston) is a potent, orally activeprogestogen indicated in a wide variety of gynaecologicalconditions related to progesterone deficiency.
Bioactivity: Elagolix sodium is a human ( )GnRH receptor GnRHRantagonist with an and of 0.25 and 3.7 nM,IC50 Kirespectively.
Bioactivity: Epiandrosterone is a steroid hormone with weak androgenicactivity. Epiandrosterone is naturally produced by the enzyme5α-reductase from the adrenal hormone DHEA.
Bioactivity: Eprotirome is a liver-selective thyroid hormone receptoragonist.
Bioactivity: Equilin is one of the estrogens present in the mixture ofestrogens isolated from horse urine.
Bioactivity: Estradiol is a steroid sex hormone vital to the maintenance offertility and secondary sexual characteristics in females.
Bioactivity: Estradiol benzoate is a synthetic ester, is the first form ofestrogen to be marketed.
Bioactivity: Estradiol cypionate is a 17 β-cyclopentylpropinate ester ofestradiol, inhibits ET-1 synthesis via estrogen receptor IC50value: Target: estrogen receptor Estradiol cypionate is asynthetic ester, is a estrogen. Compared to other commonlyused estradiol esters, via the intramuscular route, Estradiol…
6 Tel: 609-228-6898 Fax: 609-228-5909 Email: [email protected]
Diphenmanil methylsulfate (Diphemanil mesylate) Cat. No.: HY-16171
Drospirenone (Dihydrospirorenone) Cat. No.: HY-B0111
Dydrogesterone Cat. No.: HY-B0257A
Elagolix sodium (NBI-56418 sodium) Cat. No.: HY-14369
Epiandrosterone (3β-Androsterone; trans-Androsterone; iso-Androsterone) Cat. No.: HY-I0352
Eprotirome (KB2115) Cat. No.: HY-10473
Equilin (7-Dehydroestrone) Cat. No.: HY-B1176
Estradiol (β-Estradiol; E2; 17β-Estradiol; 17β-Oestradiol) Cat. No.: HY-B0141
Estradiol benzoate Cat. No.: HY-B1192
Estradiol cypionate Cat. No.: HY-B1100
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Purity: 99.86%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
10 mg, 50 mg, 100 mg
Purity: >98%Clinical Data: No Development ReportedSize: 250 mg, 500 mg
Purity: >98%Clinical Data: No Development ReportedSize: 250 mg, 500 mg
Purity: 98.52%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
10 mg, 50 mg, 100 mg, 200 mg
Purity: >98%Clinical Data: No Development ReportedSize: 1 mg, 5 mg, 10 mg, 20 mg
Purity: >98%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
1 mg, 5 mg, 10 mg
Purity: 99.40%Clinical Data: Phase 4Size: 10mM x 1mL in DMSO,
100 mg, 500 mg
Purity: 98.02%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
500 mg
Purity: 99.02%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
10 mg, 50 mg
Purity: 99.86%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
1 g, 5 g, 10 g
Bioactivity: Estrone is an estrogenic hormone. Target: EstrogenReceptor/ERR Estrone (E1) is an estrogenic hormone secreted bythe ovary as well as adipose tissue with the chemical name of3-hydroxyestra-1,3,5(10)-triene-17-one and the chemicalformula C18H22O2. Estrone is one of several natural estrogens,…
Bioactivity: Estropipate is a form of estrogen, used to treat symptoms ofmenopause, also used to prevent osteoporosis.
Bioactivity: Ethynodiol diacetate is a steroidal progestin which is used asa hormonal contraceptive, it has relatively little or nopotency as an androgen,has significant estrogenic effects.
Bioactivity: Ethynyl estradiol is an orally bio-active estrogen used inalmost all modern formulations of combined oral contraceptivepills. Target: Estrogen Receptor Ethinyl estradiol (EE), alsosometimes written as ethinylestradiol, ethynyl estradiol, orethinyl estradiol, is a derivative of 17β-estradiol (E2), the…
Bioactivity: Eurycomanone could increases spermatogenesis by inhibiting theactivity of phosphodiesterase and aromatase insteroidogenesis.
Bioactivity: Falintolol, (Z)-, a new antagonist, isβ-adrenergiccharacterized by the presence of an oxime function.
Bioactivity: Forskolin is a potent activator, with andadenylate cyclase IC50 of 41 nM and 0.5 μM for ,EC50 type I adenylyl cyclase
respectively.
