2017 EAB Members - Elsevier€¦ ·  · 2017-01-112017 EAB Members EAB Member Primary E-mail...

Preview:

Citation preview

2017 EAB Members

EAB Member Primary E-mail Address KeywordsAgrawal, Anjali anjali.agrawal@boehringer-ingelheim.com Calorimetry (DSC)

FormulationFormulation vehicleGlass transitionGranulationPolymeric drug delivery systemsPolymersSolid Dosage form TabletingWater in solidsWater sorptioncoating of solid dosage formextrusion spheronization

Ai, Hua huaai@scu.edu.cn BiocompatibilityBiodegradable polymersBiomaterialsControlled deliveryDrug deliveryImaging methodsMacromolecular drug deliverymagnetic resonance imagingMicelleMolecular ImagingMultidrug resistance-associated proteinsNanobiomaterialsNanoparticlesPolymeric drug delivery systems

Akita, Hidetaka akita@pharm.hokudai.ac.jp AntisenseBiodegradable polymersBiomaterialsCationic lipidsControlled deliveryControlled releaseDNA/oligonucleotide deliveryGene deliveryGene therapyIn situ hybridizationIntracellular traffickingsiRNA

Alvarez-Lorenzo, Carmen carmen.alvarez.lorenzo@usc.es BiomaterialsBiomimeticsCalorimetry (DSC)Controlled releaseCyclodextrinsGlass transitionMicelleMultidrug resistance transportersPolymeric biomaterialsPolymeric drug carrierResponsive delivery systemsThermal analysis

Alvarez-Nunez, Fernando faalvare@amgen.com AmorphousCrystal engineeringCrystalsCyclodextrinsDrug delivery systemsDrug targetingExtrusionGlass transitionGranulationLog PMaterials scienceMechanical propertiesNanotechnologyPoorly water-soluable drugsSolid StateSolid dispersionSolid dosage formSolubilitySurface chemistry

Amidon, Gregory geamidon@umich.edu CompactionDissolutionFormulationMechanical propertiesSolid dosage formtableting

2017 EAB Members

EAB Member Primary E-mail Address KeywordsAn, Guohua guohuaan@cop.ufl.edu ADME

Cancer chemotherapyIn vitro/in vivo correlations (IVIVC)Interspecies scalingLC-MSMultidrug resistancePharmacokinetic/pharmacodynamic modelsPharmacokinetics/pharmacodynamicsPopulation pharmacokineticsTransportersmembrane transporteroncology; drug metabolism;

Anchordoquy, Thomas J. tom.anchordoquy@ucdenver.edu AmorphousDNA deliveryliposomeslyophilizationMacromolecular drug deliveryNon-viral gene deliveryOligonucleotidesPhospholipidsPhysical stabilityPlasmid DNASolid state stabilityStabilityStabilization

Andrews, Gavin Paul g.andrews@qub.ac.uk Drug Delivery SystemsGelsPowder technologyRheologySolid dispersionSolid dosage formTabletingThermal analysisViscosity

Annaert, Pieter Pieter.Annaert@pharm.kuleuven.be ADMEBile acid transportersBiliary excretionCell cultureClearanceDrug interactionsHepatic transportHepatobiliary dispositionHepatocytesOrganic anion-transporting polypeptide transportersP-glycoproteinPediatricPermeabilityPharmacokineticsPreclinical pharmacokineticsTransportershepatocytespreclinical pharmacokinetics

Artursson, Per per.artursson@farmaci.uu.se ABC transportersActive transportADMECaco-2 cellsIntestinal absorptionMDCK cellsMucosal drug deliveryPermeabilityQSPR

Augustijns, Patrick F patrick.augustijns@pharm.kuleuven.be BiopharmacyCaco-2 usingDrug absorptionDrug transportEfflux CarriersIntestinal metabolism

Aungst, Bruce J. bruce.aungst@qps.com AbsorptionDrug transportEfflux pumpsEpithelial delivery/permeabilityFormulation vehicleGastrointestinal

2017 EAB Members

EAB Member Primary E-mail Address KeywordsAyala, Alejandro Pedro ayala@fisica.ufc.br Co-crystals

Crystal engineeringCrystal growthCrystal polymorphismCrystallographyInfrared spectroscopyMaterials scienceNear-infrared spectroscopyPhysicochemical propertiesPolymorphismPseudopolymorphismRaman spectroscopySolid stateThermal analysisX-ray powder diffractometry

Baertschi, Steve swbaertschi@aol.com Reactive oxygen speciesstabilitySolid state stabilityseparation sciencephotodegradationoxidationdegradation productsforced conditionsphoto chemistryDrug-excipient interaction

Bai, Jane jane.bai@fda.hhs.gov ApoptosisBiopharmaceutics classification system (BCS)Computational biologyDisease effectsDrug effectsDrug transportEpithelialGenetic polymorphismsGenomicsMathematical modelRegulatory science

Bak, Annette annette_bak@merck.com AbsorptionBioavailabilityBiopharmaceutics classification system (BCS)Chemical stabilityCo-crystalsCrystallinityPhysical stabilityPhysicochemical PropertiesPolymorphismPreformulationSolid stateTox formulations

Balthasar, Joseph P jb@buffalo.edu Cancer chemotherapyDrug targetingmonoclonal antibodiesPharamcokineticsPharmacodynamicsPharmacokinetics/pharmacodynamicsPhysiological modelPreclinical pharmacokinetics

Balu-Iyer, Sathy V svb@buffalo.edu Biophysical modelsBiotechnologyCircular dichroismFluorescence spectroscopyImmunologyLiposomesNanoparticlesPharmacokinetics/pharmacodynamicsProtein deliveryProtein formulation

Bann, James Jim.bann@wichita.edu Protein structureMembrane translocationProtein bindingProtein folding/refoldingProtein aggregationCircular dichroismVaccinesNMR spectroscopyPhysicochemical propertiesGlycosylation

2017 EAB Members

EAB Member Primary E-mail Address KeywordsBansal, Arvind K. akbansal@niper.ac.in Amorphous

Calorimetry (DSC)CompactionCrystal engineeringDrug-excipient interactionFormulationGlassGlass transitionMechanical propertiesMobilityOral drug deliveryPhysical stabilityPhysicochemical propertiesPolymorphismRelaxation timeSolid state

Bee, Jared S jaredsbee@gmail.com Analytical biochemistrybiopharmaceuticals characterizationBiotechnologyColloidFluorescence spectroscopyMicroparticlesNanoparticlesProtein aggregationProtein FormulationProtein structureProteinsStabilitySurface chemistry

Bergstrom, Christel ABC transportersAbsorptionSolubilityADMEBiopharmaceutics classification system (BCS)Caco-2 cellsComputational ADMEDissolution Dissolution rateDrug transport

Berkland, Cory berkland@ku.edu chemical engineeringDrug DeliverymicroparticlenanoparticlePLGA

Bernstein, Joel yoel@bgu.ac.il Crystal engineeringCrystal structureCrystallographycrystallographyCrystalsHydratehydrogen bondingPolymorphPolymorphismPseudopolymorphismSolid stateX-ray powder diffractometry

Bhatnagar, Bakul Bakul.bhatnagar@pfizer.com AmorphousCalorimetry (DSC)CrystallizationFreeze drying/lyophilizationFreeze-dryingGlass transitionLyophillization, frozen stateMaterials scienceMobilityPhase diagramPhysical characterizationPreformulationProtein formulationProtein stablizationSolid state stabilityThermal analysisX-ray powder diffractometry

