1
2008 Indole derivatives R 0140 Microwave-Assisted Synthesis of Tetrahydroindoles. — Aminolysis of carboxylic acid (I) gives the desired heterocyclic skeleton; however, in all cases the carboxylic group is lost. Protection as methyl ester or amide function is not successful. — (PIRAS, L.; GHIRON, C.; MINETTO, G.; TADDEI*, M.; Tetrahedron Lett. 49 (2008) 3, 459-462; Dip. Farm. Chim. Tecnol., Univ. Siena, I-53100 Siena, Italy; Eng.) — Mais 18- 106

ChemInform Abstract: Microwave-Assisted Synthesis of Tetrahydroindoles

Embed Size (px)

Citation preview

2008

Indole derivativesR 0140 Microwave-Assisted Synthesis of Tetrahydroindoles. — Aminolysis of carboxylic

acid (I) gives the desired heterocyclic skeleton; however, in all cases the carboxylic group is lost. Protection as methyl ester or amide function is not successful. — (PIRAS, L.; GHIRON, C.; MINETTO, G.; TADDEI*, M.; Tetrahedron Lett. 49 (2008) 3, 459-462; Dip. Farm. Chim. Tecnol., Univ. Siena, I-53100 Siena, Italy; Eng.) — Mais

18- 106