Bioactivity: FR-167653 is a selective inhibitor.p38 MAPK
Bioactivity: FR-167653 is a selective inhibitor.p38 MAPK Bioactivity: Gestodene(SHB 331;WL 70) is a progestogen hormonalcontraceptive.
Estrone (E1; Oestrone) Cat. No.: HY-B0234
Estropipate (Piperazine estrone sulfate; Estrone sulfate
piperazine salt) Cat. No.: HY-B1361
Ethynodiol diacetate (Ethynodiol acetate) Cat. No.: HY-B1089
Ethynyl Estradiol (17α-Ethynylestradiol; Ethynylestradiol) Cat. No.: HY-B0216
Eurycomanone (Pasakbumin A) Cat. No.: HY-N5012
Falintolol, (Z)- Cat. No.: HY-U00283
Forskolin (Coleonol; Colforsin) Cat. No.: HY-15371
FR 167653 (FR 167653 sulfate) Cat. No.: HY-18754A
FR 167653 free base Cat. No.: HY-18754
Gestodene (SHB 331; WL 70) Cat. No.: HY-B0110
Purity: 98.0%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg
Purity: 96.08%Clinical Data: No Development ReportedSize: 10 mg, 25 mg
Purity: 99.83%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
1 mg, 2 mg, 5 mg, 10 mg, 25 mg, 50 mg, 100 mg
Purity: 96.13%Clinical Data: Phase 2Size: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg, 500 mg
Purity: 98.07%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
2 mg, 5 mg, 10 mg, 50 mg, 100 mg
Purity: 99.96%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg
Purity: >98%Clinical Data: LaunchedSize: 10 mg
Purity: 98.74%Clinical Data: Phase 4Size: 10mM x 1mL in DMSO,
10 mg, 50 mg, 100 mg
Purity: 99.55%Clinical Data: No Development ReportedSize: 1 mg, 5 mg, 10 mg, 25 mg
Purity: 99.39%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
50 mg, 100 mg
Bioactivity: Gliquidone is an anti-diabetic drug in the sulfonylurea class,used in the treatment of diabetes mellitus type 2.
Bioactivity: GnRH-I is a small 10 amino acid long peptide (decapeptide)from the hypothalamus, acts at the hypophysis to cause anincrease in release of biologically activeFollicle-Stimulating Hormone (FSH) and Luteinizing Hormone(LH) in the blood. Sequence:…
Bioactivity: Gonadorelin acetate is a man-made protein that is like ahormone in the body called gonadotropin-releasing hormone(GnRH).
Bioactivity: Goserelin(ICI 118630) is an injectable gonadotropin releasinghormone superagonist (GnRH agonist). IC50 value: Target: GnRHagonist Goserelin is used to treat hormone-sensitive cancersof the breast (in pre- and peri- menopausal women) andprostate, and some benign gynaecological disorders…
Bioactivity: Goserelin (ICI 118630) acetate is an injectable gonadotropinreleasing hormone superagonist (GnRH agonist).
Bioactivity: GSK583 is a highly potent and selective inhibitor of RIP2, with of 5 nM.Kinase IC50
Bioactivity: Ibutamoren (Mesylate) is a potent, non-peptide Growth agonist.hormone secretagogue receptor (GHSR)
Bioactivity: Iloprost (ZK 36374) is a synthetic analogue of prostacyclinPGI2.
Bioactivity: Impurity of Doxercalciferol is an impurity of doxercalciferol,which is a synthetic analog of ergocalciferol (vitamin D2),used as a drug for secondary hyperparathyroidism and metabolicbone disease, and it suppresses parathyroid synthesis andsecretion.