2017 EAB Members

EAB Member Primary E-mail Address KeywordsBlaber, Michael Michael.blaber@med.fsu.edu Biotechnology

Calorimetry (DSC)CrystallographyProtein folding/refoldingProteinsPegylationProtein structurePhysical stabilityProteaseProtein aggregation

Boateng, Joshua Siaw J.S.Boateng@greenwich.ac.uk BuccalDrug delivery systemsFormulationFreeze drying/lyophilizationMacromolecular drug deliveryMucosal deliveryMucosal drug deliveryNovel Drug Delivery SystemsPeptide deliveryPharmaceutical FormulationPolymeric drug delivery systemsPreformulationProtein formulationProteomicsWound healing

Bogner, Robin robin.bogner@uconn.edu AmorphousDissolutiondrug releaseIsothermal calorimetryLyophilizationMechanical activationpharmaceutical manufacturing sciencePreformulationSolid dosage formSolubilitysolubility enhancementSupersaturation

Boyd, Ben ben.boyd@vcp.monash.edu.au ColloidColloid scienceLipidsNanoparticlesOral absorptionOral drug deliverySurfactants

Brodin, Birger birger.brodin@sund.ku.dk Blood brain barrierBlood-brain barrierABC transportersP-glycoproteinCaco-2 cells

Brouwer, Kenneth R. kennethbrouwer@qualyst.com ABC transportersAbsorptionADMEBile acid transportersBiliary recyclingBlood brain barrierBlood cerebrospinal fluid barrierCancerDispositionDrug interactionsDrug MetabolismDrug TransportPharmacokinetics

Buckner, Ira Shea buckneri@duq.edu AmorphousCalorimetryChemical stabilityCompactionCompressionHardnessMechanical activationMechanical propertiesPhysicochemical propertiesPowder technologySolid stateSolution calorimetryThermodynamicscalorimetry

2017 EAB Members

EAB Member Primary E-mail Address KeywordsButler, James james.m.butler@gsk.com Dissolution

BCSSolid dispersionOral absorption

Byrn, Stephen sbyrn@pharmacy.purdue.edu AmorphousCrystallizationCrystallographyCrystalsDesolvationDissolutionPolymorphPolymorphismSolid stateSolid state NMRsolid state chemistry

Caira, Mino R. Mino.Caira@uct.ac.za cyclodextrin inclusionPolymorphismPseudopolymorphismSolid state chemistry of drugsThermal analysisx-ray diffraction

Caramella, Carla M. carla.caramella@unipv.it dissolution and bioavailabilityhydrophilic matrix tabletshydrophilic polymer characterizationin vivo- in vitro correlationMicromeriticsmucoadhesion and mucoadhesive systemspharmaceutics/biopharmaceuticsrheology of semisolidstransmucosal delivery

Chadwick, Jennifer S. Analytical biochemistryAnalytical ultra-centrifugationEnzymesMolecular modelingMutationnmrNMR spectroscopyOxidationPhysical stabilityProtein bindingprotein stabilityProtein structure

Chaudhuri, Bodhisattwa bodhi.chaudhuri@uconn.edu Ab initio calculationsAerosolsBlood flowCFDCompactionDEMDryingExcipientsIn silico modelingIontophoresisMathematical modelNeural networksNot AgreeProcess Modeling

Chen, Xiaodong xiaodong.chen@bms.com BilayerBiophysical modelsComputational AnalysisLyophilizationMaterials scienceMathematical modelMechanical EngineeringMechanical propertiesPulmonary drug deliveryPulmonary systemSimulationsTabletingThermodynamics

Cheng, Wei chengwe@umich.edu Analytical ultra-centrifugationEnzyme kineticsEnzymologyFluorescence spectroscopyHIV/AIDSKineticsProtein aggregationProtein bindingprotein stability.

2017 EAB Members

EAB Member Primary E-mail Address KeywordsCheng, Woei Ping w.p.cheng3@herts.ac.uk Macromolecular drug delivery

NanoparticlesNanotechnologyNon-viral gene deliveryOral drug deliveryPeptide deliveryPolymeric biomaterialsPolymeric drug delivery systemsPoorly water-soluable drugsProtein deliverydrug deliverynanotechnologypolymer drug delivery systemssiRNA

Chiang, Po-Chang Chiang.pochang@gene.com ADMEAbsorptionAbsorption potentialBio-analyticalBioavailabilityFormulationFormulation vehicleGastrointestinal transitOral absorptionPharamcokineticsPhysical characterizationPhysicochemical propertiesPreclinical pharmacokineticsPreformulation

Coker, Adeola O. grillo@uiwtx.edu BiotechnologyCircular dichroismFTIRFluorescence spectroscopyBiotechnology, Formulation DevelopmentProtein aggregationProtein folding/refoldingProtein formulationProtein structure

Craig, Duncan d.craig@uea.ac.uk Drug deliveryMaterials SciencePolymeric drug delivery systemsPolymorphismSolid dispersionSolid stateThermal analysis

Crowe, John jhcrowe@ucdavis.edu Freeze-dryingLiposomesProteinsStabilizationsugarstrehalosewater replacement theory

Darrington, Richard Todd todd.darrington@boehringer-ingelheim.com Biopharmaceutics classification system (BCS)Blood brain barrierBlood-brain barrierChemical stabilityCo-crystalsCompactionComplexationControlled deliveryControlled releaseCyclodextrinsPhysical Pharmaceutics

Dave, Rutesh Hemant rutesh.dave@liu.edu BuccalCoatingColonic drug deliveryControlled releaseDissolutionDissolution rateFactorial designFormulationIn vitro modelsMicromeriticsOral drug deliveryPhysicochemical propertiesPowder technologyPreformulationSolid dispersionSolid dosage formTablet

2017 EAB Members

EAB Member Primary E-mail Address KeywordsDave, Vivek S viveksdave@gmail.com Compaction

CompressionControlled releaseDissolutionDissolution rateDrug delivery systemsExcipientsFormulationGranulation

Davies, Martyn martyn.davies@nottingham.ac.uk Biodegradable polymersBiomaterialsControlled deliveryDrug DeliveryImaging methodsMacromolecular drug deliveryMaterials scienceNanotechnologyPhysical characterizationPolymeric drug delivery systemsSurface chemistrySurface propertiescharaceterisation of dosage forms

de Jong, Henk J. henkdejong@orange.fr Analytical chemistryBioanalysisChromatographyCyclodextrinsExcipientsHPLC (high-performance/pressure liquid chromatography)Hydrates/solvatesNasal drug deliveryPreformulationRegulatory science

De Villiers, Melgardt M. mmdevilliers@pharmacy.wisc.edu CalorimetryChemical stabilityCrystal polymorphismDendrimersDissolutionFormulationNanocapsulesNanoparticlesNanospheresNanotechnologyPolymorphismPowder technologySolid dosage formSolubility

Deferme, Sven sven.deferme@pharmaxl.net ABC transportersAbsorptionAbsorption enhancerActive transportADMECaco-2 cellsCytochrome P450Drug resistanceDrug transportIn vitro/in vivo correlations (IVIVC)

Deguchi, Yoshiharu deguchi@pharm.teikyo-u.ac.jp biopharmaceuticsBlood brain barrierblood-brain barrier transportMembrane transportMembrane transporterMicrodialysisPeptide deliveryPharmacokinetics