Bioactivity: INT-777 is a potent agonist with an of 0.82 μM.TGR5 EC50
8 Tel: 609-228-6898 Fax: 609-228-5909 Email: [email protected]
Gliquidone Cat. No.: HY-B1114
GnRH-I Cat. No.: HY-P0292
Gonadorelin acetate Cat. No.: HY-12555
Goserelin (ICI 118630) Cat. No.: HY-13673
Goserelin acetate (ICI-118630 acetate) Cat. No.: HY-13673A
GSK583 Cat. No.: HY-100339
Ibutamoren Mesylate (MK-677; MK-0677) Cat. No.: HY-50844
Iloprost (Ciloprost; ZK 36374) Cat. No.: HY-A0096
Impurity of Doxercalciferol Cat. No.: HY-76937
INT-777 (S-EMCA) Cat. No.: HY-15677
www.MedChemExpress.com 9
Purity: 99.62%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg
Purity: 99.85%Clinical Data: Phase 4Size: 10mM x 1mL in DMSO,
500 mg, 1 g
Purity: 98.0%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
500 mg, 1 g
Purity: 98.0%Clinical Data: Phase 3Size: 10mM x 1mL in DMSO,
5 g
Purity: >98%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
10 mg, 50 mg, 100 mg
Purity: 99.62%Clinical Data: No Development ReportedSize: 1 mg, 5 mg
Purity: >98%Clinical Data: LaunchedSize: 5 mg, 10 mg, 50 mg, 100 mg
Purity: >98%Clinical Data: LaunchedSize: 5 mg, 10 mg, 50 mg, 100 mg
Purity: 99.75%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg
Purity: 98.0%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
100 mg
Bioactivity: Iopanoic acid is an inhibitor of and also an5'-Deiodinaseiodinated contrast medium.
Bioactivity: Ivacaftor is a potent and orally bioavailable CFTRpotentiator, targeting G551D-CFTR and F508del-CFTR with
s of 100 nM and 25 nM, respectively.EC50
Bioactivity: Ivacaftor benzenesulfonate is an orally bioavailable CFTRpotentiator, used for cystic fibrosis treatment.
Bioactivity: Ivacaftor hydrate is an orally bioavailable potentiator,CFTRused for cystic fibrosis treatment.
Bioactivity: Kisspeptin-10 Trifluoroacetate is the trifluoroacetate saltform of Kisspeptin-10. Kisspeptin-10, the minimal kisspeptinSequence: Tyr-Asn-Trp-Asn-Ser-Phe-Gly-Leu-Arg-Phe-NH2.
Bioactivity: KM11060 is a novel corrector of the F508del-CFTR traffickingdefect.
Bioactivity: L-lysine hydrochloride is an essential amino acid for humanswith various benefits including treating herpes, increasingcalcium absorption, reducing diabetes-related illnesses andimproving gut health.
Bioactivity: L-Thyroxine (Levothyroxine; T4) is a synthetic hormone in thetreatment of hypothyroidism. DIO enzymes convert biologicallyactive thyroid hormone (Triiodothyronine,T3) from L-Thyroxine(T4).
Bioactivity: L-Thyroxine sodium salt pentahydrate (Levothyroxine; T4) is asynthetic hormone in the treatment of hypothyroidism. DIOenzymes convert biologically active thyroid hormone(Triiodothyronine,T3) from L-Thyroxine (T4).
Bioactivity: Lasofoxifene Tartrate is a non-steroidal selective estrogenreceptor modulator (SERM).
Iopanoic acid Cat. No.: HY-B1664
Ivacaftor (VX-770) Cat. No.: HY-13017
Ivacaftor benzenesulfonate (VX-770 benzenesulfonate) Cat. No.: HY-13017A
Ivacaftor hydrate (VX-770 hydrate) Cat. No.: HY-13017B
Kisspeptin-10 Trifluoroacetate Cat. No.: HY-P0254A
KM11060 Cat. No.: HY-19970
L-Lysine hydrochloride Cat. No.: HY-N0470
L-Thyroxine (Levothyroxine; T4) Cat. No.: HY-18341
L-Thyroxine sodium salt pentahydrate (Sodium levothyroxine pentahydrate) Cat. No.: HY-18341A
Lasofoxifene Tartrate (CP-336156) Cat. No.: HY-A0038
Purity: 97.31%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg
Purity: 99.0%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
1 g, 5 g
Purity: 99.31%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
100 mg
Purity: >98%Clinical Data: No Development ReportedSize: 1 mg, 5 mg
Purity: 98.0%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
1 g, 5 g
Purity: 99.02%Clinical Data: Phase 4Size: 10mM x 1mL in DMSO,
100 mg, 500 mg
Purity: 94.09%Clinical Data: No Development ReportedSize: 5 mg, 10 mg
Purity: >98%Clinical Data: No Development ReportedSize: 5 mg, 10 mg, 25 mg
Purity: 98.27%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 25 mg, 50 mg, 100 mg
Purity: 99.88%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg
Bioactivity: Leuprolide acetate (Leuprorelin) is a GnRH analog; leuprolideacetate acts as an agonist at pituitary GnRH receptors. IC50Value: Target: GnRH receptor By interrupting the normalpulsatile stimulation of, and thus desensitizing, the GnRHreceptors, it indirectly downregulates the secretion of…
Bioactivity: LGD-3303 is a selective androgen receptor modulator ().SARM
Bioactivity: Luteinizing Hormone Releasing Hormone (LH-RH), human ishypothalamic neuropeptide which plays a key role in thecontrol of reproductive functions.