DePaz, Roberto depazr@medimmune.com LyophilizationProtein FormulationProtein aggregationProtein formulationProteinsStabilizationVaccinesViral vectorsbiopharmaceuticals characterization

Derendorf, Hartmut hartmut@cop.ufl.edu BioavailabilityClinical pharmacokineticspharmacodynamicsPharmacokinetic/pharmacodynamic modelspharmacokinetics

2017 EAB Members

EAB Member Primary E-mail Address KeywordsDiNunzio, James C. james.dinunzio@merck.com Amorphous

BioavailabilityCoatingCompressionControlled releaseDissolutionExtrusionFluid-bedGlass transition

Dressman, Jennifer dressman@em.uni-frankfurt.de BioequivalenceBiopharmaceutics classification system (BCS)DissolutionFood effectsIn vitro/in vivo correlations (IVIVC)Oral absorption

Dufès, Christine c.dufes@strath.ac.uk Blood brain barrierBrain deliveryCNSCancerCancer chemotherapyCancer therapyControlled deliveryDNA/oligonucleotide deliveryDendrimersDrug delivery systemsDrug targetingGene therapyNanotechnologyNon-viral gene deliveryTargeted drug delivery

Elder, David David.P.Elder@gsk.com AbsorptionAlginateAlkylatorsAmorphousAnalysisAnalytical chemistryBioavailabilityBioequivalenceBiopharmaceutics classification system (BCS)Blood brain barrierGenotoxic Impurities/degradantsSolid state (version/form)

Etzler, Frank M fetzler@lecom.edu Calorimetry (DSC)ColloidCompactionContact anglesFormulationMaterials scienceParticle sizePhysical characterizationPhysicochemical propertiesPorosityPowder technologyPulmonary drug deliveryQuality by design (QBD)Surface chemistry

Fattal, Elias elias.fattal@u-psud.fr Colonic drug deliveryDNA/oligonucleotide deliveryDrug DeliveryGene deliveryLipoplexesLiposomesMicroparticlesNanoparticlesNanotechnologiesPeptide deliveryPoly(lactic/glycolic) acid (PLGA or PLA)Pulmonary delivery/absorption

Finnin, Barrie C. barrie.finnin@vcp.monash.edu.au Absorption enhancerBuccalSkinTransdermal drug deliverytransdermal drug delivery

Fisher, Mark Mfisher1@kumc.edu Protein aggregationprotein foldingProtein stabilizationprotein unfoldingprotein-protein interactions

2017 EAB Members

EAB Member Primary E-mail Address KeywordsFoppoli, Anastasia Dissolution rate

Thermal analysisSolid state stabilityPsuedopolymorphismPolymorphismExcipients

Gamble, John john.gamble@bms.com CompactionExcipientsFormulationGranulationIGCImage analysisMaterial scienceMaterials scienceMorphologyPATParticle sizePhysical characterization

Gokarn, Yatin R. yatin_gokarn@yahoo.com Analytical ultra-centrifugationBiophysical modelsBiotechnologyNanoparticlesPegylationPreformulationProtein aggregationProtein folding/refoldingProtein formulationViscositybiopharmaceuticals characterization

Goldfarb, David J. david.goldfarb@merck.com compressionEncapsulationfluid-bedformulationgranulationMechanical propertiesparticle sizePowder technologyrheologySemi-solids

Gonda, Igor gondai@aradigm.com AerosolsDrug DeliveryInhalationLiposomesLung metabolismMacromolecular drug deliveryNasal absorptionNasal drug deliveryPeptide deliveryPulmonaryPulmonary delivery/absorptionPulmonary drug deliveryTransdermal

Goteti, Kosalaram gotetik@medimmune.com ClearanceIn vitro/in vivo correlationsMathematical modelPharmacokinetic/pharmacodynamic modelsPharmacokineticsPharmacokinetics/pharmacodynamicsPhysiological modelPreclinical pharmacokineticsSimulationsTissue partition

Green, Henrik henrik.green@liu.se ABC transportersCYP enzymesClinical PharmacologyDrug metabolizing enzymesDrug transportLiquid chromatographyMass spectrometryPharamcokineticsPharmacogeneticsPharmacogenomics

Guy, Richard H. r.h.guy@bath.ac.uk Iontophoresisnoninvasive clinical monitoringpermeation enhancementskin absorptiontransdermal deliverytransdermal drug delivery

2017 EAB Members

EAB Member Primary E-mail Address KeywordsHadgraft, Jonathan jonathan.hadgraft@btinternet.com Drug delivery systems

enhancersIn vitro modelsskin penetrationTransdermal

Hammarlund-Udenaes, Margareta mhu@farmbio.uu.se ABC transportersADMEBlood-brain barrierCNSDrug transportPharmacodynamicsPharmacokineticsPharmacokinetics/pharmacodynamicsPreclinical pharmacokineticsTransporters

Harris, David david.harris@spcorp.com AerosolsBuccalGastrointestinal transitMucosal drug deliveryOral absorptionPermeation enhancersPulmonary drug deliveryScintigraphySemi-solids

Hauss, David J David.hauss@rcn.com AbsorptionAbsorption enhancerAbsorption potentialBioavailabilityBiopharmaceuticsBiotechnologyControlled deliveryControlled releaseDrug DeliveryDrug delivery systemsGene deliveryLipids

He, Yan yan.he2@sanofi.com Acid-base equilibriaCyclodextrinsDrug-like propertiesMicellePhysicochemical propertiesPoorly water-soluable drugsPrecipitationPreformulationSolubilitySurfactants

Heng, Jerry Yong Yew jerry.heng@imperial.ac.uk AerosolsCrystal polymorphismCrystallizationMaterials scienceNucleationPhysical characterizationPhysicochemical propertiesPowder technologySurface energyWetting and contact angleparticle characterizationparticle engineeringsurface properties

Heng, Paul W.S. phapaulh@nus.edu.sg CoatingDissolution rateDrug delivery systemsFluid-bedGranulationPharmaceutical technologyPhysical characterizationSolid dosage formTabletcontrolled drug delivery systemsmiroencapsulationpelletisatisationpercutaneous delivery

2017 EAB Members

EAB Member Primary E-mail Address KeywordsHickey, Anthony J. ahickey@rti.org Aerosols

AntiinfectivesColloidHygroscopicityMicroparticlesMucosal immunizationParticle sizePowder technologyPulmonary delivery/absorptionPulmonary drug delivery

Higaki, Kazutaka higaki@pharm.okayama-u.ac.jp ADMEAbsorptionAbsorption enhancerAgreeBioavailabilityCaco-2 cellsDissolutionGastrointestinal transitIn vitro/in vivo correlations (IVIVC)Intestinal absorptionIntestinal secretion/transportMicroemulsionOral drug deliveryPharmacokineticsSelf-emulsifyingbiopharmaceutics

Hook, Sarah cell cultureformulationgene deliveryimmunologyliposomes

Hosoya, Ken-ichi hosoyak@pha.u-toyama.ac.jp barrier transportBlood-brain barrierblood-ocular barrierefflux transportocular drug deliverytransporter

Hussain, Munir A. munir.hussain@bms.com Degradation productsDrug delivery systemsDrug-excipient interactionFormulationPreformulation

Inoue, Katsuhisa kinoue@toyaku.ac.jp AbsorptionExcretion

High throughput technologies

Membrane transport

Transporters

membrane transport

molecular Pharmaceutics

pharmacokinetics

Ishida, Tatsuhiro ishida@tokushima-u.ac.jp Cancer chemotherapyCationic lipidsControlled deliveryControlled releaseDNA/oligonucleotide deliveryDrug delivery systemsDrug targetingEncapsulationGene deliveryGene therapydrug delivery system

Ito, Kousei ABC transportersLiver ABC transporterbiliaryHepatobiliary dispositionLactationTransportersToxicityToxicologyImmune ResponseHepatocytesbile acid tansporters

2017 EAB Members

EAB Member Primary E-mail Address KeywordsIwao, Yasunori yasuiwao@u-shizuoka-ken.ac.jp ADME

AbsorptionAlbuminAntioxidantsBiodegradable polymersCalorimetry (DSC)ClearanceColonControlled releaseDiffusionPharmaceutics

Izutsu, Ken-ichi izutsu@nihs.go.jp AmorphousCrystallizationFormulationFreeze drying/lyophilizationProtein formulation

Jiskoot, Wim w.jiskoot@lacdr.leidenuniv.nl biopharmaceuticals characterizationBiotechnologyLiposomesMucosal immunizationMucosal vaccinationProtein aggregationProtein deliveryProtein formulationprotein immunogenicityVaccine adjuvantsVaccine delivery

Johnson, Kevin C. kjohnson29@snet.net Absorptionabsorption rate constantdissolution, content uniformity, computer simulationGITSModellingnifedipinePharmacokineticsPrecipitationsimulationwater absorption

Jones Braun, LaToya Latoya.JonesBraun@ucdenver.edu 2-dimensional gel electrophoresisFormulationPhysical stabilityPreformulationProtein aggregationProtein formulationSurfactantsVaccine adjuvantsVaccine deliveryVaccines

Jones, David Simon d.jones@qub.ac.uk BiomaterialsExtrusionGelsHydrogelsMaterials sciencePolymersRelaxation timeSemi-solidsThermal analysisViscosity

Joubert, Marisa K mjoubert@amgen.com BiotechnologyFTIRIgG antibodyImmune ResponseIn vitro modelsParticle sizeProtein aggregationProtein structureProteinsbiopharmaceuticals characterization

Kalonia, Devendra S. kalonia@uconn.edu Peptide degradationpeptide oxidationProtein aggregationProtein BiophysicsProtein Characterizationprotein excipient interactionsProtein formulationprotein unfolding

2017 EAB Members

EAB Member Primary E-mail Address KeywordsKasting, Gerald B. Gerald.Kasting@uc.edu Diffusion

IontophoresisIsothermal calorimetryMathematical modelPercutaneousPermeabilityPhysicochemical propertiesSkinskin permeabilitytransdermal deliveryTransdermal drug deliveryWater sorption

Kato, Yukio ykato@p.kanazawa-u.ac.jp ABC transportersActive transportCell biologyDrug transportHepatic transportMembrane transportOrganic anion transporters (OAT)Organic cation transporters (OCT)PharmacokineticsTransporters

Kerwin, Bruce A bkerwin@amgen.com Analytical biochemistryBiotechnologyDeamidationExcipientsFTIRFluorescence spectroscopyFormulationHPLC (high-performance/pressure liquid chromatography)Liquid chromatographyMacromolecular prodrugsProtein formulation, structure, biochemistry

Kesisoglou, Filippos filippos_kesisoglou@merck.com ADMEAbsorptionAbsorption ModelingBioavailabilityBiopharmaceuticsBiopharmaceutics classification system (BCS)IVIVCIn silico modelingIn vitro/in vivo correlations (IVIVC)Intestinal absorptionPharamcokinetics

Khutoryanskiy, Vitaliy v.khutoryanskiy@reading.ac.uk ChitosanColloidComplexationDNA deliveryHydrogelsMucosal drug deliveryNanoparticlesPharmaceuticsPolyelectrolytesPolymer chemistryPolymer-biopolymer interactionsPolymeric biomaterials

Kleinebudde, Peter kleinebudde@uni-duesseldorf.de coating processextrusion/ spheronisationmicrocrystalline cellulosepelletsroll compactionsolid dosage forms

Knipp, Gregory T gknipp@purdue.edu ADMEAbsorptionActive transportBioavailabilityBlood brain barrierCaco-2 cellsCell cultureDrug transportEpithelial delivery/permeabilityFatty acid transport and regulationGastrointestinalPeptide TransportersPlacental Transort

2017 EAB Members

EAB Member Primary E-mail Address KeywordsKobayashi, Kaoru kaoruk@faculty.chiba-u.jp drug metabolism

ADME

cytochrome P50

nuclear receptor

drug-drug interaction

humanized animal

Koe, Janet G. koejanet@gmail.com BiotechnologyLipoplexesLiposomesNon-viral gene deliveryPhysical characterizationPhysical stabilityPhysicochemical propertiesPlasmid DNAStabilityTargeted drug delivery

Kubo, Yoshiyuki ABC transportersMembrane transportMembrane transporterBlood brain barriersolute transportersOrganic cation transporters (OCT)Intestinal absorptionRenal absorption

Kumru, Ozan S. okumru@ku.edu FormulationParticle sizePhysical stabilityProtein aggregationPreformulationProtein folding/refoldingproteinsvaccines

Kusuhara, Hiroyuki kusuhara@mol.f.u-tokyo.ac.jp ABC transportersBlood-brain barrierBlood-CSF barrierbraineffluxkidneyorganic anionpharmacokineticsRenal clearanceRenal excretiontransporter

Lai, Yurong laiyurong@gmail.com pharmacokineticsmembrane transporter

metabolism

hepatic clearance

hepatobiliary disposition

drug interactions

bioavailability

ABC transporters

bile acid tansporters

in vitro/in vivo correlation

Lambert, William J lambertw@medimmune.com Chemical stabilityFormulationFreeze drying/lyophilizationKineticsLiposomesPeptide deliverypharmaceuticsProtein deliveryProtein formulationSolubility

Landis, Margaret Sue margaret.s.landis@pfizer.com Chemical stabilityExcipientsNasal absorptionNasal drug deliveryOrganic chemistryPermeation enhancersPhotochemistryProdrugsSolid dosage formSolid state stabilityStabilityphotochemistry

2017 EAB Members

EAB Member Primary E-mail Address KeywordsLane, Majella E majella.lane@btinternet.com Biophysical models

Dermal deliveryDrug transportGastrointestinalSkinTransdermalTransdermal deliveryTransdermal drug delivery

Langer, Robert drug delivery systemsLaw, Devalina Amorphous

Polymorphismcrystal engineeringOral drug deliverydrug-like propertiestabletingPhysicochemical propertiessolid dispersionsalts/salt selectionPolymeric drug delivery systems

Lechuga-Ballesteros, David dlechuga@pearltherapeutics.com Co-crystalsCrystal engineeringinhalation technologyLiposomesNanotechnologypreformulationSolid dispersionSolid statesolid state characterizationSolid state stabilitySpray dryingSupercritical fluidsSurface chemistry

Loftsson, Thorsteinn thorstlo@hi.is ComplexationCyclodextrinsInclusion compoundsInclusionsPermeabilitySolubilityStability