Bioactivity: Mapracorat is a novel non-steroidal selective glucocorticoid agonist.receptor
Bioactivity: Medroxyprogesterone acetate is a progestin, a syntheticvariant of the human hormone progesterone and a potentprogesterone receptor agonist. Target: Progesterone ReceptorMedroxyprogesterone acetate(MPA) is a steroidal progestin, asynthetic variant of the human hormone progesterone. It is…
Bioactivity: Megestrol Acetate is a synthetic progesteronal agent with anIC50 of 260 μM for the inhibition of HegG2. Target:Progesterone Receptor Megestrol acetate, also known as17α-acetoxy-6-dehydro-6-methylprogesterone, and sometimesabbreviated as MGA or MA, is a steroidal progestin and…
Bioactivity: Mepixanox is an analeptic drug used in respiratory andcardiorespiratory insufficiency.
Bioactivity: Mestranol is the 3-methyl ether of ethinylestradiol. It wasthe estrogen used in many of the first oral contraceptives.
Bioactivity: Methimazole(Tapazole, Northyx) is an antithyroid medicine. Bioactivity: Metiamide is a histamine H2-receptor antagonist developed fromanother H2 antagonist, burimamide.
10 Tel: 609-228-6898 Fax: 609-228-5909 Email: [email protected]
Leuprolide Acetate (Leuprorelin acetate) Cat. No.: HY-13665
LGD-3303 Cat. No.: HY-103576
Luteinizing Hormone Releasing Hormone (LH-RH), human Cat. No.: HY-P1500
Mapracorat (ZK-245186; BOL-303242X) Cat. No.: HY-14864
Medroxyprogesterone (acetate) (Medroxyprogesterone 17-acetate; MPA) Cat. No.: HY-B0469
Megestrol Acetate Cat. No.: HY-13676
Mepixanox (Pimexone) Cat. No.: HY-100150
Mestranol Cat. No.: HY-B0390
Methimazole Cat. No.: HY-B0208
Metiamide Cat. No.: HY-15540
www.MedChemExpress.com 11
Purity: 99.33%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
100 mg, 500 mg
Purity: 99.41%Clinical Data: Phase 3Size: 10mM x 1mL in DMSO,
10 mg, 50 mg
Purity: 95.0%Clinical Data: Phase 1Size: 10mM x 1mL in DMSO,
1 mg, 5 mg, 10 mg, 50 mg
Purity: 95.0%Clinical Data: Phase 1Size: 1 mg, 5 mg, 10 mg, 50 mg
Purity: 99.12%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg
Purity: 99.48%Clinical Data: Phase 2Size: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg
Purity: 99.0%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg
Purity: 98.17%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
100 mg, 500 mg
Purity: 99.94%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
100 mg, 500 mg
Purity: 98.23%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
100 mg, 500 mg
Bioactivity: Metoclopramide is a dopamine D2 antagonist that is used as anantiemetic.
Bioactivity: Metoclopramide hydrochloride hydrate is a dopamine D2antagonist that is used as an antiemetic.
Bioactivity: Mifepristone is a ( ) andprogesterone receptor PR ( ) antagonist with s of 0.2 nMglucocorticoid receptor GR IC50
and 2.6 nM in assay.in vitro
Bioactivity: Misoprostol(SC29333) is a synthetic prostaglandin E1 (PGE1)analog that is used to prevent gastric ulcers, to treat missedmiscarriage, to induce labor, and to induce abortion.
Bioactivity: MK-0773 is a selective androgen receptor modulators (SARMs)that binds to AR with an of 6.6 nM.IC50
Bioactivity: ML224(NCGC00242364; ANTAG3) is a selective TSHR inverseagonist; inhibits TSH-stimulated cAMP production with an IC50= 2.3 μM.
Bioactivity: MSI-1436 is a selective, non-competitive inhibitor of theenzyme , with an protein tyrosine phosphatase 1B (PTB-1B) IC50of appr 1 μM, 200-fold preference over TC-PTP (IC , 22450μM).