Mach, Henryk henryk_mach@merck.com analytical ultracentrifugationvaccine stabilityUVderivative spectroscopyprotein deliveryProtein formulation

Maeda, Kazuya kmaeda@mol.f.u-tokyo.ac.jp transportersdrug interactionsgenetic polymorphismspharmacokinetic/pharmacodynamic modelsin vitro/in vivo correlations (IVIVC)hepatic transport

Mahler, Hanns-Christian hanns-christian.mahler@roche.com BiotechnologyCalorimetryCircular dichroismDrug deliveryFTIRFormulationFreeze drying/lyophilizationFreeze-dryingProtein aggregationProtein formulationProteinsSterile manufacturing

2017 EAB Members

EAB Member Primary E-mail Address KeywordsMansour, Heidi M. mansour@pharmacy.arizona.edu Aerosols

ColloidControlled releaseLiposomesNanotechnologyNot AgreePhospholipidsPulmonaryPulmonary drug deliverySurface chemistryWater sorption

Marini, Amedeo amedeo.marini@unipv.it CalorimetryCalorimetry (DSC)Chemical stabilityCo-crystalsco-crystals preparation and characterizationCrystal polymorphismCrystallinityCyclodextrinsDehydrationdrug - eccipient interactionsDrug interactionsdrug-excipient compatibility studiesFTIRGlass transitionHydrates/solvatesInclusion compoundsInfrared spectroscopyInteractionIsothermal calorimetryKineticsMaterials sciencePhysical Chemistryphysico-chemical characterization of drugsphysico-chemical characterization of solid statePhysicochemical propertiesPolymorphismSolid State ReactionsX-ray powder diffractometry

Maroni, Alessandra alessandra.maroni@unimi.it Oral drug deliverydrug delivery systems

Marsac, Patrick patrick.marsac@uky.edu AbsorptionAmorphousCalorimetryImage AnalysisRaman SpectroscopySolid State NMRSolubilitySpray dryingSpray freeze-dryingThermodynamics

Maruyama, Toru tomaru@gpo.kumamoto-u.ac.jp albuminalpha-1-acidglycoproteinantioxidantsprotein deliveryprotein structureprotein folding/refoldingprotein bindingreactive oxygen speciestargeted drug deliverycontrolled delivery

Maurin, Michael B. mmaurin30@gmail.com AbsorptionAnalysisBioavailabilityCalorimetry (DSC)Chemical stabilityComplexationControlled deliveryFormulationPhysicochemical propertiesSolubility

2017 EAB Members

EAB Member Primary E-mail Address KeywordsMcAllister, Mark mark.mcallister@pfizer.com Bioavailability

Biopharmaceutics classification system (BCS)DissolutionDrug delivery systemsIntestinal absorptionOral absorptionOral drug deliveryPreformulationSite-specific absorptionExtrusion

McGeorge, Gary gary.mcgeorge@bms.com FTIRImage analysisImaging methodsInfrared spectroscopyMultivariate analysisNear-infrared spectroscopyPATpolymorphismPrincipal component analysisRaman spectroscopySolid state NMRSpectroscopy

McNamara, Patrick pmcnamar@email.uky.edu DistributionDrug transportEfflux pumpsLactationMembrane transportMembrane transporterParacellular transportPharmacokineticsProtein bindingTransporters

Medlicott, Natalie natalie.medlicott@otago.ac.nz Macromolecular drug deliveryPrincipal component analysisPharmacokineticsProtein aggregationProtein formulationSpectroscopyChromatographyDrug-excipient interactionClinical PharmacokineticsInfrared spectroscopy

Miller, Danforth dan.miller@novartis.com AerosolsAmorphousAmorphous MaterialsCalorimetryChemometricsGlass transitionMoisture sorptionPharmaceuticsPhysical characterizationPhysical stabilityPolymorphPowder technologyPulmonaryRelaxationRelaxation timeSolid stateSolid-state pharmaceuticsSpectroscopySpray dryingX-ray powder diffractometry

Moeschwitzer, Jan info@janmoeschwitzer.de Absorption enhancerbiopharmaceuticals characterizationBlood brain barrierCrystal engineeringDissolutionDrug delivery systemsDrug NanocrystalsNanotechnologyParticle sizePoorly Soluble DrugsSolid dispersionSpray freeze-drying

Morris, Marilyn Emily memorris@buffalo.edu Hepatobiliary dispositionMonocarboxylate transportersMultidrug resistance transportersRenal clearanceRenal reabsorption

2017 EAB Members

EAB Member Primary E-mail Address KeywordsMüllertz, Anette amu@farma.ku.dk Absorption

AdsorptionBilayerBioequivalenceBiopharmaceutics classification system (BCS)Biophysical modelsCaco-2 cellsIn vitro/in vivo correlations (IVIVC)Light scattering (dynamic)Lipidspoorly soluble drugspredictive in vitro models

Munson, Eric J. eric.munson@uky.edu AmorphousAnalytical chemistryBiodegradable polymersCo-crystalsCrystallinityExcipientsHydrates/solvatesMobilityNMR spectroscopyPhysical characterization

Murthy, Narasimha S murthy@olemiss.edu ElectroporationIontophoresisMicrodialysisMicrospheresMucosal drug deliveryNanoparticlesNasal drug deliveryTransdermal drug delivery

Nail, Steven L steven_nail@baxter.com AmorphousCalorimetry (DSC)DryingFreeze drying/lyophilizationFreezing/Freeze-DryingGlass transitionMaterials sciencePharmaceutical Technology - ParenteralPhysical stabilityThermal AnalysisThermal analysis

Nakajima, Miki nmiki@p.kanazawa-u.ac.jp Cytochrome P450Drug metabolizing enzymesGenetic polymorphismsGlucuronosyltransferases (UGT)Metabolism

Nakanishi, Takeo nakanish@p.kanazawa-u.ac.jp ABC transporters5-Aminolevulinic AcidADMEToxicityDrug resistanceDrug transportAbsorptionDrug interactionsTransportersOrganic anion-transporting polypeptide transporters

Nangia, Ashwini ashwini.nangia@gmail.com ClathratesCo-crystalsCrystal engineeringCrystal structureCrystallizationHydrates/solvatesInclusion compoundsPolymorphPseudopolymorphThermal analysis

Narhi, Linda O. lnarhi@amgen.com aggregationBiophysical characterization of proteinsCalorimetry (DSC)Circular dichroismFluorescence spectroscopyFTIRLight scattering (dynamic)nonconformance investigationsProtein aggregationProtein folding/refoldingRaman spectroscopyStability

2017 EAB Members

EAB Member Primary E-mail Address KeywordsNebuloni, Marino Nebu.mari@yahoo.it Analytical chemistry

CalorimetryCrystal structurePhysical characterizationParticle sizesolid dosage formsPolymorphismThermal analysisX-ray powder diffractometry

Newman, Ann ann@seventhstreetdev.com AmorphousCo-crystalsCrystallinityCrystalsDesolvationHydrates/SolvatesPolymorphismPhysicochemical propertiesPhysical characterization

Nicolazzo, Joseph Anthony joseph.nicolazzo@monash.edu Absorption enhancerAlzheimer's diseaseBlood brain barrierBlood cerebrospinal fluid barrierblood-brain barrierBuccalbuccal mucosal drug deliveryCell cultureCNSDrug transportEfflux pumpsEpithelial delivery/permeabilityMembrane transporter

Nielson, Hanne Morck Hanne.morck@sund.ku.dk AbsorptionBiodegradable polymersBiophysical modelsProtein formulationCell culturePeptide deliveryDrug transportEncapsulationMucosal drug deliveryLipoplexes

Ogawa, Noriko noriko30@dpc.agu.ac.jp CyclodextrinsInclusion compoundsPoorly water-soluable drugsSolid dispersionSpray dryingforumulationspoorly water-soluable drugs

Ogihara, Takuo togihara@takasaki-u.ac.jp AbsorptionADMEABC transportersTransportersCaco-2 cellsBlood brain barrierEfflux pumpsP-glycoproteinPharmacokinetics/pharmacodynamicsMultidrug resistance

Ohtake, Satoshi satoshi.ohtake@pfizer.com AntiinfectivesBilayerDryingExcipientsFormulationFreeze-dryingGlassProcessingProtein formulationSolid stateVaccines

2017 EAB Members

EAB Member Primary E-mail Address KeywordsOhtsuki, Sumio sohtsuki@ohtsuki-lab.jp ABC transporters

Blood brain barrierBlood cerebrospinal fluid barrierBlood-CSF barrierBrain BarrierCell biologyEfflux pumpsEndothelialMass spectrometryMembrane transportMembrane transporterTransporter

Okuda, Tomoyuki tokuda@meijo-u.ac.jp AerosolsFreeze drying/lyophilizationLiposomesNon-viral gene deliveryPowder technologyPulmonary delivery/absorptionPulmonary drug deliverySpray dryingSpray freeze-dryingsiRNA

Okura, Takashi okura@pharm.teikyo-u.ac.jp blood-brain barrierblood-CSF barrierpharmacodynamicspharmacokinetics/pharmacodynamicsmembrane transporterstransporters

Ozeki, Tetsuya ozekit@phar.nagoya-cu.ac.jp Drug delivery systemsGene deliveryLipoplexesLiposomesNanoparticlesOral absorptionPowder TechnologyPowder technologyPulmonary delivery/absorptionWater-insoluble drugs

Panyam, Jayanth jpanyam@umn.edu BiomaterialsDNA/oligonucleotide deliveryDrug DeliveryDrug resistanceGene therapyIntracellular traffickingLocal deliveryMicroparticlesNanoparticlesNanotechnologyrestenosisSustained Release

Pauletti, Giovanni gm.pauletti@uc.edu Cell CultureDrug TransportPharmacokineticsProdrugs

Perrie, Yvonne y.perrie@aston.ac.uk Gene deliveryGene therapyGene vectorsdrug deliveryLiposomesVaccine deliveryVaccines

Pikal, Michael J. michael.pikal@uconn.edu AmorphousCalorimetry (DSC)CrystallinityFreeze drying/lyophilizationGlass transitionIsothermal calorimetryMobilityProtein aggregationSolid state stability

Porter, Christopher J.H. chris.porter@monash.edu ADMEAbsorptionDrug deliveryintestinal permeabilityLipid based drug delivery systemsLymphatic transport

2017 EAB Members

EAB Member Primary E-mail Address KeywordsPrankerd, Richard Richard.Prankerd@pharm.monash.edu.au Analytical chemistry

CalorimetryChemical stabilityCrystal structureDissolutionFormulationHydrates/solvatesLight-scatteringPhysicochemical propertiesSpectroscopy

Qian, Feng AmorphousFormulationSolid dispersionMaterials scienceOral drug deliveryPeptide deliveryPolymeric biomaterialsPolymeric drug delivery systems

Rajewski, Roger A rajewski@ku.edu ComplexationCyclodextrinsFreeze drying/lyophilizationPharamcokineticsPharmacodynamics

Randolph, Theodore W. theodore.randolph@colorado.edu Biodegradable polymersNanoparticlesProtein aggregationProtein folding/refoldingProtein formulationSpray dryingStabilityStabilizationThermodynamics

Rantanen, Jukka jukka.rantanen@sund.ku.dk CrystallizationDehydrationPolymorphismprocess analytical technology (PAT)ProcessingSolid statesolid state propertiesSolid state stabilitySolvateSpectroscopyspectroscopy (near infrared NIR & Raman)Water in solidsX-ray powder diffractometry

Reutzel-Edens, Susan M. reutzel@lilly.com Calorimetry (DSC)PolymorphismSolid stateSolid state NMRSolvateSpectroscopyStructure-property relationship (SPR)Water in solidsWater sorptionX-ray powder diffractometry

Rice, Kevin G. kevin-rice@uiowa.edu DNAGlycoproteinGlycoproteins/glycoprotein receptorsGlycosylationMacromolecular drug deliveryOligonucleotidesPegylationPeptidesPlasmid DNATargeted drug delivery

Roberts, Christopher Glass transitionMolecular modelingProtein aggregationProtein folding/refoldingProtein formulationstabilitythermodynamics/statistical mechanics

Rodríguez-Hornedo, Naír nrh@umich.edu ClathratesCo-crystalsCrystal engineeringCrystal shapeCrystallizationHydrates/solvatesPolymorphism

2017 EAB Members

EAB Member Primary E-mail Address KeywordsRogge, Mark mark.rogge1@biogenidec.com ADME

AbsorptionBiopharmaceuticsBiotechnologyClinical pharmacokineticsCYP enzymesDistributionDrug effectsDrug interactionsEliminationFood interactionsPharmacokinetics

Rosenberg, Amy amy.rosenberg@fda.hhs.gov BiotechnologyEnzymesGlycosylationImmunologyImmunology/Immunogenicity of Therapeutic ProteinsProtein aggregationProteinsVaccines

Rumondor, Alfred rumondor@gmail.com AmorphousFormulationPhysical stabilityPoorly water-soluable drugsPreformulationSolid dispersion

Sahajwalla, Chandra chandrahas.sahajwalla@fda.hhs.gov ADMEAbsorptionActive transportBiliary excretionBioavailabilityBioequivalenceBiopharmaceutics classification system (BCS)CNSClearanceClinical pharmacokinetics

SAI, YOSHIMICHI sai-ys@staff.kanazawa-u.ac.jp Intestinal secretion/transportMembrane TransportMembrane transportOral absorptionPeptide transportersSolute transportersTranscellular transportTransporters

Sampath Kumar, Krishnan Krishnan.Sampathkumar@hospira.com FormulationBiotechnologyFreeze drying/lyophilizationStabilizationHPLC (high-performance/pressure liquid chromatography)FTIRChemical stabilityProtein aggregationProtein formulationProteins

Sandler, Niklas niklas.sandler@abo.fi Fluid-bedImage analysisMechanical activationMechanical propertiesMoisture sorptionNeural networksPartial least squaresParticle sizePhysical characterizationRoller Compactionparticle and bulk characterisationpowder technology and related processingsolid-state characterisation

Sandri, Giuseppina Absorption enhancerbiocompatibilityCell Culturewound healingbuccalMucosal drug deliveryBiomaterialsPermeation enhancersPolymeric drug delivery systemsEpithelial delivery/permeability

2017 EAB Members

EAB Member Primary E-mail Address KeywordsSasaki, Hitoshi sasaki@net.nagasaki-u.ac.jp Clinical pharmacokinetics

Controlled deliveryDrug targetingGene deliveryIndividualized drug therapyMucosal deliveryPharmacokinetics/pharmacodynamicsPolymeric drug delivery systemsProdrugsTransdermal drug delivery