Bioactivity: MSI-1436 lactate is a selective, non-competitive inhibitor ofthe enzyme ( ), with anprotein tyrosine phosphatase 1B PTB-1B
of 1 μM, 200-fold preference over TC-PTP ( of 224IC50 IC50μM).
Bioactivity: Nestoron(ST1435; Elcometrine) is a 19-norprogesteronederivative and steroidal progestin which is used as a hormonalcontraceptive; a high-affinity agonist of the progesteronereceptor.
Bioactivity: Norethindrone acetate is a female progestin approved by FDAfor the treatment of endometriosis, uterine bleeding caused byabnormal hormone levels, and secondary amenorrhea.
Metoclopramide Cat. No.: HY-17382
Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) Cat. No.: HY-17382A
Mifepristone (RU486; RU 38486) Cat. No.: HY-13683
Misoprostol (SC-29333) Cat. No.: HY-B0610
MK-0773 (PF-05314882) Cat. No.: HY-11027
ML224 (NCGC00242364; ANTAG3) Cat. No.: HY-12381
MSI-1436 (Trodusquemine; Aminosterol-1436) Cat. No.: HY-12219
MSI-1436 lactate (Trodusquemine lactate; Aminosterol-1436 lactate) Cat. No.: HY-12219A
Nestoron (Elcometrine; Nestorone; ST-1435) Cat. No.: HY-13071
Norethindrone acetate (19-Norethindrone acetate) Cat. No.: HY-B1710
Purity:Clinical Data: No Development ReportedSize: 100 mg
Purity: 99.79%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg, 200 mg, 500 mg
Purity: 98.68%Clinical Data: LaunchedSize: 5 mg, 10 mg
Purity: >98%Clinical Data: No Development ReportedSize: 250 mg, 500 mg
Purity: >98%Clinical Data: No Development ReportedSize: 250 mg, 500 mg
Purity: >98%Clinical Data: No Development ReportedSize: 250 mg, 500 mg
Purity: 95.09%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg
Purity: >98%Clinical Data: No Development ReportedSize: 1 mg, 5 mg, 10 mg
Purity: >98%Clinical Data: No Development ReportedSize: 500 mg, 250 mg
Purity: 98.05%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
2 mg, 5 mg, 10 mg, 25 mg, 50 mg, 100 mg
Bioactivity: NVP-BAW2881 (BAW2881) is a potent and selective VEGFR2inhibitor with an of 4 nM.IC50
Bioactivity: OBE022 is an oral and selective prostaglandin F ( )2α PGF2αreceptor antagonist, with of 1 nM, 26 nM for human and ratK siFP receptors, respectively.
Bioactivity: Org41841 is a partial agonist of both luteinizinghormone/chorionic gonadotropin receptor ( ) andLHCGRthyroid-stimulating hormone receptor ( ) with s ofTSHR EC500.2 and 7.7 μM, respectively.
Bioactivity: ORM-15341 is a potent and full antagonist for human AR (hAR)with IC50 values of 38 nM as shown by transactivation assaysin AR-HEK293 cells stably expressing full-length hAR and anandrogen-responsive luciferase reporter gene construct.
Bioactivity: OT antagonist 1 (Compound 4) is a potent, selective Oxytocinantagonist with a of 50 nM.Ki
Bioactivity: OT antagonist 1 demethyl derivative is the demethyl derivativeof OT antagonist 1. OT antagonist 1 (Compound 4) is a potent,selective antagonist with a of 50 nM.Oxytocin Ki
Bioactivity: OT antagonist 3 is an (OT) antagonist extracted fromoxytocinpatent WO2007017752A1.
Bioactivity: Oxytocin (α-Hypophamine) is a mammalian neurohypophysialhormone; its actions are mediated by specific, high-affinityoxytocin receptors; ligand of oxytocin receptor.
Bioactivity: Oxytocin (α-Hypophamine) acetate is a mammalianneurohypophysial hormone; its actions are mediated byspecific, high-affinity oxytocin receptors; ligand of oxytocinreceptor.
Bioactivity: Pancreatin is the porcine pancreas extract (PPE) whichcontains the main pancreatic digestive enzymes.