Schöneich, Christian schoneic@ku.edu antioxidantFree radicalsOxidationproteinSolid stateStability

Serajuddin, Abu T. M. serajuda@stjohns.edu AbsorptionBioavailabilityChemical stabilityControlled releaseDissolutionLipids; Solid Dispersion; Amorphous Drug SubstancesMicroemulsionPhysicochemical propertiesPreformulationSolid dispersionSolubility

Shen, Danny D. ds@u.washington.edu ABC transportersMetabolismMonocarboxylate transportersMultidrug resistance transportersOrganic anion transporters (OAT)PharmacokineticsPharmacokinetics/pharmacodynamicsPhase I metabolismPreclinical pharmacokineticsTransporters

Siahaan, Teruna J. siahaan@ku.edu adheren junctionsCadherinCell adhesionCell adhesion proteins and peptidesdrug deliveryDrug TargetingICAMIntercellular JunctionsLFA-1PeptidesProdrugsProteins

Singh, Satish Kumar satish.singh@pfizer.com AggregationBiophysical modelsCalorimetryCircular dichroismColloidColloidsGlass transitionProtein aggregationProtein binding

Protein delivery

Protein folding/refolding

Protein structure

Proteins

Souillac, Pierre Olivier pierre_souillac@eisai.com Calorimetry (DSC)

Circular dichroism

FTIR

Fluorescence spectroscopy

Formulation

Freeze drying/lyophilization

Polymorphism

Preformulation

Protein aggregation

Protein formulation

2017 EAB Members

EAB Member Primary E-mail Address KeywordsSpencer, David spencerd@medimmune.com Analytical biochemistry

Deamidation

Glycoprotein

Glycosaminoglycans

Glycosylation

IgG antibody

Liquid chromatography

Mass spectrometry

Oxidation

Physicochemical properties

Protein characterization

Proteins

biopharmaceuticals characterization

Stella, Valentino J. stella@ku.edu Chemical stability

Cyclodextrins

Kinetics

Macromolecular prodrugs

Physical stability

Prodrugs

Solubility

Stability

Stephenson, Gregory A Stephenson_Gregory_A@lilly.com Crystal structure

Crystallization

Crystallography

Solid state

Solid state NMR

solid state NMR

solid-state chemistry

Solubility

Spectroscopy

X-ray powder diffractometry

Stinchcomb, Audra L astinchc@rx.umaryland.edu Epithelial delivery/permeability

HPLC (high-performance/pressure liquid chromatography)

In vitro/in vivo correlations (IVIVC)

Nasal absorption

Nasal drug delivery

Near-infrared spectroscopy

Percutaneous

Prodrugs

topical

Transdermal

Transdermal drug delivery

Straubinger, Robert M. rms@buffalo.edu Liposomes

drug delivery

gene arrays

liposomes, drug delivery, gene arrays

Pharmacogenomics

Strickley, Robert rstrickley@gilead.com Formulation

Solid state stability

Kinetics

Injectables

Pediatric

Oral drug delivery

Physical stability

Physicochemical properties

Preformulation

Prodrugs

Sun, Changquan Calvin sunx0053@umn.edu Amorphous

Co-crystals

Compaction

Crystal engineering

Crystallization

Formulation

Granulation

Materials science

Polymorphism

Solid-state characterization, powder flow and compaction

Solubility

Tablet formulation

2017 EAB Members

EAB Member Primary E-mail Address KeywordsSuryanarayanan, Raj surya001@umn.edu Co-crystals

Crystal engineering

Crystallinity

Crystals

Desolvation

Dissolution

Dissolution rate

Formulation

Freeze drying/lyophilization

Freeze-drying

Tachikawa, Masanori tachikaw@m.tohoku.ac.jp ABC transporters

Active transport

Barrier

Blood-CSF barrier

Blood-brain barrier

Brain

CNS

Cell biology

Cerebrospinal fluid

Tachikawa, Masanori tachikaw@m.tohoku.ac.jp Choroid plexus

Drug transport

Endothelial

Transporter

Taft, David R. dtaft@liu.edu Erythrocyte distribution

pharmacokinetics

Pharmacokinetics

Preclinical pharmacokinetics

Renal excretion

Renal transport

Takano, Mikihisa takanom@hiroshima-u.ac.jp Biopharmaceutics

Intestinal absorption

Intestinal secretion/transport

Membrane transport

Membrane transporter

P-glycoprotein

Renal transport

Tam, Yun K. ytam@sinoveda.com Absorption

Clearance

Drug Metabolism

Food interactions

Hepatic metabolism

Intestinal absorption

Intestinal metabolism

Natural products

Oral absorption

Pharamcokinetics

Pharmacokinetic/pharmacodynamic models

Pharmacokinetics

Tamai, Ikumi tamai@p.kanazawa-u.ac.jp Absorption

biliary elimination

Blood-brain barrier

membrane transport

Membrane transport

Renal excretion

transporter

Taylor, Lynne S lstaylor@purdue.edu Amorphous

Bioavailability

Calorimetry (DSC)

Crystallinity

Crystallization

Hydrates/solvates

Infrared spectroscopy

Moisture sorption

Physical stability

Polymorphism

Raman spectroscopy

2017 EAB Members

EAB Member Primary E-mail Address KeywordsTempleton, Allen allen_templeton@merck.com Analytical chemistry

Bioavailability

Biopharmaceutics classification system (BCS)

Chemical stability

Chromatography

Co-crystals

Drug stability

Oxidation

Pharmaceutical analysis

Photodegradation

Physical characterization

Preformulation

Thakker, Dhiren R. dhiren_thakker@unc.edu Absorption

Absorption enhancer

Blood brain barrier

Caco-2 cells

Clinical pharmacokinetics

Cytochrome P450

Drug interactions

Drug Metabolism

Drug metabolizing enzymes

Theil, Frank-Peter theilfdrk@gmail.com Modeling & Simulation

Monte Carlo

PBPK

PKPD

Pharmacodynamics

Pharmacokinetic/pharmacodynamic models

Pharmacokinetics

Pharmacokinetics/pharmacodynamics

Physiological model

Population pharmacokinetics

Population pharmacokinetics/pharmacodynamics

Preclinical pharmacokinetics

Simulations

Tobyn, Mike mike.tobyn@bms.com Inhaler

aerosol

dry powder

excipient

microcrystalline cellulose

tablet

Tomi, Masatoshi tomi-ms@pha.keio.ac.jp placenta

pregnancy

drug transport

membrane transporter

ophthalmic drug delivery

disposition

blood brain barrier

pharmacokinetics

Torchilin, Vladimir v.torchilin@neu.edu Drug delivery systems

micelle

liposomes

Drug Targeting

cancer

cancer immunology

imaging agents

Tsutsumi, Yasuo ytsutsumi@phs.osaka-u.ac.jp DDS

DNA delivery

Drug transport

Polymeric drug carrier

Polymeric drug delivery systems

Polymeric drugs

Protein delivery

Protein structure

Proteomics

Toxicity

Toxicology

drug delivery

2017 EAB Members

EAB Member Primary E-mail Address KeywordsUchiyama, Susumu suchi@bio.eng.osaka-u.ac.jp Physicochemical properties