12 Tel: 609-228-6898 Fax: 609-228-5909 Email: [email protected]
NVP-BAW2881 (BAW2881) Cat. No.: HY-100394
OBE022 Cat. No.: HY-112284
Org41841 Cat. No.: HY-100271
ORM-15341 Cat. No.: HY-19337
OT antagonist 1 Cat. No.: HY-103650
OT antagonist 1 demethyl derivative Cat. No.: HY-103651
OT antagonist 3 Cat. No.: HY-103649
Oxytocin (α-Hypophamine; Oxytocic hormone) Cat. No.: HY-17571
Oxytocin acetate (α-Hypophamine acetate; Oxytocic hormone acetate) Cat. No.: HY-17571A
Pancreatin Cat. No.: HY-B2118
www.MedChemExpress.com 13
Purity: 99.58%Clinical Data: Phase 3Size: 10mM x 1mL in DMSO,
10 mg, 50 mg, 100 mg
Purity: >98%Clinical Data: Phase 3Size: 10 mg
Purity: 99.16%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
100 mg, 500 mg
Purity: 98.0%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
1 g, 5 g
Purity: 99.85%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg
Purity: >98%Clinical Data: No Development ReportedSize: 250 mg, 500 mg
Purity: >98%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
1 mg, 5 mg, 10 mg
Purity: 95.06%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
1 mg, 5 mg, 10 mg
Purity: >98%Clinical Data: LaunchedSize: 1 mg, 5 mg, 10 mg
Purity: 99.96%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
1 g
Bioactivity: Paroxypropione is a manufactured, nonsteroidal estrogen whichhas been used medically as an antigonadotropin.
Bioactivity: Pasireotide(SOM 230) is a stable cyclohexapeptide somatostatinmimic that exhibits unique high-affinity binding to humansomatostatin receptors (subtypes sst1/2/3/4/5,pKi=8.2/9.0/9.1/<7.0/9.9 respectively). IC50 value:8.2/9.0/9.1/<7.0/9.9(pKi, sst1/2/3/4/5) [1] in vitro:…
Bioactivity: Pasireotide (ditrifluoroacetate) is a stable cyclohexapeptidesomatostatin mimic that exhibits unique high-affinity bindingto human (subtypes sst1/2/3/4/5,somatostatin receptors
=8.2/9.0/9.1/<7.0/9.9, respectively).pKi
Bioactivity: Pasireotide(SOM 230) is a stable cyclohexapeptide somatostatinmimic that exhibits unique high-affinity binding to humansomatostatin receptors (subtypes sst1/2/3/4/5,pKi=8.2/9.0/9.1/<7.0/9.9 respectively). IC50 value:8.2/9.0/9.1/<7.0/9.9(pKi, sst1/2/3/4/5) [1] in vitro:…
Bioactivity: PCO371 is an orally active full agonist of parathyroid hormone, with no effect on PTH type 2 receptor.receptor 1 (PTHR1)
Bioactivity: PF-3274167 is a high-affinity nonpeptide oxytocin receptor(OTR) antagonist, with Ki of 9.5 nM. IC50 value: 9.5 nM [1]Target: oxytocin receptor (OTR)
Bioactivity: Prednisolone is a glucocorticoid with the general propertiesof the corticosteroids.
Bioactivity: Propylthiouracil(6-Propyl-2-thiouracil) is a thyroperoxidaseand 5'-deiodinase inhibitor.
Bioactivity: Protirelin is a highly conserved neuropeptide that exerts thehormonal control of thyroid-stimulating hormone (TSH) levelsas well as neuromodulatory functions.
Bioactivity: Protirelin Acetate is a highly conserved neuropeptide thatexerts the hormonal control of thyroid-stimulating hormone(TSH) levels as well as neuromodulatory functions.
Paroxypropione (4'-Hydroxypropiophenone) Cat. No.: HY-B1353
Pasireotide (SOM 230; SOM 320) Cat. No.: HY-16381
Pasireotide ditrifluoroacetate (SOM230 ditrifluoroacetate; Pasireotide TFA salt) Cat. No.: HY-79135
Pasireotide L-aspartate salt (SOM230 L-aspartate) Cat. No.: HY-79136
PCO371 Cat. No.: HY-100856
PF-3274167 (cligosiban) Cat. No.: HY-15023
Prednisolone Cat. No.: HY-17463
Propylthiouracil (6-n-Propylthiouracil; 6-Propyl-2-thiouracil; PTU) Cat. No.: HY-B0346
Protirelin (Synthetic thyrotropin-releasing factor; Synthetic
thyrotropin-releasing hormone; TRF; TRH; TSH-RF; …) Cat. No.: HY-P0002
Protirelin Acetate (TRF Acetate; TRH Acetate; TSH-RF Acetate) Cat. No.: HY-P0002A
Purity: >98%Clinical Data: No Development ReportedSize: 1 mg, 5 mg, 10 mg
Purity: >98%Clinical Data: No Development ReportedSize: 10 mg
Purity: 99.71%Clinical Data: Phase 4Size: 1 mg, 5 mg
Purity: 98.0%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
100 mg
Purity: 99.96%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
10 mg, 50 mg, 100 mg
Purity: 99.60%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 25 mg, 50 mg, 100 mg
Purity: 98.16%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
10 mg, 50 mg
Purity: 99.64%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
50 mg, 100 mg
Purity: 99.53%Clinical Data: Phase 1Size: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg
Purity: 99.59%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
100 mg, 500 mg
Bioactivity: Quinestrol is a synthetic estrogen, used in hormonereplacement therapy, and occasionally to treat breast cancerand prostate cancer
Bioactivity: RAD140 is a potent, orally bioavailable, nonsteroidalselective androgen receptor modulator (SARM).
Bioactivity: RaloxifeneHcl(LY156758 Hcl) is a second generation selectiveestrogen receptor antagonist. Target: Estrogen receptorApproved: September 14, 2007 Raloxifene activates TGF beta 3promoter as a full agonist at nanomolar concentrations, andraloxifene inhibits the estrogen response element-containing…
Bioactivity: RU 58841 is a specific androgen receptor antagonist oranti-androgen; RU 58841 has a dramatic effect on hairregrowth. IC50 value: Target: androgen receptor
Bioactivity: SecinH3 is an antagonist of with s of 5.4 μM,cytohesins IC502.4 μM, 5.4 μM, 5.6 μM, 5.6 μM and 65 μM for , ,hCyh1 hCyh2
, , and ,mCyh3 hCyh3 drosophila steppke yGea2-S7respectively.
Bioactivity: Silodosin (Rapaflo; KMD-3213) is an α1-adrenoceptor antagonistwith high uroselectivity; In treatment of dysuria.
Bioactivity: Sodium tauroglycocholate is an inhibitor of the biliary acidtransporting system of the hepatocyte and also a surfactantused as a chemical permeation enhancer.
Bioactivity: Somatostatin is a tetradecapeptide which can suppress thegrowth hormone (GH) secretion and control the pituitaryhormone secretion in human CNS. Sequence: H-Ala-Gly-Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Thr-Ser-Cys-OH(Disulfide bridge:Cys3-Cys14).
Bioactivity: Statine is an unusual amino acid that occurs twice in thesequence of pepstatin, a protease inhibitor that is activeagainst and other .pepsin acid proteases
Bioactivity: Substituted piperidines-1 is a compound that can promote therelease of growth hormone in humans and animals.
14 Tel: 609-228-6898 Fax: 609-228-5909 Email: [email protected]
Quinestrol (W-3566) Cat. No.: HY-B1012
RAD140 Cat. No.: HY-14383
Raloxifene hydrochloride (LY156758 hydrochloride) Cat. No.: HY-13738A
RU 58841 (PSK-3841; HMR-3841) Cat. No.: HY-10561
SecinH3 Cat. No.: HY-100559
Silodosin (KAD 3213; KMD 3213) Cat. No.: HY-10122
Sodium tauroglycocholate (Tauroglycocholic acid sodium salt) Cat. No.: HY-B2119
Somatostatin Cat. No.: HY-P0015
Statine ((3S,4S)-Statine; (S,S)-Statine) Cat. No.: HY-101877
Substituted piperidines-1 Cat. No.: HY-100305
www.MedChemExpress.com 15
Purity: >98%Clinical Data: No Development ReportedSize: 100 mg
Purity: 99.43%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg
Purity: 99.76%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
10 mg, 50 mg, 100 mg, 200 mg
Purity: 99.35%Clinical Data: Phase 3Size: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg
Purity: 99.87%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
10 mg, 50 mg
Purity: 98.02%Clinical Data: LaunchedSize: 100 mg
Purity: 99.85%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
100 mg
Purity: 98.99%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg
Purity: 99.97%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg, 100 mg
Purity: 98.64%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 25 mg, 50 mg, 100 mg
Bioactivity: Sufugolix (TAK-013) is a highly potent and orally availableluteinizing hormone-releasing hormone ( ) receptorLHRHantagonist with an of 0.1 nM.IC50
Bioactivity: TAK-438 is an orally active potassium-competitive acid which inhibits H , K -ATPase activity with an blocker + + IC50
of 19 nM.