Analytical ultra-centrifugation

biopharmaceuticals characterization

Calorimetry

Protein formulation

Chromatin

Formulation

Hydration

Particle size

Mass spectrometry

Van Speybroeck, Michiel michiel.vanspeybroeck@formacpharma.com AdsorptionBio-ceramicsBioavailabilityDesorptionDissolutionFormulationIn vitro/in vivo correlations (IVIVC)LipidsMesoporous silica SBA-15

Physical characterization

Physical stability

Poor solubility

Silica

Solid dosage form

Solubility

Supersaturation

Surface chemistry

van de Weert, Marco marco.vandeweert@sund.ku.dk Calorimetry (DSC)

Circular dichroism

FTIR

Fluorescence spectroscopy

Follow-on biologics

Freeze drying/lyophilization

Pegylation

Polymeric drug delivery systems

Protein aggregation

Protein delivery

Van den Mooter, Guy guy.vandenmooter@pharm.kuleuven.be Calorimetry (DSC)

Physical characterization

physical pharmacy

Physicochemical

Polymorphism

preformulation

Solid dispersion

Supersaturation

Verreck, Geert gverreck@its.jnj.com Amorphous

Controlled release

Extrusion

Glass

melt extrusion

Nanotechnology

Oral drug delivery

Solid dispersion

Spray drying

Supercritical fluids

Supersaturation

Vert, Michel vertm@univ-montp1.fr Biodegradable polymers

Controlled delivery

Drug targeting

Hydrogels

Macromolecular prodrugs

Poly(lactic/glycolic) acid (PLGA or PLA)

Polymeric biomaterials

Polymeric drug delivery systems

Tissue engineering

2017 EAB Members

EAB Member Primary E-mail Address KeywordsVolkin, David B volkin@ku.edu Analytical biochemistry

Biotechnology

Deamidation

Formulation

Freeze drying/lyophilization

Oxidation

Protein delivery

Protein folding/refolding

Solubility

Vaccines

Wahlstrom, Dr. Jan janw@amgen.com ADME

CYP enzymes

Cytochrome P450

Drug Metabolism

Drug interactions

Drug metabolizing enzymes

Glucuronosyltransferases (UGT)

Metabolism

Pharmacokinetics

Phase I metabolism

Phase II metabolism

Warne, Nicholas Nicholas.warne@pfizer.com Freeze drying/lyophilization

Lyophilization

Protein aggregation

Protein Delivery

Protein formulation

Proteins

Wiedmann, Timothy S. wiedm001@umn.edu AbsorptionColloid

Diffusion

Hydrogels

Lipids

Micelle

Monolayer

NMR spectroscopy

Pulmonary drug delivery

Surfactants

Williams, Adrian C. a.c.williams@reading.ac.uk Amorphouspermeation

Raman spectroscopy

Skin

Topical

Transdermal

Transdermal drug delivery / solid state pharmaceuticals

Williams, Desmond B Des.Williams@unisa.edu.au ADME

Absorption

Acid-base equilibria

Analytical chemistry

Bioavailability

Biopharmaceutics classification system (BCS)

Chemical stability

Controlled release

Drug delivery systems

Food effects

Gastrointestinal

Intestinal absorption

Oral drug delivery

Pharmaceutics

Pharmacokinetics

Physicochemical properties

Poorly water-soluable drugs

Prodrugs

pH

Winter, Gerhard gerhard.winter@lrz.uni-muenchen.de biologicals, proteinsControlled release

Drug delivery systems

freeze drying

lyophilisation, protein stability,

Protein formulation

Proteins

2017 EAB Members

EAB Member Primary E-mail Address KeywordsYalkowsky, Samuel H. yalkowsky@pharmacy.arizona.edu Solubility

melting point

physical properties

Yamamoto, Akira yamamoto@mb.kyoto-phu.ac.jp Absorption enhancer

Colonic drug delivery

Intestinal absorption

Intestinal secretion/transport

Mucosal drug delivery

P-glycoprotein

Paracellular transport

Peptide delivery

Pulmonary delivery/ absorption

Tight junction

Yamashita, Fumiyoshi yama@pharm.kyoto-u.ac.jp biophysical models

computational ADME

drug-like properties

in silico modeling

mathematical model

multivariate analysis

pharmacokinetic/pharmacodynamic models

physiological model

QSPR

structure-property relationship (SPR)

Yamashita, Shinji shinji@pharm.setsunan.ac.jp Caco-2 cells

Computational ADME

Drug transport

In vitro/in vivo correlations (IVIVC)

Intestinal absorption

Membrane transport

Oral absorption

Oral drug delivery

Paracellular transport

Permeability

Yamazaki, Hiroshi hyamazak@ac.shoyaku.ac.jp Cytochrome P450Enzyme kinetics

Flavin monooxygenases (FMO)

Genetic polymorphisms

Hepatic metabolism

Metabolism

Microsomes

Pharmacogenetics

Phase I enzyme

Toxicology

Yang, Jian jyang74@jhmi.edu Cancer ChemotherapyChromatography

combinatorial chemistry

drug design

Drug targeting

NMR spectroscopy

Non-viral gene delivery

Polymeric drug delivery systems

structure-activity relationship (SAR)

Yazdanian, Mehran mehran.yazdanian@tevapharm.com Bioavailability

Biopharmaceutics classification system (BCS)

Caco-2 cells

Drug transport

Drug-like properties

Efflux pumps

Passive diffusion/transport

Permeability

Physicochemical properties

Preformulation

Solubility

Stability

Transport

Yoshinari, Kouichi yoshinari@m.tohoku.ac.jp Cytochrome P450

Sulfotransferases (ST)

2017 EAB Members

EAB Member Primary E-mail Address KeywordsYuasa, Hiroaki yuasa@phar.nagoya-cu.ac.jp Bioavailability

First-pass metabolism

Gastrointestinal transit

Intestinal absorption

Intestinal metabolism

Intestinal secretion/transport

Oral absorption

Oral drug delivery

Zeitler, Axel jaz22@cam.ac.uk THz

Terahertz

Amorphous

Crystal defects

Crystallinity

Dehydration

Infrared spectroscopy

Polymorphism

Raman spectroscopy

Solid state

Zema, Lucia lucia.zema@unimi.it ExtrusionColonic drug delivery

Drug delivery systems

Granulation

Oral drug delivery

Zentner, Gaylen M. gaylen.zentner@gmail.com Biodegradable polymersCoating

Colloid

Controlled delivery

Controlled release

Diffusion

Hydrogels

Microparticles

Microspheres

Osmotic pumps

Zhang, Ming mzhang25@buffalo.edu Drug interactionsNonlinear pharmacokineticsPharamcokinetics

Pharmacodynamics

Pharmacokinetic/pharmacodynamic models

Pharmacokinetics

Pharmacokinetics/pahrmacodynamics

Population pharmacokinetics

Population pharmacokinetics/pharmacodynamics

Preclinical pharmacokinetics

ZHOU, QI (Tony) qi.zhou@sydney.edu.au Aerosols

Coating

Materials science

Microparticles

Physical characterization

Physicochemical properties

Powder technology

Pulmonary drug delivery

Spray drying

Surface chemistry

aerosol

powder technology

Zimmerman, Cheryl L zimme005@umn.edu ADME

Bioavailability

Cancer chemoprevention

drug metabolism

Drug metabolizing enzymes

Hepatic clearance

Intestinal absorption

Intestinal metabolism

Metabolite kinetics

Oral absorption

Pharamcokinetics

Population pharmacokinetics/pharmacodynamics