Bioactivity: Tanaproget(NSP989) is a novel nonsteroidal progesteronereceptor agonist which can bind to the PR from various specieswith a higher relative affinity than reference steroidalprogestins.
Bioactivity: Terazosin Hydrochloride dihydrate is a selectivealpha1-antagonist used for treatment of symptoms of benignprostatic hyperplasia (BPH).
Bioactivity: Tiratricol is a thyroid hormone analog with hepatic, has beenused to suppress pituitary TSH secretion, with attenuation ofextrapituitary thyromimetic effects.
Bioactivity: Tolazamide is an oral blood glucose lowering drug used forpeople with Type 2 diabetes.
Bioactivity: Torcetrapib(CP-529414) is a CETP inhibitor with IC50 of 37 nM,elevates HDL-C and reduces nonHDL-C in plasma.
Bioactivity: Trilostane(Win 24540; Modrastane) is an inhibitor of 3β-hydroxysteroid dehydrogenase used in the treatment ofCushing's syndrome.
Bioactivity: Ulipristal (acetate) is a novel selective progesterone receptor for the treatment of benign gynecologicalmodulator (SPRM)
conditions such as uterine myoma.
Bioactivity: Vanitiolide is a choleretics.
Sufugolix (TAK-013) Cat. No.: HY-100209
TAK-438 (Vonoprazan Fumarate) Cat. No.: HY-15295
Tanaproget (NSP-989) Cat. No.: HY-15606
Terazosin hydrochloride dihydrate Cat. No.: HY-B0371A
Tiratricol (3,3',5-Triiodothyroacetic acid) Cat. No.: HY-B1201
Tolazamide (U-17835) Cat. No.: HY-B0920
Torcetrapib (CP-529414) Cat. No.: HY-12089
Trilostane (Win 24540) Cat. No.: HY-14281
Ulipristal acetate (CDB-2914) Cat. No.: HY-16508
Vanitiolide (Vanitiolid) Cat. No.: HY-B1034
Purity: 98.0%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
1 g, 5 g
Purity: 95.64%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
100 mg
Purity: 99.0%Clinical Data: No Development ReportedSize: 10mM x 1mL in DMSO,
5 mg, 10 mg, 50 mg
Purity: >98%Clinical Data: No Development ReportedSize: 1 mg, 5 mg, 10 mg, 20 mg
Purity: 99.33%Clinical Data: LaunchedSize: 10mM x 1mL in DMSO,
50 mg, 100 mg
Purity: >98%Clinical Data: LaunchedSize: 100 mg, 200 mg
Bioactivity: Vardenafil is a PDE5 inhibitor used for treating erectiledysfunction.
Bioactivity: TAK-438 (free base) is a novel P-CAB (potassium-competitiveacid blocker) that reversibly inhibits H+/K+ ATPase with IC50of 19 nM (pH 6.5), controls gastric acid secretion. IC50value: 19 nM [1] Target: H+/K+ ATPase in vitro: TAK-438 is apyrrole derivative with a chemical structure that is…
Bioactivity: YM-46303 is an antagonist which exhibits the highestmAChRaffinities for M1 and M3 receptors, and selectivity for M3over M2 receptor.
Bioactivity: Zaltidine(CP-57361) is a H2-receptor antagonist, which has theantisecretory action.
Bioactivity: β-Estradiol 17-acetate is a metabolite of estradiol. Bioactivity: β-estradiol 17-valerate (EV) is a synthetic estrogen widelyused in combination with other steroid hormones in hormonereplacement therapy drugs.
16 Tel: 609-228-6898 Fax: 609-228-5909 Email: [email protected]
Vardenafil Cat. No.: HY-B0442
Vonoprazan (TAK-438) Cat. No.: HY-100007
YM-46303 Cat. No.: HY-U00104
Zaltidine (CP-57361) Cat. No.: HY-15541
β-Estradiol 17-acetate (1,3,5(10)-Estratriene-3,17β-diol 17-acetate) Cat. No.: HY-B0708
β-Estradiol 17-valerate (Estradiol valerianate) Cat. No.: HY-B0672
